9H-Pyrido[3,4-b]indole-3-carboxylicacid, ethyl ester
| Title | Journal |
|---|---|
| Remarkable selectivity of the in vivo binding of [3H]Ro15-4513 to α5 subtype of benzodiazepine receptor in the living mouse brain. | Synapse (New York, N.Y.) 20101201 |
| Alcohol- and alcohol antagonist-sensitive human GABAA receptors: tracking δ subunit incorporation into functional receptors. | Molecular pharmacology 20101101 |
| Design, synthesis, and subtype selectivity of 3,6-disubstituted β-carbolines at Bz/GABA(A)ergic receptors. SAR and studies directed toward agents for treatment of alcohol abuse. | Bioorganic & medicinal chemistry 20101101 |
| Relative potency and effectiveness of flunitrazepam, ethanol, and beta-CCE for disrupting the acquisition and retention of response sequences in rats. | Behavioural pharmacology 20090201 |
| 3D and quantum QSAR of non-benzodiazepine compounds. | European journal of medicinal chemistry 20081101 |
| Selective influence on contextual memory: physiochemical properties associated with selectivity of benzodiazepine ligands at GABAA receptors containing the alpha5 subunit. | Journal of medicinal chemistry 20080710 |
| Efficacy and the discriminative stimulus effects of negative GABAA modulators, or inverse agonists, in diazepam-treated rhesus monkeys. | The Journal of pharmacology and experimental therapeutics 20060801 |
| Microsphere-based protease assays and screening application for lethal factor and factor Xa. | Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501 |
| Negative GABA(A) modulators attenuate the discriminative stimulus effects of benzodiazepines and the neuroactive steroid pregnanolone in rhesus monkeys. | Psychopharmacology 20051001 |
| Identification of a residue in the gamma-aminobutyric acid type A receptor alpha subunit that differentially affects diazepam-sensitive and -insensitive benzodiazepine site binding. | Journal of neurochemistry 20040301 |
| The discovery of tadalafil: a novel and highly selective PDE5 inhibitor. 1: 5,6,11,11a-tetrahydro-1H-imidazo[1',5':1,6]pyrido[3,4-b]indole-1,3(2H)-dione analogues. | Journal of medicinal chemistry 20031009 |
| Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach. | Journal of medicinal chemistry 20000113 |
| Synthesis and evaluation of analogues of the partial agonist 6-(propyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester (6-PBC) and the full agonist 6-(benzyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester (Zk 93423) at wild type and recombinant GABAA receptors. | Journal of medicinal chemistry 19980702 |
| Increasing-current electroshock seizure test: a new method for assessment of anti- and pro-convulsant activities of drugs in mice. | Journal of pharmacological and toxicological methods 19960201 |
| Enhanced sensitivity to beta-carboline inverse agonists in rats chronically treated with FG 7142. | Brain research bulletin 19870901 |
| Chlordiazepoxide enhances the anxiogenic action of CGS 8216 in the social interaction test: evidence for benzodiazepine withdrawal? | Pharmacology, biochemistry, and behavior 19850701 |
| Isoniazid-induced convulsions in rats: effects of Ro 15-1788 and beta-CCE. | European journal of pharmacology 19850619 |
| Evidence for an involvement of GABA receptors in the mediation of the proconvulsant action of ethyl-beta-carboline-3-carboxylate. | Neuropharmacology 19840301 |