7-[[(11R)-3-chloro-6-methyl-5,5-dioxo-11H-benzo[c][2,1]benzothiazepin-11-yl]amino]heptanoic acid
Title | Journal |
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Changes in the cannabinoids receptors in rats following treatment with antidepressants. | Neurotoxicology 20171201 |
Both cholestatic and steatotic drugs trigger extensive alterations in the mRNA level of biliary transporters in rat hepatocytes: Application to develop new predictive biomarkers for early drug development. | Toxicology letters 20161130 |
Advantageous use of HepaRG cells for the screening and mechanistic study of drug-induced steatosis. | Toxicology and applied pharmacology 20160701 |
Synthetic and Receptor Signaling Explorations of the Mitragyna Alkaloids: Mitragynine as an Atypical Molecular Framework for Opioid Receptor Modulators. | Journal of the American Chemical Society 20160601 |
A simple transcriptomic signature able to predict drug-induced hepatic steatosis. | Archives of toxicology 20140401 |
Chronic antidepressant treatment impairs the acquisition of fear extinction. | Biological psychiatry 20130601 |
Chronic social defeat stress model: behavioral features, antidepressant action, and interaction with biological risk factors. | Psychopharmacology 20121101 |
The same antidepressant elicits contrasting patterns of synaptic changes in the amygdala vs hippocampus. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20121101 |
Antidepressants for depression in stage 3-5 chronic kidney disease: a systematic review of pharmacokinetics, efficacy and safety with recommendations by European Renal Best Practice (ERBP). | Nephrology, dialysis, transplantation : official publication of the European Dialysis and Transplant Association - European Renal Association 20121001 |
Anxiety- rather than depression-like behavior is associated with adult neurogenesis in a female mouse model of higher trait anxiety- and comorbid depression-like behavior. | Translational psychiatry 20121001 |
In vitro inhibition of mitochondrial respiratory rate by antidepressants. | Toxicology letters 20120918 |
Outpatient treatment of children and adolescents with antidepressants in Croatia. | International journal of psychiatry in clinical practice 20120901 |
Tianeptine vs amitriptyline for the treatment of irritable bowel syndrome with diarrhea: a multicenter, open-label, non-inferiority, randomized controlled study. | Neurogastroenterology and motility : the official journal of the European Gastrointestinal Motility Society 20120901 |
Sildenafil, a phosphodiesterase type 5 inhibitor, enhances the activity of two atypical antidepressant drugs, mianserin and tianeptine, in the forced swim test in mice. | Progress in neuro-psychopharmacology & biological psychiatry 20120807 |
The effect of pH on polymorph formation of the pharmaceutically active compound tianeptine. | International journal of pharmaceutics 20120801 |
Tianeptine treatment induces antidepressive-like effects and alters BDNF and energy metabolism in the brain of rats. | Behavioural brain research 20120801 |
Tianeptine's effects on spontaneous and Ca2+-induced uterine smooth muscle contraction. | Acta physiologica Hungarica 20120601 |
Tianeptine: more cases of dependence. | Prescrire international 20120501 |
The antinociceptive effects of intravenous tianeptine in colorectal distension-induced visceral pain in rats: the role of 5-HT₃ receptors. | European journal of pharmacology 20120415 |
Assessment of abuse of tianeptine from a reimbursement database using 'doctor-shopping' as an indicator. | Fundamental & clinical pharmacology 20120401 |
Factors influencing the choice of antidepressants: a study of antidepressant prescribing practice at University Psychiatric Clinic in Belgrade. | Vojnosanitetski pregled 20120401 |
Tricyclic antidepressants for autism spectrum disorders (ASD) in children and adolescents. | The Cochrane database of systematic reviews 20120314 |
The analgesic activity of intrathecal tianeptine, an atypical antidepressant, in a rat model of inflammatory pain. | Anesthesia and analgesia 20120301 |
Usefulness of LDAEP to predict tolerability to SSRIs in major depressive disorder: a case report. | Psychiatry investigation 20120301 |
Emotional memory impairments in a genetic rat model of depression: involvement of 5-HT/MEK/Arc signaling in restoration. | Molecular psychiatry 20120201 |
Chronic fluoxetine treatment in middle-aged rats induces changes in the expression of plasticity-related molecules and in neurogenesis. | BMC neuroscience 20120101 |
Stress leads to contrasting effects on the levels of brain derived neurotrophic factor in the hippocampus and amygdala. | PloS one 20120101 |
Dynamic regulation of NMDAR function in the adult brain by the stress hormone corticosterone. | Frontiers in cellular neuroscience 20120101 |
Restraint Stress Intensifies Interstitial K(+) Accumulation during Severe Hypoxia. | Frontiers in pharmacology 20120101 |
GluA1 phosphorylation alters evoked firing pattern in vivo. | Neural plasticity 20120101 |
Treatment-resistant depression: therapeutic trends, challenges, and future directions. | Patient preference and adherence 20120101 |
Stress-induced changes of hippocampal NMDA receptors: modulation by duloxetine treatment. | PloS one 20120101 |
Preclinical and clinical evidence of antioxidant effects of antidepressant agents: implications for the pathophysiology of major depressive disorder. | Oxidative medicine and cellular longevity 20120101 |
Tianeptine in combination with monoamine oxidase inhibitors for major depressive disorder. | BMJ case reports 20120101 |
Tianeptine reverses stress-induced asymmetrical hippocampal volume and N-acetylaspartate loss in rats: an in vivo study. | Psychiatry research 20111230 |
Tianeptine potentiates AMPA receptors by activating CaMKII and PKA via the p38, p42/44 MAPK and JNK pathways. | Neurochemistry international 20111201 |
Translating clinical findings into knowledge in drug safety evaluation--drug induced liver injury prediction system (DILIps). | PLoS computational biology 20111201 |
Efficacy of antidepressants for late-life depression: a meta-analysis and meta-regression of placebo-controlled randomized trials. | The Journal of clinical psychiatry 20111201 |
Neurotrophins role in depression neurobiology: a review of basic and clinical evidence. | Current neuropharmacology 20111201 |
cGMP Signaling, Phosphodiesterases and Major Depressive Disorder. | Current neuropharmacology 20111201 |
The protective effect of tianeptine on Gp120-induced apoptosis in astroglial cells: role of GS and NOS, and NF-κB suppression. | British journal of pharmacology 20111101 |
Epidemiological characterization of drug overconsumption: the example of antidepressants. | Journal of addictive diseases 20111001 |
[Depressive disorder, treatment and sexual dysfunction--part II]. | Polski merkuriusz lekarski : organ Polskiego Towarzystwa Lekarskiego 20111001 |
Effect of tianeptine on cognitive functions in patients with depressive disorders during a 3-month observation. | Psychiatria Danubina 20110901 |
Tianeptine in the combined treatment of combat related posttraumatic stress disorder. | Psychiatria Danubina 20110901 |
Antidepressant prescribing patterns in Korea: results from the clinical research center for depression study. | Psychiatry investigation 20110901 |
Absence of psychostimulant effects of a supratherapeutic dose of tianeptine: a placebo-controlled study versus methylphenidate in young healthy volunteers. | Journal of clinical psychopharmacology 20110801 |
[Evaluation of the influence of tianeptine on the psychosomatic status of patients with ulcerative colitis in remission]. | Polski merkuriusz lekarski : organ Polskiego Towarzystwa Lekarskiego 20110801 |
Collapsin response mediator protein-2: an emerging pathologic feature and therapeutic target for neurodisease indications. | Molecular neurobiology 20110601 |
Effects of tryptophan depletion and tryptophan loading on the affective response to high-dose CO2 challenge in healthy volunteers. | Psychopharmacology 20110601 |
Baseline lipid levels and acute treatment response to paroxetine and tianeptine in depressed women. | Journal of clinical psychopharmacology 20110601 |
Biomarkers in development of psychotropic drugs. | Dialogues in clinical neuroscience 20110601 |
Fluoxetine Up-Regulates Bcl-xL Expression in Rat C6 Glioma Cells. | Psychiatry investigation 20110601 |
Efficacy of antidepressants for dysthymia: a meta-analysis of placebo-controlled randomized trials. | The Journal of clinical psychiatry 20110401 |
Importance of neuroplasticity changes in mood disorder. | The Journal of the American Osteopathic Association 20110401 |
Effect of quercetin on lipopolysaccharide induced-sickness behavior and oxidative stress in rats. | Indian journal of pharmacology 20110401 |
Duloxetine-related panic attacks. | Psychiatria Danubina 20110301 |
Tablet potency of Tianeptine in coated tablets by near infrared spectroscopy: model optimisation, calibration transfer and confidence intervals. | Journal of pharmaceutical and biomedical analysis 20110220 |
The effects of antidepressants on mitochondrial function in a model cell system and isolated mitochondria. | Neurochemical research 20110201 |
Does personality disorder co-morbidity impact treatment outcome for patients with major depression? A multi-level analysis. | Journal of personality disorders 20110201 |
Psychotropic medication use among elderly nursing home residents in Slovenia: cross-sectional study. | Croatian medical journal 20110201 |
Systemic chemical desensitization of peptidergic sensory neurons with resiniferatoxin inhibits experimental periodontitis. | The open dentistry journal 20110101 |
Necessity of hippocampal neurogenesis for the therapeutic action of antidepressants in adult nonhuman primates. | PloS one 20110101 |
Activation of mitogen-activated protein kinase in descending pain modulatory system. | Journal of signal transduction 20110101 |
One universal common endpoint in mouse models of amyotrophic lateral sclerosis. | PloS one 20110101 |
Modulation of cortisol responses to the DEX/CRH test by polymorphisms of the interleukin-1beta gene in healthy adults. | Behavioral and brain functions : BBF 20110101 |
Influence of Pre-Training Predator Stress on the Expression of c-fos mRNA in the Hippocampus, Amygdala, and Striatum Following Long-Term Spatial Memory Retrieval. | Frontiers in behavioral neuroscience 20110101 |
Diffusion-weighted MRI and quantitative biophysical modeling of hippocampal neurite loss in chronic stress. | PloS one 20110101 |
Development and validation of stability indicating method for determination of sertraline following ICH guidlines and its determination in pharmaceuticals and biological fluids. | Chemistry Central journal 20110101 |
Lithium monotherapy increases ACTH and cortisol response in the DEX/CRH test in unipolar depressed subjects. A study with 30 treatment-naive patients. | PloS one 20110101 |
Chronic stress induces sex-specific alterations in methylation and expression of corticotropin-releasing factor gene in the rat. | PloS one 20110101 |
NMDA and AMPA receptors are involved in the antidepressant-like activity of tianeptine in the forced swim test in mice. | Pharmacological reports : PR 20110101 |
Neurosteroids reduce social isolation-induced behavioral deficits: a proposed link with neurosteroid-mediated upregulation of BDNF expression. | Frontiers in endocrinology 20110101 |
A predictive ligand-based Bayesian model for human drug-induced liver injury. | Drug metabolism and disposition: the biological fate of chemicals 20101201 |
Amitriptyline and tianeptine poisoning treated by naloxone. | Human & experimental toxicology 20100901 |
Formulation of a novel tianeptine sodium orodispersible film. | AAPS PharmSciTech 20100901 |
Tianeptine reduces morphine antinociceptive tolerance and physical dependence. | Behavioural pharmacology 20100901 |
Acute effects of serotonergic antidepressants on tryptophan metabolism and corticosterone levels in rats. | Pakistan journal of pharmaceutical sciences 20100701 |
Computational analysis of the impact of chronic stress on intrinsic and synaptic excitability in the hippocampus. | Journal of neurophysiology 20100601 |
The decrease in JNK- and p38-MAP kinase activity is accompanied by the enhancement of PP2A phosphate level in the brain of prenatally stressed rats. | Journal of physiology and pharmacology : an official journal of the Polish Physiological Society 20100401 |
The neurobiological properties of tianeptine (Stablon): from monoamine hypothesis to glutamatergic modulation. | Molecular psychiatry 20100301 |
Tianeptine may be a therapeutic option for Tourette's syndrome. | Contemporary clinical trials 20100301 |
[Effects of amitriptyline, fluoxetine, and tianeptine on the content of monoamines and their metabolites in Wistar rat brain structures]. | Eksperimental'naia i klinicheskaia farmakologiia 20100301 |
Neurotrophic effects of tianeptine on hippocampal neurons: a proteomic approach. | Journal of proteome research 20100205 |
Knockdown of brain-derived neurotrophic factor in specific brain sites precipitates behaviors associated with depression and reduces neurogenesis. | Molecular psychiatry 20100101 |
Interaction of the human plasma membrane monoamine transporter (hPMAT) with antidepressants and antipsychotics. | Naunyn-Schmiedeberg's archives of pharmacology 20100101 |
Antidepressants are a rational complementary therapy for the treatment of Alzheimer's disease. | Molecular neurodegeneration 20100101 |
Effect of venlafaxine on bone loss associated with ligature-induced periodontitis in Wistar rats. | Journal of negative results in biomedicine 20100101 |
Activities of respiratory chain complexes and citrate synthase influenced by pharmacologically different antidepressants and mood stabilizers. | Neuro endocrinology letters 20100101 |
Adherence to antidepressant therapy for major depressive patients in a psychiatric hospital in Thailand. | BMC psychiatry 20100101 |
Innovative approaches to treatment - refractory depression: The ketamine story. | Indian journal of psychiatry 20100101 |
Role of paliperidone extended-release in treatment of schizoaffective disorder. | Neuropsychiatric disease and treatment 20100101 |
A new strategy for antidepressant prescription. | Frontiers in neuroscience 20100101 |
Acute stress induces contrasting changes in AMPA receptor subunit phosphorylation within the prefrontal cortex, amygdala and hippocampus. | PloS one 20100101 |
Inhibition of monoamine oxidase activity by antidepressants and mood stabilizers. | Neuro endocrinology letters 20100101 |
Neural pathways in allergic inflammation. | Journal of allergy 20100101 |
[Affective disorders in acute myocardial infarction and possibilities of their correction with tianeptin]. | Terapevticheskii arkhiv 20100101 |
[Antiviral therapy in a patient with chronic hepatitis C, metabolic syndrome and interferon-induced depression]. | Klinicheskaia meditsina 20100101 |
Chronic stress effects on hippocampal structure and synaptic function: relevance for depression and normalization by anti-glucocorticoid treatment. | Frontiers in synaptic neuroscience 20100101 |
Anorexia nervosa depends on adrenal sympathetic hyperactivity: opposite neuroautonomic profile of hyperinsulinism syndrome. | Diabetes, metabolic syndrome and obesity : targets and therapy 20100101 |
Research on antidepressants in India. | Indian journal of psychiatry 20100101 |
Addictive potential of Tianeptine - the threatening reality. | Georgian medical news 20090901 |
The neurotrophic and neuroprotective effects of psychotropic agents. | Dialogues in clinical neuroscience 20090901 |
Re-exposure to endotoxin induces differential cytokine gene expression in the rat hypothalamus and spleen. | Brain, behavior, and immunity 20090801 |
Comparative study on the gastroprotective potential of some antidepressants in indomethacin-induced ulcer in rats. | Chemico-biological interactions 20090715 |
The effect of antidepressant drugs on the HPA axis activity, glucocorticoid receptor level and FKBP51 concentration in prenatally stressed rats. | Psychoneuroendocrinology 20090701 |
Comparison of antidepressant effects of azafan, tianeptine, and paroxetine. | Bulletin of experimental biology and medicine 20090701 |
Effect of a single dose of citalopram on amygdala response to emotional faces. | The British journal of psychiatry : the journal of mental science 20090601 |
Efficacy, tolerability and safety of tianeptine in special populations of depressive patients. | Psychiatria Danubina 20090601 |
Antidepressant action of tianeptine is connected with acceleration of serotonin turnover in the synapse: a hypothesis. | Neuropsychopharmacologia Hungarica : a Magyar Pszichofarmakologiai Egyesulet lapja = official journal of the Hungarian Association of Psychopharmacology 20090601 |
Different effects of tianeptine pretreatment in rats exposed to acute stress and repeated severe stress. | Methods and findings in experimental and clinical pharmacology 20090401 |
Protective effects of melatonin against oxidative stress in Fmr1 knockout mice: a therapeutic research model for the fragile X syndrome. | Journal of pineal research 20090301 |
Antidepressants reverse the attenuation of the neurotrophic MEK/MAPK cascade in frontal cortex by elevated platform stress; reversal of effects on LTP is associated with GluA1 phosphorylation. | Neuropharmacology 20090101 |
Use of Coaxil (tianeptine) in elderly patients with combined mild cognitive and depressive-anxiety disorders. | Neuroscience and behavioral physiology 20090101 |
[Myocardial infarction and depression: clinical-functional relationships and possibilities of correction of left ventricular remodeling with antidepressant tianeptine]. | Kardiologiia 20090101 |
The combined dexamethasone/CRH Test (DEX/CRH test) and prediction of acute treatment response in major depression. | PloS one 20090101 |
Stress and depression: preclinical research and clinical implications. | PloS one 20090101 |
[Experience of application of tianeptine in anxiety-depressive disorders comorbid with climacteric syndrome]. | Kardiologiia 20090101 |
Impaired interleukin-1beta and c-Fos expression in the hippocampus is associated with a spatial memory deficit in P2X(7) receptor-deficient mice. | PloS one 20090101 |
5-hydroxytryptamine modulates migration, cytokine and chemokine release and T-cell priming capacity of dendritic cells in vitro and in vivo. | PloS one 20090101 |
[Changes in the brain neuroplasticity at the stress background and its correction in cardiological patients]. | Kardiologiia 20090101 |
[Misuse of substances theoretically without abuse potential--case series]. | Przeglad lekarski 20090101 |
Prenatal stress decreases glycogen synthase kinase-3 phosphorylation in the rat frontal cortex. | Pharmacological reports : PR 20090101 |
[Dynamics of depressive disorders, endothelial dysfunction, and phagocytic activity of neutrophils in patients with chronic inflammation under influence of treatment with tianeptine]. | Kardiologiia 20090101 |
Tianeptine influence on plasmatic catecholamine levels and anxiety index in rats under variable chronic stress after early maternal separation. | The International journal of neuroscience 20090101 |
[Current views on the pathogenesis of depression and approaches to antidepressive therapy (in case of coaxil)]. | Terapevticheskii arkhiv 20090101 |
Possible Role of Platelet GluR1 Receptors in Comorbid Depression and Cardiovascular Disease. | Cardiovascular psychiatry and neurology 20090101 |
Tianeptine treating narcolepsy. Case report. | Neuro endocrinology letters 20090101 |
[Peptic ulcer in patients with neurotic and affective disorders: comorbidity, clinicoendoscopic and psychopathological features, approaches to therapy]. | Terapevticheskii arkhiv 20090101 |
New approaches to the pharmacological management of major depressive disorder. | Advances in pharmacology (San Diego, Calif.) 20090101 |
[The clinical picture and treatment of depression spectrum disorders in patients with cardiovascular disease]. | Terapevticheskii arkhiv 20090101 |
Amantadine reduces glucagon and enhances insulin secretion throughout the oral glucose tolerance test: central plus peripheral nervous system mechanisms. | Diabetes, metabolic syndrome and obesity : targets and therapy 20090101 |
Mind, brain and psychotherapy. | Indian journal of psychological medicine 20090101 |
The effect of tianeptine in the prevention of radiation-induced neurocognitive impairment. | Medical hypotheses 20081201 |
A new spectrophotometric method for the determination of tianeptine in tablets using ion-pair reagents. | Chemical & pharmaceutical bulletin 20081201 |
Cellular and molecular mechanisms in the long-term action of antidepressants. | Dialogues in clinical neuroscience 20081201 |
['Atypical' antidepressive mechanisms: glutamatergic modulation and neuroplasticity in case of tianeptine]. | Neuropsychopharmacologia Hungarica : a Magyar Pszichofarmakologiai Egyesulet lapja = official journal of the Hungarian Association of Psychopharmacology 20081201 |
Tianeptine: an antidepressant with memory-protective properties. | Current neuropharmacology 20081201 |
Stimulus properties of venlafaxine in a conditioned taste aversion procedure. | European journal of pharmacology 20081031 |
Neuronal NOS inhibitor 1-(2-trifluoromethylphenyl)-imidazole augment the effects of antidepressants acting via serotonergic system in the forced swimming test in rats. | Pharmacology, biochemistry, and behavior 20081001 |
Planned complex suicide: an unusual case. | Journal of forensic sciences 20080701 |
Dimensional personality traits and treatment outcome in patients with major depressive disorder. | Journal of affective disorders 20080601 |
Tianeptine: potential influences on neuroplasticity and novel pharmacological effects. | Progress in neuro-psychopharmacology & biological psychiatry 20080515 |
The immobility produced by intermittent swim stress is not mediated by serotonin. | Pharmacology, biochemistry, and behavior 20080501 |
Inhibition by tianeptine of neuronally mediated contractions in the rat isolated gastrointestinal tract. | Pharmacological research 20080501 |
Psychopharmacology of aggression in children and adolescents with autism: a critical review of efficacy and tolerability. | Journal of child and adolescent psychopharmacology 20080401 |
The enduring effects of an adolescent social stressor on synaptic density, part II: Poststress reversal of synaptic loss in the cortex by adinazolam and MK-801. | Synapse (New York, N.Y.) 20080301 |
Effect of some antidepressants on the low corticosterone concentration-induced gene transcription in LMCAT fibroblast cells. | Journal of physiology and pharmacology : an official journal of the Polish Physiological Society 20080301 |
Pre-training administration of tianeptine, but not propranolol, protects hippocampus-dependent memory from being impaired by predator stress. | European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20080201 |
Association analysis between variants of the interleukin-1beta and the interleukin-1 receptor antagonist gene and antidepressant treatment response in major depression. | Neuropsychiatric disease and treatment 20080201 |
Serotonergic anti-depressants and ethanol withdrawal syndrome: a review. | Alcohol and alcoholism (Oxford, Oxfordshire) 20080101 |
Neurobiological and clinical effects of the antidepressant tianeptine. | CNS drugs 20080101 |
Post-traumatic stress disorder in different types of stress (clinical features and treatment). | Neuroscience and behavioral physiology 20080101 |
Diverse antidepressants increase CDP-diacylglycerol production and phosphatidylinositide resynthesis in depression-relevant regions of the rat brain. | BMC neuroscience 20080101 |
[Dynamics of biochemical parameters in patients with anxious depression treated with serotonergic antidepressants with different mechanisms of action]. | Zhurnal nevrologii i psikhiatrii imeni S.S. Korsakova 20080101 |
[The use of coaxil (tianeptine) in the treatment of aged people with combined mild cognitive impairment and depressive-anxiety disorders]. | Zhurnal nevrologii i psikhiatrii imeni S.S. Korsakova 20080101 |
Neurotrophins and cytokines in neuronal plasticity. | Novartis Foundation symposium 20080101 |
[Tianeptin (coaxil) in therapy of depression in cardiovascular patients]. | Terapevticheskii arkhiv 20080101 |
Antidepressant treatments-induced modifications of glutamatergic transmission in rat frontal cortex. | Pharmacological reports : PR 20080101 |
Effects of co-administration of fluoxetine or tianeptine with metyrapone on immobility time and plasma corticosterone concentration in rats subjected to the forced swim test. | Pharmacological reports : PR 20080101 |
Effect of two behavioral tests on corticosterone level in plasma of mice lacking the noradrenaline transporter. | Pharmacological reports : PR 20080101 |
Information Processing Bias in Post-traumatic Stress Disorder. | The open neuroimaging journal 20080101 |
Cough up for just a cup of coffee: Pharmacoeconomics of depression. | Indian journal of psychiatry 20080101 |
Psychological factors in asthma. | Allergy, asthma, and clinical immunology : official journal of the Canadian Society of Allergy and Clinical Immunology 20080101 |
Involvement of AMPA receptor phosphorylation in antidepressant actions with special reference to tianeptine. | The European journal of neuroscience 20071201 |
Acute selective serotonin reuptake inhibitors increase conditioned fear expression: blockade with a 5-HT(2C) receptor antagonist. | Biological psychiatry 20071115 |
Tianeptine abuse: yet again. | Prescrire international 20071001 |
Modulation of antidepressant-like activity of magnesium by serotonergic system. | Journal of neural transmission (Vienna, Austria : 1996) 20070901 |
Fatal intoxication with tianeptine (Stablon). | Forensic science international 20070806 |
High-performance liquid chromatographic stability indicating assay method of tianeptine sodium with simultaneous fluorescence and UV detection. | Journal of chromatographic science 20070701 |
Tianeptine increases brain-derived neurotrophic factor expression in the rat amygdala. | European journal of pharmacology 20070622 |
The effects of antidepressants on cyclic AMP-response element-driven gene transcription in a model cell system. | Biochemical pharmacology 20070615 |
Coaxil (tianeptine) in the treatment of depression in Parkinson's disease. | Neuroscience and behavioral physiology 20070501 |
Polycystic ovary syndrome and hyperprolactinemia are distinct entities. | Gynecological endocrinology : the official journal of the International Society of Gynecological Endocrinology 20070501 |
Acute stress-mediated increases in extracellular glutamate levels in the rat amygdala: differential effects of antidepressant treatment. | The European journal of neuroscience 20070501 |
Is it possible to be dependent to Tianeptine, an antidepressant? A case report. | Progress in neuro-psychopharmacology & biological psychiatry 20070413 |
Effects of tianeptine on onset time of pentylenetetrazole-induced seizures in mice: possible role of adenosine A1 receptors. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20070201 |
Is hippocampal atrophy a future drug target? | Medical hypotheses 20070101 |
[Comparative study of the effects of amitriptyline, fluoxetine, and tianeptine on the amplitude of transcallosal evoked potentials]. | Eksperimental'naia i klinicheskaia farmakologiia 20070101 |
Anti-inflammatory properties of desipramine and fluoxetine. | Respiratory research 20070101 |
Determination of tianeptine in tablets by high-performance liquid chromatography with fluorescence detection. | Journal of AOAC International 20070101 |
The temporal dynamics model of emotional memory processing: a synthesis on the neurobiological basis of stress-induced amnesia, flashbulb and traumatic memories, and the Yerkes-Dodson law. | Neural plasticity 20070101 |
Hippocampal neurogenesis, depressive disorders, and antidepressant therapy. | Neural plasticity 20070101 |
Stress and memory: behavioral effects and neurobiological mechanisms. | Neural plasticity 20070101 |
[Clinico-epidemiological characteristics of elderly patients with cardiovascular diseases comorbid with depression (results of a multicenter prospective trial COORDINATA)]. | Terapevticheskii arkhiv 20070101 |
Effects of repetitive administration of tianeptine, zinc hydroaspartate and electroconvulsive shock on the reactivity of 5-HT(7) receptors in rat hippocampus. | Pharmacological reports : PR 20070101 |
[Pharmacologic correction of psycho-emotive disorders in the rehabilitation of patients after removal of brain tumors]. | Voprosy onkologii 20070101 |
Long-term voluntary exercise and the mouse hypothalamic-pituitary-adrenocortical axis: impact of concurrent treatment with the antidepressant drug tianeptine. | Journal of neuroendocrinology 20061201 |
Common efficacy of psychotropic drugs in restoring stress-induced impairment of prefrontal plasticity. | Neurotoxicity research 20061201 |
Protective and damaging effects of stress mediators: central role of the brain. | Dialogues in clinical neuroscience 20061201 |
Traumatic stress: effects on the brain. | Dialogues in clinical neuroscience 20061201 |
Sertraline, escitalopram and tianeptine related abnormal movements but not with bupropion: a case report. | Progress in neuro-psychopharmacology & biological psychiatry 20060930 |
Tianeptine can be effective in men with depression and erectile dysfunction. | The journal of sexual medicine 20060901 |
New directions for drug discovery. | Dialogues in clinical neuroscience 20060901 |
[Tianeptine-induced weight gain in adolescents suffering from autism]. | Minerva pediatrica 20060801 |
Enhanced susceptibility to periodontitis in an animal model of depression: reversed by chronic treatment with the anti-depressant tianeptine. | Journal of clinical periodontology 20060701 |
Differential pulse, square wave and adsorptive stripping voltammetric quantification of tianeptine in tablets. | Journal of pharmaceutical and biomedical analysis 20060616 |
Effects of repeated tianeptine treatment on CRF mRNA expression in non-stressed and chronic mild stress-exposed rats. | Neuropharmacology 20060601 |
Antidepressants: general practitioners' opinions and clinical practice. | Acta psychiatrica Scandinavica 20060601 |
Treatments in depression. | Dialogues in clinical neuroscience 20060601 |
Acute and chronic tianeptine treatments attenuate ethanol withdrawal syndrome in rats. | Progress in neuro-psychopharmacology & biological psychiatry 20060501 |
Determination of tianeptine in human plasma using high-performance liquid chromatography with fluorescence detection. | Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20060413 |
A comparative study of fluoxetine, moclobemide, and tianeptine in the treatment of posttraumatic stress disorder following an earthquake. | European psychiatry : the journal of the Association of European Psychiatrists 20060401 |
Acute effects of tianeptine on circulating neurotransmitters and cardiovascular parameters. | Progress in neuro-psychopharmacology & biological psychiatry 20060301 |
Biochemical profile in patients with anxious depression under the treatment with serotonergic antidepressants with different mechanisms of action. | Human psychopharmacology 20060301 |
Benefit of tianeptine and morphine in a transgenic model of familial amyotrophic lateral sclerosis. | Amyotrophic lateral sclerosis : official publication of the World Federation of Neurology Research Group on Motor Neuron Diseases 20060301 |
Differential effects of predator stress and the antidepressant tianeptine on physiological plasticity in the hippocampus and basolateral amygdala. | Stress (Amsterdam, Netherlands) 20060301 |
Regulation of hippocampal gene expression is conserved in two species subjected to different stressors and antidepressant treatments. | Biological psychiatry 20060201 |
Neonatal dexamethasone and chronic tianeptine treatment inhibit ligature-induced periodontitis in adult rats. | Journal of periodontal research 20060201 |
Evident exception in clinical practice not sufficient to break traditional hypothesis. | PLoS medicine 20060201 |
Tyr-95 and Ile-172 in transmembrane segments 1 and 3 of human serotonin transporters interact to establish high affinity recognition of antidepressants. | The Journal of biological chemistry 20060127 |
Discriminative stimulus properties of tianeptine. | Psychopharmacology 20060101 |
Evidence that serotonin reuptake modulators increase the density of serotonin innervation in the forebrain. | Journal of neurochemistry 20060101 |
[A case of tianeptine abuse]. | Turk psikiyatri dergisi = Turkish journal of psychiatry 20060101 |
[Coaxil (tianeptine) in the treatment of depression in Parkinson's disease]. | Zhurnal nevrologii i psikhiatrii imeni S.S. Korsakova 20060101 |
[Depression in cardiological practice: pilot results from a multicenter clinico-epidemiological trial in hypertensive patients with ischemic heart disease (koordinata)]. | Terapevticheskii arkhiv 20060101 |
[Treatment of depression in patients with myocardial infarction with tianeptine]. | Kardiologiia 20060101 |
[Effects of antidepressants in models of brain self-stimulation and place preference after prolong social isolation and alcoholization]. | Eksperimental'naia i klinicheskaia farmakologiia 20060101 |
[Trends in heart rate variability in patients with ischemic heart disease and depression treated with antidepressant tianeptine]. | Terapevticheskii arkhiv 20060101 |
[A double-blind controlled study of the efficacy and acceptability of tianeptine in comparison with fluvoxamine in the treatment of depressed alcoholic patients]. | Psychiatria polska 20060101 |
[Anabolic-catabolic balance in depression: an effect of coaxil]. | Zhurnal nevrologii i psikhiatrii imeni S.S. Korsakova 20060101 |
[A comparative study of efficacy and tolerability of antidepressants from different classes in mild and moderate depression]. | Zhurnal nevrologii i psikhiatrii imeni S.S. Korsakova 20060101 |
[Effect of depressive state on parameters of heart rate variability in patients with ischemic heart disease and correction of revealed disturbances with antidepressant tianeptine]. | Kardiologiia 20060101 |
[Experience in application of various antidepressants in gerontology]. | Klinicheskaia meditsina 20060101 |
Tianeptine: a novel atypical antidepressant that may provide new insights into the biomolecular basis of depression. | Recent patents on CNS drug discovery 20060101 |
Control of ACTH secretion by excitatory amino acids: functional significance and clinical implications. | Endocrine 20051201 |
Contribution of sleep research to the development of new antidepressants. | Dialogues in clinical neuroscience 20051201 |
Sleep disturbances, psychiatric disorders, and psychotropic drugs. | Dialogues in clinical neuroscience 20051201 |
[Trends in pharmacotherapy of unipolar depression at the beginning of the century in Hungary]. | Neuropsychopharmacologia Hungarica : a Magyar Pszichofarmakologiai Egyesulet lapja = official journal of the Hungarian Association of Psychopharmacology 20051201 |
[Attention deficit hyperactivity: tianeptine open trial]. | Minerva pediatrica 20051001 |
The pharmacological management of depression. | Dialogues in clinical neuroscience 20050901 |
Neuroendocrine predictors of the evolution of depression. | Dialogues in clinical neuroscience 20050901 |
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Investigation of the effects of tianeptine and fluoxetine on pentylenetetrazole-induced seizures in rats. | Journal of psychiatric research 20050301 |
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The effects of tianeptine or paroxetine on 35% CO2 provoked panic in panic disorder. | Journal of psychopharmacology (Oxford, England) 20041201 |
Treatment of bronchial asthma with tianeptine. | Methods and findings in experimental and clinical pharmacology 20041101 |
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Chronic administration of tianeptine balances lipopolysaccharide-induced expression of cytokines in the spleen and hypothalamus of rats. | Psychoneuroendocrinology 20040701 |
Untreated depression and hippocampal volume loss. | The American journal of psychiatry 20040701 |
The selective serotonin reuptake inhibitor citalopram increases fear after acute treatment but reduces fear with chronic treatment: a comparison with tianeptine. | Biological psychiatry 20040615 |
Behavioral and neuroendocrine changes during mental stress and repeated treatment with antidepressants in healthy men. | Annals of the New York Academy of Sciences 20040601 |
Cellular consequences of stress and depression. | Dialogues in clinical neuroscience 20040601 |
Structural plasticity of the adult brain: how animal models help us understand brain changes in depression and systemic disorders related to depression. | Dialogues in clinical neuroscience 20040601 |
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Antidepressant treatment with tianeptine reduces apoptosis in the hippocampal dentate gyrus and temporal cortex. | Biological psychiatry 20040415 |
Regulation of the human corticotropin-releasing-hormone gene promoter activity by antidepressant drugs in Neuro-2A and AtT-20 cells. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20040401 |
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Refractory pain-depression syndrome treated with tianeptine: a case report. | The Australian and New Zealand journal of psychiatry 20040301 |
Current perspectives in the management of treatment-resistant depression. | Dialogues in clinical neuroscience 20040301 |
Acute stress-induced changes in hippocampal/prefrontal circuits in rats: effects of antidepressants. | Cerebral cortex (New York, N.Y. : 1991) 20040201 |
Tianeptine: a new exploratory therapy for asthma. | Chest 20040101 |
Tianeptine as a slightly effective therapeutic option for attention-deficit hyperactivity disorder. | Neuropsychobiology 20040101 |
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Thyroid hormones in the rat amygdala as common targets for antidepressant drugs, mood stabilizers, and sleep deprivation. | Biological psychiatry 20031115 |
Prenatal stress in rats predicts immobility behavior in the forced swim test. Effects of a chronic treatment with tianeptine. | Brain research 20031107 |
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Evaluation of cognitive function of fluoxetine, sertraline and tianeptine in isolation and chronic unpredictable mild stress-induced depressive Wistar rats. | Indian journal of experimental biology 20031101 |
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Inhibition of microsomal triglyceride transfer protein: another mechanism for drug-induced steatosis in mice. | Hepatology (Baltimore, Md.) 20030701 |
Tianeptine: a novel strategy of psychopharmacological treatment of children with autistic disorder. | Human psychopharmacology 20030701 |
Switching to tianeptine in patients with antidepressant-induced sexual dysfunction. | Human psychopharmacology 20030601 |
Alcohol, nicotine, caffeine, and mental disorders. | Dialogues in clinical neuroscience 20030601 |
Broken heart: depression in cardiovascular disease. | Dialogues in clinical neuroscience 20030601 |
Neuroprotective properties of tianeptine: interactions with cytokines. | Neuropharmacology 20030501 |
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Clinical and neurobiological effects of tianeptine and paroxetine in major depression. | Journal of clinical psychopharmacology 20030401 |
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Behavioral disturbances in dementia. | Dialogues in clinical neuroscience 20030301 |
State markers of depression in sleep EEG: dependency on drug and gender in patients treated with tianeptine or paroxetine. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20030201 |
Treatment of major depression and anxiety with the selective serotonin re-uptake enhancer tianeptine in the outpatient psychiatric care setting of India. | Journal of the Indian Medical Association 20030201 |
Tianeptine, plasma serotonin, and pulmonary hypertension. | Lancet (London, England) 20030104 |
Local, but not systemic, administration of serotonergic antidepressants decreases hippocampal nitric oxide synthase activity. | Brain research 20030103 |
Chronic treatment with the antidepressant tianeptine attenuates lipopolysaccharide-induced Fos expression in the rat paraventricular nucleus and HPA axis activation. | Psychoneuroendocrinology 20030101 |
Tianeptine may be a useful adjunct in the treatment of alcohol dependence of adolescents. | Alcoholism, clinical and experimental research 20030101 |
Neuropharmacological study of hetero[2,1]benzothiazepine derivatives analogues of tianeptine. | Farmaco (Societa chimica italiana : 1989) 20030101 |
Psychopharmacological effects of tianeptine analogous hetero[2,1] benzothiazepine derivatives. | Arzneimittel-Forschung 20030101 |
The ELIXIR study: evaluation of sexual dysfunction in 4557 depressed patients in France. | Current medical research and opinion 20030101 |
Effect of antidepressants on the phospholipase A2 activity in plasma membranes of the rat brain cortex. | Polish journal of pharmacology 20030101 |
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Mss4 gene is up-regulated in rat brain after chronic treatment with antidepressant and down-regulated when rats are anhedonic. | Molecular pharmacology 20021201 |
The effects of paroxetine and tianeptine on peripheral biochemical markers in major depression. | Progress in neuro-psychopharmacology & biological psychiatry 20021201 |
Sleep-wake mechanisms and drug discovery: sleep EEG as a tool for the development of CNS-acting drugs. | Dialogues in clinical neuroscience 20021201 |
Modulation of tianeptine on ion currents induced by inhibitory neurotransmitters in acutely dissociated dorsal raphe neurons of Sprague-Dawley rats. | European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20021001 |
Enhancement of stress-induced pituitary hormone release and cardiovascular activation by antidepressant treatment in healthy men. | Journal of psychopharmacology (Oxford, England) 20020901 |
The antidepressant tianeptine persistently modulates glutamate receptor currents of the hippocampal CA3 commissural associational synapse in chronically stressed rats. | The European journal of neuroscience 20020901 |
Psychopharmacology of anxiety disorders. | Dialogues in clinical neuroscience 20020901 |
Tianeptine and fluoxetine in major depression: a 6-week randomised double-blind study. | Human psychopharmacology 20020801 |
Synaptic plasticity and tianeptine: structural regulation. | European psychiatry : the journal of the Association of European Psychiatrists 20020701 |
Structural plasticity and tianeptine: cellular and molecular targets. | European psychiatry : the journal of the Association of European Psychiatrists 20020701 |
A meta-analysis of randomized controlled trials of tianeptine versus SSRI in the short-term treatment of depression. | European psychiatry : the journal of the Association of European Psychiatrists 20020701 |
Overcoming the effects of stress on synaptic plasticity in the intact hippocampus: rapid actions of serotonergic and antidepressant agents. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20020501 |
Tianeptine: 5-HT uptake sites and 5-HT(1-7) receptors modulate memory formation in an autoshaping Pavlovian/instrumental task. | Neuroscience and biobehavioral reviews 20020501 |
Effect of tianeptine and fluoxetine on the levels of Met-enkephalin and mRNA encoding proenkephalin in the rat. | Journal of physiology and pharmacology : an official journal of the Polish Physiological Society 20020301 |
Effect of repeated treatment with tianeptine and fluoxetine on central dopamine D(2) /D(3) receptors. | Behavioural pharmacology 20020301 |
Pathophysiology of depression and mechanisms of treatment. | Dialogues in clinical neuroscience 20020301 |
The clinical pharmacology of depressive states. | Dialogues in clinical neuroscience 20020301 |
Enhancing synaptic plasticity and cellular resilience to develop novel, improved treatments for mood disorders. | Dialogues in clinical neuroscience 20020301 |
Efficacy and safety of tianeptine in major depression: evidence from a 3-month controlled clinical trial versus paroxetine. | CNS drugs 20020101 |
[The level of 8-iso-prostaglandin F2 alpha, 4-hydroxynonenal and malondialdehyde in alcohol dependent men during combined therapy]. | Psychiatria polska 20020101 |
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Effect of antidepressant drugs on the human corticotropin-releasing-hormone gene promoter activity in neuro-2A cells. | Polish journal of pharmacology 20020101 |
Asthma, asthma medication and autonomic nervous system dysfunction. | Clinical physiology (Oxford, England) 20011101 |
Tianeptine versus fluoxetine in the treatment of depression complicating Alzheimer's disease. | International journal of geriatric psychiatry 20011101 |
Effect of repeated treatment with tianeptine and fluoxetine on the central alpha(1)-adrenergic system. | Neuropharmacology 20010901 |
Hormonal and behavioural abnormalities induced by stress in utero: an animal model for depression. | Stress (Amsterdam, Netherlands) 20010901 |
Tianeptine and its enantiomers: effects on spatial memory in rats with medial septum lesions. | Neuropharmacology 20010801 |
Effects of tianeptine and mianserin on car driving skills. | Psychopharmacology 20010401 |
Current trends in the development of new antidepressants. | Current medicinal chemistry 20010201 |
Chronic treatment with the atypical antidepressant tianeptine attenuates sickness behavior induced by peripheral but not central lipopolysaccharide and interleukin-1beta in the rat. | Psychopharmacology 20010201 |
Tianeptine: a review of its use in depressive disorders. | CNS drugs 20010101 |
Metyrapone reveals that previous chronic stress differentially impairs hippocampal-dependent memory. | Stress (Amsterdam, Netherlands) 20010101 |
Although chemically related to amineptine, the antidepressant tianeptine is not a dopamine uptake inhibitor. | Pharmacology, biochemistry, and behavior 19990601 |
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