N-(Cis-1-benzyl-2-methylpyrrolidin-3-yl)-5-chloro-2-methoxy-4-(methylamino)benzamide
| Title | Journal |
|---|---|
| Schizophrenia-like features in transgenic mice overexpressing human HO-1 in the astrocytic compartment. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20120808 |
| Loss of Mecp2 in substantia nigra dopamine neurons compromises the nigrostriatal pathway. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20110831 |
| Dopamine D₁ and D₂ receptor subtypes functional regulation in corpus striatum of unilateral rotenone lesioned Parkinson's rat model: effect of serotonin, dopamine and norepinephrine. | Neurological research 20101101 |
| Dopamine D1 and D2 receptor functional down regulation in the cerebellum of hypoxic neonatal rats: neuroprotective role of glucose and oxygen, epinephrine resuscitation. | Pharmacological research 20100201 |
| [(3)H]-YM-09151-2 binding sites in human brain postmortem. | Neurochemistry international 20091201 |
| Differences among conventional, atypical and novel putative D(2)/5-HT(1A) antipsychotics on catalepsy-associated behaviour in cynomolgus monkeys. | Behavioural brain research 20091105 |
| Dopamine released by dendritic cells polarizes Th2 differentiation. | International immunology 20090601 |
| Clozapine reverses schizophrenia-related behaviours in the metabotropic glutamate receptor 5 knockout mouse: association with N-methyl-D-aspartic acid receptor up-regulation. | The international journal of neuropsychopharmacology 20090201 |
| A new entry into cis-3-amino-2-methylpyrrolidines via ring expansion of 2-(2-hydroxyethyl)-3-methylaziridines. | Organic & biomolecular chemistry 20090107 |
| 3-Aminopyrrolidines from alpha-aminoacids: total synthesis of (+)-nemonapride from D-alanine. | The Journal of organic chemistry 20080201 |
| Partial agonist actions of aripiprazole and the candidate antipsychotics S33592, bifeprunox, N-desmethylclozapine and preclamol at dopamine D(2L) receptors are modified by co-transfection of D(3) receptors: potential role of heterodimer formation. | Journal of neurochemistry 20070801 |
| Catalytic asymmetric phase-transfer Michael reaction and Mannich-type reaction of glycine Schiff bases with tartrate-derived diammonium salts. | Chemistry, an Asian journal 20070604 |
| F15063, a potential antipsychotic with dopamine D(2)/D(3) antagonist, 5-HT(1A) agonist and D(4) partial agonist properties: (IV) duration of brain D2-like receptor occupancy and antipsychotic-like activity versus plasma concentration in mice. | Naunyn-Schmiedeberg's archives of pharmacology 20070601 |
| Presence of D4 dopamine receptors in human prefrontal cortex: a postmortem study. | Revista brasileira de psiquiatria (Sao Paulo, Brazil : 1999) 20070601 |
| Decreased [3H] YM-09151-2 binding to dopamine D2 receptors in the hypothalamus, brainstem and pancreatic islets of streptozotocin-induced diabetic rats. | European journal of pharmacology 20070227 |
| 5-HT1A receptor agonist properties of antipsychotics determined by [35S]GTPgammaS binding in rat hippocampal membranes. | Clinical and experimental pharmacology & physiology 20070101 |
| In vivo occupancy of dopamine D2 receptors by antipsychotic drugs and novel compounds in the mouse striatum and olfactory tubercles. | Naunyn-Schmiedeberg's archives of pharmacology 20060901 |
| Topographical resolution of jaw movements mediated by cyclase- vs. non-cyclase-coupled dopamine D(1)-like receptors: studies with SK&F 83822. | European journal of pharmacology 20060524 |
| Investigation of cooperativity in the binding of ligands to the D(2) dopamine receptor. | Molecular pharmacology 20060101 |
| Differential in vivo inhibition of [3H]nemonapride binding by atypical antipsychotics in rat striatum, olfactory lobes, and frontal cortex. | Pharmacology 20051001 |
| Increased brain dopamine D4-like binding after chronic ethanol is not associated with behavioral sensitization in mice. | Alcohol (Fayetteville, N.Y.) 20051001 |
| Strain differences of dopamine receptor levels and dopamine related behaviors in rats. | Brain research bulletin 20050430 |
| Subthalamic nucleus lesions alter basal and dopamine agonist stimulated electrophysiological output from the rat basal ganglia. | Synapse (New York, N.Y.) 20041101 |
| Ethologically based resolution of D2-like dopamine receptor agonist-versus antagonist-induced behavioral topography in dopamine- and adenosine 3',5'-monophosphate-regulated phosphoprotein of 32 kDa 'knockout' mutants congenic on the C57BL/6 genetic background. | The Journal of pharmacology and experimental therapeutics 20040901 |
| Early adoption modifies the effects of prenatal stress on dopamine and glutamate receptors in adult rat brain. | Journal of neuroscience research 20040515 |
| The inhibitory role of methylation on the binding characteristics of dopamine receptors and transporter. | Neuroscience research 20040301 |
| SK&F 83822 distinguishes adenylyl cyclase from phospholipase C-coupled dopamine D1-like receptors: behavioural topography. | European journal of pharmacology 20040223 |
| Dopamine transmission in DYT1 dystonia. | Advances in neurology 20040101 |
| Pharmacological actions of a novel and selective dopamine D3 receptor antagonist, KCH-1110. | Pharmacological research 20031201 |
| Potent activation of dopamine D3/D2 heterodimers by the antiparkinsonian agents, S32504, pramipexole and ropinirole. | Journal of neurochemistry 20031101 |
| The effects of chronic L-DOPA therapy on pharmacodynamic parameters in a rat model of motor response fluctuations. | Experimental neurology 20031101 |
| Characterization of dopamine D2 receptor gene expression and binding sites in human placenta amniotic epithelial cells. | Placenta 20030701 |
| Sigma1 and dopamine D2 receptor occupancy in the mouse brain after a single administration of haloperidol and two dopamine D2-like receptor ligands. | Nuclear medicine and biology 20030501 |
| Suppression of cocaine- and food-maintained behavior by the D2-like receptor partial agonist terguride in squirrel monkeys. | Psychopharmacology 20030301 |
| Constitutive coupling of a chimeric dopamine D2/alpha 1B receptor to the phospholipase C pathway: inverse agonism to silent antagonism by neuroleptic drugs. | The Journal of pharmacology and experimental therapeutics 20030101 |
| Congenic D1A dopamine receptor mutants: ethologically based resolution of behavioural topography indicates genetic background as a determinant of knockout phenotype. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20030101 |
| The impact of stereotactic pallidal surgery on the dopamine D2 receptor in Parkinson disease: a positron emission tomography study. | Journal of neurosurgery 20030101 |
| N-methyl-D-aspartate-R1 receptor antisense oligodeoxynucleotide modulates pre- and postsynaptic expression of D2 dopamine receptors in the rat. | Neuroscience letters 20021219 |
| Increased sensitivity in dopamine D(2)-like brain receptors from 2,4-dichlorophenoxyacetic acid (2,4-D)-exposed and amphetamine-challenged rats. | Annals of the New York Academy of Sciences 20020601 |
| Functional and autoradiographic characterization of dopamine D2-like receptors in the guinea pig heart. | Canadian journal of physiology and pharmacology 20020601 |
| Positron emission tomography and ex vivo and in vitro autoradiography studies on dopamine D2-like receptor degeneration in the quinolinic acid-lesioned rat striatum: comparison of [11C]raclopride, [11C]nemonapride and [11C]N-methylspiperone. | Nuclear medicine and biology 20020401 |
| Effects of individual and concurrent stimulation of striatal D1 and D2 dopamine receptors on electrophysiological and behavioral output from rat basal ganglia. | The Journal of pharmacology and experimental therapeutics 20020301 |
| Associations between side effects of nemonapride and plasma concentrations of the drug and prolactin. | Progress in neuro-psychopharmacology & biological psychiatry 20020201 |
| (-)S amisulpride binds with high affinity to cloned dopamine D(3) and D(2) receptors. | European journal of pharmacology 20011207 |
| Agonist-independent and -dependent oligomerization of dopamine D(2) receptors by fusion to fluorescent proteins. | FEBS letters 20011019 |
| Extended treatment with typical and atypical antipsychotic drugs differential effects on the densities of dopamine D2-like and GABAA receptors in rat striatum. | Life sciences 20010803 |
| The -141C Ins/Del polymorphism in the dopamine D2 receptor gene promoter region is associated with anxiolytic and antidepressive effects during treatment with dopamine antagonists in schizophrenic patients. | Pharmacogenetics 20010801 |
| No relationship between--141C Ins/Del polymorphism in the promoter region of dopamine D2 receptor and extrapyramidal adverse effects of selective dopamine D2 antagonists in schizophrenic patients: a preliminary study. | Psychiatry research 20010214 |
| Possible pharmacokinetic and pharmacodynamic factors affecting parkinsonism inducement by cinnarizine and flunarizine. | Biochemical pharmacology 19951109 |
| Differential effects of [3H]nemonapride and [3H]spiperone binding on human dopamine D4 receptors. | Neuroscience letters 19950217 |
| Low density of dopamine D4 receptors in Parkinson's, schizophrenia, and control brain striata. | Synapse (New York, N.Y.) 19930801 |
| Influence of (-)-sulpiride and YM-09151-2 on stereotyped behavior in chicks and catalepsy in rats. | Japanese journal of pharmacology 19870201 |