Ethene,1,1'-sulfonylbis-
Title | Journal |
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Inhibition of cathepsin S induces autophagy and apoptosis in human glioblastoma cell lines through ROS-mediated PI3K/AKT/mTOR/p70S6K and JNK signaling pathways. | Toxicology letters 20140804 |
An endoperoxide-based hybrid approach to deliver falcipain inhibitors inside malaria parasites. | ChemMedChem 20130901 |
Turnover-dependent covalent inactivation of Staphylococcus aureus coenzyme A-disulfide reductase by coenzyme A-mimetics: mechanistic and structural insights. | Biochemistry 20121002 |
Effects of calcium salts of acidic monomers on mineral induction of phosphoprotein immobilized to agarose beads. | Journal of biomedical materials research. Part A 20121001 |
A general approach to the synthesis of enantiopure 19-nor-vitamin D3 and its C-2 phosphate analogs prepared from cyclohexadienyl sulfone. | Chemical communications (Cambridge, England) 20120918 |
Synthesis of trans-disubstituted alkenes by cobalt-catalyzed reductive coupling of terminal alkynes with activated alkenes. | Chemistry (Weinheim an der Bergstrasse, Germany) 20120910 |
Novel cruzain inhibitors for the treatment of Chagas' disease. | Chemical biology & drug design 20120901 |
Nanostructured PEG-based hydrogels with tunable physical properties for gene delivery to human mesenchymal stem cells. | Biomaterials 20120901 |
Magnetic bead cellulose as a suitable support for immobilization of α-chymotrypsin. | Applied biochemistry and biotechnology 20120901 |
Biofunctional paper via the covalent modification of cellulose. | Langmuir : the ACS journal of surfaces and colloids 20120731 |
Fluoride-mediated elimination of allyl sulfones: application to the synthesis of a 2,4-dimethyl-A-ring vitamin D3 analogue. | The Journal of organic chemistry 20120601 |
Vinyl sulfone functionalization: a feasible approach for the study of the lectin-carbohydrate interactions. | Bioconjugate chemistry 20120418 |
Novel cyanine dyes with vinylsulfone group for labeling biomolecules. | Bioconjugate chemistry 20120321 |
Stereocontrolled fluorobenzylation of vinyl sulfones and α,β-unsaturated esters mediated by a remote sulfinyl group. Synthesis of functionalized enantiomerically pure benzylic fluorides. | The Journal of organic chemistry 20120316 |
Expedient enantioselective synthesis of cermizine D. | Organic letters 20120316 |
One-step 'click' method for generating vinyl sulfone groups on hydroxyl-containing water-soluble polymers. | Biomacromolecules 20120312 |
Effect of vinyl sulfone inhibitors of cysteine proteinases on Tritrichomonas foetus infection. | International journal of antimicrobial agents 20120301 |
An organophosphonate strategy for functionalizing silicon photonic biosensors. | Langmuir : the ACS journal of surfaces and colloids 20120214 |
Accelerated identification of proteins by mass spectrometry by employing covalent pre-gel staining with Uniblue A. | PloS one 20120101 |
AFM Specific Identification of Bacterial Cell Fragments on Biofunctional Surfaces. | The open microbiology journal 20120101 |
Novel magnetic fibrin hydrogel scaffolds containing thrombin and growth factors conjugated iron oxide nanoparticles for tissue engineering. | International journal of nanomedicine 20120101 |
Electrocoagulation treatment of simulated floor-wash containing Reactive Black 5 using iron sacrificial anode. | Journal of hazardous materials 20111215 |
Structural basis for inhibition of cathepsin B drug target from the human blood fluke, Schistosoma mansoni. | The Journal of biological chemistry 20111014 |
In situ forming physical hydrogels for three-dimensional tissue morphogenesis. | Macromolecular bioscience 20111010 |
Targeting ligand-functionalized and redox-sensitive heparin-Pluronic nanogels for intracellular protein delivery. | Biomedical materials (Bristol, England) 20111001 |
Enhanced toxicity of the protein cross-linkers divinyl sulfone and diethyl acetylenedicarboxylate in comparison to related monofunctional electrophiles. | Chemical research in toxicology 20110919 |
Heparin-decorated, hyaluronic acid-based hydrogel particles for the controlled release of bone morphogenetic protein 2. | Acta biomaterialia 20110801 |
Molecular docking and 3D-quantitative structure activity relationship analyses of peptidyl vinyl sulfones: Plasmodium Falciparum cysteine proteases inhibitors. | Journal of computer-aided molecular design 20110801 |
Controlling the facial selectivity of asymmetric [4+2] cyclo-additions: a concise synthesis of the cis-decalin core structure of superstolides A and B. | Organic letters 20110715 |
Highly enantioselective organocascade intermolecular iminium/enamine Michael addition on enals. | Chemical communications (Cambridge, England) 20110707 |
Development of novel peptidomimetics containing a vinyl sulfone moiety as proteasome inhibitors. | ChemMedChem 20110704 |
Apatite-coated hyaluronan for bone regeneration. | Journal of dental research 20110701 |
Occupational Asthma Induced by the Reactive Dye Synozol Red-K 3BS. | Allergy, asthma & immunology research 20110701 |
Aspartic vinyl sulfones: inhibitors of a caspase-3-dependent pathway. | European journal of medicinal chemistry 20110601 |
Coupling of gelatin to inner surfaces of pore walls in spongy alginate-based scaffolds facilitates the adhesion, growth and differentiation of human bone marrow mesenchymal stromal cells. | Journal of materials science. Materials in medicine 20110601 |
2,6-Dichloro-1-[(1E)-2-(phenyl-sulfon-yl)ethen-yl]benzene. | Acta crystallographica. Section E, Structure reports online 20110501 |
Site-specific conjugation of monodispersed DOTA-PEGn to a thiolated diabody reveals the effect of increasing peg size on kidney clearance and tumor uptake with improved 64-copper PET imaging. | Bioconjugate chemistry 20110420 |
Biodegradable and biocompatible synthetic saccharide-Peptide hydrogels for three-dimensional stem cell culture. | Biomacromolecules 20110314 |
Targeting adenovirus gene delivery to activated tumour-associated vasculature via endothelial selectins. | Journal of controlled release : official journal of the Controlled Release Society 20110310 |
Palladium-catalyzed conjugate addition to electron-deficient alkynes with benzenesulfinic acid derived from 1,2-bis(phenylsulfonyl)ethane: selective synthesis of (E)-vinyl sulfones. | The Journal of organic chemistry 20110204 |
A versatile method for functionalizing surfaces with bioactive glycans. | Bioconjugate chemistry 20110119 |
Effects of surface pre-reacted glass-ionomer fillers on mineral induction by phosphoprotein. | Journal of dentistry 20110101 |
Structure-activity relationship of cinnamaldehyde analogs as inhibitors of AI-2 based quorum sensing and their effect on virulence of Vibrio spp. | PloS one 20110101 |
Diversity in protein glycosylation among insect species. | PloS one 20110101 |
Affinity purification of specific anti-Listeria monocytogenes egg yolk antibodies (IgY) using amino-activated cells as receptors. | Journal of immunoassay & immunochemistry 20110101 |
Hyaluronic acid dermal fillers: can adjunctive lidocaine improve patient satisfaction without decreasing efficacy or duration? | Patient preference and adherence 20110101 |
Convection-enhanced delivery of methotrexate-loaded maghemite nanoparticles. | International journal of nanomedicine 20110101 |
Mining the Active Proteome of Arabidopsis thaliana. | Frontiers in plant science 20110101 |
Nature of pharmacophore influences active site specificity of proteasome inhibitors. | The Journal of biological chemistry 20101217 |
Stereocontrolled creation of all-carbon quaternary stereocenters by organocatalytic conjugate addition of oxindoles to vinyl sulfone. | Angewandte Chemie (International ed. in English) 20101011 |
Synthesis and evaluation of vinyl sulfones as caspase-3 inhibitors. A structure-activity study. | European journal of medicinal chemistry 20100901 |
Biodegradable poly(ethylene glycol) hydrogels based on a self-elimination degradation mechanism. | Biomaterials 20100901 |
In vitro and in vivo studies of the trypanocidal properties of WRR-483 against Trypanosoma cruzi. | PLoS neglected tropical diseases 20100901 |
The impact of hyaluronic acid oligomer content on physical, mechanical, and biologic properties of divinyl sulfone-crosslinked hyaluronic acid hydrogels. | Journal of biomedical materials research. Part A 20100801 |
Vinyl sulfone bifunctional tag reagents for single-point modification of proteins. | The Journal of organic chemistry 20100618 |
First synthesis and antiprotozoal activities of divinyl sulfone-modified carbohydrates. | Bioorganic & medicinal chemistry letters 20100615 |
A novel Entamoeba histolytica cysteine proteinase, EhCP4, is key for invasive amebiasis and a therapeutic target. | The Journal of biological chemistry 20100611 |
Sulfones: new reagents in organocatalysis. | Chemical Society reviews 20100601 |
Crystal Structures of TbCatB and rhodesain, potential chemotherapeutic targets and major cysteine proteases of Trypanosoma brucei. | PLoS neglected tropical diseases 20100601 |
Long acting hyaluronate--exendin 4 conjugate for the treatment of type 2 diabetes. | Biomaterials 20100501 |
Computational identification of uncharacterized cruzain binding sites. | PLoS neglected tropical diseases 20100501 |
Chiral primary amine mediated conjugate addition of branched aldehydes to vinyl sulfone: asymmetric generation of quaternary carbon centers. | Chemical communications (Cambridge, England) 20100407 |
Anti-inflammatory compounds parthenolide and Bay 11-7082 are direct inhibitors of the inflammasome. | The Journal of biological chemistry 20100326 |
Tandem Ir-catalyzed allylic substitution reaction of allyl sulfinates and isomerization. | Organic letters 20100219 |
Effect of cross-linking reagents for hyaluronic acid hydrogel dermal fillers on tissue augmentation and regeneration. | Bioconjugate chemistry 20100217 |
Vinyl sulfone: a versatile function for simple bioconjugation and immobilization. | Organic & biomolecular chemistry 20100207 |
Dihydroxylation of vinyl sulfones: stereoselective synthesis of (+)- and (-)-febrifugine and halofuginone. | The Journal of organic chemistry 20100115 |
An experimental and theoretical study on the remarkable influence of protecting groups on the selectivity of addition of amines to vinyl sulfone-modified hex-2-enopyranosides. | The Journal of organic chemistry 20100115 |
The efficiency of contact lens care regimens on protein removal from hydrogel and silicone hydrogel lenses. | Molecular vision 20100101 |
Chitin deacetylases: properties and applications. | Marine drugs 20100101 |
Therapeutic utility and medicinal chemistry of cathepsin C inhibitors. | Current topics in medicinal chemistry 20100101 |
Soft tissue augmentation in dermatology - 2009 update. | Journal of cutaneous and aesthetic surgery 20100101 |
Detection of ubiquityl-calmodulin conjugates with a novel high-molecular weight ubiquitylprotein-isopeptidase in rabbit tissues. | European journal of medical research 20100101 |
Column-switching HPLC determination of mexiletine using tris(bipyridine)ruthenium(III) electrogenerated chemiluminescence and precolumn derivatization with divinylsulfone. | Analytical sciences : the international journal of the Japan Society for Analytical Chemistry 20100101 |
Synthesis and characterization of recombinant factor VIIa-conjugated magnetic iron oxide nanoparticles for hemophilia treatment. | Journal of biomedical materials research. Part A 20091215 |
Addition of amines and carbon nucleophiles to vinyl sulfone-modified 6-deoxy-hex-3-enopyranoside: a case of nucleophile dependent diastereoselectivity. | Carbohydrate research 20091123 |
Purification of the 90 kDa heat shock protein (hsp90) and simultaneous purification of hsp70/hsc70, hsp90 and hsp96 from mammalian tissues and cells using thiophilic interaction chromatography. | Biomedical chromatography : BMC 20091101 |
Chemically crosslinkable thermosensitive polyphosphazene gels as injectable materials for biomedical applications. | Biomaterials 20091001 |
Vinyl sulfones as antiparasitic agents and a structural basis for drug design. | The Journal of biological chemistry 20090918 |
Design, syntheses, and evaluation of Taspase1 inhibitors. | Bioorganic & medicinal chemistry letters 20090901 |
Stimuli-responsive coacervate induced in binary functionalized poly(N-isopropylacrylamide) aqueous system and novel method for preparing semi-ipn microgel using the coacervate. | Langmuir : the ACS journal of surfaces and colloids 20090818 |
Two approaches to discovering and developing new drugs for Chagas disease. | Memorias do Instituto Oswaldo Cruz 20090701 |
Artemisinin-dipeptidyl vinyl sulfone hybrid molecules: design, synthesis and preliminary SAR for antiplasmodial activity and falcipain-2 inhibition. | Bioorganic & medicinal chemistry letters 20090615 |
Evolving organic synthesis fostered by the pluripotent phenylsulfone moiety. | Chemical reviews 20090601 |
SmCL3, a gastrodermal cysteine protease of the human blood fluke Schistosoma mansoni. | PLoS neglected tropical diseases 20090601 |
The liberation of fractalkine in the dorsal horn requires microglial cathepsin S. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20090527 |
Enantioselective conjugate addition of nitroalkanes to vinyl sulfone: an organocatalytic access to chiral amines. | Organic letters 20090416 |
Potential use of cotton plant wastes for the removal of Remazol Black B reactive dye. | Journal of hazardous materials 20090415 |
Efficient isolation of immunoglobulin G by paramagnetic polymer beads modified with 2-mercapto-4-mythyl-pyrimidine. | Journal of immunological methods 20090415 |
A diastereoselective unique route to cyclopropanes functionalized at all three ring carbon atoms from acyclic vinyl sulfone-modified carbohydrates. | The Journal of organic chemistry 20090403 |
Probing of the cis-5-phenyl proline scaffold as a platform for the synthesis of mechanism-based inhibitors of the Staphylococcus aureus sortase SrtA isoform. | Bioorganic & medicinal chemistry 20090401 |
Evidence for bidentate substrate binding as the basis for the K48 linkage specificity of otubain 1. | Journal of molecular biology 20090306 |
Designer discodermolide segments via ozonolysis of vinyl phosphonates. | Organic letters 20090205 |
Densely functionalized chiral pyrroles from endocyclic, exocyclic, and acyclic vinyl sulfone-modified carbohydrates. | The Journal of organic chemistry 20090116 |
Micelles and polymersomes obtained by self-assembly of dextran and polystyrene based block copolymers. | Biomacromolecules 20090112 |
Enantioselective organocatalytic conjugate addition of aldehydes to vinyl sulfones and vinyl phosphonates as challenging Michael acceptors. | Chemistry (Weinheim an der Bergstrasse, Germany) 20090101 |
The efficient and specific isolation of the antibodies from human serum by thiophilic paramagnetic polymer nanospheres. | Biotechnology progress 20090101 |
Hemoglobin cleavage site-specificity of the Plasmodium falciparum cysteine proteases falcipain-2 and falcipain-3. | PloS one 20090101 |
Identification and developmental expression of Xenopus laevis SUMO proteases. | PloS one 20090101 |
Asymmetric organocatalytic Michael addition of ketones to vinyl sulfone. | Chemical communications (Cambridge, England) 20081221 |
The effective and specific isolation of antibodies from human serum by using thiophilic paramagnetic polymer beads. | Colloids and surfaces. B, Biointerfaces 20081201 |
Hyaluronic acid gel (Juvéderm) preparations in the treatment of facial wrinkles and folds. | Clinical interventions in aging 20081201 |
Organocatalytic Michael addition of aldehydes to vinyl sulfones: enantioselective alpha-alkylations of aldehydes and their derivatives. | Organic letters 20081106 |
Physical properties of crosslinked hyaluronic acid hydrogels. | Journal of materials science. Materials in medicine 20081101 |
Hydrogels for potential colon drug release by thiol-ene conjugate addition of a new inulin derivative. | Macromolecular bioscience 20081008 |
Kinetics and products of the gas-phase reactions of divinyl sulfoxide with OH and NO3 radicals and O3. | The journal of physical chemistry. A 20080918 |
Hyaluronan-tethered opioid depots: synthetic strategies and release kinetics in vitro and in vivo. | Bioconjugate chemistry 20080901 |
A vinyl sulfone-modified carbohydrate mediated new route to aminosugars and branched-chain sugars. | Carbohydrate research 20080811 |
Nonpeptidic vinyl and allyl phosphonates as falcipain-2 inhibitors. | ChemMedChem 20080701 |
Unusual addition of amines to C-2 of vinyl sulfone-modified-beta-D-pent-2-enofuranosyl carbohydrates: synthesis of a new class of beta-anomeric 2-amino-2,3-dideoxy-D-threo-pentofuranosides. | Carbohydrate research 20080609 |
Catalytic enantioselective addition of diorganozinc reagents to vinyl sulfones. | Organic letters 20080605 |
Conjugation to hyperbranched polyglycerols improves RGD-mediated inhibition of platelet function in vitro. | Bioconjugate chemistry 20080601 |
Identification of a new class of nonpeptidic inhibitors of cruzain. | Journal of the American Chemical Society 20080521 |
Studies on the synthesis and unusual behavior of vinyl sulfone-modified hexenopyranosylthymines. | Carbohydrate research 20080519 |
Fasciola gigantica: evaluation of the effect of phenyl vinyl sulfone in vitro. | Experimental parasitology 20080501 |
Highly enantioselective asymmetric 1,3-dipolar cycloaddition of azomethine ylide catalyzed by a copper(I)/ClickFerrophos complex. | Organic letters 20080501 |
'Click' synthesis of small-molecule inhibitors targeting caspases. | Organic & biomolecular chemistry 20080307 |
Laccase immobilization on the tailored cellulose-based Granocel carriers. | International journal of biological macromolecules 20080301 |
Vinyl sulfones. | Acta crystallographica. Section C, Crystal structure communications 20080301 |
Hyaluronic acid gel fillers in the management of facial aging. | Clinical interventions in aging 20080301 |
Development of peptidomimetics with a vinyl sulfone warhead as irreversible falcipain-2 inhibitors. | Journal of medicinal chemistry 20080227 |
Interaction of pepsin with aromatic amino acids and their derivatives immobilized to Sepharose. | Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20080215 |
Carbon nanotubes as structural nanofibers for hyaluronic acid hydrogel scaffolds. | Biomacromolecules 20080201 |
Application and properties of butyl acrylate/pentaerythrite triacrylate copolymers and cellulose-based Granocel as carriers for trypsin immobilization. | Colloids and surfaces. B, Biointerfaces 20080115 |
Potency and selectivity of P2/P3-modified inhibitors of cysteine proteases from trypanosomes. | Bioorganic & medicinal chemistry letters 20080115 |
Fabrication and characterization of cross-linkable hydrogel particles based on hyaluronic acid: potential application in vocal fold regeneration. | Journal of biomaterials science. Polymer edition 20080101 |
The AAA+ superfamily of functionally diverse proteins. | Genome biology 20080101 |
[Procedure for obtaining and catalytic properties of trypsin immobilized in cryogels of polyvinyl alcohol]. | Prikladnaia biokhimiia i mikrobiologiia 20080101 |
[Subtilisin Carlsberg in complex with sodium dodecyl sulfate--an effective catalyst for the solid phase segment coupling of peptides on polyvinyl alcohol cryogel]. | Bioorganicheskaia khimiia 20080101 |
Comprehensive study of proteasome inhibitors against Plasmodium falciparum laboratory strains and field isolates from Gabon. | Malaria journal 20080101 |
Dipeptidyl alpha-fluorovinyl Michael acceptors: synthesis and activity against cysteine proteases. | Bioorganic & medicinal chemistry letters 20071201 |
Tandem conjugate addition-elimination for the diastereoselective synthesis of 4E-alkenyl syn-1,3-diols. | Organic letters 20071011 |
Michael acceptors as cysteine protease inhibitors. | Mini reviews in medicinal chemistry 20071001 |
Release of model proteins and basic fibroblast growth factor from in situ forming degradable dextran hydrogels. | Journal of controlled release : official journal of the Controlled Release Society 20070911 |
Use of hyaluronic acid fillers for the treatment of the aging face. | Clinical interventions in aging 20070901 |
Diastereoselective C-C bond formation at C-5 of vinyl sulfone-modified hex-5-enofuranosyl carbohydrates: diversity-oriented synthesis of branched-chain sugars and beyond. | The Journal of organic chemistry 20070720 |
A smart membrane based on an antigen-responsive hydrogel. | Biotechnology and bioengineering 20070701 |
Use of recombinant Entamoeba histolytica cysteine proteinase 1 to identify a potent inhibitor of amebic invasion in a human colonic model. | Eukaryotic cell 20070701 |
Evaluation of man-tailored cellulose-based carriers in glucoamylase immobilization. | Carbohydrate research 20070611 |
The vinyl-sulfonium bond in human myeloperoxidase: impact on compound I formation and reduction by halides and thiocyanate. | Biochemical and biophysical research communications 20070504 |
Rapidly in situ-forming degradable hydrogels from dextran thiols through Michael addition. | Biomacromolecules 20070501 |
Activity-based fingerprinting and inhibitor discovery of cysteine proteases in a microarray. | Chemical communications (Cambridge, England) 20070421 |
Effects of gamma-irradiation on physical and biologic properties of crosslinked hyaluronan tissue engineering scaffolds. | Tissue engineering 20070301 |
Schistosomiasis mansoni: novel chemotherapy using a cysteine protease inhibitor. | PLoS medicine 20070101 |
A highly selective synthesis of dialkenyl sulfones via cross-metathesis of divinyl sulfone. | Organic letters 20061207 |
Principles of soft tissue augmentation for the aging face. | Clinical interventions in aging 20061201 |
3,3'-bimorpholine derivatives as a new class of organocatalysts for asymmetric Michael addition. | Organic letters 20060608 |
Enantioselective construction of quaternary carbon centre catalysed by bifunctional organocatalyst. | Organic & biomolecular chemistry 20060607 |
Physical matrices stabilized by enzymatically sensitive covalent crosslinks. | Acta biomaterialia 20060501 |
Cobalt-catalyzed reductive coupling of saturated alkyl halides with activated alkenes. | The Journal of organic chemistry 20060120 |
Reuse of reactive dyes for dyeing of jute fabric. | Bioresource technology 20060101 |
Three-dimensional domain-swapped oligomers of ribonuclease A: identification of a fifth tetramer, pentamers and hexamers, and detection of trace heptameric, octameric and nonameric species. | Biochimica et biophysica acta 20060101 |
Inhibitors of cysteine proteases. | Current topics in medicinal chemistry 20060101 |
Functional inhibition of NF-kappaB signal transduction in alphavbeta3 integrin expressing endothelial cells by using RGD-PEG-modified adenovirus with a mutant IkappaB gene. | Arthritis research & therapy 20060101 |
A new antibody immobilization strategy based on electrodeposition of nanometer-sized hydroxyapatite for label-free capacitive immunosensor. | Talanta 20051115 |
Novel synthesis of 2-aryl and 2,3-disubstituted indoles by modified double elimination protocol. | Organic letters 20051013 |
A diastereoselective and general route to 5-amino-5-deoxysugars: influence of C-3 substitution on the addition of amines to C-5 of vinyl sulfone-modified hex-5-enofuranosyl carbohydrates. | The Journal of organic chemistry 20050930 |
Zn/CuI-mediated coupling of alkyl halides with vinyl sulfones, vinyl sulfonates, and vinyl sulfonamides. | The Journal of organic chemistry 20050819 |
Response of intestinal cells and macrophages to an orally administered cellulose-PEG based polymer as a potential treatment for intractable edemas. | Biomaterials 20050701 |
Effect of shear on intramolecular and intermolecular association during cross-linking of hydroxyethylcellulose in dilute aqueous solutions. | The journal of physical chemistry. B 20050630 |
Kinetics of degradation of sulphur mustard on impregnated carbons. | Journal of hazardous materials 20050520 |
Thiophilic paramagnetic particles as a batch separation medium for the purification of antibodies from various source materials. | Analytical biochemistry 20050315 |
Recombinant protein-co-PEG networks as cell-adhesive and proteolytically degradable hydrogel matrixes. Part I: Development and physicochemical characteristics. | Biomacromolecules 20050101 |
Synthesis and evaluation of hydrolyzable hyaluronan-tethered bupivacaine delivery systems. | Bioconjugate chemistry 20050101 |
Screening for selective small molecule inhibitors of the proteasome using activity-based probes. | Methods in enzymology 20050101 |
Reactions of sulphur mustard on impregnated carbons. | Journal of hazardous materials 20041231 |
Inhibitors of the eukaryotic 20S proteasome core particle: a structural approach. | Biochimica et biophysica acta 20041129 |
Peptidyl allyl sulfones: a new class of inhibitors for clan CA cysteine proteases. | Bioorganic & medicinal chemistry 20041001 |
Oligomerization of ribonuclease A: two novel three-dimensional domain-swapped tetramers. | The Journal of biological chemistry 20040827 |
Mercaptoheterocyclic ligands grafted on a poly(ethylene vinyl alcohol) membrane for the purification of immunoglobulin G in a salt independent thiophilic chromatography. | Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20040825 |
Selection of cysteine protease inhibitor-resistant malaria parasites is accompanied by amplification of falcipain genes and alteration in inhibitor transport. | The Journal of biological chemistry 20040820 |
Design and evaluation of inhibitors for dipeptidyl peptidase I (Cathepsin C). | Archives of biochemistry and biophysics 20040715 |
Divinyl sulfone as a postdigestion modifier for enhancing the a(1) Ion in MS/MS and postsource decay: potential applications in proteomics. | Analytical chemistry 20040715 |
Two stage biological treatment of a diazo reactive textile dye and the fate of the dye metabolites. | Chemosphere 20040701 |
Vinyl sulfones: inhibitors of SrtA, a transpeptidase required for cell wall protein anchoring and virulence in Staphylococcus aureus. | Journal of the American Chemical Society 20040324 |
Identification and biochemical characterization of vivapains, cysteine proteases of the malaria parasite Plasmodium vivax. | The Biochemical journal 20040301 |
Affinity chromatography of porcine pepsin and pepsinogen using immobilized ligands derived from the specific substrate for this enzyme. | Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20040205 |
Comparative study of thiophilic functionalised matrices for polyclonal F(ab')2 purification. | Journal of chromatography. A 20040102 |
Cellulose derivative-hyaluronic acid-based microporous hydrogels cross-linked through divinyl sulfone (DVS) to modulate equilibrium sorption capacity and network stability. | Biomacromolecules 20040101 |
Anti-inflammatory drug delivery from hyaluronic acid hydrogels. | Journal of biomaterials science. Polymer edition 20040101 |
Biomedical application of a superabsorbent hydrogel for body water elimination in the treatment of edemas. | Journal of biomedical materials research. Part A 20031201 |
Stereospecific rearrangements during the synthesis of pyrrolidines and related heterocycles from cyclizations of amino alcohols with vinyl Sulfones. | The Journal of organic chemistry 20031128 |
Combinatorial synthesis of a small-molecule library based on the vinyl sulfone scaffold. | Organic letters 20031113 |
Sortase from Staphylococcus aureus does not contain a thiolate-imidazolium ion pair in its active site. | The Journal of biological chemistry 20030905 |
Determination of aromatic and branched-chain amino acids in plasma by HPLC with electrogenerated Ru(bpy)3(3+) chemiluminescence detection. | Chemical & pharmaceutical bulletin 20030901 |
Phenylsulfonyl ene-allenes as efficient precursors to bicyclic systems via intramolecular [2 + 2]-cycloaddition reactions. | The Journal of organic chemistry 20030808 |
Identification and characterization of DEN1, a deneddylase of the ULP family. | The Journal of biological chemistry 20030801 |
Ultraviolet light-induced modification of crosslinked hyaluronan gels. | Journal of biomedical materials research. Part A 20030801 |
Structure and reactivity of an asymmetric complex between HslV and I-domain deleted HslU, a prokaryotic homolog of the eukaryotic proteasome. | Journal of molecular biology 20030704 |
Relative rates of Michael reactions of 2'-(phenethyl)thiol with vinyl sulfones, vinyl sulfonate esters, and vinyl sulfonamides relevant to vinyl sulfonyl cysteine protease inhibitors. | Organic letters 20030529 |
Anomeric configuration-directed diastereoselective C-C bond formation in vinyl sulfone-modified carbohydrates: a general route to branched-chain sugars. | Organic letters 20030417 |
Specificity determinants of human cathepsin s revealed by crystal structures of complexes. | Biochemistry 20030325 |
Vibrational frequencies and structural determinations of di-vinyl sulfone. | Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20030301 |
Lead discovery of alpha,beta-unsaturated sulfones from a combinatorial library as inhibitors of inducible VCAM-1 expression. | Bioorganic & medicinal chemistry letters 20030224 |
[Divinyl sulfone as a cross-linking reagent for oligomeric proteins]. | Bioorganicheskaia khimiia 20030101 |
Physical polymer matrices based on affinity interactions between peptides and polysaccharides. | Biomacromolecules 20030101 |
Expression, purification, crystallization and preliminary X-ray diffraction studies of human cathepsin F complexed with an irreversible vinyl sulfone inhibitor. | Acta crystallographica. Section D, Biological crystallography 20021201 |
Basic and reductive sulfone-directed ring-opening reactions of difluorinated oxa[2.2.1]bicycloheptanes. | Organic letters 20021114 |
The crystal structure of human cathepsin F and its implications for the development of novel immunomodulators. | Journal of molecular biology 20020920 |
Versatile 'traceless' sulfone linker for SPOS: preparation of isoxazolinopyrrole 2-carboxylates. | The Journal of organic chemistry 20020906 |
Regioselective reduction of 3-sulfonyl glutarimides to 3,4-dihydro-5-sulfonylpyridin-2-ones. Formal synthesis of the indolizidine 8a-epi-dendroprimine. | The Journal of organic chemistry 20020712 |
Double elimination protocol for synthesis of 5,6,11,12-tetradehydrodibenzo[a,e]cyclooctene. | Chemistry (Weinheim an der Bergstrasse, Germany) 20020503 |
Crystal structure of HslUV complexed with a vinyl sulfone inhibitor: corroboration of a proposed mechanism of allosteric activation of HslV by HslU. | Journal of molecular biology 20020503 |
Probing structural determinants distal to the site of hydrolysis that control substrate specificity of the 20S proteasome. | Chemistry & biology 20020501 |
Lectin-mediated drug delivery: binding and uptake of BSA-WGA conjugates using the Caco-2 model. | International journal of pharmaceutics 20020426 |
Aromatic amino acids and their derivatives as ligands for the isolation of aspartic proteinases. | Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20020425 |
Smooth muscle cell adhesion on crosslinked hyaluronan gels. | Journal of biomedical materials research 20020401 |
Homology modeling of falcipain-2: validation, de novo ligand design and synthesis of novel inhibitors. | Journal of biomolecular structure & dynamics 20020401 |
Vinyl sulfone bifunctional derivatives of DOTA allow sulfhydryl- or amino-directed coupling to antibodies. Conjugates retain immunoreactivity and have similar biodistributions. | Bioconjugate chemistry 20020101 |
Synthesis of sulfhydryl cross-linking poly(ethylene glycol)-peptides and glycopeptides as carriers for gene delivery. | Bioconjugate chemistry 20020101 |
Towards tissue engineering of a composite aortic valve. | Biomedical sciences instrumentation 20020101 |
Photoswitching of ligand association with a photoresponsive polymer-protein conjugate. | Bioconjugate chemistry 20020101 |
Heterogeneity of IgE epitopes of vinyl sulphone reactive dye: human serum albumin that react with IgE. | Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology 20011101 |
Active site mapping, biochemical properties and subcellular localization of rhodesain, the major cysteine protease of Trypanosoma brucei rhodesiense. | Molecular and biochemical parasitology 20011101 |
Extended peptide-based inhibitors efficiently target the proteasome and reveal overlapping specificities of the catalytic beta-subunits. | Chemistry & biology 20010901 |
Vinyl sulfones in solid-phase synthesis: preparation of 4,5,6,7-tetrahydroisoindole derivatives. | The Journal of organic chemistry 20010810 |
The major cysteine proteinase of Trypanosoma cruzi: a valid target for chemotherapy of Chagas disease. | Current pharmaceutical design 20010801 |
Role of skin prick test and serological measurement of specific IgE in the diagnosis of occupational asthma resulting from exposure to vinyl sulphone reactive dyes. | Occupational and environmental medicine 20010601 |
Affinity chromatography of porcine pepsin on different types of immobilized 3,5-diiodo-L-tyrosine. | Journal of chromatography. A 20010316 |
Cysteine protease activity is up-regulated in inflamed ankle joints of rats with adjuvant-induced arthritis and decreases with in vivo administration of a vinyl sulfone cysteine protease inhibitor. | Arthritis and rheumatism 20010301 |
Use of ion-exchange chromatography and hydrophobic interaction chromatography in the preparation and recovery of polyethylene glycol-linked proteins. | Journal of chromatography. A 20010126 |
Mechanistic investigation of smart polymer-protein conjugates. | Bioconjugate chemistry 20010101 |
Dipeptide vinyl sulfones suitable for intracellular inhibition of dipeptidyl peptidase I. | International immunopharmacology 20010101 |