Delamanid
| Title | Journal |
|---|---|
| Pentacyclic nitrofurans with in vivo efficacy and activity against nonreplicating Mycobacterium tuberculosis. | PloS one 20140101 |
| Tuberculosis: the drug development pipeline at a glance. | European journal of medicinal chemistry 20120501 |
| Structure-activity relationships for amide-, carbamate-, and urea-linked analogues of the tuberculosis drug (6S)-2-nitro-6-{[4-(trifluoromethoxy)benzyl]oxy}-6,7-dihydro-5H-imidazo[2,1-b][1,3]oxazine (PA-824). | Journal of medicinal chemistry 20120112 |
| Substrate specificity of the deazaflavin-dependent nitroreductase from Mycobacterium tuberculosis responsible for the bioreductive activation of bicyclic nitroimidazoles. | The FEBS journal 20120101 |
| Structure-activity relationships of antitubercular nitroimidazoles. 3. Exploration of the linker and lipophilic tail of ((s)-2-nitro-6,7-dihydro-5H-imidazo[2,1-b][1,3]oxazin-6-yl)-(4-trifluoromethoxybenzyl)amine (6-amino PA-824). | Journal of medicinal chemistry 20110825 |
| A microbiological assessment of novel nitrofuranylamides as anti-tuberculosis agents. | The Journal of antimicrobial chemotherapy 20081101 |
| Synthesis and antitubercular activity of 7-(R)- and 7-(S)-methyl-2-nitro-6-(S)-(4-(trifluoromethoxy)benzyloxy)-6,7-dihydro-5H-imidazo[2,1-b][1,3]oxazines, analogues of PA-824. | Bioorganic & medicinal chemistry letters 20080401 |
| [Some new antitubercular agents]. | Revue medicale suisse 20080319 |
| New anti-tuberculosis drugs with novel mechanisms of action. | Current medicinal chemistry 20080101 |
| Bactericidal activity of OPC-67683 against drug-tolerant Mycobacterium tuberculosis. | The Journal of antimicrobial chemotherapy 20071101 |
| Advances in the treatment of tuberculosis. | Clinical pharmacology and therapeutics 20071101 |
| [Recent progress in mycobacteriology]. | Kekkaku : [Tuberculosis] 20071001 |
| Synthesis and antituberculosis activity of a novel series of optically active 6-nitro-2,3-dihydroimidazo[2,1-b]oxazoles. | Journal of medicinal chemistry 20061228 |
| OPC-67683, a nitro-dihydro-imidazooxazole derivative with promising action against tuberculosis in vitro and in mice. | PLoS medicine 20061101 |