eperezolid
Title | Journal |
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Response of methicillin-resistant Staphylococcus aureus to amicoumacin A. | PloS one 20120101 |
4-(o-Tol-yl)piperazin-1-ium chloride. | Acta crystallographica. Section E, Structure reports online 20111101 |
Production of icaADBC-encoded polysaccharide intercellular adhesin and therapeutic failure in pediatric patients with Staphylococcal device-related infections. | BMC infectious diseases 20100101 |
Pharmacokinetics of Linezolid and Ertapenem in experimental parapneumonic pleural effusion. | Journal of inflammation (London, England) 20100101 |
Clinical outcomes of antimicrobial lock solutions used in a treatment modality: a retrospective case series analysis. | Clinical pharmacology : advances and applications 20100101 |
Synthesis and antibacterial activities of eperezolid analogs with glycinyl substitutions. | Archiv der Pharmazie 20090701 |
Linezolid (ZYVOX), the first member of a completely new class of antibacterial agents for treatment of serious gram-positive infections. | Journal of medicinal chemistry 20080410 |
Synthesis and in vitro antibacterial activities of novel oxazolidinones. | European journal of medicinal chemistry 20080401 |
Synthesis and in vitro antibacterial activity of novel methylamino piperidinyl oxazolidinones. | Bioorganic & medicinal chemistry letters 20070915 |
Evaluation of a basic physiologically based pharmacokinetic model for simulating the first-time-in-animal study. | European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20070701 |
High-performance liquid chromatographic method for simple and rapid determination of linezolid in human plasma. | Biomedical chromatography : BMC 20060801 |
Novel 4-N-substituted aryl pent-2-ene-1,4-dione derivatives of piperazinyloxazolidinones as antibacterials. | Bioorganic & medicinal chemistry letters 20060315 |
Synthesis and SAR of novel oxazolidinones: discovery of ranbezolid. | Bioorganic & medicinal chemistry letters 20051001 |
Synthesis and antibacterial activity of dihydro-1,2-oxazine and 2-pyrazoline oxazolidinones: novel analogs of linezolid. | Bioorganic & medicinal chemistry letters 20050602 |
In vitro activity of vancomycin, quinupristin/dalfopristin, and linezolid against intact and disrupted biofilms of staphylococci. | Annals of clinical microbiology and antimicrobials 20050101 |
Novel tetrahydro-thieno pyridyl oxazolidinone: an antibacterial agent. | Bioorganic & medicinal chemistry 20040901 |
Simple method for the assay of eperezolid in brain heart infusion broth by high-performance liquid chromatography. | Journal of pharmaceutical and biomedical analysis 20040629 |
Oxazolidinone: search for highly potent antibacterial. | Bioorganic & medicinal chemistry letters 20040621 |
Simple method for the assay of linezolid in Brain Heart Infusion broth by high-performance liquid chromatography. | Biomedical chromatography : BMC 20040101 |
Identification of phenylisoxazolines as novel and viable antibacterial agents active against Gram-positive pathogens. | Journal of medicinal chemistry 20030116 |
Oxazolidinone antibacterial agents: a critical review. | Current topics in medicinal chemistry 20030101 |
Carbon-carbon-linked (pyrazolylphenyl)oxazolidinones with antibacterial activity against multiple drug resistant gram-positive and fastidious gram-negative bacteria. | Bioorganic & medicinal chemistry 20011201 |
The discovery of linezolid, the first oxazolidinone antibacterial agent. | Current drug targets. Infectious disorders 20010801 |
Novel piperidinyloxy oxazolidinone antimicrobial agents. | Bioorganic & medicinal chemistry letters 20010723 |
RU-79115 (Aventis Pharma). | Current opinion in investigational drugs (London, England : 2000) 20010601 |
Oxazolidinones: a review. | Drugs 20000101 |
Activities of several novel oxazolidinones against Mycobacterium tuberculosis in a murine model. | Antimicrobial agents and chemotherapy 19990501 |
In vitro activities of U-100592 and U-100766, novel oxazolidinone antibacterial agents. | Antimicrobial agents and chemotherapy 19960401 |
Synthesis and antibacterial activity of U-100592 and U-100766, two oxazolidinone antibacterial agents for the potential treatment of multidrug-resistant gram-positive bacterial infections. | Journal of medicinal chemistry 19960202 |