JNJ 5207852 dihydrochloride
Title | Journal |
---|---|
Radiofluorinated histamine H₃ receptor antagonist as a potential probe for in vivo PET imaging: radiosynthesis and pharmacological evaluation. | Bioorganic & medicinal chemistry 20120501 |
Novel and highly potent histamine H3 receptor ligands. Part 2: exploring the cyclohexylamine-based series. | Bioorganic & medicinal chemistry letters 20110915 |
Histamine H3 receptor as a drug discovery target. | Journal of medicinal chemistry 20110113 |
Indole- and benzothiophene-based histamine H3 antagonists. | Bioorganic & medicinal chemistry letters 20101101 |
Novel substituted pyrrolidines are high affinity histamine H3 receptor antagonists. | Bioorganic & medicinal chemistry letters 20100501 |
Acidic elements in histamine H(3) receptor antagonists. | Bioorganic & medicinal chemistry letters 20100301 |
Heterocyclic replacement of the central phenyl core of diamine-based histamine H3 receptor antagonists. | European journal of medicinal chemistry 20091101 |
5-hydroxyindole-2-carboxylic acid amides: novel histamine-3 receptor inverse agonists for the treatment of obesity. | Journal of medicinal chemistry 20090709 |
Fluorinated non-imidazole histamine H3 receptor antagonists. | Bioorganic & medicinal chemistry letters 20090415 |
2-Aryloxymethylmorpholine histamine H(3) antagonists. | Bioorganic & medicinal chemistry letters 20081101 |
Diamine derivatives containing imidazolidinylidene propanedinitrile as a new class of histamine H3 receptor antagonists. Part I. | Bioorganic & medicinal chemistry letters 20080401 |
Lead identification of acetylcholinesterase inhibitors-histamine H3 receptor antagonists from molecular modeling. | Bioorganic & medicinal chemistry 20080315 |
Benzylamine histamine H(3) antagonists and serotonin reuptake inhibitors. | Bioorganic & medicinal chemistry letters 20070901 |
A new class of histamine H3 receptor antagonists derived from ligand based design. | Bioorganic & medicinal chemistry letters 20070701 |
Histamine H3 receptor antagonists: from target identification to drug leads. | Biochemical pharmacology 20070415 |
4-[6-(2-Aminoethyl)naphthalen-2-yl]benzonitriles are potent histamine H3 receptor antagonists with high CNS penetration. | Bioorganic & medicinal chemistry letters 20070301 |
Microsphere-based protease assays and screening application for lethal factor and factor Xa. | Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501 |
Effects of histamine H(3) antagonists and donepezil on learning and mnemonic deficits induced by pentylenetetrazol kindling in weanling mice. | Neuropharmacology 20060301 |
Aplysamine-1 and related analogs as histamine H3 receptor antagonists. | Bioorganic & medicinal chemistry letters 20060215 |
4-phenoxypiperidines: potent, conformationally restricted, non-imidazole histamine H3 antagonists. | Journal of medicinal chemistry 20050324 |
2-(4-alkylpiperazin-1-yl)quinolines as a new class of imidazole-free histamine H3 receptor antagonists. | Journal of medicinal chemistry 20050113 |
Acute wake-promoting actions of JNJ-5207852, a novel, diamine-based H3 antagonist. | British journal of pharmacology 20041101 |
A new class of diamine-based human histamine H3 receptor antagonists: 4-(aminoalkoxy)benzylamines. | Journal of medicinal chemistry 20030828 |