Zatebradine
Title | Journal |
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Why are most phospholipidosis inducers also hERG blockers? | Archives of toxicology 20171201 |
The effects of jaspamide on human cardiomyocyte function and cardiac ion channel activity. | Toxicology in vitro : an international journal published in association with BIBRA 20130301 |
Application of human stem cell-derived cardiomyocytes in safety pharmacology requires caution beyond hERG. | Journal of molecular and cellular cardiology 20120501 |
Characterization of HCN and cardiac function in a colonial ascidian. | Journal of experimental zoology. Part A, Ecological genetics and physiology 20111001 |
Design, synthesis, and preliminary biological evaluation of new isoform-selective f-current blockers. | Journal of medicinal chemistry 20100923 |
8-OH-DPAT prevents cardiac arrhythmias and attenuates tachycardia during social stress in rats. | Physiology & behavior 20090216 |
[Effects of zatebradine on the course of experimental myocardial infarction under long-term treatment conditions in rats]. | Eksperimental'naia i klinicheskaia farmakologiia 20080101 |
A pharmacological model for calcium overload-induced tachycardia in isolated rat left atria. | European journal of pharmacology 20071208 |
Three different bradycardic agents, zatebradine, diltiazem and propranolol, distinctly modify heart rate variability and QT-interval variability. | Pharmacology 20070101 |
Bradycardic and proarrhythmic properties of sinus node inhibitors. | Molecular pharmacology 20060401 |
[Selective I(f) channel inhibition: an alternative for treating coronary artery disease?]. | Herz 20060201 |
Characterization of the human HCN1 channel and its inhibition by capsazepine. | British journal of pharmacology 20041001 |
Role of force--frequency relation during AV-block, sinus node block and beta-adrenoceptor block in conscious animals. | Basic research in cardiology 20040901 |
Heart rate reduction by zatebradine reduces infarct size and mortality but promotes remodeling in rats with experimental myocardial infarction. | American journal of physiology. Heart and circulatory physiology 20040401 |
The impact of organic inhibitors of the hyperpolarization activated current (Ih) on the electroretinogram (ERG) of rodents. | Archives italiennes de biologie 20040301 |
A simulation analysis on mechanisms of damped oscillation in retinal rod photoreceptor cells. | Vision research 20030901 |
(+/-)-2-(3-Piperidyl)-1,2,3,4-tetrahydroisoquinolines as a new class of specific bradycardic agents. | Bioorganic & medicinal chemistry letters 20030707 |
Sinus tachyarrhythmias and the specific bradycardic agents: a marriage made in heaven? | Journal of cardiovascular pharmacology and therapeutics 20030601 |
Effects of changing heart rate on electrophysiological and hemodynamic function in the dog. | Life sciences 20030314 |
Multiple inhibitory effects of zatebradine (UL-FS 49) on the electrophysiological properties of retinal rod photoreceptors. | Pflugers Archiv : European journal of physiology 20020201 |
Parallel solid-phase synthesis of zatebradine analogues as potential I(f) channel blockers. | Bioorganic & medicinal chemistry letters 20010903 |
Intraretinal analysis of the a-wave of the electroretinogram (ERG) in dark-adapted intact cat retina. | Visual neuroscience 20010101 |
Increases in inotropic state without change in heart rate: combined use of dobutamine and zatebradine in conscious dogs. | European journal of pharmacology 19961205 |
Effects of zatebradine on ouabain-, two-stage coronary ligation- and epinephrine-induced ventricular tachyarrhythmias. | European journal of pharmacology 19960411 |
Addition of zatebradine, a direct sinus node inhibitor, provides no greater exercise tolerance benefit in patients with angina taking extended-release nifedipine: results of a multicenter, randomized, double-blind, placebo-controlled, parallel-group study. The Zatebradine Study Group. | Journal of the American College of Cardiology 19950801 |
Zatebradine attenuates cyclic AMP-related positive chronotropic but not inotropic responses in isolated, perfused right atria of the dog. | Clinical and experimental pharmacology & physiology 19950101 |
Zatebradine, a specific bradycardic agent, enhances the positive inotropic actions of dobutamine in ischemic myocardium. | Journal of the American College of Cardiology 19940101 |
Effect of zatebradine on contractility, relaxation and coronary blood flow. | Journal of the American College of Cardiology 19930201 |
Specific bradycardic agents, a new therapeutic modality for anesthesiology: hemodynamic effects of UL-FS 49 and propranolol in conscious and isoflurane-anesthetized dogs. | Anesthesiology 19871101 |
Cardiovascular characterization of UL-FS 49, 1,3,4,5-tetrahydro-7,8-dimethoxy-3-[3-][2-(3,4-dimethoxyphenyl)ethyl] methylimino]propyl]-2H-3-benzazepin-2-on hydrochloride, a new 'specific bradycardic agent'. | European journal of pharmacology 19840903 |