[Sar-9, Met(O2)-11]-Substance P
| Title | Journal |
|---|---|
| Synthesis and structure-activity relationship studies in serotonin 5-HT(1A) receptor agonists based on fused pyrrolidone scaffolds. | European journal of medicinal chemistry 20130501 |
| Evidence for regulatory diversity and auto-regulation at the TAC1 locus in sensory neurones. | Journal of neuroinflammation 20110101 |
| Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: design, synthesis, and structure-activity relationships. | Bioorganic & medicinal chemistry 20101101 |
| Substance P sensitizes P2X3 in nociceptive trigeminal neurons. | Journal of dental research 20101001 |
| The neurokinin-1 receptor modulates the methamphetamine-induced striatal apoptosis and nitric oxide formation in mice. | Journal of neurochemistry 20091101 |
| Neurokinin receptor modulation of respiratory activity in the rabbit. | The European journal of neuroscience 20080601 |
| Expression and coupling of neurokinin receptor subtypes to inositol phosphate and calcium signaling pathways in human airway smooth muscle cells. | American journal of physiology. Lung cellular and molecular physiology 20080301 |
| Pharmacological characterization of T-2328, 2-fluoro-4'-methoxy-3'-[[[(2S,3S)-2-phenyl-3-piperidinyl]amino]methyl]-[1,1'-biphenyl]-4-carbonitrile dihydrochloride, as a brain-penetrating antagonist of tachykinin NK1 receptor. | Journal of pharmacological sciences 20080101 |
| Effect of melatonin on the vasopressin secretion as influenced by tachykinin NK-1 receptor agonist and antagonist: in vivo and in vitro studies. | Journal of physiology and pharmacology : an official journal of the Polish Physiological Society 20071201 |
| Substance P excites globus pallidus neurons in vivo. | The European journal of neuroscience 20071001 |
| Role for NK(1) and NK(2) receptors in the motor activity in mouse colon. | European journal of pharmacology 20070910 |
| Neurokinin-1 receptor activation in Botzinger complex evokes bradypnoea. | The Journal of physiology 20060915 |
| Characteristics of substance P transport across the blood-brain barrier. | Pharmaceutical research 20060601 |
| Upregulation of tachykinin NK-1 and NK-3 receptor binding sites in the spinal cord of spontaneously hypertensive rat: impact on the autonomic control of blood pressure. | British journal of pharmacology 20060501 |
| Ava[L-Pro9,N-MeLeu10] substance P(7-11) (GR 73632) and Sar9, Met(O2)11 increase distention-induced peristalsis through activation of neurokinin-1 receptors on smooth muscle and interstitial cells of cajal. | The Journal of pharmacology and experimental therapeutics 20060401 |
| Neurokinin-1 receptor in peripheral nerve terminals mediates thermal hyperalgesia. | Biochemical and biophysical research communications 20060106 |
| Activation of central neurokinin-1 receptors induces reinstatement of cocaine-seeking behavior. | Neuroscience letters 20051216 |
| The ventral tegmental area as a putative target for tachykinins in cardiovascular regulation. | British journal of pharmacology 20050701 |
| Elimination of rat spinal neurons expressing neurokinin 1 receptors reduces bladder overactivity and spinal c-fos expression induced by bladder irritation. | American journal of physiology. Renal physiology 20050301 |
| A model of organotypic rat spinal slice culture and biolistic transfection to elucidate factors that drive the preprotachykinin-A promoter. | Brain research. Brain research reviews 20041001 |
| Neurokinin-1 and -3 receptor blockade inhibits slow excitatory synaptic transmission in myenteric neurons and reveals slow inhibitory input. | Neuroscience 20040101 |
| Substance P modulates localized calcium transients and membrane current responses in murine colonic myocytes. | British journal of pharmacology 20030401 |
| Evidence for a GABA(B) receptor component in the spinal action of Substance P (SP) on arterial blood pressure in the awake rat. | British journal of pharmacology 20020801 |
| Chemical coding and electrophysiology of enteric neurons expressing neurofilament 145 in guinea pig gastrointestinal tract. | The Journal of comparative neurology 20020114 |
| Permissive role of neurokinin NK(3) receptors in NK(1) receptor-mediated activation of the locus coeruleus revealed by SR 142801. | Synapse (New York, N.Y.) 20020101 |
| Assessing the emetic potential of PDE4 inhibitors in rats. | British journal of pharmacology 20020101 |
| Peripheral inflammation reduces the response of spinal dorsal horn neurons to an NK3 receptor agonist. | Neuroscience letters 20010727 |
| Priming effects of substance P on calcium changes evoked by interleukin-8 in human neutrophils. | Journal of leukocyte biology 20010601 |
| Effect of the long-acting tachykinin NK(1) receptor antagonist MEN 11467 on tracheal mucus secretion in allergic ferrets. | British journal of pharmacology 20010101 |
| Treatment of gastric ulcers and diarrhea with the Amazonian herbal medicine sangre de grado. | American journal of physiology. Gastrointestinal and liver physiology 20000701 |
| NK1-receptor activation prevents hydrocarbon-induced lung injury in mice. | The American journal of physiology 19990201 |