1H-Indole-3-carboxylic acid amide
| Title | Journal |
|---|---|
| Synthesis of retinoid enhancers based on 2-aminobenzothiazoles for anti-cancer therapy. | Bioorganic & medicinal chemistry 20121201 |
| Palladium-catalyzed mono- and double-carbonylation of indoles with amines controllably leading to amides and α-ketoamides. | Chemical communications (Cambridge, England) 20121118 |
| Exploring the substructural space of indole-3-carboxamide derivatives binding to renin: a novel active-site spatial partitioning approach. | Journal of molecular modeling 20120901 |
| Detailed structure-activity relationship of indolecarboxamides as H4 receptor ligands. | European journal of medicinal chemistry 20120801 |
| Alkaloids from the root of Isatis indigotica. | Journal of natural products 20120622 |
| Preclinical pharmacology of novel indolecarboxamide ML-970, an investigative anticancer agent. | Cancer chemotherapy and pharmacology 20120601 |
| Induction of VMAT-1 and TPH-1 expression induces vesicular accumulation of serotonin and protects cells and tissue from cooling/rewarming injury. | PloS one 20120101 |
| Novel indole and azaindole (pyrrolopyridine) cannabinoid (CB) receptor agonists: design, synthesis, structure-activity relationships, physicochemical properties and biological activity. | European journal of medicinal chemistry 20111001 |
| New indole amide derivatives as potent CRTH2 receptor antagonists. | Bioorganic & medicinal chemistry letters 20110601 |
| KDR inhibitor with the intramolecular non-bonded interaction: conformation-activity relationships of novel indole-3-carboxamide derivatives. | Bioorganic & medicinal chemistry letters 20110315 |
| From SOMAmer-based biomarker discovery to diagnostic and clinical applications: a SOMAmer-based, streamlined multiplex proteomic assay. | PloS one 20110101 |
| Synthesis and pharmacological properties of novel hydrophilic 5-HT4 receptor antagonists. | Bioorganic & medicinal chemistry 20101215 |
| Indoleamine 2,3-dioxygenase, an immunomodulatory protein, is suppressed by (-)-epigallocatechin-3-gallate via blocking of gamma-interferon-induced JAK-PKC-delta-STAT1 signaling in human oral cancer cells. | Journal of agricultural and food chemistry 20100127 |
| (1)H, (15)N, and (13)C chemical shift assignments of neuronal calcium sensor-1 homolog from fission yeast. | Biomolecular NMR assignments 20091201 |
| Single-flask synthesis of N-acylated indoles by catalytic dehydrogenative coupling with primary alcohols. | Organic letters 20090402 |
| Structural insights for design of potent spleen tyrosine kinase inhibitors from crystallographic analysis of three inhibitor complexes. | Chemical biology & drug design 20090401 |
| Reduction of pyrrolyl- and indolylamides with BH3 x THF: cyclodeoxygenation versus deoxygenation. | The Journal of organic chemistry 20081107 |
| Antimicrobial and antiviral screening of novel indole carboxamide and propanamide derivatives. | Zeitschrift fur Naturforschung. C, Journal of biosciences 20080101 |
| QSAR study on permeability of hydrophobic compounds with artificial membranes. | Bioorganic & medicinal chemistry 20070601 |
| Bioactivity of glycogen phosphorylase inhibitors that bind to the purine nucleoside site. | Bioorganic & medicinal chemistry 20061201 |
| Low molecular weight indole fragments as IMPDH inhibitors. | Bioorganic & medicinal chemistry letters 20060501 |
| Microsphere-based protease assays and screening application for lethal factor and factor Xa. | Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501 |
| Antitubercular sterols from Thalia multiflora Horkel ex Koernicke. | Phytotherapy research : PTR 20051001 |
| Exploration of a binding mode of indole amide analogues as potent histone deacetylase inhibitors and 3D-QSAR analyses. | Bioorganic & medicinal chemistry 20050915 |
| Increased potency and efficacy of combined phosphorylase inactivation and glucokinase activation in control of hepatocyte glycogen metabolism. | Diabetes 20050301 |
| Synthesis, molecular modeling, and evaluation of nonphenolic indole analogs of mycophenolic acid. | Bioorganic & medicinal chemistry 20040601 |
| Homology modeling, force field design, and free energy simulation studies to optimize the activities of histone deacetylase inhibitors. | Journal of computer-aided molecular design 20040601 |
| Oxidative cross-linking of tryptophan to glycine restrains matrix metalloproteinase activity: specific structural motifs control protein oxidation. | The Journal of biological chemistry 20040220 |
| Indole amide hydroxamic acids as potent inhibitors of histone deacetylases. | Bioorganic & medicinal chemistry letters 20030602 |
| Isolation and insecticidal activity of mellamide from Aspergillus melleus. | Journal of industrial microbiology & biotechnology 20030401 |