ethenesulfonamide
Title | Journal |
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Synthesis of a unique isoindoline/tetrahydroisoquinoline-based tricyclic sultam library utilizing a Heck-aza-Michael strategy. | ACS combinatorial science 20120312 |
Automated synthesis of a 184-member library of thiadiazepan-1,1-dioxide-4-ones. | ACS combinatorial science 20110509 |
In vitro and in vivo studies of the trypanocidal properties of WRR-483 against Trypanosoma cruzi. | PLoS neglected tropical diseases 20100901 |
Designed semisynthetic protein inhibitors of Ub/Ubl E1 activating enzymes. | Journal of the American Chemical Society 20100217 |
'Click, click, cyclize': a DOS approach to sultams utilizing vinyl sulfonamide linchpins. | Organic letters 20090205 |
A versatile synthesis of 2,4-substituted oxazoles. | Chemical communications (Cambridge, England) 20080828 |
Indium-mediated tandem radical addition-cyclization-trap reactions in aqueous media. | Organic letters 20031016 |
Evaluation of vinylsulfamides as sulfhydryl selective alkylation reagents in protein modification. | Bioorganic & medicinal chemistry letters 20030210 |
omega-(Imidazol-4-yl)alkane-1-sulfonamides: a new series of potent histamine H(3) receptor antagonists. | Bioorganic & medicinal chemistry 20020201 |
Synthesis and structure-activity relationships in a series of ethenesulfonamide derivatives, a novel class of endothelin receptor antagonists. | Chemical & pharmaceutical bulletin 20011201 |
Ethenesulfonamide and ethanesulfonamide derivatives, a novel class of orally active endothelin-A receptor antagonists. | Bioorganic & medicinal chemistry 20011101 |
Potent second generation vinyl sulfonamide inhibitors of the trypanosomal cysteine protease cruzain. | Bioorganic & medicinal chemistry letters 20011022 |
Ethenesulfonamide derivatives, a novel class of orally active endothelin-A receptor antagonists. | Chemical & pharmaceutical bulletin 20010501 |
Tyrosine kinase inhibitors. 18. 6-Substituted 4-anilinoquinazolines and 4-anilinopyrido[3,4-d]pyrimidines as soluble, irreversible inhibitors of the epidermal growth factor receptor. | Journal of medicinal chemistry 20010201 |