PIBOSEROD,2H-(1,3)OXAZINO(3,2-A)INDOLE-10-CARBOXAMIDE, N-((1-BUTYL-4-PIPERIDINYL)METHYL)-3,4-DIHYDRO-
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Identification of potent Yes1 kinase inhibitors using a library screening approach. | Bioorganic & medicinal chemistry letters 20130801 |
Synthesis and pharmacological properties of novel hydrophilic 5-HT4 receptor antagonists. | Bioorganic & medicinal chemistry 20101215 |
Effect of piboserod, a 5-HT4 serotonin receptor antagonist, on left ventricular function in patients with symptomatic heart failure. | European journal of heart failure 20090801 |
Novel antagonists of serotonin-4 receptors: synthesis and biological evaluation of pyrrolothienopyrazines. | Bioorganic & medicinal chemistry 20090315 |
Measurement of 5-HT4 receptor-mediated esophageal responses by digital sonomicrometry in the anesthetized rat. | Journal of pharmacological and toxicological methods 20060101 |
Piboserod (SB 207266), a selective 5-HT4 receptor antagonist, reduces serotonin potentiation of neurally-mediated contractile responses of human detrusor muscle. | World journal of urology 20050601 |
Identification of a 5-HT4 receptor antagonist clinical candidate through side-chain modification. | Bioorganic & medicinal chemistry letters 20050315 |
The 5-HT4 receptor agonist, tegaserod, is a potent 5-HT2B receptor antagonist in vitro and in vivo. | British journal of pharmacology 20041101 |
Trials of new antiarrhythmic drugs for maintenance of sinus rhythm in patients with atrial fibrillation. | Journal of interventional cardiac electrophysiology : an international journal of arrhythmias and pacing 20040101 |
Regulatory role of 5-HT and muscarinic receptor antagonists on the migrating myoelectric complex in rats. | European journal of pharmacology 20030425 |
5-HT4 receptor ligands: applications and new prospects. | Journal of medicinal chemistry 20030130 |
Synthesis and pharmacological activity of metabolites of the 5-HT(4) receptor antagonist SB-207266. | Bioorganic & medicinal chemistry 20010801 |
Serotonin-4 receptor antagonists reverse cocaine-induced cardiac arrhythmia. | Life sciences 19980101 |
Cloning and expression of human 5-HT4S receptors. Effect of receptor density on their coupling to adenylyl cyclase. | Neuroreport 19971020 |