Spiperone
Title | Journal |
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Pharmacokinetic and pharmacodynamic evaluation of 5-methoxy-2-aminoindane (MEAI): A new binge-mitigating agent. | Toxicology and applied pharmacology 20180315 |
The herbicide glyphosate causes behavioral changes and alterations in dopaminergic markers in male Sprague-Dawley rat. | Neurotoxicology 20150101 |
Role of somatodendritic and postsynaptic 5-HT₁A receptors on learning and memory functions in rats. | Neurochemical research 20121001 |
Syntheses and in vitro evaluation of decalinvesamicol analogues as potential imaging probes for vesicular acetylcholine transporter (VAChT). | Bioorganic & medicinal chemistry 20120815 |
Design, synthesis, and pharmacological evaluation of novel tetrahydroprotoberberine derivatives: selective inhibitors of dopamine D₁ receptor. | Bioorganic & medicinal chemistry 20120801 |
Pharmacokinetic-pharmacodynamic modeling of the D₂ and 5-HT (2A) receptor occupancy of risperidone and paliperidone in rats. | Pharmaceutical research 20120701 |
The restructuring of dopamine receptor subtype gene transcripts in c-fos KO mice. | Brain research bulletin 20120410 |
A novel G protein-coupled receptor of Schistosoma mansoni (SmGPR-3) is activated by dopamine and is widely expressed in the nervous system. | PLoS neglected tropical diseases 20120201 |
Synthesis, biological activities and bioavailability of moschamine, a safflomide-type phenylpropenoic acid amide found in Centaurea cyanus. | Natural product research 20120101 |
The influence of dopamine receptor d4 polymorphism on resting EEG in healthy young females. | The open neuroimaging journal 20120101 |
Distinct neurobehavioural effects of cannabidiol in transmembrane domain neuregulin 1 mutant mice. | PloS one 20120101 |
Dopamine D(2) Receptor-Mediated Heterologous Sensitization of AC5 Requires Signalosome Assembly. | Journal of signal transduction 20120101 |
Serotonin receptors in hippocampus. | TheScientificWorldJournal 20120101 |
Studies of olfactory system neural plasticity: the contribution of the unilateral naris occlusion technique. | Neural plasticity 20120101 |
Development of a bivalent dopamine D₂ receptor agonist. | Journal of medicinal chemistry 20111124 |
Dopamine as an anorectic neuromodulator in the cockroach Rhyparobia maderae. | The Journal of experimental biology 20111115 |
Involvement of the first transmembrane segment of human α(2) -adrenoceptors in the subtype-selective binding of chlorpromazine, spiperone and spiroxatrine. | British journal of pharmacology 20111101 |
Dopamine antagonists and brief vision distinguish lens-induced- and form-deprivation-induced myopia. | Experimental eye research 20111101 |
Roles of Non-cholinergic Intrapancreatic Nerves, Serotonergic Nerves, on Pancreatic Exocrine Secretion in the Isolated Perfused Rat Pancreas. | The Korean journal of physiology & pharmacology : official journal of the Korean Physiological Society and the Korean Society of Pharmacology 20111001 |
Absolute abundances and affinity states of dopamine receptors in mammalian brain: A review. | Synapse (New York, N.Y.) 20110901 |
Profiling of a prescription drug library for potential renal drug-drug interactions mediated by the organic cation transporter 2. | Journal of medicinal chemistry 20110714 |
Postnatal manganese exposure alters the expression of D2L and D2S receptor isoforms: relationship to PKA activity and Akt levels. | Synapse (New York, N.Y.) 20110701 |
Participation of cyclooxygenase pathway in the vasoconstriction induced by 5-HT in the in situ autoperfused kidney of long-term diabetic rats. | European journal of pharmacology 20110520 |
Wnt5a-dopamine D2 receptor interactions regulate dopamine neuron development via extracellular signal-regulated kinase (ERK) activation. | The Journal of biological chemistry 20110506 |
Melittin stimulates fatty acid release through non-phospholipase-mediated mechanisms and interacts with the dopamine transporter and other membrane-spanning proteins. | European journal of pharmacology 20110115 |
In vitro effects of both dopaminergic and enkephalinergic antagonists on the ovarian growth of Cherax quadricarinatus (Decapoda, Parastacidae), at different periods of the reproductive cycle. | Comparative biochemistry and physiology. Part A, Molecular & integrative physiology 20110101 |
Decreased striatal dopamine receptor binding in primary focal dystonia: a D2 or D3 defect? | Movement disorders : official journal of the Movement Disorder Society 20110101 |
Synthesis and SAR study of diphenylbutylpiperidines as cell autophagy inducers. | Bioorganic & medicinal chemistry letters 20110101 |
Molecular characterization of novel sulfotransferases from the tick, Ixodes scapularis. | BMC biochemistry 20110101 |
A novel role of protein tyrosine kinase2 in mediating chloride secretion in human airway epithelial cells. | PloS one 20110101 |
Serotonin and dopamine protect from hypothermia/rewarming damage through the CBS/H2S pathway. | PloS one 20110101 |
No evidence for strong recent positive selection favoring the 7 repeat allele of VNTR in the DRD4 gene. | PloS one 20110101 |
Dopamine and octopamine influence avoidance learning of honey bees in a place preference assay. | PloS one 20110101 |
Inverse agonism and its therapeutic significance. | Indian journal of pharmacology 20110101 |
Honey bee dopamine and octopamine receptors linked to intracellular calcium signaling have a close phylogenetic and pharmacological relationship. | PloS one 20110101 |
Inhibition of experimental myopia by a dopamine agonist: different effectiveness between form deprivation and hyperopic defocus in guinea pigs. | Molecular vision 20110101 |
Sequential mechanisms underlying concentration invariance in biological olfaction. | Frontiers in neuroengineering 20110101 |
Development of a microfluidic confocal fluorescence detection system for the hyphenation of nano-LC to on-line biochemical assays. | Analytical and bioanalytical chemistry 20101201 |
Dopaminergic agonists that result in ocular growth inhibition also elicit transient increases in choroidal thickness in chicks. | Experimental eye research 20101101 |
Synthesis and SAR studies of 1,4-benzoxazine MenB inhibitors: novel antibacterial agents against Mycobacterium tuberculosis. | Bioorganic & medicinal chemistry letters 20101101 |
The effect of bright light on lens compensation in chicks. | Investigative ophthalmology & visual science 20101001 |
Amphetamine regulates NR2B expression in Go2α knockout mice and thereby sustains behavioral sensitization. | Journal of neurochemistry 20101001 |
[(3)H]-F13640, a novel, selective and high-efficacy serotonin 5-HT(1A) receptor agonist radioligand. | Naunyn-Schmiedeberg's archives of pharmacology 20101001 |
Pharmacological profile of 5-hydroxytryptamine-induced inhibition on the pressor effect elicited by sympathetic stimulation in long-term diabetic pithed rats. | European journal of pharmacology 20100915 |
Dopamine beta-hydroxylase-deficient mice have normal densities of D(2) dopamine receptors in the high-affinity state based on in vivo PET imaging and in vitro radioligand binding. | Synapse (New York, N.Y.) 20100901 |
Dopamine inhibition of glycine release in the rat trigeminal nucleus pars caudalis: possible involvement of trace amine receptors. | Journal of neurochemistry 20100901 |
Inhibition of aldehyde dehydrogenase-2 suppresses cocaine seeking by generating THP, a cocaine use-dependent inhibitor of dopamine synthesis. | Nature medicine 20100901 |
Haloperidol, spiperone, pimozide and aripiprazole reduce intracellular dopamine content in PC12 cells and rat mesencephalic cultures: Implication of inhibition of vesicular transport. | European journal of pharmacology 20100825 |
Further delineation of hydrophobic binding sites in dopamine D(2)/D(3) receptors for N-4 substituents on the piperazine ring of the hybrid template 5/7-{[2-(4-aryl-piperazin-1-yl)-ethyl]-propyl-amino}-5,6,7,8-tetrahydro-naphthalen-2-ol. | Bioorganic & medicinal chemistry 20100801 |
Dopamine receptor alterations in female rats with diet-induced decreased brain docosahexaenoic acid (DHA): interactions with reproductive status. | Nutritional neuroscience 20100801 |
Increased 5-HT2A receptors in the temporal cortex of parkinsonian patients with visual hallucinations. | Movement disorders : official journal of the Movement Disorder Society 20100730 |
Leptin increases striatal dopamine D2 receptor binding in leptin-deficient obese (ob/ob) mice. | Synapse (New York, N.Y.) 20100701 |
Non-competitive interaction between raclopride and spiperone on human D-receptors in intact Chinese hamster ovary cells. | Fundamental & clinical pharmacology 20100601 |
Antagonist-D2S-dopamine receptor interactions in intact recombinant Chinese hamster ovary cells [corrected]. | Fundamental & clinical pharmacology 20100601 |
A 5-HT1A-like receptor is involved in the regulation of the embryonic rotation of Lymnaea stagnalis L. | Comparative biochemistry and physiology. Toxicology & pharmacology : CBP 20100601 |
Concentration of receptor and ligand revisited in a modified receptor binding protocol for high-affinity radioligands: [3H]Spiperone binding to D2 and D3 dopamine receptors. | Journal of neuroscience methods 20100430 |
Discovery of 4-(4-(2-((5-Hydroxy-1,2,3,4-tetrahydronaphthalen-2-yl)(propyl)amino)ethyl)piperazin-1-yl)quinolin-8-ol and its analogues as highly potent dopamine D2/D3 agonists and as iron chelator: in vivo activity indicates potential application in symptomatic and neuroprotective therapy for Parkinson's disease. | Journal of medicinal chemistry 20100311 |
Development of (S)-N6-(2-(4-(isoquinolin-1-yl)piperazin-1-yl)ethyl)-N6-propyl-4,5,6,7-tetrahydrobenzo[d]-thiazole-2,6-diamine and its analogue as a D3 receptor preferring agonist: potent in vivo activity in Parkinson's disease animal models. | Journal of medicinal chemistry 20100211 |
Effects of SCH23390 and spiperone administered into medial striatum and intermediate medial mesopallium on rewarding effects of morphine in day-old chicks. | European journal of pharmacology 20100210 |
JL13 has clozapine-like actions on thermoregulatory cutaneous blood flow in rats: Involvement of serotonin 5-HT1A and 5-HT2A receptor mechanisms. | Progress in neuro-psychopharmacology & biological psychiatry 20100201 |
Evidence for dopamine involvement in ambulation promoted by pulegone in mice. | Pharmacology, biochemistry, and behavior 20100201 |
Competition between 11C-raclopride and endogenous dopamine in Parkinson's disease. | Nuclear medicine communications 20100201 |
Serotonin regulates an acyl-CoA-binding protein (ACBP) gene expression in the midgut of Rhodnius prolixus. | Insect biochemistry and molecular biology 20100201 |
MDMA-evoked changes in the binding of dopamine D(2) receptor ligands in striatum of rats with unilateral serotonin depletion. | Synapse (New York, N.Y.) 20100101 |
Serotonin receptors are involved in the spinal mediation of descending facilitation of surgical incision-induced increase of Fos-like immunoreactivity in rats. | Molecular pain 20100101 |
Altered ratio of D1 and D2 dopamine receptors in mouse striatum is associated with behavioral sensitization to cocaine. | PloS one 20100101 |
Identification of a circadian clock-controlled neural pathway in the rabbit retina. | PloS one 20100101 |
Impact of RNA editing on functions of the serotonin 2C receptor in vivo. | Frontiers in neuroscience 20100101 |
Roles of aminergic neurons in formation and recall of associative memory in crickets. | Frontiers in behavioral neuroscience 20100101 |
Adverse drug effects in hospitalized elderly: data from the healthcare cost and utilization project. | Clinical pharmacology : advances and applications 20100101 |
Neuroprotective effects of pramipexole against tunicamycin-induced cell death in PC12 cells. | Clinical and experimental pharmacology & physiology 20091201 |
Microglial responses to dopamine in a cell culture model of Parkinson's disease. | Neurobiology of aging 20091101 |
Investigation of a dopamine receptor in Schistosoma mansoni: functional studies and immunolocalization. | Molecular and biochemical parasitology 20091101 |
Characterization of the contractile 5-hydroxytryptamine receptor in the autoperfused kidney of L-NAME hypertensive rats. | European journal of pharmacology 20091012 |
Physical binding pocket induction for affinity prediction. | Journal of medicinal chemistry 20091008 |
Mutant 5-hydroxytryptamine 1A receptor D116A is a receptor activated solely by synthetic ligands with a rich pharmacology. | The Journal of pharmacology and experimental therapeutics 20091001 |
Dopamine D2, D3, and D4 selective phenylpiperazines as molecular probes to explore the origins of subtype specific receptor binding. | Journal of medicinal chemistry 20090813 |
Rats self-administer intravenous nicotine delivered in a novel smoking-relevant procedure: effects of dopamine antagonists. | The Journal of pharmacology and experimental therapeutics 20090801 |
Overexpression of 5-HT2C receptors in forebrain leads to elevated anxiety and hypoactivity. | The European journal of neuroscience 20090701 |
Automated on-line in-tube solid-phase microextraction coupled with HPLC/MS/MS for the determination of butyrophenone derivatives in human plasma. | Analytical and bioanalytical chemistry 20090601 |
Platelet dopamine: D2 receptor binding in patients with migraine. | Cephalalgia : an international journal of headache 20090501 |
Role of the serotoninergic system in the development of diseases of the intestinal and biliferous tracts. | Bulletin of experimental biology and medicine 20090501 |
Early deprivation leads to long-term reductions in motivation for reward and 5-HT1A binding and both effects are reversed by fluoxetine. | Neuropharmacology 20090301 |
Pulp and paper mill effluents contain neuroactive substances that potentially disrupt neuroendocrine control of fish reproduction. | Environmental science & technology 20090301 |
Activation of serotonin 5-HT1-receptors decreased gripping-induced immobility episodes in taiep rats. | Neuroscience letters 20090109 |
Evidence for dopamine involvement in ambulation promoted by menthone in mice. | Pharmacology, biochemistry, and behavior 20090101 |
Spiperone, identified through compound screening, activates calcium-dependent chloride secretion in the airway. | American journal of physiology. Cell physiology 20090101 |
Species differences in the relative densities of D1- and D2-like dopamine receptor subtypes in the Japanese quail and rats: an in vitro quantitative receptor autoradiography study. | Brain, behavior and evolution 20090101 |
The importance of brain banks for molecular neuropathological research: The New South Wales Tissue Resource Centre experience. | International journal of molecular sciences 20090101 |
5-HT-induced depression of the spinal monosynaptic reflex potential utilizes different types of 5-HT receptors depending on Mg2+ availability. | Pharmacological reports : PR 20090101 |
The role of dopamine in Drosophila larval classical olfactory conditioning. | PloS one 20090101 |
Roles of octopaminergic and dopaminergic neurons in appetitive and aversive memory recall in an insect. | BMC biology 20090101 |
Selective deletion of PTEN in dopamine neurons leads to trophic effects and adaptation of striatal medium spiny projecting neurons. | PloS one 20090101 |
Spiperone enhances intracellular calcium level and inhibits the Wnt signaling pathway. | BMC pharmacology 20090101 |
Serotomide and safflomide modulate forskolin-stimulated cAMP formation via 5-HT1 receptor. | Phytomedicine : international journal of phytotherapy and phytopharmacology 20081201 |
The antipsychotic spiperone attenuates inflammatory response in cultured microglia via the reduction of proinflammatory cytokine expression and nitric oxide production. | Journal of neurochemistry 20081201 |
Targeting liver myofibroblasts: a novel approach in anti-fibrogenic therapy. | Hepatology international 20081201 |
Chemical substructures that enrich for biological activity. | Bioinformatics (Oxford, England) 20081101 |
Effects of selective serotonin2 ligands on behaviors evoked by stress in the rat. | Pharmacology, biochemistry, and behavior 20081001 |
Dopamine D1 receptor inhibition of NMDA receptor currents mediated by tyrosine kinase-dependent receptor trafficking in neonatal rat striatum. | The Journal of physiology 20081001 |
Altered dopamine D2-like receptor binding in rats with behavioral sensitization to quinpirole: effects of pre-treatment with Ro 41-1049. | European journal of pharmacology 20080911 |
Characterization of contractile 5-hydroxytryptamine receptor subtypes in the in situ autoperfused kidney in the anaesthetized rat. | European journal of pharmacology 20080911 |
Serotonin receptors contribute to the promnesic effects of P. olacoides (Marapuama). | Physiology & behavior 20080903 |
11C-NMSP/ 18F-FDG microPET to monitor neural stem cell transplantation in a rat model of traumatic brain injury. | European journal of nuclear medicine and molecular imaging 20080901 |
Selective alterations of brain dopamine D(2) receptor binding in cirrhotic patients: results of a (11)C-N-methylspiperone PET study. | Metabolic brain disease 20080901 |
Induction of ovarian growth in Aegla platensis (Crustacea, Aeglidae) by means of neuroregulators incorporated to food. | Revista de biologia tropical 20080901 |
Increased dopamine after mating impairs olfaction and prevents odor interference with pregnancy. | Nature neuroscience 20080801 |
Serotoninergic system in the development of pyloric stenosis and pancreatitis. | Bulletin of experimental biology and medicine 20080801 |
When administered to rats in a cold environment, 3,4-methylenedioxymethamphetamine reduces brown adipose tissue thermogenesis and increases tail blood flow: effects of pretreatment with 5-HT1A and dopamine D2 antagonists. | Neuroscience 20080717 |
Synthesis and pharmacological investigation of novel 2-aminothiazole-privileged aporphines. | Bioorganic & medicinal chemistry 20080715 |
Dopamine receptors in the anterior insular cortex modulate long-term nociception in the rat. | European journal of pain (London, England) 20080701 |
Mechanisms for metoclopramide-mediated sensitization and haloperidol-induced catalepsy in rats. | European journal of pharmacology 20080610 |
Antagonist-radioligand binding to D2L-receptors in intact cells. | Biochemical pharmacology 20080601 |
Bioisosteric heterocyclic versions of 7-{[2-(4-phenyl-piperazin-1-yl)ethyl]propylamino}-5,6,7,8-tetrahydronaphthalen-2-ol: identification of highly potent and selective agonists for dopamine D3 receptor with potent in vivo activity. | Journal of medicinal chemistry 20080522 |
Dopamine determines the vulnerability of striatal neurons to the N-terminal fragment of mutant huntingtin through the regulation of mitochondrial complex II. | Human molecular genetics 20080515 |
Dopamine D4 receptors regulate intracellular calcium concentration in cultured chicken cone photoreceptor cells: relationship to dopamine receptor-mediated inhibition of cAMP formation. | Brain research 20080501 |
Dopamine D2(High) receptors on intact cells. | Synapse (New York, N.Y.) 20080401 |
Characterization of functional roles of DRY motif in the 2nd intracellular loop of dopamine D2 and D3 receptors. | Archives of pharmacal research 20080401 |
PET analysis of the 5-HT2A receptor inverse agonist ACP-103 in human brain. | The international journal of neuropsychopharmacology 20080301 |
Pergolide protects CA1 neurons from apoptosis in a gerbil model of global cerebral ischemia. | Neurological research 20080201 |
Further structure-activity relationships study of hybrid 7-{[2-(4-phenylpiperazin-1-yl)ethyl]propylamino}-5,6,7,8-tetrahydronaphthalen-2-ol analogues: identification of a high-affinity D3-preferring agonist with potent in vivo activity with long duration of action. | Journal of medicinal chemistry 20080110 |
Food restriction markedly increases dopamine D2 receptor (D2R) in a rat model of obesity as assessed with in-vivo muPET imaging ([11C] raclopride) and in-vitro ([3H] spiperone) autoradiography. | Synapse (New York, N.Y.) 20080101 |
A review of imaging techniques for systems biology. | BMC systems biology 20080101 |
The neuropharmacology of (-)-stepholidine and its potential applications. | Current neuropharmacology 20071201 |
Possible involvement of endogenous 5-HT in aggravation of cerulein-induced acute pancreatitis in mice. | Journal of pharmacological sciences 20071101 |
Chronic SKF83959 induced less severe dyskinesia and attenuated L-DOPA-induced dyskinesia in 6-OHDA-lesioned rat model of Parkinson's disease. | Neuropharmacology 20070701 |
Dopamine D2 receptor stimulation inhibits cold-initiated thermogenesis in brown adipose tissue in conscious rats. | Neuroscience 20070615 |
Frontal-subcortical circuitry and behavior. | Dialogues in clinical neuroscience 20070601 |
Dopamine stimulates 45Ca2+ uptake through cAMP, PLC/PKC, and MAPKs in renal proximal tubule cells. | Journal of cellular physiology 20070501 |
Activation of dopamine D2 receptors in the CNS inhibits sympathetic cutaneous vasomotor alerting responses (SCVARs), contributing to clozapine's SCVAR-inhibiting action. | Progress in neuro-psychopharmacology & biological psychiatry 20070330 |
Acute and chronic administration of the cannabinoid receptor agonist CP 55,940 attenuates tumor-evoked hyperalgesia. | European journal of pharmacology 20070308 |
Native rat hippocampal 5-HT1A receptors show constitutive activity. | Molecular pharmacology 20070301 |
Screening of 5-HT1A receptor antagonists using molecularly imprinted polymers. | Journal of the American Chemical Society 20070214 |
Striatal serotonin depletion facilitates rat egocentric learning via dopamine modulation. | European journal of pharmacology 20070205 |
Changes in levels of D1, D2, or NMDA receptors during withdrawal from brief or extended daily access to IV cocaine. | Brain research 20070202 |
Aversive learning in honeybees revealed by the olfactory conditioning of the sting extension reflex. | PloS one 20070101 |
[Implication of serotonin in the regulation of hemostasis in the experiment]. | Anesteziologiia i reanimatologiia 20070101 |
Tracer coupling between fish rod horizontal cells: modulation by light and dopamine but not the retinal circadian clock. | Visual neuroscience 20070101 |
Synthesis of two potential NK1-receptor ligands using [1-11C]ethyl iodide and [1-11C]propyl iodide and initial PET-imaging. | BMC medical imaging 20070101 |
[The role of the serotoninergic system in the pathogenesis of experimental ulcerous colitis]. | Vestnik Rossiiskoi akademii meditsinskikh nauk 20070101 |
A positron emission tomography study on the role of nigral lesions in parkinsonism in patients with amyotrophic lateral sclerosis. | Archives of neurology 20061201 |
Ptychodiscus brevis toxin-induced depression of spinal reflexes involves 5-HT via 5-HT3 receptors modulated by NMDA receptor. | Neuroscience letters 20061127 |
Naloxone-blocked depriming effect of anxiolytic selank on apomorphine-induced behavioral manifestations of hyperfunction of dopamine system. | Bulletin of experimental biology and medicine 20061101 |
Perospirone is a new generation antipsychotic: evidence from a positron emission tomography study of serotonin 2 and D2 receptor occupancy in the living human brain. | Journal of clinical psychopharmacology 20061001 |
Roles of octopaminergic and dopaminergic neurons in mediating reward and punishment signals in insect visual learning. | The European journal of neuroscience 20061001 |
Dopamine D2 receptor-mediated G protein activation assessed by agonist-stimulated [35S]guanosine 5'-O-(gamma-thiotriphosphate) binding in rat striatal membranes. | Progress in neuro-psychopharmacology & biological psychiatry 20060930 |
Association of caffeine to MDMA does not increase antinociception but potentiates adverse effects of this recreational drug. | Brain research 20060921 |
Sympathetic neurotransmission in the rat testicular capsule: functional characterization and identification of mRNA encoding alpha1-adrenoceptor subtypes. | European journal of pharmacology 20060814 |
Fluorescence studies reveal heterodimerization of dopamine D1 and D2 receptors in the plasma membrane. | Biochemistry 20060725 |
Dopaminergic regulation of ion transport in gills of the euryhaline semiterrestrial crab Chasmagnathus granulatus: interaction between D1- and D2-like receptors. | The Journal of experimental biology 20060701 |
Effects of dopamine D1-like receptor agonists on food-maintained operant behavior in rats. | Behavioural pharmacology 20060601 |
Comparison of rat dopamine D2 receptor occupancy for a series of antipsychotic drugs measured using radiolabeled or nonlabeled raclopride tracer. | Life sciences 20060522 |
Microsphere-based protease assays and screening application for lethal factor and factor Xa. | Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501 |
Serotonin receptor antagonists discriminate between PKA- and PKC-mediated plasticity in aplysia sensory neurons. | Journal of neurophysiology 20060401 |
Pharmacological characterization of 5-hydroxytryptamine-induced contraction in the chicken gastrointestinal tract. | Autonomic & autacoid pharmacology 20060401 |
Dopamine D(2) receptor activation modulates perceived odor intensity. | Behavioral neuroscience 20060401 |
Potential vascular alpha1-adrenoceptor blocking properties of an array of 5-HT receptor ligands in the rat. | European journal of pharmacology 20060327 |
Transient and selective overexpression of dopamine D2 receptors in the striatum causes persistent abnormalities in prefrontal cortex functioning. | Neuron 20060216 |
Dopamine, oxytocin, and vasopressin receptor binding in the medial prefrontal cortex of monogamous and promiscuous voles. | Neuroscience letters 20060213 |
Simultaneous analysis of haloperidol, its three metabolites and two other butyrophenone-type neuroleptics by high performance liquid chromatography with dual ultraviolet detection. | Biomedical chromatography : BMC 20060201 |
D2-like receptors mediate the expulsion phase of ejaculation elicited by 8-hydroxy-2-(di-N-propylamino)tetralin in rats. | The Journal of pharmacology and experimental therapeutics 20060201 |
Synthesis and binding profile of constrained analogues of N-[4-(4-arylpiperazin-1-yl)butyl]-3-methoxybenzamides, a class of potent dopamine D3 receptor ligands. | The Journal of pharmacy and pharmacology 20060201 |
Differential effects of cocaine-induced seizures and lethality on M(1)-like muscarinic and dopaminergic D (1)- and D (2)-like binding receptors in mice brain. | Cellular and molecular neurobiology 20060201 |
Investigation of the alternatively spliced insert region of the D2L dopamine receptor by epitope substitution. | Neuroscience letters 20060130 |
Investigation of cooperativity in the binding of ligands to the D(2) dopamine receptor. | Molecular pharmacology 20060101 |
Structural determinants of pharmacological specificity between D(1) and D(2) dopamine receptors. | Molecular pharmacology 20060101 |
Pramipexole protects against H2O2-induced PC12 cell death. | Naunyn-Schmiedeberg's archives of pharmacology 20060101 |
Influence of human B-casomorphin-7 on specific binding of 3H-spiperone to the 5-HT2-receptors of rat brain frontal cortex. | Protein and peptide letters 20060101 |
Serotonin 5-HT2A and 5-HT6 receptors in the prefrontal cortex of Alzheimer and normal aging patients. | BMC neuroscience 20060101 |
Dopamine presynaptically and heterogeneously modulates nucleus accumbens medium-spiny neuron GABA synapses in vitro. | BMC neuroscience 20060101 |
Interaction between different parts of the autonomic nervous system in the regulation of smooth muscles in the femoral artery and trachea. | Bulletin of experimental biology and medicine 20060101 |
Dibenzazecine compounds with a novel dopamine/5HT2A receptor profile and 3D-QSAR analysis. | BMC pharmacology 20060101 |
Review of F-FDG Synthesis and Quality Control. | Biomedical imaging and intervention journal 20060101 |
Modifications in muscarinic, dopaminergic and serotonergic receptors concentrations in the hippocampus and striatum of epileptic rats. | Life sciences 20051205 |
Reactions between beta-casomorphins-7 and 5-HT2-serotonin receptors. | Bulletin of experimental biology and medicine 20051101 |
8-(Heteroaryl)phenalkyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-ones as opioid receptor modulators. | Medicinal chemistry (Shariqah (United Arab Emirates)) 20051101 |
Differential in vivo inhibition of [3H]nemonapride binding by atypical antipsychotics in rat striatum, olfactory lobes, and frontal cortex. | Pharmacology 20051001 |
Competitive MS binding assays for dopamine D2 receptors employing spiperone as a native marker. | Chembiochem : a European journal of chemical biology 20051001 |
KKHA-761, a potent D3 receptor antagonist with high 5-HT1A receptor affinity, exhibits antipsychotic properties in animal models of schizophrenia. | Pharmacology, biochemistry, and behavior 20051001 |
Participation of octopaminergic reward system and dopaminergic punishment system in insect olfactory learning revealed by pharmacological study. | The European journal of neuroscience 20050901 |
Cognitive effects of dopaminergic and glutamatergic blockade in nucleus accumbens in pigeons. | Pharmacology, biochemistry, and behavior 20050801 |
N1/P2 component of auditory evoked potential reflect changes of the brain serotonin biosynthesis in rats. | Nutritional neuroscience 20050801 |
2-[4-(3,4-Dimethylphenyl)piperazin-1-ylmethyl]-1H benzoimidazole (A-381393), a selective dopamine D4 receptor antagonist. | Neuropharmacology 20050701 |
Reciprocal mutations in TM2/TM3 in a D2 dopamine receptor background confirms the importance of this microdomain as a selective determinant of para-halogenated 1,4-disubstituted aromatic piperazines. | Archiv der Pharmazie 20050601 |
Chirospecific and subtype selective dopamine receptor binding of heterocyclic methoxynaphthamide analogs. | Archiv der Pharmazie 20050601 |
Effects of mercury on neurochemical receptors in wild river otters (Lontra canadensis). | Environmental science & technology 20050515 |
Enhanced binding of dopamine D1 receptors in caudate-putamen subregions in High-Yawning Sprague-Dawley rats. | Synapse (New York, N.Y.) 20050501 |
Mechanisms of inverse agonist action at D2 dopamine receptors. | British journal of pharmacology 20050501 |
Dopamine D2 receptor stimulation of mitogen-activated protein kinases mediated by cell type-dependent transactivation of receptor tyrosine kinases. | Journal of neurochemistry 20050501 |
Dopamine receptor activation in bovine pinealocyte via a cAMP-dependent transcription pathway. | Journal of pineal research 20050401 |
The role of the phosphatidyinositol-linked D1 dopamine receptor in the pharmacology of SKF83959. | Pharmacology, biochemistry, and behavior 20050401 |
Estrogen mediated inhibition of dopamine transport in the striatum: regulation by G alpha i/o. | European journal of pharmacology 20050328 |
Stimulation of 5-HT1A receptor with 8-OH-DPAT inhibits hydrogen peroxide-induced neurotoxicity in cultured rat cortical cells. | Pharmacological research 20050301 |
Modeling the similarity and divergence of dopamine D2-like receptors and identification of validated ligand-receptor complexes. | Journal of medicinal chemistry 20050210 |
Developmental neurotoxicity of pyrethroid insecticides: critical review and future research needs. | Environmental health perspectives 20050201 |
Distribution of D1-like and D2-like dopamine receptors in the brain of genetic epileptic WAG/Rij rats. | Epilepsy research 20050201 |
Effect of dopamine injection into caudate nucleus on immune responsiveness in rats: a pilot study. | Immunology letters 20050115 |
Synthesis and structure-activity relationships of 1-aralkyl-4-benzylpiperidine and 1-aralkyl-4-benzylpiperazine derivatives as potent sigma ligands. | Journal of medicinal chemistry 20050113 |
Effects of long-term biogenic amine transporter blockade on receptor/G-protein coupling in rat brain. | Neuropharmacology 20050101 |
Prenatal ethanol preferentially enhances reactivity of the dopamine D1 but not D2 or D3 receptors in offspring. | Neurotoxicology and teratology 20050101 |
Evidence for 5-HT2B and 5-HT7 receptor-mediated relaxation in pulmonary arteries of weaned pigs. | Naunyn-Schmiedeberg's archives of pharmacology 20050101 |
Behavioral and neurochemical effects on rat offspring after prenatal exposure to ethanol. | Neurotoxicology and teratology 20050101 |
Biphasic firing response of nucleus accumbens neurons elicited by THPB-18 and its correlation with DA receptor subtypes. | Acta pharmacologica Sinica 20041201 |
Aglycemia and ischemia depress monosynaptic and polysynaptic reflexes in neonatal rat spinal cord in vitro by involving different types of 5-hydroxytryptamine receptors. | Neuroscience letters 20041130 |
Atypical properties of several classes of antipsychotic drugs on the basis of differential induction of Fos-like immunoreactivity in the rat brain. | Life sciences 20041126 |
Targeted mutation of CCK(2) receptor gene antagonises behavioural changes induced by social isolation in female, but not in male mice. | Behavioural brain research 20041105 |
The influence of G protein subtype on agonist action at D2 dopamine receptors. | Neuropharmacology 20041101 |
Reduced hypophagic effects of d-fenfluramine and the 5-HT2C receptor agonist mCPP in 5-HT1B receptor knockout mice. | Psychopharmacology 20041001 |
Cloned human 5-HT1A receptor pharmacology determined using agonist binding and measurement of cAMP accumulation. | The Journal of pharmacy and pharmacology 20041001 |
MDMA-evoked changes in [11C]raclopride and [11C]NMSP binding in living pig brain. | Synapse (New York, N.Y.) 20040915 |
Cerebral D2 and 5-HT2 receptor occupancy in Schizophrenic patients treated with olanzapine or clozapine. | Journal of psychopharmacology (Oxford, England) 20040901 |
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors. | Naunyn-Schmiedeberg's archives of pharmacology 20040801 |
Novel regulatory properties of human type 9 adenylate cyclase. | The Journal of pharmacology and experimental therapeutics 20040701 |
Electrostatic surface potential calculation on several new halogenated benzimidazole-like dopaminergic ligands. | Archiv der Pharmazie 20040701 |
Early administration of tiapride to young rats without long-lasting changes in the development of the dopaminergic system. | Pharmacopsychiatry 20040701 |
Lack of restraint-induced increases of brain serotonin metabolism in rats treated with spiperone: relationship with restraint-induced behavioral deficits. | Pakistan journal of pharmaceutical sciences 20040701 |
Vasoconstrictor responses to 5-hydroxytryptamine in the autoperfused hindquarters of spontaneously hypertensive rats. | Pharmacology 20040601 |
Measurement of dopamine D2-like receptors in postmortem CNS and pituitary: differential regional changes in schizophrenia. | Life sciences 20040507 |
Investigation of the mechanism of agonist and inverse agonist action at D2 dopamine receptors. | Biochemical pharmacology 20040501 |
Antipsychotic drugs influence transport of the beta-adrenergic antagonist [3H]-dihydroalprenolol into neuronal and blood cells. | The world journal of biological psychiatry : the official journal of the World Federation of Societies of Biological Psychiatry 20040401 |
Micro-positron emission tomography imaging of cardiac gene expression in rats using bicistronic adenoviral vector-mediated gene delivery. | Circulation 20040323 |
Evidence that alpha(1B)-adrenoceptors are involved in noradrenaline-induced contractions of rat tail artery. | European journal of pharmacology 20040319 |
Pharmacological properties of serotonin receptor subtypes mediating contraction of bovine inferior alveolar arteries. | Archives of oral biology 20040301 |
Opposing effects of D1 and D2 receptor activation on odor discrimination learning. | Behavioral neuroscience 20040201 |
Cocaine treatment causes early and long-lasting changes in muscarinic and dopaminergic receptors. | Cellular and molecular neurobiology 20040201 |
A circadian clock in the fish retina regulates dopamine release via activation of melatonin receptors. | The Journal of physiology 20040115 |
Sensitization of neuronal A2A adenosine receptors after persistent D2 dopamine receptor activation. | The Journal of pharmacology and experimental therapeutics 20040101 |
Postnatal haloperidol eliminates the deficit in circling behavior produced by prenatal exposure to the same drug. | Neurotoxicology and teratology 20040101 |
Comparison of brain activity between dopamine D2 receptor-knockout and wild mice in response to dopamine agonist and antagonist assessed by fMRI. | Neuro-Signals 20040101 |
Optimization of the pharmacophore model for 5-HT7R antagonism. Design and synthesis of new naphtholactam and naphthosultam derivatives. | Journal of medicinal chemistry 20031218 |
Direct activation by dopamine of recombinant human 5-HT1A receptors: comparison with human 5-HT2C and 5-HT3 receptors. | Synapse (New York, N.Y.) 20031215 |
Absence of circadian clock regulation of horizontal cell gap junctional coupling reveals two dopamine systems in the goldfish retina. | The Journal of comparative neurology 20031208 |
Elevated neuronal nitric oxide synthase expression in chronic haloperidol-treated rats. | Neuropharmacology 20031201 |
Pharmacological characterization of a serotonin receptor (5-HT7) stimulating cAMP production in human corneal epithelial cells. | Investigative ophthalmology & visual science 20031101 |
Human umbilical vein vasoconstriction induced by epinephrine acting on alpha1B-adrenoceptor subtype. | American journal of obstetrics and gynecology 20031101 |
[Effects of D1 and D2 dopamine receptor agonists and antagonists on cerebral ischemia/reperfusion injury]. | Sheng li xue bao : [Acta physiologica Sinica] 20031025 |
Molecular modeling of the three-dimensional structure of dopamine 3 (D3) subtype receptor: discovery of novel and potent D3 ligands through a hybrid pharmacophore- and structure-based database searching approach. | Journal of medicinal chemistry 20031009 |
Effects of D1- and D2-dopamine receptor activation on melatonin synthesis in bovine pinealocytes. | Journal of pineal research 20031001 |
Pilocarpine-induced seizures in adult rats: monoamine content and muscarinic and dopaminergic receptor changes in the striatum. | Comparative biochemistry and physiology. Toxicology & pharmacology : CBP 20031001 |
Dopamine displaces [3H]domperidone from high-affinity sites of the dopamine D2 receptor, but not [3H]raclopride or [3H]spiperone in isotonic medium: Implications for human positron emission tomography. | Synapse (New York, N.Y.) 20030915 |
Comparison of hippocampal G protein activation by 5-HT(1A) receptor agonists and the atypical antipsychotics clozapine and S16924. | Naunyn-Schmiedeberg's archives of pharmacology 20030901 |
Pharmacologic identification of putative D1 dopamine receptors in feline kidneys. | Journal of veterinary pharmacology and therapeutics 20030801 |
Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7). | Journal of medicinal chemistry 20030703 |
Characterization of dopamine D2 receptor gene expression and binding sites in human placenta amniotic epithelial cells. | Placenta 20030701 |
Pharmacological analysis of a dopamine D(2Short):G(alphao) fusion protein expressed in Sf9 cells. | FEBS letters 20030619 |
Distinct effects of amantadine and memantine on dopaminergic transmission in the rat striatum. | Neuroscience letters 20030612 |
Pharmacological and functional characterisation of dopamine D4 receptors in the rat retina. | Neuropharmacology 20030601 |
Sigma1 and dopamine D2 receptor occupancy in the mouse brain after a single administration of haloperidol and two dopamine D2-like receptor ligands. | Nuclear medicine and biology 20030501 |
5-HT(2A) receptor binding is reduced in drug-naive and unchanged in SSRI-responder depressed patients compared to healthy controls: a PET study. | Psychopharmacology 20030401 |
Interaction of the D2short dopamine receptor with G proteins: analysis of receptor/G protein selectivity. | Biochemical pharmacology 20030401 |
Photic regulation of heme oxygenase activity in the golden hamster retina: involvement of dopamine. | Journal of neurochemistry 20030401 |
Effect of sabcomeline on muscarinic and dopamine receptor binding in intact mouse brain. | Annals of nuclear medicine 20030401 |
Biphasic role of dopamine on female sexual behaviour via D2 receptors in the mediobasal hypothalamus. | Neuropharmacology 20030301 |
Pharmacological characterization of an adenylyl cyclase-coupled 5-HT receptor in aplysia: comparison with mammalian 5-HT receptors. | Journal of neurophysiology 20030301 |
5-HT7 receptor-mediated relaxation of the oviduct in nonpregnant proestrus pigs. | European journal of pharmacology 20030214 |
In vivo evidence for dopamine-mediated internalization of D2-receptors after amphetamine: differential findings with [3H]raclopride versus [3H]spiperone. | Molecular pharmacology 20030201 |
GABA(A) alpha 1 subunit knock-out mice do not show a hyperlocomotor response following amphetamine or cocaine treatment. | Neuropharmacology 20030201 |
CCK2 receptor-deficient mice have increased sensitivity of dopamine D2 receptors. | Neuropeptides 20030201 |
5-HT(2) receptor-mediated phosphoinositide hydrolysis in bovine ciliary epithelium. | Journal of ocular pharmacology and therapeutics : the official journal of the Association for Ocular Pharmacology and Therapeutics 20030201 |
Evidence for the involvement of dopamine in ambulation promoted by menthol in mice. | Journal of pharmacological sciences 20030201 |
Characterization of the 5-hydroxytryptamine receptors mediating contraction in the pig isolated intravesical ureter. | British journal of pharmacology 20030101 |
Corticotropin-releasing factor as well as opioid and dopamine are involved in tail-pinch-induced food intake of rats. | Neuroscience 20030101 |
Behavioral response profiles following drug challenge with dopamine receptor subtype agonists and antagonists in developing rat. | Neurotoxicology and teratology 20030101 |
Axonal degeneration and progressive neurologic disability in multiple sclerosis. | Neurotoxicity research 20030101 |
Kinetics of synaptic transfer from rods and cones to horizontal cells in the salamander retina. | Neuroscience 20030101 |
Targeted molecular imaging. | Korean journal of radiology 20030101 |
The role of catecholamines in retention performance of a partially baited radial eight-arm maze for rats. | The Chinese journal of physiology 20021231 |
Novel (bisarylmethoxy)butylpiperidine analogues as neurotransmitter transporter inhibitors with activity at dopamine receptor sites. | Bioorganic & medicinal chemistry 20021201 |
Inhibition of protein tyrosine/mitogen-activated protein kinase phosphatase activity is associated with D2 dopamine receptor supersensitivity in a rat model of Parkinson's disease. | Molecular pharmacology 20021201 |
Characterization of 5-HT receptor subtypes mediating contraction in human umbilical vein. 1. Evidence of involvement of 5-HT2A receptors using functional and radioligand binding assays. | Naunyn-Schmiedeberg's archives of pharmacology 20021201 |
Functional cooperation between neurosteroids and D2 dopamine antagonists on KCl-evoked [3H]noradrenaline release: modulation by calcium channel blockers. | Journal of neuroendocrinology 20021201 |
Serotonin-induced MMP-13 production is mediated via phospholipase C, protein kinase C, and ERK1/2 in rat uterine smooth muscle cells. | The Journal of biological chemistry 20021108 |
Dopamine mediates circadian clock regulation of rod and cone input to fish retinal horizontal cells. | The Journal of physiology 20021101 |
In vivo serotonin 5HT(2A) receptor binding and personality traits in healthy subjects: a positron emission tomography study. | NeuroImage 20021101 |
Changes in electrophysiological properties of lamprey spinal motoneurons during fictive swimming. | Journal of neurophysiology 20021101 |
Spreading depression: imaging and blockade in the rat neocortical brain slice. | Journal of neurophysiology 20021101 |
Apomorphine induces trophic factors that support fetal rat mesencephalic dopaminergic neurons in cultures. | The European journal of neuroscience 20021101 |
Effect of nooglutil on benzodiazepine withdrawal syndrome and binding of 3H-spiperone with D2 receptors in rat striatum. | Bulletin of experimental biology and medicine 20021101 |
Synthesis and structure-activity relationship of the isoindolinyl benzisoxazolpiperidines as potent, selective, and orally active human dopamine D4 receptor antagonists. | Chembiochem : a European journal of chemical biology 20021004 |
Antibody capture assay reveals bell-shaped concentration-response isotherms for h5-HT(1A) receptor-mediated Galpha(i3) activation: conformational selection by high-efficacy agonists, and relationship to trafficking of receptor signaling. | Molecular pharmacology 20020901 |
Development of an automated system for synthesizing 18F-labeled compounds using [18F]fluoroethyl bromide as a synthetic precursor. | Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine 20020901 |
Effects of rolipram on in vivo dopamine receptor binding. | Journal of neural transmission (Vienna, Austria : 1996) 20020901 |
Metachlorophenylpiperazine (m-CPP) induced intracavernous pressure responses in anaesthetized rats. | International journal of impotence research 20020801 |
Aripiprazole, a novel antipsychotic, is a high-affinity partial agonist at human dopamine D2 receptors. | The Journal of pharmacology and experimental therapeutics 20020701 |
Effects of intrathecal injection of diatrizoate on dopamine receptors. | Academic radiology 20020701 |
Ketanserin and spiperone as templates for novel serotonin 5-HT(2A) antagonists. | Current topics in medicinal chemistry 20020601 |
Effect of dopamine receptor agonists on sensory nerve activity: possible therapeutic targets for the treatment of asthma and COPD. | British journal of pharmacology 20020601 |
Adenosinergic modulation of the discriminative-stimulus effects of methamphetamine in rats. | Psychopharmacology 20020601 |
Functional screening of G protein-coupled receptors by measuring intracellular calcium with a fluorescence microplate reader. | Journal of biomolecular screening 20020601 |
Serotonin antagonist profiling on 5HT2A and 5HT2C receptors by nonequilibrium intracellular calcium response using an automated flow-through fluorescence analysis system, HT-PS 100. | Journal of biomolecular screening 20020601 |
Design and synthesis of a piperazinylalkylisoxazole library for subtype selective dopamine receptor ligands. | Bioorganic & medicinal chemistry letters 20020520 |
Hemiparkinsonism associated with a mesencephalic tumor. | Journal of the neurological sciences 20020515 |
Contrasting effects of dopamine antagonists and frequency reduction on Fos expression induced by lateral hypothalamic stimulation. | Behavioural brain research 20020514 |
Enhanced detection of receptor constitutive activity in the presence of regulators of G protein signaling: applications to the detection and analysis of inverse agonists and low-efficacy partial agonists. | Molecular pharmacology 20020501 |
Brain neurotransmitter receptor binding and nootropic studies on Indian Hypericum perforatum Linn. | Phytotherapy research : PTR 20020501 |
Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells. | The Journal of biological chemistry 20020419 |
Physiologically identified 5-HT2-like receptors at the crayfish neuromuscular junction. | Brain research 20020405 |
Hypothalamic paraventricular 5-hydroxytryptamine: receptor-specific inhibition of NPY-stimulated eating and energy metabolism. | Pharmacology, biochemistry, and behavior 20020401 |
Neuropharmacological profile of a novel potential atypical antipsychotic drug Y-931 (8-fluoro-12-(4-methylpiperazin-1-yl)- 6H-[1]benzothieno[2,3-b][1,5] benzodiazepine maleate). | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20020401 |
(+)-[76Br]A-69024: a non-benzazepine radioligand for studies of dopamine D1 receptors using PET. | Nuclear medicine and biology 20020401 |
Positron emission tomography and ex vivo and in vitro autoradiography studies on dopamine D2-like receptor degeneration in the quinolinic acid-lesioned rat striatum: comparison of [11C]raclopride, [11C]nemonapride and [11C]N-methylspiperone. | Nuclear medicine and biology 20020401 |
Timing is everything: the effects of putative dopamine antagonists on metamorphosis vary with larval age and experimental duration in the prosobranch gastropod Crepidula fornicata. | The Biological bulletin 20020401 |
The atypical 5-HT2 receptor mediating tachycardia in pithed rats: pharmacological correlation with the 5-HT2A receptor subtype. | British journal of pharmacology 20020301 |
The human 5-HT7 serotonin receptor splice variants: constitutive activity and inverse agonist effects. | British journal of pharmacology 20020301 |
A novel series of hybrid compounds derived by combining 2-aminotetralin and piperazine fragments: binding activity at D2 and D3 receptors. | Bioorganic & medicinal chemistry letters 20020225 |
In vitro evidence that 5-hydroxytryptamine increases efflux of glial glutamate via 5-HT(2A) receptor activation. | Journal of neuroscience research 20020201 |
Effects of some steroids and other compounds on ovarian growth of the red swamp crayfish, Procambarus clarkii, during early vitellogenesis. | The Journal of experimental zoology 20020101 |
Implementation and evaluation of a 3D one-step late reconstruction algorithm for 3D positron emission tomography brain studies using median root prior. | European journal of nuclear medicine and molecular imaging 20020101 |
Atmospheric pressure laser desorption/chemical ionization mass spectrometry: a new ionization method based on existing themes. | Rapid communications in mass spectrometry : RCM 20020101 |
Decreased [(3)H]spiperone binding in the anterior cingulate cortex of schizophrenia patients: an autoradiographic study. | Neuroscience 20020101 |
[Dopamine antibodies as neuromodulators of behavioral reactions in mice of different genotypes]. | Zhurnal vysshei nervnoi deiatelnosti imeni I P Pavlova 20020101 |
The effects of dopamine synthesis inhibitors and dopamine antagonists on regeneration in the hydra Hydra attenuata. | Neuroscience and behavioral physiology 20020101 |
Occurrence of dopaminergic (D(2)) receptors within the rabbit pulmonary circulation. | Pulmonary pharmacology & therapeutics 20020101 |
Nad-299 antagonises 5-HT-stimulated and spiperone-inhibited [35S]GTPgammaS binding in cloned 5-HT1A receptors. | Journal of receptor and signal transduction research 20020101 |
(-)S amisulpride binds with high affinity to cloned dopamine D(3) and D(2) receptors. | European journal of pharmacology 20011207 |
Expression of catecholaminergic mRNAs in the hyperactive mouse mutant coloboma. | Brain research. Molecular brain research 20011130 |
Modulation of [3H]quinpirole binding at striatal D2 dopamine receptors by a monoamine oxidaseA-like site: evidence from radioligand binding studies and D2 receptor- and MAO(A)-deficient mice. | Life sciences 20011130 |
Effects of endogenous neurotransmitters on the in vivo binding of dopamine and 5-HT radiotracers in mice. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20011101 |
Modulation of dopamine uptake in rat nucleus accumbens: effect of specific dopamine receptor antagonists and sigma ligands. | Neuroscience letters 20011026 |
Noninvasive, quantitative imaging in living animals of a mutant dopamine D2 receptor reporter gene in which ligand binding is uncoupled from signal transduction. | Gene therapy 20011001 |
Benzamide bioisosteres incorporating dihydroheteroazole substructures: EPC synthesis and SAR leading to a selective dopamine D4 receptor partial agonist (FAUC 179). | Bioorganic & medicinal chemistry letters 20010917 |
Determination of dopamine D(4) receptor density in rat striatum using PB12 as a probe. | European journal of pharmacology 20010907 |
New 1-aryl-4-(biarylmethylene)piperazines as potential atypical antipsychotics sharing dopamine D(2)-receptor and serotonin 5-HT(1A)-receptor affinities. | Bioorganic & medicinal chemistry letters 20010903 |
Dosing time-dependent tolerance of catalepsy by repetitive administration of haloperidol in mice. | The Journal of pharmacology and experimental therapeutics 20010901 |
Dopamine inhibits vasopressin action in the rat inner medullary collecting duct via alpha(2)-adrenoceptors. | The Journal of pharmacology and experimental therapeutics 20010901 |
Agonist regulation of D(2) dopamine receptor/G protein interaction. Evidence for agonist selection of G protein subtype. | The Journal of biological chemistry 20010803 |
Direct correlation between positron emission tomographic images of two reporter genes delivered by two distinct adenoviral vectors. | Gene therapy 20010701 |
Pharmacological evaluation of (+)-2- [123I]A-69024: a radioligand for in vivo studies of dopamine D1 receptors. | Life sciences 20010629 |
Dopamine D2 receptor dimer formation: evidence from ligand binding. | The Journal of biological chemistry 20010622 |
Hypericum perforatum as a nootropic drug: enhancement of retrieval memory of a passive avoidance conditioning paradigm in mice. | Journal of ethnopharmacology 20010601 |
The cloned human 5-HT7 receptor splice variants: a comparative characterization of their pharmacology, function and distribution. | Naunyn-Schmiedeberg's archives of pharmacology 20010601 |
Stimulation of sodium-dependent inorganic phosphate transport by activation of Gi/o-protein-coupled receptors by epinephrine in MC3T3-E1 osteoblast-like cells. | Bone 20010601 |
Affinity of serotonin receptor antagonists and agonists to recombinant and native alpha1-adrenoceptor subtypes. | Japanese journal of pharmacology 20010601 |
Pharmacological characterization of the D1- and D2-like dopamine receptors from the brain of the leopard frog, Rana pipiens. | Brain, behavior and evolution 20010601 |
Differential effects of 5-HT1A receptor deletion upon basal and fluoxetine-evoked 5-HT concentrations as revealed by in vivo microdialysis. | Brain research 20010525 |
Reversible decrease of dopamine D2 receptor density in the striatum of rats with acute hepatic failure. | Brain research 20010504 |
D2 but not D3 receptors are elevated after 9 or 11 months chronic haloperidol treatment: influence of withdrawal period. | Synapse (New York, N.Y.) 20010501 |
D(3) dopamine receptors in rat spinal cord: implications for sensory and motor function. | Neuroscience letters 20010427 |
Effects of dopaminergic agents on carrageenan hyperalgesia after intrathecal administration to rats. | European journal of pharmacology 20010420 |
Cis- and trans-N-benzyl-octahydrobenzo[g]quinolines. Adrenergic and dopaminergic activity studies. | Bioorganic & medicinal chemistry letters 20010409 |
Characterization of the serotonin receptor mediating contraction in the mouse thoracic aorta and signal pathway coupling. | The Journal of pharmacology and experimental therapeutics 20010401 |
Mechanisms of inverse agonism of antipsychotic drugs at the D(2) dopamine receptor: use of a mutant D(2) dopamine receptor that adopts the activated conformation. | Journal of neurochemistry 20010401 |
The role of D2-like dopamine receptors in the locomotor stimulant effects of cocaine in mice. | Psychopharmacology 20010401 |
Alteration of dopamine transport in the striatum and nucleus accumbens of ovariectomized and estrogen-primed rats following N-(p-isothiocyanatophenethyl) spiperone (NIPS) treatment. | Brain research bulletin 20010401 |
S 14506: novel receptor coupling at 5-HT(1A) receptors. | Neuropharmacology 20010301 |
Failure of AH11110A to functionally discriminate between alpha(1)-adrenoceptor subtypes A, B and D or between alpha(1)- and alpha(2)-adrenoceptors. | European journal of pharmacology 20010301 |
Stimulus properties of 7-OH-DPAT versus auto- and postsynaptic receptor-specific doses of quinpirole. | Pharmacology, biochemistry, and behavior 20010301 |
Effects of intrastriatal infusion of D2 and D3 dopamine receptor preferring antagonists on dopamine release in rat dorsal striatum (in vivo microdialysis study). | Pharmacological research 20010301 |
Increased 5-hydroxytryptamine-2 receptor binding in the frontal cortex of depressed patients responding to paroxetine treatment: a positron emission tomography scan study. | Journal of clinical psychopharmacology 20010201 |
The effect of nicotine and haloperidol co-treatment on nicotinic receptor levels in the rat brain. | Brain research. Molecular brain research 20010131 |
Modulation of 5-HT(1A) receptor activation by its interaction with wild-type and mutant g(alphai3) proteins. | Neuropharmacology 20010101 |
Differential modulation by GTPgammaS of agonist and inverse agonist binding to h5-HT(1A) receptors revealed by [3H]-WAY100,635. | British journal of pharmacology 20010101 |
Dopaminergic activity in transgenic mice underexpressing glucocorticoid receptors: effect of antidepressants. | Neuroscience 20010101 |
Recent advances in imaging endogenous or transferred gene expression utilizing radionuclide technologies in living subjects: applications to breast cancer. | Breast cancer research : BCR 20010101 |
A consideration of the dopamine D2 receptor monomer-dimer equilibrium and the anomalous binding properties of the dopamine D2 receptor ligand, N-methyl spiperone. | Journal of neural transmission (Vienna, Austria : 1996) 20010101 |
Effects of lithium on dopamine D2 receptor expression in the rat brain striatum. | Journal of neural transmission (Vienna, Austria : 1996) 20010101 |
Dopamine depletion with 6-OHDA enhances dopamine D1-receptor modulation of potassium currents in retinal bipolar cells. | Visual neuroscience 20010101 |
Patterns of cyclic AMP formation by coexpressed D1 and D2L dopamine receptors in HEK 293 cells. | Receptors & channels 20010101 |
Differential modes of agonist binding to 5-hydroxytryptamine(2A) serotonin receptors revealed by mutation and molecular modeling of conserved residues in transmembrane region 5. | Molecular pharmacology 20001101 |
Inverse agonist activity of atypical antipsychotic drugs at human 5-hydroxytryptamine2C receptors. | The Journal of pharmacology and experimental therapeutics 20001001 |
Regulation of human D(1), d(2(long)), d(2(short)), D(3) and D(4) dopamine receptors by amiloride and amiloride analogues. | British journal of pharmacology 20000701 |
The effects of benzamide analogues on cocaine self-administration in rhesus monkeys. | Psychopharmacology 19991101 |
Enhanced striatal dopamine D(2) receptor-induced [35S]GTPgammaS binding after haloperidol treatment. | European journal of pharmacology 19991008 |
Synthesis and preliminary pharmacological investigations of 1-(1,2-dihydro-2-acenaphthylenyl)piperazine derivatives as potential atypical antipsychotic agents in mice. | Farmaco (Societa chimica italiana : 1989) 19990830 |
Zinc modulates antagonist interactions with D2-like dopamine receptors through distinct molecular mechanisms. | The Journal of pharmacology and experimental therapeutics 19990501 |
High-affinity agonist binding correlates with efficacy (intrinsic activity) at the human serotonin 5-HT2A and 5-HT2C receptors: evidence favoring the ternary complex and two-state models of agonist action. | Journal of neurochemistry 19990501 |
Characterization of alpha1-adrenoceptor subtypes mediating noradrenaline-induced contraction of rat epididymal vas deferens in calcium-free medium. | Life sciences 19990101 |
Agonist and antagonist actions of antipsychotic agents at 5-HT1A receptors: a [35S]GTPgammaS binding study. | European journal of pharmacology 19980821 |
Creation of a constitutively activated state of the 5-hydroxytryptamine2A receptor by site-directed mutagenesis: inverse agonist activity of antipsychotic drugs. | The Journal of pharmacology and experimental therapeutics 19980701 |
Labelling of recombinant human and native rat serotonin 5-HT1A receptors by a novel, selective radioligand, [3H]-S 15535: definition of its binding profile using agonists, antagonists and inverse agonists. | Naunyn-Schmiedeberg's archives of pharmacology 19980301 |
[3H]Rauwolscine: an antagonist radioligand for the cloned human 5-hydroxytryptamine2b (5-HT2B) receptor. | Naunyn-Schmiedeberg's archives of pharmacology 19980101 |
Cloning, expression and pharmacology of a truncated splice variant of the human 5-HT7 receptor (h5-HT7b). | British journal of pharmacology 19970901 |
Zinc allosterically modulates antagonist binding to cloned D1 and D2 dopamine receptors. | Journal of neurochemistry 19970501 |
Bromocriptine transcriptionally activates the multidrug resistance gene (pgp2/mdr1b) by a novel pathway. | The Journal of biological chemistry 19970425 |
The behavioural effects of pramipexole, a novel dopamine receptor agonist. | European journal of pharmacology 19970411 |
Synthesis and biological profile of the enantiomers of [4-(4-amino-6,7-dimethoxyquinazolin-2-yl)-cis-octahydroquinoxalin- 1-yl]furan-2-ylmethanone (cyclazosin), a potent competitive alpha 1B- adrenoceptor antagonist. | Journal of medicinal chemistry 19961108 |
Nefiracetam (DM-9384) reverses apomorphine-induced amnesia of a passive avoidance response: delayed emergence of the memory retention effects. | Neurochemical research 19960601 |
Critical reevaluation of spiperone and benzamide binding to dopamine D2 receptors: evidence for identical binding sites. | European journal of pharmacology 19960506 |
Radiolabelling of the human 5-HT2A receptor with an agonist, a partial agonist and an antagonist: effects on apparent agonist affinities. | Biochemical pharmacology 19960112 |
ABT-431: the diacetyl prodrug of A-86929, a potent and selective dopamine D1 receptor agonist: in vitro characterization and effects in animal models of Parkinson's disease. | The Journal of pharmacology and experimental therapeutics 19960101 |
Roxindole, a potential antidepressant. I. Effect on the dopamine system. | Journal of neural transmission (Vienna, Austria : 1996) 19960101 |
Neurochemical and functional characterization of the preferentially selective dopamine D3 agonist PD 128907. | The Journal of pharmacology and experimental therapeutics 19951201 |
Functional correlates of dopamine D3 receptor activation in the rat in vivo and their modulation by the selective antagonist, (+)-S 14297: 1. Activation of postsynaptic D3 receptors mediates hypothermia, whereas blockade of D2 receptors elicits prolactin secretion and catalepsy. | The Journal of pharmacology and experimental therapeutics 19951101 |
Alpha- and beta-adrenoceptors: from the gene to the clinic. 1. Molecular biology and adrenoceptor subclassification. | Journal of medicinal chemistry 19950901 |
Pramipexole binding and activation of cloned and expressed dopamine D2, D3 and D4 receptors. | European journal of pharmacology 19950623 |
Behavioral and biochemical changes after bilateral electrolytic lesions of the red nucleus of rat. | Pharmacology, biochemistry, and behavior 19950501 |
Differential effects of [3H]nemonapride and [3H]spiperone binding on human dopamine D4 receptors. | Neuroscience letters 19950217 |
Is clozapine selective for the dopamine D4 receptor? | Life sciences 19950101 |
Some behavioral effects of CNQX AND NBQX, AMPA receptor antagonists. | Polish journal of pharmacology 19950101 |
Elimination of cocaine-induced hyperactivity and dopamine-mediated neurophysiological effects in dopamine D1 receptor mutant mice. | Cell 19941216 |
Molecular cloning, functional expression, and mRNA tissue distribution of the human 5-hydroxytryptamine2B receptor. | Molecular pharmacology 19940801 |
Binding of typical and atypical antipsychotic agents to 5-hydroxytryptamine-6 and 5-hydroxytryptamine-7 receptors. | The Journal of pharmacology and experimental therapeutics 19940301 |
Characterization of the human dopamine D3 receptor expressed in transfected cell lines. | European journal of pharmacology 19940101 |
Some central effects of kynurenic acid, 7-chlorokynurenic acid and 5,7- dichloro-kynurenic acid, glycine site antagonists. | Polish journal of pharmacology 19940101 |
Pharmacological and functional characterization of D2, D3 and D4 dopamine receptors in fibroblast and dopaminergic cell lines. | The Journal of pharmacology and experimental therapeutics 19940101 |
Dopamine D2 and serotonin S2 receptors in susceptibility to methamphetamine psychosis detected by positron emission tomography. | Psychiatry research 19931201 |
Cloning of a novel human serotonin receptor (5-HT7) positively linked to adenylate cyclase. | The Journal of biological chemistry 19931105 |
Molecular cloning, characterization, and localization of a high-affinity serotonin receptor (5-HT7) activating cAMP formation. | Proceedings of the National Academy of Sciences of the United States of America 19930915 |
Low density of dopamine D4 receptors in Parkinson's, schizophrenia, and control brain striata. | Synapse (New York, N.Y.) 19930801 |
Molecular cloning of a mammalian serotonin receptor that activates adenylate cyclase. | Molecular pharmacology 19930801 |
Strain differences in clonidine-induced aggressiveness in mice and its interaction with the dopamine system. | Pharmacology, biochemistry, and behavior 19930401 |
The role of receptor binding in drug discovery. | Journal of natural products 19930401 |
Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor. | Molecular pharmacology 19930301 |
Cloning of another human serotonin receptor (5-HT1F): a fifth 5-HT1 receptor subtype coupled to the inhibition of adenylate cyclase. | Proceedings of the National Academy of Sciences of the United States of America 19930115 |
Pharmacological profile of AD-5423, a novel antipsychotic with both potent dopamine-D2 and serotonin-S2 antagonist properties. | The Journal of pharmacology and experimental therapeutics 19930101 |
High-level stable expression of recombinant 5-HT1A 5-hydroxytryptamine receptors in Chinese hamster ovary cells. | The Biochemical journal 19920801 |
Upregulation of postsynaptic dopamine receptors in the striatum does not influence haloperidol-induced catalepsy in mice. | Pharmacology, biochemistry, and behavior 19920801 |
Human serotonin 1D receptor is encoded by a subfamily of two distinct genes: 5-HT1D alpha and 5-HT1D beta. | Proceedings of the National Academy of Sciences of the United States of America 19920415 |
Mouse 5HT1B serotonin receptor: cloning, functional expression, and localization in motor control centers. | Proceedings of the National Academy of Sciences of the United States of America 19920401 |
Effect of mesulergine on prolactin secretion and dopamine D2 receptors-adaptive changes in diethylstilbestrol-induced hyperplasia of the rat anterior pituitary. | Endocrine regulations 19920301 |
Fluorescent probes for dopamine receptors: synthesis and characterization of fluorescein and 7-nitrobenz-2-oxa-1,3-diazol-4-yl conjugates of D-1 and D-2 receptor ligands. | Journal of medicinal chemistry 19911101 |
Primary structure and functional characterization of a human 5-HT1D-type serotonin receptor. | Molecular pharmacology 19910801 |
Reduced D2 dopamine and muscarinic cholinergic receptor densities in caudate specimens from fluctuating parkinsonian patients. | Annals of neurology 19910801 |
Cloning of the gene for a human dopamine D5 receptor with higher affinity for dopamine than D1. | Nature 19910418 |
Cloning of the gene for a human dopamine D4 receptor with high affinity for the antipsychotic clozapine. | Nature 19910418 |
Simultaneous quantitation of loxapine, amoxapine and their 7- and 8-hydroxy metabolites in plasma by high-performance liquid chromatography. | Journal of chromatography 19910308 |
Behavioural and electoencephalographic interactions between haloperidol and PCP/sigma ligands in the rat. | Psychopharmacology 19910101 |
Antidopaminergic effects of the stereoisomers of N-[(1-alkyl-2- pyrrolidinyl)methyl]-5-sulfamoylbenzamides and -2,3-dihydrobenzofuran-7-carboxamides. | Journal of medicinal chemistry 19910101 |
On the selection of mice for haloperidol response and non-response. | Psychopharmacology 19910101 |
Effects of subchronic amphetamine or amfonelic acid on rat brain dopaminergic and serotonergic function. | Journal of neural transmission. General section 19910101 |
[3H]-DOB(4-bromo-2,5-dimethoxyphenylisopropylamine) and [3H] ketanserin label two affinity states of the cloned human 5-hydroxytryptamine2 receptor. | Molecular pharmacology 19901101 |
Modulation of dopamine receptors by cations in 7315a, MtTW15 and estradiol-induced pituitary tumors. | Biochemical pharmacology 19900915 |
Molecular cloning and characterization of a novel dopamine receptor (D3) as a target for neuroleptics. | Nature 19900913 |
Evidence that central 5-HT1A-receptors play a role in the von Bezold-Jarisch reflex in the rat. | British journal of pharmacology 19900801 |
Pharmacological actions of SM-9018, a new neuroleptic drug with both potent 5-hydroxytryptamine2 and dopamine2 antagonistic actions. | Japanese journal of pharmacology 19900701 |
Dopamine receptor agonists: selectivity and dopamine D1 receptor efficacy. | European journal of pharmacology 19900612 |
Dihydrexidine, a novel selective high potency full dopamine D-1 receptor agonist. | European journal of pharmacology 19890704 |
Dopamine blockade and clinical response: evidence for two biological subgroups of schizophrenia. | The American journal of psychiatry 19890701 |
Cloning and expression of a rat D2 dopamine receptor cDNA. | Nature 19881201 |
In vitro estrogen-like effects of 7,12-dimethylbenz(a)anthracene on anterior pituitary dopamine receptors of rats. | Cancer research 19881115 |
Receptor mechanisms of nicotine-induced locomotor hyperactivity in chronic nicotine-treated rats. | European journal of pharmacology 19880802 |
Alpha 2-adrenoceptors as a target for formamidine pesticides: in vitro and in vivo studies in mice. | Toxicology and applied pharmacology 19880401 |
High doses of morphine do not change characteristics of the cerebral catecholamine receptors in the rat. | Polish journal of pharmacology and pharmacy 19880101 |
Antagonism by neuroleptics of serotonin 5-HT1A and 5-HT2 receptors of normal human brain in vitro. | European journal of pharmacology 19871110 |
MPTP-induced parkinsonism in the monkey: neurochemical pathology, complications of treatment and pathophysiological mechanisms. | The Canadian journal of neurological sciences. Le journal canadien des sciences neurologiques 19870801 |
Experimental study on resting tremor and L-dopa-induced dyskinesia. | European neurology 19870101 |
The selective dopamine D2 receptor antagonist raclopride discriminates between dopamine-mediated motor functions. | Psychopharmacology 19860101 |
Simultaneous catalepsy and apomorphine-induced stereotypic behavior in mice. | Life sciences 19851104 |
Prenatal exposure of rats to antidepressants enhances agonist affinity of brain dopamine receptors and dopamine-mediated behaviour. | European journal of pharmacology 19851022 |
Repeated treatment with imipramine or amitriptyline increases the locomotor response of rats to (+)-amphetamine given into the nucleus accumbens. | The Journal of pharmacy and pharmacology 19850501 |
The role of the GABA mechanisms of the globus pallidus in mediating catalepsy, stereotypy and locomotor activity. | Pharmacology, biochemistry, and behavior 19841201 |
[Effect of repeated haloperidol and apomorphine administration on the development of tolerance for catalepsy and dopamine receptor hypersensitivity in mice]. | Biulleten' eksperimental'noi biologii i meditsiny 19841001 |
Sigma opiates and certain antipsychotic drugs mutually inhibit (+)-[3H] SKF 10,047 and [3H]haloperidol binding in guinea pig brain membranes. | Proceedings of the National Academy of Sciences of the United States of America 19840901 |
Dopamine receptors in rat pituitary and estradiol-induced pituitary tumor: effect of chronic treatment with bromocriptine. | Biochemical and biophysical research communications 19840830 |
Remoxipride, a new potential antipsychotic compound with selective antidopaminergic actions in the rat brain. | European journal of pharmacology 19840720 |
Interactions of neurotensin with brain dopamine systems: biochemical and behavioral studies. | The Journal of pharmacology and experimental therapeutics 19830501 |
CGS 7525A, a new, centrally active alpha 2 adrenoceptor antagonist. | Life sciences 19830124 |
Assessment of the antidepressant activity of dothiepin and its metabolites by preclinical tests. | Journal of affective disorders 19820901 |
Possible involvement of serotonergic neurons in the reduction of locomotor hyperactivity caused by amphetamine in neonatal rats depleted of brain dopamine. | Brain research 19820722 |
Cataleptogenic doses of morphine suppress 3H-spiroperidol binding to striatal membranes. | Naunyn-Schmiedeberg's archives of pharmacology 19820501 |
Septo-hippocampal system: target for substituted benzamides. | European journal of pharmacology 19820423 |
Central neurotropic activity of homovanillic acid. | Acta physiologica Polonica 19810101 |
Chronic treatment with antidepressant drugs: potentiation of apomorphine-induced aggressive behaviour in rats. | Neuroscience letters 19790801 |
On the anticataleptic action of cyproheptadine. | Pharmacology, biochemistry, and behavior 19760801 |
Influence of WA-335, a factor which blocks serotonin receptors, on neuroleptic-induced catalepsy. | Archivum immunologiae et therapiae experimentalis 19760101 |
Antagonistic effect of cyproheptadine on neuroleptic-induced catalepsy. | Pharmacology, biochemistry, and behavior 19750101 |
The effect of 5-hydroxytrytamine synthesis inhibitors on neuroleptic-induced catalepsy in rats. | Archivum immunologiae et therapiae experimentalis 19750101 |