Home Other Building Blocks Benzimidamide

Benzimidamide

CAS No.:
618-39-3
Catalog Number:
AG003O0K
Molecular Formula:
C7H8N2
Molecular Weight:
120.1518
Pack Size
Purity
Availability
Location
Price(USD)
Quantity
  
250mg
95+%
1 week
United States
$88
- +
1g
95%
1 week
United States
$117
- +
Product Description
Catalog Number:
AG003O0K
Chemical Name:
Benzimidamide
CAS Number:
618-39-3
Molecular Formula:
C7H8N2
Molecular Weight:
120.1518
MDL Number:
MFCD00042826
IUPAC Name:
benzenecarboximidamide
InChI:
InChI=1S/C7H8N2/c8-7(9)6-4-2-1-3-5-6/h1-5H,(H3,8,9)
InChI Key:
PXXJHWLDUBFPOL-UHFFFAOYSA-N
SMILES:
NC(=N)c1ccccc1
EC Number:
210-546-3
UNII:
KUE3ZY3J1F
NSC Number:
243704
Properties
Complexity:
104  
Compound Is Canonicalized:
Yes
Covalently-Bonded Unit Count:
1  
Defined Atom Stereocenter Count:
0
Defined Bond Stereocenter Count:
0
Exact Mass:
120.069g/mol
Formal Charge:
0
Heavy Atom Count:
9  
Hydrogen Bond Acceptor Count:
1  
Hydrogen Bond Donor Count:
2  
Isotope Atom Count:
0
Molecular Weight:
120.155g/mol
Monoisotopic Mass:
120.069g/mol
Rotatable Bond Count:
1  
Topological Polar Surface Area:
49.9A^2
Undefined Atom Stereocenter Count:
0
Undefined Bond Stereocenter Count:
0
XLogP3:
0.7  
Literature
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Functional incorporation of sorghum small subunit increases the catalytic turnover rate of Rubisco in transgenic rice. Plant physiology 20110701
Defining the specificity of cotranslationally acting chaperones by systematic analysis of mRNAs associated with ribosome-nascent chain complexes. PLoS biology 20110701
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A magnetic adsorbent-based process for semi-continuous PEGylation of proteins. Biotechnology journal 20110401
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Solution structure of a repeated unit of the ABA-1 nematode polyprotein allergen of Ascaris reveals a novel fold and two discrete lipid-binding sites. PLoS neglected tropical diseases 20110401
Mechanism of neuroprotective mitochondrial remodeling by PKA/AKAP1. PLoS biology 20110401
Protein phosphatase 2A controls ethylene biosynthesis by differentially regulating the turnover of ACC synthase isoforms. PLoS genetics 20110401
Effect of PI3K- and mTOR-specific inhibitors on spontaneous B-cell follicular lymphomas in PTEN/LKB1-deficient mice. British journal of cancer 20110329
Small molecule AKAP-protein kinase A (PKA) interaction disruptors that activate PKA interfere with compartmentalized cAMP signaling in cardiac myocytes. The Journal of biological chemistry 20110318
Synthesis and biological evaluation of L-valine-amidoximeesters as double prodrugs of amidines. Bioorganic & medicinal chemistry 20110315
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Congeneric but still distinct: how closely related trypsin ligands exhibit different thermodynamic and structural properties. Journal of molecular biology 20110204
Structural basis of the 9-fold symmetry of centrioles. Cell 20110204
Anthrolysin O and fermentation products mediate the toxicity of Bacillus anthracis to lung epithelial cells under microaerobic conditions. FEMS immunology and medical microbiology 20110201
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Lead dysregulates serine/threonine protein phosphatases in human neurons. Neurochemical research 20110201
ERK/p90(RSK)/14-3-3 signalling has an impact on expression of PEA3 Ets transcription factors via the transcriptional repressor capicúa. The Biochemical journal 20110201
PERK activation at low glucose concentration is mediated by SERCA pump inhibition and confers preemptive cytoprotection to pancreatic β-cells. Molecular endocrinology (Baltimore, Md.) 20110201
Modulation of aberrant CDK5 signaling rescues impaired neurogenesis in models of Alzheimer's disease. Cell death & disease 20110201
The C-terminal domain of the Arabinosyltransferase Mycobacterium tuberculosis EmbC is a lectin-like carbohydrate binding module. PLoS pathogens 20110201
Recognition and specificity determinants of the human cbx chromodomains. The Journal of biological chemistry 20110107
S-Petasin, the Main Sesquiterpene of Petasites formosanus, Inhibits Phosphodiesterase Activity and Suppresses Ovalbumin-Induced Airway Hyperresponsiveness. Evidence-based complementary and alternative medicine : eCAM 20110101
Restoration of photosystem II photochemistry and carbon assimilation and related changes in chlorophyll and protein contents during the rehydration of desiccated Xerophyta scabrida leaves. Journal of experimental botany 20110101
Molecular mechanism analysis of Gloydius shedaoensis venom gloshedobin interaction with inhibitors by homology modeling. International journal of biological macromolecules 20110101
Rationale for possible targeting of histone deacetylase signaling in cancer diseases with a special reference to pancreatic cancer. Journal of biomedicine & biotechnology 20110101
A structural basis for Staphylococcal complement subversion: X-ray structure of the complement-binding domain of Staphylococcus aureus protein Sbi in complex with ligand C3d. Molecular immunology 20110101
Beneficial effect of Sparassis crispa on stroke through activation of Akt/eNOS pathway in brain of SHRSP. Journal of natural medicines 20110101
Rubisco activity in Mediterranean species is regulated by the chloroplastic CO2 concentration under water stress. Journal of experimental botany 20110101
Palmitoylethanolamide reduces granuloma-induced hyperalgesia by modulation of mast cell activation in rats. Molecular pain 20110101
Characterization of ERK docking domain inhibitors that induce apoptosis by targeting Rsk-1 and caspase-9. BMC cancer 20110101
Malate plays a crucial role in starch metabolism, ripening, and soluble solid content of tomato fruit and affects postharvest softening. The Plant cell 20110101
Endogenous plasma activated protein C levels and the effect of enoxaparin and drotrecogin alfa (activated) on markers of coagulation activation and fibrinolysis in pulmonary embolism. Critical care (London, England) 20110101
Targets downstream of Cdk8 in Dictyostelium development. BMC developmental biology 20110101
Identification and regulation of c-Myb target genes in MCF-7 cells. BMC cancer 20110101
A single acidic residue can guide binding site selection but does not govern QacR cationic-drug affinity. PloS one 20110101
IκB kinase β regulates epithelium migration during corneal wound healing. PloS one 20110101
MAP4K3 is a component of the TORC1 signalling complex that modulates cell growth and viability in Drosophila melanogaster. PloS one 20110101
Temporal and tissue specific regulation of RP-associated splicing factor genes PRPF3, PRPF31 and PRPC8--implications in the pathogenesis of RP. PloS one 20110101
Sustained delivery of activated Rho GTPases and BDNF promotes axon growth in CSPG-rich regions following spinal cord injury. PloS one 20110101
Protein-protein interactions within late pre-40S ribosomes. PloS one 20110101
Purification and biochemical characterization of a secreted group IIA chicken intestinal phospholipase A₂. Lipids in health and disease 20110101
Dot1 binding induces chromatin rearrangements by histone methylation-dependent and -independent mechanisms. Epigenetics & chromatin 20110101
Lymphocyte deficiency limits Epstein-Barr virus latent membrane protein 1 induced chronic inflammation and carcinogenic pathology in vivo. Molecular cancer 20110101
Serotonin transporter (SERT) and translocator protein (TSPO) expression in the obese ob/ob mouse. BMC neuroscience 20110101
Peripheral delivery of a CNS targeted, metalo-protease reduces aβ toxicity in a mouse model of Alzheimer's disease. PloS one 20110101
The level of claudin-7 is reduced as an early event in colorectal carcinogenesis. BMC cancer 20110101
Characterization of the proteases involved in the N-terminal clipping of glucagon-like-peptide-1-antibody fusion proteins. Biotechnology progress 20110101
Mechanisms underlying Actinobacillus pleuropneumoniae exotoxin ApxI induced expression of IL-1β, IL-8 and TNF-α in porcine alveolar macrophages. Veterinary research 20110101
Purification and biochemical characterization of pancreatic phospholipase A2 from the common stingray Dasyatis pastinaca. Lipids in health and disease 20110101
TGFβ1 enhances MAD1 expression and stimulates promoter-bound Pol II phosphorylation: basic functions of C/EBP, SP and SMAD3 transcription factors. BMC molecular biology 20110101
Dramatic repositioning of c-Myb to different promoters during the cell cycle observed by combining cell sorting with chromatin immunoprecipitation. PloS one 20110101
Increased expression of interleukin-6 family members and receptors in urinary bladder with cyclophosphamide-induced bladder inflammation in female rats. Frontiers in neuroscience 20110101
Sperm proteasomes degrade sperm receptor on the egg zona pellucida during mammalian fertilization. PloS one 20110101
Acinetobacter baumannii secretes cytotoxic outer membrane protein A via outer membrane vesicles. PloS one 20110101
Crystal structure of an integron gene cassette-associated protein from Vibrio cholerae identifies a cationic drug-binding module. PloS one 20110101
The regulatory subunit of PKA-I remains partially structured and undergoes β-aggregation upon thermal denaturation. PloS one 20110101
Purification and biochemical properties of a cytochrome bc complex from the aerobic hyperthermophilic archaeon Aeropyrum pernix. BMC microbiology 20110101
Increased Cell-Cell Coupling Increases Infarct Size and Does not Decrease Incidence of Ventricular Tachycardia in Mice. Frontiers in physiology 20110101
Endurance exercise training reduces cardiac sodium/calcium exchanger expression in animals susceptible to ventricular fibrillation. Frontiers in physiology 20110101
A mutation in synaptojanin 2 causes progressive hearing loss in the ENU-mutagenised mouse strain Mozart. PloS one 20110101
Cross-sample validation provides enhanced proteome coverage in rat vocal fold mucosa. PloS one 20110101
Biochanin a, a phytoestrogenic isoflavone with selective inhibition of phosphodiesterase 4, suppresses ovalbumin-induced airway hyperresponsiveness. Evidence-based complementary and alternative medicine : eCAM 20110101
Differential levels of glutamate dehydrogenase 1 (GLUD1) in Balb/c and C57BL/6 mice and the effects of overexpression of the Glud1 gene on glutamate release in striatum. ASN neuro 20110101
Altered gene expression in pulmonary tissue of tryptophan hydroxylase-1 knockout mice: implications for pulmonary arterial hypertension. PloS one 20110101
Unexpected long-term protection of adult offspring born to high-fat fed dams against obesity induced by a sucrose-rich diet. PloS one 20110101
Pro-inflammatory endothelial cell dysfunction is associated with intersectin-1s down-regulation. Respiratory research 20110101
Comparative analysis of Erk phosphorylation suggests a mixed strategy for measuring phospho-form distributions. Molecular systems biology 20110101
Foxp3 interacts with c-Rel to mediate NF-κB repression. PloS one 20110101
Role of endothelial Nox2 NADPH oxidase in angiotensin II-induced hypertension and vasomotor dysfunction. Basic research in cardiology 20110101
Modeling the TNFα-induced apoptosis pathway in hepatocytes. PloS one 20110101
Photodynamic treatment induces an apoptotic pathway involving calcium, nitric oxide, p53, p21-activated kinase 2, and c-Jun N-terminal kinase and inactivates survival signal in human umbilical vein endothelial cells. International journal of molecular sciences 20110101
High-throughput protein expression using a combination of ligation-independent cloning (LIC) and infrared fluorescent protein (IFP) detection. PloS one 20110101
Systemically administered ligands of Toll-like receptor 2, -4, and -9 induce distinct inflammatory responses in the murine lung. Mediators of inflammation 20110101
Biochemical properties of pancreatic colipase from the common stingray Dasyatis pastinaca. Lipids in health and disease 20110101
The stress response factors Yap6, Cin5, Phd1, and Skn7 direct targeting of the conserved co-repressor Tup1-Ssn6 in S. cerevisiae. PloS one 20110101
Is aboriginal food less allergenic? Comparing IgE-reactivity of eggs from modern and ancient chicken breeds in a cohort of allergic children. PloS one 20110101
The rate of NF-κB nuclear translocation is regulated by PKA and A kinase interacting protein 1. PloS one 20110101
Phosphorylation of the Twist1-family basic helix-loop-helix transcription factors is involved in pathological cardiac remodeling. PloS one 20110101
The chromatin remodelling complex B-WICH changes the chromatin structure and recruits histone acetyl-transferases to active rRNA genes. PloS one 20110101
The effect of anandamide on uterine nitric oxide synthase activity depends on the presence of the blastocyst. PloS one 20110101
Geminin overexpression prevents the completion of topoisomerase IIα chromosome decatenation, leading to aneuploidy in human mammary epithelial cells. Breast cancer research : BCR 20110101
Crystal structure of alkyl hydroperoxidase D like protein PA0269 from Pseudomonas aeruginosa: homology of the AhpD-like structural family. BMC structural biology 20110101
Binding of ATP to vascular endothelial growth factor isoform VEGF-A165 is essential for inducing proliferation of human umbilical vein endothelial cells. BMC biochemistry 20110101
Functional characterization of a lipoprotein-encoding operon in Campylobacter jejuni. PloS one 20110101
Calpain-catalyzed proteolysis of human dUTPase specifically removes the nuclear localization signal peptide. PloS one 20110101
Immunohistochemical localization of hepatopancreatic phospholipase A2 in Hexaplex trunculus digestive cells. Lipids in health and disease 20110101
Regulation of petrobactin and bacillibactin biosynthesis in Bacillus anthracis under iron and oxygen variation. PloS one 20110101
RyRCa2+ leak limits cardiac Ca2+ window current overcoming the tonic effect of calmodulinin mice. PloS one 20110101
Coordinated gene expression of Th17- and Treg-associated molecules correlated with resolution of the monophasic experimental autoimmune uveitis. Molecular vision 20110101
The nucleosome (histone-DNA complex) is the TLR9-specific immunostimulatory component of Plasmodium falciparum that activates DCs. PloS one 20110101
Structure of catalytic domain of Matriptase in complex with Sunflower trypsin inhibitor-1. BMC structural biology 20110101
Importance of post-translational modifications for functionality of a chloroplast-localized carbonic anhydrase (CAH1) in Arabidopsis thaliana. PloS one 20110101
Increased sensitivity to broadly neutralizing antibodies of end-stage disease R5 HIV-1 correlates with evolution in Env glycosylation and charge. PloS one 20110101
Neurite outgrowth of mature retinal ganglion cells and PC12 cells requires activity of CK1δ and CK1ε. PloS one 20110101
In vivo versus in vitro protein abundance analysis of Shigella dysenteriae type 1 reveals changes in the expression of proteins involved in virulence, stress and energy metabolism. BMC microbiology 20110101
The actions of exogenous leucine on mTOR signalling and amino acid transporters in human myotubes. BMC physiology 20110101
Modulation of myocardial mitochondrial mechanisms during severe polymicrobial sepsis in the rat. PloS one 20110101
Characterizing the role of cell-wall β-1,3-exoglucanase Xog1p in Candida albicans adhesion by the human antimicrobial peptide LL-37. PloS one 20110101
Zoledronic acid inhibits vasculogenic mimicry in murine osteosarcoma cell line in vitro. BMC musculoskeletal disorders 20110101
PP1 forms an active complex with TLRR (lrrc67), a putative PP1 regulatory subunit, during the early stages of spermiogenesis in mice. PloS one 20110101
Alendronate (ALN) combined with osteoprotegerin (OPG) significantly improves mechanical properties of long bone than the single use of ALN or OPG in the ovariectomized rats. Journal of orthopaedic surgery and research 20110101
Plasmodium falciparum glutamate dehydrogenase a is dispensable and not a drug target during erythrocytic development. Malaria journal 20110101
Quantification of mRNA and protein and integration with protein turnover in a bacterium. Molecular systems biology 20110101
Aerobic exercise training adaptations are increased by postexercise carbohydrate-protein supplementation. Journal of nutrition and metabolism 20110101
A new chymotrypsin-like serine protease involved in dietary protein digestion in a primitive animal, Scorpio maurus: purification and biochemical characterization. Lipids in health and disease 20110101
Production of recombinant human DNA polymerase delta in a Bombyx mori bioreactor. PloS one 20110101
Proteolytic cleavage of stingray phospholipase A2: isolation and biochemical characterization of an active N-terminal form. Lipids in health and disease 20110101
Caspase-3, myogenic transcription factors and cell cycle inhibitors are regulated by leukemia inhibitory factor to mediate inhibition of myogenic differentiation. Skeletal muscle 20110101
Zinc-regulated DNA binding of the yeast Zap1 zinc-responsive activator. PloS one 20110101
Inhibition of IGF-1 signalling enhances the apoptotic effect of AS602868, an IKK2 inhibitor, in multiple myeloma cell lines. PloS one 20110101
Influence of a probiotic soy product on fecal microbiota and its association with cardiovascular risk factors in an animal model. Lipids in health and disease 20110101
Role of epithelial integrin-linked kinase in promoting intestinal inflammation: effects on CCL2, fibronectin and the T cell repertoire. BMC immunology 20110101
HrpA, a DEAH-box RNA helicase, is involved in global gene regulation in the Lyme disease spirochete. PloS one 20110101
Contribution of Alanine-76 and Serine Phosphorylation in α-Synuclein Membrane Association and Aggregation in Yeasts. Parkinson's disease 20110101
In vitro activation and enzyme kinetic analysis of recombinant midgut serine proteases from the Dengue vector mosquito Aedes aegypti. BMC biochemistry 20110101
Upregulation of HYAL1 expression in breast cancer promoted tumor cell proliferation, migration, invasion and angiogenesis. PloS one 20110101
Differential effects of TNF (TNFSF2) and IFN-γ on intestinal epithelial cell morphogenesis and barrier function in three-dimensional culture. PloS one 20110101
Increased muscle stress-sensitivity induced by selenoprotein N inactivation in mouse: a mammalian model for SEPN1-related myopathy. PloS one 20110101
Berberine radiosensitizes human esophageal cancer cells by downregulating homologous recombination repair protein RAD51. PloS one 20110101
Relative Expression Levels Rather Than Specific Activity Plays the Major Role in Determining In Vivo AKT Isoform Substrate Specificity. Enzyme research 20110101
Purification of tropomyosin, paramyosin, actin, tubulin, troponin and kinases for chemiproteomics and its application to different scientific fields. PloS one 20110101
[Inhibition mechanism of trypsin by Schiff base metal chelate inhibitors]. Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan 20110101
Phosphorylation provides a negative mode of regulation for the yeast Rab GTPase Sec4p. PloS one 20110101
Global gene expression analysis of fission yeast mutants impaired in Ser-2 phosphorylation of the RNA pol II carboxy terminal domain. PloS one 20110101
Effects of RNA interference-mediated gene silencing of JMJD2A on human breast cancer cell line MDA-MB-231 in vitro. Journal of experimental & clinical cancer research : CR 20110101
Resveratrol inhibits growth of orthotopic pancreatic tumors through activation of FOXO transcription factors. PloS one 20110101
The effect of OPA1 on mitochondrial Ca²⁺ signaling. PloS one 20110101
The amino-terminus of nitric oxide sensitive guanylyl cyclase α₁ does not affect dimerization but influences subcellular localization. PloS one 20110101
Systemic remodeling of the redox regulatory network due to RNAi perturbations of glutaredoxin 1, thioredoxin 1, and glucose-6-phosphate dehydrogenase. BMC systems biology 20110101
Structural and biochemical studies of human 4-hydroxy-2-oxoglutarate aldolase: implications for hydroxyproline metabolism in primary hyperoxaluria. PloS one 20110101
Low concentrations of methamphetamine can protect dopaminergic cells against a larger oxidative stress injury: mechanistic study. PloS one 20110101
Pallidal hyperdopaminergic innervation underlying D2 receptor-dependent behavioral deficits in the schizophrenia animal model established by EGF. PloS one 20110101
Neonatal lethality in knockout mice expressing the kinase-dead form of the gefitinib target GAK is caused by pulmonary dysfunction. PloS one 20110101
Characteristics of stem cells derived from the degenerated human intervertebral disc cartilage endplate. PloS one 20110101
The minimal domain of adipose triglyceride lipase (ATGL) ranges until leucine 254 and can be activated and inhibited by CGI-58 and G0S2, respectively. PloS one 20110101
Polyamidoamine (PAMAM) dendrimer conjugate specifically activates the A3 adenosine receptor to improve post-ischemic/reperfusion function in isolated mouse hearts. BMC pharmacology 20110101
Liquid facets-related (lqfR) is required for egg chamber morphogenesis during Drosophila oogenesis. PloS one 20110101
Differential roles of hyperglycemia and hypoinsulinemia in diabetes induced retinal cell death: evidence for retinal insulin resistance. PloS one 20110101
Generation and characterization of transgenic mice expressing mitochondrial targeted red fluorescent protein selectively in neurons: modeling mitochondriopathy in excitotoxicity and amyotrophic lateral sclerosis. Molecular neurodegeneration 20110101
Differential pattern of glycogen accumulation after protein phosphatase 1 glycogen-targeting subunit PPP1R6 overexpression, compared to PPP1R3C and PPP1R3A, in skeletal muscle cells. BMC biochemistry 20110101
Modularity and hormone sensitivity of the Drosophila melanogaster insulin receptor/target of rapamycin interaction proteome. Molecular systems biology 20110101
TOPAZ1, a novel germ cell-specific expressed gene conserved during evolution across vertebrates. PloS one 20110101
Substance P is a mechanoresponsive, autocrine regulator of human tenocyte proliferation. PloS one 20110101
N-terminal arginines modulate plasma-membrane localization of Kv7.1/KCNE1 channel complexes. PloS one 20110101
RpkA, a highly conserved GPCR with a lipid kinase domain, has a role in phagocytosis and anti-bacterial defense. PloS one 20110101
Hesperetin-7,3'-O-dimethylether selectively inhibits phosphodiesterase 4 and effectively suppresses ovalbumin-induced airway hyperresponsiveness with a high therapeutic ratio. Journal of biomedical science 20110101
Characterizing the Escherichia coli O157:H7 proteome including protein associations with higher order assemblies. PloS one 20110101
The biology and dynamics of mammalian cortical granules. Reproductive biology and endocrinology : RB&E 20110101
Protein synthesis attenuation by phosphorylation of eIF2α is required for the differentiation of Trypanosoma cruzi into infective forms. PloS one 20110101
A newly high alkaline lipase: an ideal choice for application in detergent formulations. Lipids in health and disease 20110101
P(5A)-type ATPase Cta4p is essential for Ca2+ transport in the endoplasmic reticulum of Schizosaccharomyces pombe. PloS one 20110101
Implantation serine proteinase 1 exhibits mixed substrate specificity that silences signaling via proteinase-activated receptors. PloS one 20110101
Switch of voltage-gated K+ channel expression in the plasma membrane of chondrogenic cells affects cytosolic Ca2+-oscillations and cartilage formation. PloS one 20110101
Activation of epidermal growth factor receptor is required for NTHi-induced NF-κB-dependent inflammation. PloS one 20110101
TRESK background K(+) channel is inhibited by PAR-1/MARK microtubule affinity-regulating kinases in Xenopus oocytes. PloS one 20110101
Presence and distribution of the lubricating protein, lubricin, in the meibomian gland in rabbits. Molecular vision 20110101
Improving the catalytic activity of hyperthermophilic Pyrococcus horikoshii prolidase for detoxification of organophosphorus nerve agents over a broad range of temperatures. Archaea (Vancouver, B.C.) 20110101
Cannabidiol reduces intestinal inflammation through the control of neuroimmune axis. PloS one 20110101
Upregulation of the cell-cycle regulator RGC-32 in Epstein-Barr virus-immortalized cells. PloS one 20110101
Disruption of spectrin-like cytoskeleton in differentiating keratinocytes by PKCδ activation is associated with phosphorylated adducin. PloS one 20110101
NF-κB feedback control of JNK1 activation modulates TRPV1-induced increases in IL-6 and IL-8 release by human corneal epithelial cells. Molecular vision 20110101
A crucial role in fertility for the oyster angiotensin-converting enzyme orthologue CgACE. PloS one 20110101
Development of derivatives of 3, 3'-diindolylmethane as potent Leishmania donovani bi-subunit topoisomerase IB poisons. PloS one 20110101
The effect of arrestin conformation on the recruitment of c-Raf1, MEK1, and ERK1/2 activation. PloS one 20110101
Neuronal markers are expressed in human gliomas and NSE knockdown sensitizes glioblastoma cells to radiotherapy and temozolomide. BMC cancer 20110101
Incorporation of albumin fusion proteins into fibrin clots in vitro and in vivo: comparison of different fusion motifs recognized by factor XIIIa. BMC biotechnology 20110101
Soluble THSD7A is an N-glycoprotein that promotes endothelial cell migration and tube formation in angiogenesis. PloS one 20110101
Curative effect of 18β-glycyrrhetinic acid in experimental visceral leishmaniasis depends on phosphatase-dependent modulation of cellular MAP kinases. PloS one 20110101
Concentration-dependent effects of narciclasine on cell cycle progression in Arabidopsis root tips. BMC plant biology 20110101
Simple preparation of pacific cod trypsin for enzymatic Peptide synthesis. Journal of amino acids 20110101
Familial Parkinson's Disease Mutant E46K α-Synuclein Localizes to Membranous Structures, Forms Aggregates, and Induces Toxicity in Yeast Models. ISRN neurology 20110101
Interaction of human complement factor H variants Tyr⁴⁰² and His⁴⁰² with Leptospira spp. Frontiers in immunology 20110101
Identification, subcellular localization, biochemical properties, and high-resolution crystal structure of Trypanosoma brucei UDP-glucose pyrophosphorylase. Glycobiology 20101201
Identification of the hair cell soma-1 antigen, HCS-1, as otoferlin. Journal of the Association for Research in Otolaryngology : JARO 20101201
High-throughput chemical screen identifies a novel potent modulator of cellular circadian rhythms and reveals CKIα as a clock regulatory kinase. PLoS biology 20101201
Obatoclax induces Atg7-dependent autophagy independent of beclin-1 and BAX/BAK. Cell death & disease 20101201
Human OGA binds substrates in a conserved peptide recognition groove. The Biochemical journal 20101115
New hierarchical phosphorylation pathway of the translational repressor eIF4E-binding protein 1 (4E-BP1) in ischemia-reperfusion stress. The Journal of biological chemistry 20101105
Natural and synthetic inhibitors of kallikrein-related peptidases (KLKs). Biochimie 20101101
Protein association and dissociation regulated by extension peptide: a mode for iron control by phytoferritin in seeds. Plant physiology 20101101
Mitochondrial malate dehydrogenase lowers leaf respiration and alters photorespiration and plant growth in Arabidopsis. Plant physiology 20101101
Selective determinants of inositol 1,4,5-trisphosphate and adenophostin A interactions with type 1 inositol 1,4,5-trisphosphate receptors. British journal of pharmacology 20101101
Isolation of potent and specific trypsin inhibitors from a DNA-encoded chemical library. Bioconjugate chemistry 20101020
Discovery of small molecule inhibitors of the PH domain leucine-rich repeat protein phosphatase (PHLPP) by chemical and virtual screening. Journal of medicinal chemistry 20101014
The p38 SAPK is recruited to chromatin via its interaction with transcription factors. The Journal of biological chemistry 20101008
Efficacy of CR3294, a new benzamidine derivative, in the prevention of 5-fluorouracil-induced gastrointestinal mucositis and diarrhea in mice. Cancer chemotherapy and pharmacology 20101001
Compromized geranylgeranylation of RhoA and Rac1 in mevalonate kinase deficiency. Journal of inherited metabolic disease 20101001
The Medicago truncatula E3 ubiquitin ligase PUB1 interacts with the LYK3 symbiotic receptor and negatively regulates infection and nodulation. The Plant cell 20101001
14-3-3 binding to LRRK2 is disrupted by multiple Parkinson's disease-associated mutations and regulates cytoplasmic localization. The Biochemical journal 20100915
Bisphenol A exposure during pregnancy disrupts glucose homeostasis in mothers and adult male offspring. Environmental health perspectives 20100901
Ablation of 4E-BP1/2 prevents hyperglycemia-mediated induction of VEGF expression in the rodent retina and in Muller cells in culture. Diabetes 20100901
Activation of ASK1, downstream MAPKK and MAPK isoforms during cardiac ischaemia. Biochimica et biophysica acta 20100901
A new look at the pathogenesis of the meconium aspiration syndrome: a role for fetal pancreatic proteolytic enzymes in epithelial cell detachment. Pediatric research 20100901
Ghrelin suppresses glucose-stimulated insulin secretion and deteriorates glucose tolerance in healthy humans. Diabetes 20100901
Systems biology of coagulation initiation: kinetics of thrombin generation in resting and activated human blood. PLoS computational biology 20100901
Nitrogen-bound diazeniumdiolated amidines. Chemical communications (Cambridge, England) 20100821
Sub-picomolar relaxin signalling by a pre-assembled RXFP1, AKAP79, AC2, beta-arrestin 2, PDE4D3 complex. The EMBO journal 20100818
Purification and properties of trypsin-like enzyme from the midgut of Morimus funereus (coleoptera, cerambycidae) Larvae. Archives of insect biochemistry and physiology 20100801
Selective delivery of 2-hydroxy APA to Trypanosoma brucei using the melamine motif. Bioorganic & medicinal chemistry letters 20100801
Dynamics of Rad9 chromatin binding and checkpoint function are mediated by its dimerization and are cell cycle-regulated by CDK1 activity. PLoS genetics 20100801
The transcription factor Rbf1 is the master regulator for b-mating type controlled pathogenic development in Ustilago maydis. PLoS pathogens 20100801
Two novel Src homology 2 domain proteins interact to regulate dictyostelium gene expression during growth and early development. The Journal of biological chemistry 20100723
A medicinal chemist's guide to molecular interactions. Journal of medicinal chemistry 20100722
Characterization of a unique proline iminopeptidase from white-rot basidiomycetes Phanerochaete chrysosporium. Biochimie 20100701
Leptin deficiency causes insulin resistance induced by uncontrolled diabetes. Diabetes 20100701
1,2-ethane bis-1-amino-4-benzamidine is active against several brain insult and seizure challenges through anti-NMDA mechanisms targeting the 3H-TCP binding site and antioxidant action. European journal of medicinal chemistry 20100701
Salivary histatin 5 internalization by translocation, but not endocytosis, is required for fungicidal activity in Candida albicans. Molecular microbiology 20100701
The role of peripheral cannabinoid receptors type 1 in rats with visceral hypersensitivity induced by chronic restraint stress. Journal of neurogastroenterology and motility 20100701
AKAP79/150 interacts with AC8 and regulates Ca2+-dependent cAMP synthesis in pancreatic and neuronal systems. The Journal of biological chemistry 20100625
Bhalternin: Functional and structural characterization of a new thrombin-like enzyme from Bothrops alternatus snake venom. Toxicon : official journal of the International Society on Toxinology 20100615
Insights into the importance of hydrogen bonding in the gamma-phosphate binding pocket of myosin: structural and functional studies of serine 236. Biochemistry 20100615
Use of cells expressing gamma subunit variants to identify diverse mechanisms of AMPK activation. Cell metabolism 20100609
Serine 129 phosphorylation reduces the ability of alpha-synuclein to regulate tyrosine hydroxylase and protein phosphatase 2A in vitro and in vivo. The Journal of biological chemistry 20100604
Purification, characterization and substrate specificity of a trypsin from the Amazonian fish tambaqui (Colossoma macropomum). Biochemical and biophysical research communications 20100604
A Plasmodium falciparum transcriptional cyclin-dependent kinase-related kinase with a crucial role in parasite proliferation associates with histone deacetylase activity. Eukaryotic cell 20100601
Nitric oxide increases cyclic GMP levels, AMP-activated protein kinase (AMPK)alpha1-specific activity and glucose transport in human skeletal muscle. Diabetologia 20100601
Structural binding evidence of the trypanocidal drugs berenil and pentacarinate active principles to a serine protease model. International journal of biological macromolecules 20100601
Involvement of phospholipase D and phosphatidic acid in the light-dependent up-regulation of sorghum leaf phosphoenolpyruvate carboxylase-kinase. Journal of experimental botany 20100601
Supramolecular association in proton-transfer adducts containing benzamidinium cations. I. Four molecular salts with uracil derivatives. Acta crystallographica. Section C, Crystal structure communications 20100601
NleG Type 3 effectors from enterohaemorrhagic Escherichia coli are U-Box E3 ubiquitin ligases. PLoS pathogens 20100601
Molecular shape and medicinal chemistry: a perspective. Journal of medicinal chemistry 20100527
Trypsin from the processing waste of the lane snapper (Lutjanus synagris) and its compatibility with oxidants, surfactants and commercial detergents. Journal of agricultural and food chemistry 20100526
Physical interaction of RECQ5 helicase with RAD51 facilitates its anti-recombinase activity. The Journal of biological chemistry 20100521
The pseudophosphatase MK-STYX interacts with G3BP and decreases stress granule formation. The Biochemical journal 20100501
Purification and biochemical characterization of Eumiliin from Euphorbia milii var. hislopii latex. Phytochemistry 20100501
Rubisco activities, properties, and regulation in three different C4 grasses under drought. Journal of experimental botany 20100501
Formation of covalently bound protein adducts from the cytotoxicant naphthalene in nasal epithelium: species comparisons. Environmental health perspectives 20100501
B-cyclin/CDKs regulate mitotic spindle assembly by phosphorylating kinesins-5 in budding yeast. PLoS genetics 20100501
Conformer generation with OMEGA: algorithm and validation using high quality structures from the Protein Databank and Cambridge Structural Database. Journal of chemical information and modeling 20100426
L-Arginine stimulates proliferation and prevents endotoxin-induced death of intestinal cells. Amino acids 20100401
Bioinformatic and experimental survey of 14-3-3-binding sites. The Biochemical journal 20100401
Actin-related protein Arp6 influences H2A.Z-dependent and -independent gene expression and links ribosomal protein genes to nuclear pores. PLoS genetics 20100401
The expression of survivin and its related genes in adipocyte-derived stem cell by demethylation. Korean journal of anesthesiology 20100401
Pituitary adenylate cyclase-activating polypeptide (PACAP)/PAC1HOP1 receptor activation coordinates multiple neurotrophic signaling pathways: Akt activation through phosphatidylinositol 3-kinase gamma and vesicle endocytosis for neuronal survival. The Journal of biological chemistry 20100326
Regulation of actin polymerization and adhesion-dependent cell edge protrusion by the Abl-related gene (Arg) tyrosine kinase and N-WASp. Biochemistry 20100316
Apical surface expression of aspartic protease Plasmepsin 4, a potential transmission-blocking target of the plasmodium ookinete. The Journal of biological chemistry 20100312
Enhancement of hydrophobic interactions and hydrogen bond strength by cooperativity: synthesis, modeling, and molecular dynamics simulations of a congeneric series of thrombin inhibitors. Journal of medicinal chemistry 20100311
Expression quantitative trait loci analysis of two genes encoding rubisco activase in soybean. Plant physiology 20100301
Irreversible insertion of benzonitrile into platinum(II)-nitrogen bonds of nucleobase complexes. Synthesis and structural characterization of stable azametallacycle compounds. Inorganic chemistry 20100301
Endocytosis of the anthrax toxin is mediated by clathrin, actin and unconventional adaptors. PLoS pathogens 20100301
Biochemical study and in vitro insect immune suppression by a trypsin-like secreted protease from the nematode Steinernema carpocapsae. Parasite immunology 20100301
Formulation of immunoassay calibrators in pasteurized albumin can significantly enhance their durability. Journal of immunological methods 20100227
Architecture of the RNA polymerase II-TFIIF complex revealed by cross-linking and mass spectrometry. The EMBO journal 20100217
Calmodulin-dependent protein kinase kinase-beta activates AMPK without forming a stable complex: synergistic effects of Ca2+ and AMP. The Biochemical journal 20100215
Analysis of a new crystal form of procarboxypeptidase B: further insights into the catalytic mechanism. Biopolymers 20100201
Assessment of the enzymatic activity and inhibition using HPFA with a microreactor, trypsin, absorbed on immobilized artificial membrane. Journal of chromatographic science 20100201
Screening of benzamidine-based thrombin inhibitors via a linear interaction energy in continuum electrostatics model. Journal of computer-aided molecular design 20100201
Proteasome nuclear activity affects chromosome stability by controlling the turnover of Mms22, a protein important for DNA repair. PLoS genetics 20100201
Low muscle glycogen and elevated plasma free fatty acid modify but do not prevent exercise-induced PDH activation in human skeletal muscle. Diabetes 20100101
Partial purification and characterization of trypsin-like proteinases from insecticide-resistant and -susceptible strains of the maize weevil, Sitophilus zeamais. Comparative biochemistry and physiology. Part B, Biochemistry & molecular biology 20100101
Presynaptic external calcium signaling involves the calcium-sensing receptor in neocortical nerve terminals. PloS one 20100101
A stromal heat shock protein 70 system functions in protein import into chloroplasts in the moss Physcomitrella patens. The Plant cell 20100101
Rac1 and Cdc42 are regulators of HRasV12-transformation and angiogenic factors in human fibroblasts. BMC cancer 20100101
Identification of possible targets of the Aspergillus fumigatus CRZ1 homologue, CrzA. BMC microbiology 20100101
Structure of the HCMV UL16-MICB complex elucidates select binding of a viral immunoevasin to diverse NKG2D ligands. PLoS pathogens 20100101
Microtubules regulate migratory polarity through Rho/ROCK signaling in T cells. PloS one 20100101
Proteomic analysis of iron acquisition, metabolic and regulatory responses of Yersinia pestis to iron starvation. BMC microbiology 20100101
A mitotic phosphorylation feedback network connects Cdk1, Plk1, 53BP1, and Chk2 to inactivate the G(2)/M DNA damage checkpoint. PLoS biology 20100101
Role of plastid protein phosphatase TAP38 in LHCII dephosphorylation and thylakoid electron flow. PLoS biology 20100101
Madm (Mlf1 adapter molecule) cooperates with Bunched A to promote growth in Drosophila. Journal of biology 20100101
Selective serotonin reuptake inhibitors potentiate the rapid antidepressant-like effects of serotonin4 receptor agonists in the rat. PloS one 20100101
Whole genome analysis of p38 SAPK-mediated gene expression upon stress. BMC genomics 20100101
Scyl1 regulates Golgi morphology. PloS one 20100101
Purification and functional characterisation of rhinocerase, a novel serine protease from the venom of Bitis gabonica rhinoceros. PloS one 20100101
Hypoxia promotes glycogen accumulation through hypoxia inducible factor (HIF)-mediated induction of glycogen synthase 1. PloS one 20100101
Proteomics reveals novel oxidative and glycolytic mechanisms in type 1 diabetic patients' skin which are normalized by kidney-pancreas transplantation. PloS one 20100101
ERK1/2 signaling dominates over RhoA signaling in regulating early changes in RNA expression induced by endothelin-1 in neonatal rat cardiomyocytes. PloS one 20100101
High-fat diet-induced neuropathy of prediabetes and obesity: effect of PMI-5011, an ethanolic extract of Artemisia dracunculus L. Mediators of inflammation 20100101
Dysferlin interacts with tubulin and microtubules in mouse skeletal muscle. PloS one 20100101
Activation of rat liver microsomal glutathione transferase by hepsin. Biological & pharmaceutical bulletin 20100101
Phosphatidylinositol 3-kinase inhibitor(LY294002) induces apoptosis of human nasopharyngeal carcinoma in vitro and in vivo. Journal of experimental & clinical cancer research : CR 20100101
AKAR2-AKAP12 fusion protein 'biosenses' dynamic phosphorylation and localization of a GPCR-based scaffold. Journal of molecular signaling 20100101
A local role for the small ribosomal subunit primary binder rpS5 in final 18S rRNA processing in yeast. PloS one 20100101
Adhesion of renal carcinoma cells to endothelial cells depends on PKCmu. BMC cancer 20100101
Towards a membrane proteome in Drosophila: a method for the isolation of plasma membrane. BMC genomics 20100101
A positive feedback-based gene circuit to increase the production of a membrane protein. Journal of biological engineering 20100101
Trypsin-like serine proteases in Lutzomyia longipalpis--expression, activity and possible modulation by Leishmania infantum chagasi. PloS one 20100101
Trazodone effects on [H]-paroxetine and alpha(2)-adrenoreceptors in platelets of patients with major depression. Neuropsychiatric disease and treatment 20100101
Molecular cloning and biochemical characterization of a novel erythrose reductase from Candida magnoliae JH110. Microbial cell factories 20100101
Sterol carrier protein-x gene and effects of sterol carrier protein-2 inhibitors on lipid uptake in Manduca sexta. BMC physiology 20100101
Delta opioid receptor on equine sperm cells: subcellular localization and involvement in sperm motility analyzed by computer assisted sperm analyzer (CASA). Reproductive biology and endocrinology : RB&E 20100101
How pig sperm prepares to fertilize: stable acrosome docking to the plasma membrane. PloS one 20100101
Molecular composition of staufen2-containing ribonucleoproteins in embryonic rat brain. PloS one 20100101
Higher plant calreticulins have acquired specialized functions in Arabidopsis. PloS one 20100101
Brassinosteroid-mediated stress tolerance in Arabidopsis shows interactions with abscisic acid, ethylene and salicylic acid pathways. BMC plant biology 20100101
Increased apoptosis of myoblasts in Drosophila model for the Walker-Warburg syndrome. PloS one 20100101
Fluorescent fusion proteins of soluble guanylyl cyclase indicate proximity of the heme nitric oxide domain and catalytic domain. PloS one 20100101
Characterization of the first beta-class carbonic anhydrase from an arthropod (Drosophila melanogaster) and phylogenetic analysis of beta-class carbonic anhydrases in invertebrates. BMC biochemistry 20100101
Induction of early Purkinje cell dendritic differentiation by thyroid hormone requires RORα. Neural development 20100101
Stat3 activates the receptor tyrosine kinase like orphan receptor-1 gene in chronic lymphocytic leukemia cells. PloS one 20100101
Na+-stimulated ATPase of alkaliphilic halotolerant cyanobacterium Aphanothece halophytica translocates Na+ into proteoliposomes via Na+ uniport mechanism. BMC biochemistry 20100101
Calcineurin interacts with PERK and dephosphorylates calnexin to relieve ER stress in mammals and frogs. PloS one 20100101
Endotoxin tolerance and cross-tolerance in mast cells involves TLR4, TLR2 and FcepsilonR1 interactions and SOCS expression: perspectives on immunomodulation in infectious and allergic diseases. BMC infectious diseases 20100101
Delayed treatment with systemic (S)-roscovitine provides neuroprotection and inhibits in vivo CDK5 activity increase in animal stroke models. PloS one 20100101
Quantitative in vitro and in vivo pharmacological profile of CE-178253, a potent and selective cannabinoid type 1 (CB1) receptor antagonist. BMC pharmacology 20100101
Suppression of lung tumorigenesis by leucine zipper/EF hand-containing transmembrane-1. PloS one 20100101
Calcium regulation of EGF-induced ERK5 activation: role of Lad1-MEKK2 interaction. PloS one 20100101
Involvement of hyaluronidases in colorectal cancer. BMC cancer 20100101
Akt deficiency attenuates muscle size and function but not the response to ActRIIB inhibition. PloS one 20100101
The crystal structure of Toxoplasma gondii pyruvate kinase 1. PloS one 20100101
Self-association of the Lentivirus protein, Nef. Retrovirology 20100101
The role of growth retardation in lasting effects of neonatal dexamethasone treatment on hippocampal synaptic function. PloS one 20100101
A novel system for the efficient generation of antibodies following immunization of unique knockout mouse strains. PloS one 20100101
Quantitative phosphoproteomics of proteasome inhibition in multiple myeloma cells. PloS one 20100101
Sustained spindle-assembly checkpoint response requires de novo transcription and translation of cyclin B1. PloS one 20100101
The chondroitin/dermatan sulfate synthesizing and modifying enzymes in laryngeal cancer: expressional and epigenetic studies. Head & neck oncology 20100101
Signal transduction protein array analysis links LRRK2 to Ste20 kinases and PKC zeta that modulate neuronal plasticity. PloS one 20100101
Monomerization of cytosolic mature smac attenuates interaction with IAPs and potentiation of caspase activation. PloS one 20100101
A computational simulation study of benzamidine derivatives binding to arginine-specific gingipain (HRgpA) from periodontopathogen Porphyromonas gingivalis. International journal of molecular sciences 20100101
Expression of glycogen phosphorylase isoforms in cultured muscle from patients with McArdle's disease carrying the p.R771PfsX33 PYGM mutation. PloS one 20100101
Preclinical evaluation of novel triphenylphosphonium salts with broad-spectrum activity. PloS one 20100101
New insight into the dynamic properties and the active site architecture of H-Ras p21 revealed by X-ray crystallography at very high resolution. BMC structural biology 20100101
P130Cas Src-binding and substrate domains have distinct roles in sustaining focal adhesion disassembly and promoting cell migration. PloS one 20100101
Proteins involved in platelet signaling are differentially regulated in acute coronary syndrome: a proteomic study. PloS one 20100101
Optimizing structural modeling for a specific protein scaffold: knottins or inhibitor cystine knots. BMC bioinformatics 20100101
Classifying and scoring of molecules with the NGN: new datasets, significance tests, and generalization. BMC bioinformatics 20100101
MicroRNAs are mediators of androgen action in prostate and muscle. PloS one 20100101
Synphilin-1 enhances α-synuclein aggregation in yeast and contributes to cellular stress and cell death in a Sir2-dependent manner. PloS one 20100101
Impaired growth and force production in skeletal muscles of young partially pancreatectomized rats: a model of adolescent type 1 diabetic myopathy? PloS one 20100101
Molecularly imprinted polymers: shaping enzyme inhibitors. Nature chemistry 20100101
Fat oxidation, fitness and skeletal muscle expression of oxidative/lipid metabolism genes in South Asians: implications for insulin resistance? PloS one 20100101
Lewis Y promotes growth and adhesion of ovarian carcinoma-derived RMG-I cells by upregulating growth factors. International journal of molecular sciences 20100101
Down-regulation of phosphoglucomutase 3 mediates sulforaphane-induced cell death in LNCaP prostate cancer cells. Proteome science 20100101
Glyceraldehyde-3-phosphate dehydrogenase is largely unresponsive to low regulatory levels of hydrogen peroxide in Saccharomyces cerevisiae. BMC biochemistry 20100101
Ocular proteomics with emphasis on two-dimensional gel electrophoresis and mass spectrometry. Biological procedures online 20100101
miR-146a is critical for endotoxin-induced tolerance: IMPLICATION IN INNATE IMMUNITY. The Journal of biological chemistry 20091211
The anti-inflammatory agent bindarit inhibits neointima formation in both rats and hyperlipidaemic mice. Cardiovascular research 20091201
ON/OFF and beyond--a boolean model of apoptosis. PLoS computational biology 20091201
Intracellular autoactivation of human cationic trypsinogen mutants causes reduced trypsinogen secretion and acinar cell death. The Journal of biological chemistry 20091127
Biochemical and functional properties of a thrombin-like enzyme isolated from Bothrops pauloensis snake venom. Toxicon : official journal of the International Society on Toxinology 20091101
Nutrient stress activates inflammation and reduces glucose metabolism by suppressing AMP-activated protein kinase in the heart. Diabetes 20091101
Novel factor Xa inhibitors: a patent review. Expert opinion on therapeutic patents 20091101
The role of phosphorylated glucocorticoid receptor in mitochondrial functions and apoptotic signalling in brain tissue of stressed Wistar rats. The international journal of biochemistry & cell biology 20091101
4-Bromo-N,N'-bis-(4-methoxy-phen-yl)benzamidine. Acta crystallographica. Section E, Structure reports online 20091101
Molecularly imprinted microgels as enzyme inhibitors. Journal of the American Chemical Society 20091021
MAP kinase dependent cyclinE/cdk2 activity promotes DNA replication in early sea urchin embryos. Developmental biology 20091015
An apoptosis-inducing serine protease secreted by the entomopathogenic nematode Steinernema carpocapsae. International journal for parasitology 20091001
Regulation of type IV collagen alpha chains of glomerular epithelial cells in diabetic conditions. Journal of Korean medical science 20091001
EBNA1-mediated recruitment of a histone H2B deubiquitylating complex to the Epstein-Barr virus latent origin of DNA replication. PLoS pathogens 20091001
Clostridium difficile toxin CDT induces formation of microtubule-based protrusions and increases adherence of bacteria. PLoS pathogens 20091001
The elongator complex interacts with PCNA and modulates transcriptional silencing and sensitivity to DNA damage agents. PLoS genetics 20091001
The role of medical structural genomics in discovering new drugs for infectious diseases. PLoS computational biology 20091001
N,N-Bis-(2,6-di-methyl-phen-yl)-N-hydroxyformamidine N,N'-bis-(2,6-dimethyl-phen-yl)-N-oxidoformamidinium dichloro-methane solvate. Acta crystallographica. Section E, Structure reports online 20091001
Echinoderm phosphorylated matrix proteins UTMP16 and UTMP19 have different functions in sea urchin tooth mineralization. The Journal of biological chemistry 20090918
Gas phase stabilization of noncovalent protein complexes formed by electrospray ionization. Analytical chemistry 20090915
Cyclic olefin homopolymer-based microfluidics for protein crystallization and in situ X-ray diffraction. Acta crystallographica. Section D, Biological crystallography 20090901
Is amino acid racemization a useful tool for screening for ancient DNA in bone? Proceedings. Biological sciences 20090822
Immunocytochemical techniques reveal multiple, distinct cellular pools of PtdIns4P and PtdIns(4,5)P(2). The Biochemical journal 20090815
Three-dimensional structure of CaV3.1: comparison with the cardiac L-type voltage-gated calcium channel monomer architecture. The Journal of biological chemistry 20090814
alpha-ENaC is a functional element of the hypertonicity-induced cation channel in HepG2 cells and it mediates proliferation. Pflugers Archiv : European journal of physiology 20090801
Trypsin-ligand binding free energies from explicit and implicit solvent simulations with polarizable potential. Journal of computational chemistry 20090801
Characterization of the angiotensin (AT1b) receptor promoter and its regulation by glucocorticoids. Journal of molecular endocrinology 20090801
Casein kinase 1 isoform 2 is essential for bloodstream form Trypanosoma brucei. Molecular and biochemical parasitology 20090801
Bioactivity-guided mapping and navigation of chemical space. Nature chemical biology 20090801
Studies on the DIDS-binding site of monocarboxylate transporter 1 suggest a homology model of the open conformation and a plausible translocation cycle. The Journal of biological chemistry 20090724
Recombinant expression and affinity purification of snake venom gland parvalbumin in Escherichia coli. Comparative biochemistry and physiology. Part A, Molecular & integrative physiology 20090701
Infrared techniques for quantifying protein structural stability. Analytical biochemistry 20090701
The phosphoproteome of bloodstream form Trypanosoma brucei, causative agent of African sleeping sickness. Molecular & cellular proteomics : MCP 20090701
Ku-0063794 is a specific inhibitor of the mammalian target of rapamycin (mTOR). The Biochemical journal 20090701
Acute or chronic stress induce cell compartment-specific phosphorylation of glucocorticoid receptor and alter its transcriptional activity in Wistar rat brain. The Journal of endocrinology 20090701
Interference with hemozoin formation represents an important mechanism of schistosomicidal action of antimalarial quinoline methanols. PLoS neglected tropical diseases 20090701
Molecular dynamics of water-mediated interactions of a linear benzimidazole-biphenyl diamidine with the DNA minor groove. Journal of the American Chemical Society 20090610
Separate elements within a single IQ-like motif in adenylyl cyclase type 8 impart ca2+/calmodulin binding and autoinhibition. The Journal of biological chemistry 20090605
Amidine surface modification of poly(acrylonitrile-co-vinyl chloride) reduces platelet adhesion. Journal of biomedical materials research. Part A 20090601
GlcNAcstatins are nanomolar inhibitors of human O-GlcNAcase inducing cellular hyper-O-GlcNAcylation. The Biochemical journal 20090601
ATP and MO25alpha regulate the conformational state of the STRADalpha pseudokinase and activation of the LKB1 tumour suppressor. PLoS biology 20090601
A genome-wide screen for regulators of TORC1 in response to amino acid starvation reveals a conserved Npr2/3 complex. PLoS genetics 20090601
Prdx1 inhibits tumorigenesis via regulating PTEN/AKT activity. The EMBO journal 20090520
Blunting of AICAR-induced human skeletal muscle glucose uptake in type 2 diabetes is dependent on age rather than diabetic status. American journal of physiology. Endocrinology and metabolism 20090501
Structure of pig heart citrate synthase at 1.78 A resolution. Acta crystallographica. Section F, Structural biology and crystallization communications 20090501
Beneficial Effects of Fermented Green Tea Extract in a Rat Model of Non-alcoholic Steatohepatitis. Journal of clinical biochemistry and nutrition 20090501
Entropic cost of protein-ligand binding and its dependence on the entropy in solution. The journal of physical chemistry. B 20090430
Differential tissue-specific protein markers of vaginal carcinoma. British journal of cancer 20090421
Anthranilamide-based N,N-dialkylbenzamidines as potent and orally bioavailable factor Xa inhibitors: P4 SAR. Bioorganic & medicinal chemistry letters 20090415
Identification of the high affinity binding site in the Streptococcus intermedius toxin intermedilysin for its membrane receptor, the human complement regulator CD59. Molecular immunology 20090401
Structure and function of the human Gly1619Arg polymorphism of M6P/IGF2R domain 11 implicated in IGF2 dependent growth. Journal of molecular endocrinology 20090401
Impact of methylglyoxal and high glucose co-treatment on human mononuclear cells. International journal of molecular sciences 20090401
The trefoil factor interacting protein TFIZ1 binds the trefoil protein TFF1 preferentially in normal gastric mucosal cells but the co-expression of these proteins is deregulated in gastric cancer. The international journal of biochemistry & cell biology 20090301
Expression, purification, and characterization of recombinant human beta-amyloid42 peptide in Escherichia coli. Protein expression and purification 20090301
Overexpression of carnitine palmitoyltransferase-1 in skeletal muscle is sufficient to enhance fatty acid oxidation and improve high-fat diet-induced insulin resistance. Diabetes 20090301
Insights into the residence in lipid rafts of adenylyl cyclase AC8 and its regulation by capacitative calcium entry. American journal of physiology. Cell physiology 20090301
Detection of an L-amino acid dehydrogenase activity in Synechocystis sp. PCC 6803. Journal of experimental botany 20090301
Colouring cryo-cooled crystals: online microspectrophotometry. Journal of synchrotron radiation 20090301
An amphipathic alpha-helix controls multiple roles of brome mosaic virus protein 1a in RNA replication complex assembly and function. PLoS pathogens 20090301
Functional ryanodine receptors in the plasma membrane of RINm5F pancreatic beta-cells. The Journal of biological chemistry 20090220
DOC2B: a novel syntaxin-4 binding protein mediating insulin-regulated GLUT4 vesicle fusion in adipocytes. Diabetes 20090201
Whey protein ingestion activates mTOR-dependent signalling after resistance exercise in young men: a double-blinded randomized controlled trial. Nutrients 20090201
A role for water molecules in DNA-ligand minor groove recognition. Accounts of chemical research 20090120
Myogenic Akt signaling upregulates the utrophin-glycoprotein complex and promotes sarcolemma stability in muscular dystrophy. Human molecular genetics 20090115
C-terminal phosphorylation of LKB1 is not required for regulation of AMP-activated protein kinase, BRSK1, BRSK2, or cell cycle arrest. The Journal of biological chemistry 20090102
Intracellular amyloid formation in muscle cells of Abeta-transgenic Caenorhabditis elegans: determinants and physiological role in copper detoxification. Molecular neurodegeneration 20090101
Catalytic inhibition of topoisomerase II by a novel rationally designed ATP-competitive purine analogue. BMC chemical biology 20090101
An essential role of the universal polarity protein, aPKClambda, on the maintenance of podocyte slit diaphragms. PloS one 20090101
Alcohol-induced decrease in muscle protein synthesis associated with increased binding of mTOR and raptor: Comparable effects in young and mature rats. Nutrition & metabolism 20090101
Whi5 regulation by site specific CDK-phosphorylation in Saccharomyces cerevisiae. PloS one 20090101
The Staphylococcus aureus response to unsaturated long chain free fatty acids: survival mechanisms and virulence implications. PloS one 20090101
Cardiac force-frequency relationship and frequency-dependent acceleration of relaxation are impaired in LPS-treated rats. Critical care (London, England) 20090101
An effective docking strategy for virtual screening based on multi-objective optimization algorithm. BMC bioinformatics 20090101
miRNA-dependent translational repression in the Drosophila ovary. PloS one 20090101
Addition of a sequence from alpha2-antiplasmin transforms human serum albumin into a blood clot component that speeds clot lysis. BMC biotechnology 20090101
Preliminary evidence for cell membrane amelioration in children with cystic fibrosis by 5-MTHF and vitamin B12 supplementation: a single arm trial. PloS one 20090101
High Erk-1 activation and Gadd45a expression as prognostic markers in high risk pediatric haemolymphoproliferative diseases. Journal of experimental & clinical cancer research : CR 20090101
PP1gamma2 and PPP1R11 are parts of a multimeric complex in developing testicular germ cells in which their steady state levels are reciprocally related. PloS one 20090101
Chemically-induced RAT mesenchymal stem cells adopt molecular properties of neuronal-like cells but do not have basic neuronal functional properties. PloS one 20090101
Site directed mutagenesis of amino acid residues at the active site of mouse aldehyde oxidase AOX1. PloS one 20090101
A vault nanoparticle vaccine induces protective mucosal immunity. PloS one 20090101
Apoptosis signal-regulating kinase 1 mediates denbinobin-induced apoptosis in human lung adenocarcinoma cells. Journal of biomedical science 20090101
The Carboxy-Terminal Modulator Protein (CTMP) regulates mitochondrial dynamics. PloS one 20090101
Canine babesiosis: from molecular taxonomy to control. Parasites & vectors 20090101
Purification and characterization of a serine protease (CESP) from mature coconut endosperm. BMC research notes 20090101
Emodin targets the beta-hydroxyacyl-acyl carrier protein dehydratase from Helicobacter pylori: enzymatic inhibition assay with crystal structural and thermodynamic characterization. BMC microbiology 20090101
Knockout studies reveal an important role of Plasmodium lipoic acid protein ligase A1 for asexual blood stage parasite survival. PloS one 20090101
Expression of hyaluronan synthases (HAS1-3) and hyaluronidases (HYAL1-2) in serous ovarian carcinomas: inverse correlation between HYAL1 and hyaluronan content. BMC cancer 20090101
PfeIK1, a eukaryotic initiation factor 2alpha kinase of the human malaria parasite Plasmodium falciparum, regulates stress-response to amino-acid starvation. Malaria journal 20090101
Cereal and nonfat milk support muscle recovery following exercise. Journal of the International Society of Sports Nutrition 20090101
Conserved features of cohesin binding along fission yeast chromosomes. Genome biology 20090101
Co-ordinated stage-dependent enhancement of Plasmodium falciparum antioxidant enzymes and heat shock protein expression in parasites growing in oxidatively stressed or G6PD-deficient red blood cells. Malaria journal 20090101
Cloning and analysis of a bifunctional methyltransferase/restriction endonuclease TspGWI, the prototype of a Thermus sp. enzyme family. BMC molecular biology 20090101
Conserved threonine residues within the A-loop of the receptor NIK differentially regulate the kinase function required for antiviral signaling. PloS one 20090101
TIPT2 and geminin interact with basal transcription factors to synergize in transcriptional regulation. BMC biochemistry 20090101
Unconjugated bilirubin exposure impairs hippocampal long-term synaptic plasticity. PloS one 20090101
Lapatinib, a dual EGFR and HER2 tyrosine kinase inhibitor, downregulates thymidylate synthase by inhibiting the nuclear translocation of EGFR and HER2. PloS one 20090101
PAR1 is selectively over expressed in high grade breast cancer patients: a cohort study. Journal of translational medicine 20090101
Synovial fluid level of aggrecan ARGS fragments is a more sensitive marker of joint disease than glycosaminoglycan or aggrecan levels: a cross-sectional study. Arthritis research & therapy 20090101
Protein Never in Mitosis Gene A Interacting-1 regulates calpain activity and the degradation of cyclooxygenase-2 in endothelial cells. Journal of inflammation (London, England) 20090101
Long-term potentiation in isolated dendritic spines. PloS one 20090101
Is inflammation a consequence of extracellular hyperosmolarity? Journal of inflammation (London, England) 20090101
Gene expression profiling identifies activated growth factor signaling in poor prognosis (Luminal-B) estrogen receptor positive breast cancer. BMC medical genomics 20090101
Comparison of two label-free global quantitation methods, APEX and 2D gel electrophoresis, applied to the Shigella dysenteriae proteome. Proteome science 20090101
Host envelope glycoprotein processing proteases are indispensable for entry into human cells by seasonal and highly pathogenic avian influenza viruses. Journal of molecular and genetic medicine : an international journal of biomedical research 20090101
Structure-function analysis of nucleolin and ErbB receptors interactions. PloS one 20090101
Molt-inhibiting hormone stimulates vitellogenesis at advanced ovarian developmental stages in the female blue crab, Callinectes sapidus 2: novel specific binding sites in hepatopancreas and cAMP as a second messenger. Saline systems 20090101
Oocyte-specific deletion of Pten in mice reveals a stage-specific function of PTEN/PI3K signaling in oocytes in controlling follicular activation. PloS one 20090101
Adenylate-cyclase activity in platelets of patients with obsessive-compulsive disorder. Neuropsychiatric disease and treatment 20090101
Nucleocytoplasmic shuttling of the TACC protein Mia1p/Alp7p is required for remodeling of microtubule arrays during the cell cycle. PloS one 20090101
Phospho-ablated Id2 is growth suppressive and pro-apoptotic in proliferating myoblasts. PloS one 20090101
The excitotoxin quinolinic acid induces tau phosphorylation in human neurons. PloS one 20090101
Comparative study of the swabbing properties of seven commercially available swab materials for cleaning verification. PDA journal of pharmaceutical science and technology 20090101
Paraquat induces oxidative stress, neuronal loss in substantia nigra region and parkinsonism in adult rats: neuroprotection and amelioration of symptoms by water-soluble formulation of coenzyme Q10. BMC neuroscience 20090101
Multiple histone modifications in euchromatin promote heterochromatin formation by redundant mechanisms in Saccharomyces cerevisiae. BMC molecular biology 20090101
Hypoxia-induced transcription of dopamine D3 and D4 receptors in human neuroblastoma and astrocytoma cells. BMC neuroscience 20090101
Ligand scaffold hopping combining 3D maximal substructure search and molecular similarity. BMC bioinformatics 20090101
Suppression of experimental uveitis by a recombinant adeno-associated virus vector encoding interleukin-1 receptor antagonist. Molecular vision 20090101
Selenoprotein N is dynamically expressed during mouse development and detected early in muscle precursors. BMC developmental biology 20090101
Alpha-glucosidase promotes hemozoin formation in a blood-sucking bug: an evolutionary history. PloS one 20090101
The Sam domain of the lipid phosphatase Ship2 adopts a common model to interact with Arap3-Sam and EphA2-Sam. BMC structural biology 20090101
LKR/SDH plays important roles throughout the tick life cycle including a long starvation period. PloS one 20090101
Immature and mature species of the human Prostacyclin Receptor are ubiquitinated and targeted to the 26S proteasomal or lysosomal degradation pathways, respectively. Journal of molecular signaling 20090101
Suppression of growth, migration and invasion of highly-metastatic human breast cancer cells by berbamine and its molecular mechanisms of action. Molecular cancer 20090101
Stem cell therapy with overexpressed VEGF and PDGF genes improves cardiac function in a rat infarct model. PloS one 20090101
Effects of isoflavone-supplemented soy yogurt on lipid parameters and atherosclerosis development in hypercholesterolemic rabbits: a randomized double-blind study. Lipids in health and disease 20090101
Modified epidermal growth factor receptor (EGFR)-bearing liposomes (MRBLs) are sensitive to EGF in solution. PloS one 20090101
The goldfish SG2NA gene encodes two alpha-type regulatory subunits for PP-2A and displays distinct developmental expression pattern. Gene regulation and systems biology 20090101
Biochemical and virological analysis of the 18-residue C-terminal tail of HIV-1 integrase. Retrovirology 20090101
Infectivity of Leishmania mexicana is associated with differential expression of protein kinase C-like triggered during a cell-cell contact. PloS one 20090101
The molecular basis for stability of heterochromatin-mediated silencing in mammals. Epigenetics & chromatin 20090101
Vitamin B6 deficient plants display increased sensitivity to high light and photo-oxidative stress. BMC plant biology 20090101
Differential requirement for MEK Partner 1 in DU145 prostate cancer cell migration. Cell communication and signaling : CCS 20090101
Alterations in gene expression and sensitivity to genotoxic stress following HdmX or Hdm2 knockdown in human tumor cells harboring wild-type p53. Aging 20090101
Functional role of p-glycoprotein and binding protein effect on the placental transfer of lopinavir/ritonavir in the ex vivo human perfusion model. Obstetrics and gynecology international 20090101
Trypsin-ligand binding free energy calculation with AMOEBA. Conference proceedings : ... Annual International Conference of the IEEE Engineering in Medicine and Biology Society. IEEE Engineering in Medicine and Biology Society. Annual Conference 20090101
Structural requirements for PACSIN/Syndapin operation during zebrafish embryonic notochord development. PloS one 20090101
Depot-specific differences in perilipin and hormone-sensitive lipase expression in lean and obese. Lipids in health and disease 20090101
The Noc-domain containing C-terminus of Noc4p mediates both formation of the Noc4p-Nop14p submodule and its incorporation into the SSU processome. PloS one 20090101
Evolution of primary hemostasis in early vertebrates. PloS one 20090101
Activation of Wnt/beta-catenin signaling increases insulin sensitivity through a reciprocal regulation of Wnt10b and SREBP-1c in skeletal muscle cells. PloS one 20090101
Determinants Present in the Receptor Carboxy Tail Are Responsible for Differences in Subtype-Specific Coupling of beta-Adrenergic Receptors to Phosphoinositide 3-Kinase. International journal of cell biology 20090101
VAC14 nucleates a protein complex essential for the acute interconversion of PI3P and PI(3,5)P(2) in yeast and mouse. The EMBO journal 20081217
NFAT regulates induction of COX-2 and apoptosis of keratinocytes in response to ultraviolet radiation exposure. FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20081201
UTP and ATP increase extracellular signal-regulated kinase 1/2 phosphorylation in bovine chromaffin cells through epidermal growth factor receptor transactivation. Purinergic signalling 20081201
Seminal plasma proteins of Atlantic halibut (Hippoglossus hippoglossus L.). Fish physiology and biochemistry 20081201
Using Caenorhabditis elegans as a model organism for evaluating extracellular signal-regulated kinase docking domain inhibitors. Journal of cell communication and signaling 20081201
Anticancer alkaloid lamellarins inhibit protein kinases. Marine drugs 20081201
Use of a decoy peptide to purify p21 activated kinase-1 in cardiac muscle and identification of ceramide-related activation. Biologics : targets & therapy 20081201
DNA-small molecule chimera with responsive protein-binding ability. Journal of the American Chemical Society 20081112
Sprint training increases muscle oxidative metabolism during high-intensity exercise in patients with type 1 diabetes. Diabetes care 20081101
Aminoglycoside resistance genes sgm and kgmB protect bacterial but not yeast small ribosomal subunits in vitro despite high conservation of the rRNA A-site. Research in microbiology 20081101
rac regulates its effector phospholipase Cgamma2 through interaction with a split pleckstrin homology domain. The Journal of biological chemistry 20081031
Temporal and spatial regulation of the phosphatidate phosphatases lipin 1 and 2. The Journal of biological chemistry 20081024
Structural insights into mechanism and specificity of O-GlcNAc transferase. The EMBO journal 20081022
Synthesis of novel benzamidine- and guanidine-derived polyazamacrocycles: Selective anti-protozoal activity for human African trypanosomiasis. Bioorganic & medicinal chemistry letters 20081015
Structural analysis of the interactions between paxillin LD motifs and alpha-parvin. Structure (London, England : 1993) 20081008
Elevated toll-like receptor 4 expression and signaling in muscle from insulin-resistant subjects. Diabetes 20081001
Reductions in mesophyll and guard cell photosynthesis impact on the control of stomatal responses to light and CO2. Journal of experimental botany 20081001
Regulated expression of an essential allosteric activator of polyamine biosynthesis in African trypanosomes. PLoS pathogens 20081001
Rapid-reaction kinetic characterization of the pathway of streptokinase-plasmin catalytic complex formation. The Journal of biological chemistry 20080919
Anti-microtubule activity of tubeimoside I and its colchicine binding site of tubulin. Cancer chemotherapy and pharmacology 20080901
If the antibody fails--a mass western approach. The Plant journal : for cell and molecular biology 20080901
Development of a countergradient parking system for gradient liquid chromatography with online biochemical detection of serine protease inhibitors. Analytical chemistry 20080901
Rice XB15, a protein phosphatase 2C, negatively regulates cell death and XA21-mediated innate immunity. PLoS biology 20080901
Crystal structure of soluble domain of malaria sporozoite protein UIS3 in complex with lipid. The Journal of biological chemistry 20080829
Structure-function analysis of the C3 binding region of Staphylococcus aureus immune subversion protein Sbi. The Journal of biological chemistry 20080808
QacR-cation recognition is mediated by a redundancy of residues capable of charge neutralization. Biochemistry 20080805
Hypothalamic protein kinase C regulates glucose production. Diabetes 20080801
Cyclin-dependent kinase inhibitor p27Kip1 controls growth and cell cycle progression in human uterine leiomyoma. Journal of Korean medical science 20080801
Hormone-sensitive lipase serine phosphorylation and glycerol exchange across skeletal muscle in lean and obese subjects: effect of beta-adrenergic stimulation. Diabetes 20080701
Cytokinin deficiency causes distinct changes of sink and source parameters in tobacco shoots and roots. Journal of experimental botany 20080701
Benzamidinium tetra-hydro-penta-borate sesquihydrate. Acta crystallographica. Section E, Structure reports online 20080701
Inhibition of V3-specific cleavage of recombinant HIV-1 gp120 produced in Chinese hamster ovary cells. Protein expression and purification 20080601
Identification of a serine protease as a major allergen (Per a 10) of Periplaneta americana. Allergy 20080601
4-Ammonio-benzamidinium dichloride. Acta crystallographica. Section E, Structure reports online 20080601
Novel potent and selective thrombin inhibitors based on a central 1,4-benzoxazin-3(4H)-one scaffold. Journal of medicinal chemistry 20080508
APC promoter methylation and protein expression in hepatocellular carcinoma. Journal of cancer research and clinical oncology 20080501
Myocardial adaptation of energy metabolism to elevated preload depends on calcineurin activity : a proteomic approach. Basic research in cardiology 20080501
Structure of isochorismate synthase in complex with magnesium. Acta crystallographica. Section D, Biological crystallography 20080501
Caffeine induces cell death via activation of apoptotic signal and inactivation of survival signal in human osteoblasts. International journal of molecular sciences 20080501
Contribution of P2Y(1) receptors to ADP signalling in mouse spinal cord cultures. Neuroscience letters 20080425
Arp2/3 complex interactions and actin network turnover in lamellipodia. The EMBO journal 20080409
Isolation and structural characterization of a new fibrin(ogen)olytic metalloproteinase from Bothrops moojeni snake venom. Toxicon : official journal of the International Society on Toxinology 20080315
Reductive isoxazole ring opening of the anticoagulant razaxaban is the major metabolic clearance pathway in rats and dogs. Drug metabolism and disposition: the biological fate of chemicals 20080201
Plasmodium falciparum regulatory subunit of cAMP-dependent PKA and anion channel conductance. PLoS pathogens 20080201
Motility screen identifies Drosophila IGF-II mRNA-binding protein--zipcode-binding protein acting in oogenesis and synaptogenesis. PLoS genetics 20080201
MSPL/TMPRSS13. Frontiers in bioscience : a journal and virtual library 20080101
Evaluation of the inhibitory effects of human serum components on bactericidal activity of human beta defensin 3. Peptides 20080101
Inhibition of hyaluronan export reduces collagen degradation in interleukin-1 treated cartilage. Arthritis research & therapy 20080101
Mutational analysis of betaCOP (Sec26p) identifies an appendage domain critical for function. BMC cell biology 20080101
A prevalent variant in PPP1R3A impairs glycogen synthesis and reduces muscle glycogen content in humans and mice. PLoS medicine 20080101
Identification of a novel Leucine-rich repeat protein and candidate PP1 regulatory subunit expressed in developing spermatids. BMC cell biology 20080101
Expression of the 'stem cell marker' CD133 in pancreas and pancreatic ductal adenocarcinomas. BMC cancer 20080101
Isolation, cloning and structural characterisation of boophilin, a multifunctional Kunitz-type proteinase inhibitor from the cattle tick. PloS one 20080101
Identification and characterization of a novel Plasmodium falciparum merozoite apical protein involved in erythrocyte binding and invasion. PloS one 20080101
The orexigenic effect of ghrelin is mediated through central activation of the endogenous cannabinoid system. PloS one 20080101
Imp-L2, a putative homolog of vertebrate IGF-binding protein 7, counteracts insulin signaling in Drosophila and is essential for starvation resistance. Journal of biology 20080101
Differential expression of the catalytic subunits for PP-1 and PP-2A and the regulatory subunits for PP-2A in mouse eye. Molecular vision 20080101
TNK2 preserves epidermal growth factor receptor expression on the cell surface and enhances migration and invasion of human breast cancer cells. Breast cancer research : BCR 20080101
Mutation at tyrosine in AMLRY (GILRY like) motif of yeast eRF1 on nonsense codons suppression and binding affinity to eRF3. International journal of biological sciences 20080101
A facile route to 2,4-dihydro-1H-benzo[d][1,3]thiazines via silver-catalyzed tandem addition-cyclization reactions. Journal of combinatorial chemistry 20080101
The yeast Tor signaling pathway is involved in G2/M transition via polo-kinase. PloS one 20080101
His-tag ELISA for the detection of humoral tumor-specific immunity. BMC immunology 20080101
Identification of immune genes and proteins involved in the response of bovine mammary tissue to Staphylococcus aureus infection. BMC veterinary research 20080101
High-level expression, single-step immunoaffinity purification and characterization of human tetraspanin membrane protein CD81. PloS one 20080101
Combination of native and denaturing PAGE for the detection of protein binding regions in long fragments of genomic DNA. BMC genomics 20080101
Skeletal muscle-specific ablation of gamma(cyto)-actin does not exacerbate the mdx phenotype. PloS one 20080101
Human pregnane X receptor is expressed in breast carcinomas, potential heterodimers formation between hPXR and RXR-alpha. BMC cancer 20080101
Fragmentation of decorin, biglycan, lumican and keratocan is elevated in degenerate human meniscus, knee and hip articular cartilages compared with age-matched macroscopically normal and control tissues. Arthritis research & therapy 20080101
Fus3-triggered Tec1 degradation modulates mating transcriptional output during the pheromone response. Molecular systems biology 20080101
Novel functional view of the crocidolite asbestos-treated A549 human lung epithelial transcriptome reveals an intricate network of pathways with opposing functions. BMC genomics 20080101
Mutational analysis of highly conserved aspartate residues essential to the catalytic core of the piggyBac transposase. BMC molecular biology 20080101
Circadian control of the daily plasma glucose rhythm: an interplay of GABA and glutamate. PloS one 20080101
Effect of exercise training on calpain systems in lean and obese Zucker rats. International journal of biological sciences 20080101
NF-kappaB mediates the survival of human bronchial epithelial cells exposed to cigarette smoke extract. Respiratory research 20080101
P38 MAP kinase signaling is required for the conversion of CD4+CD25- T cells into iTreg. PloS one 20080101
Oxygen-independent stabilization of hypoxia inducible factor (HIF)-1 during RSV infection. PloS one 20080101
A role of p38 mitogen-activated protein kinase in adenosine A₁ receptor-mediated synaptic depotentiation in area CA1 of the rat hippocampus. Molecular brain 20080101
Isolation and characterization of betaA3-crystallin associated proteinase from alpha-crystallin fraction of human lenses. Molecular vision 20080101
Cutaneous tactile allodynia associated with microvascular dysfunction in muscle. Molecular pain 20080101
Small molecule, non-peptide p75 ligands inhibit Abeta-induced neurodegeneration and synaptic impairment. PloS one 20080101
Displacement affinity chromatography of protein phosphatase one (PP1) complexes. BMC biochemistry 20080101
Arabidopsis At5g39790 encodes a chloroplast-localized, carbohydrate-binding, coiled-coil domain-containing putative scaffold protein. BMC plant biology 20080101
G-protein-coupled receptor-associated A-kinase anchoring proteins AKAP5 and AKAP12: differential signaling to MAPK and GPCR recycling. Journal of molecular signaling 20080101
Evaluation of an in silico predicted specific and immunogenic antigen from the OmcB protein for the serodiagnosis of Chlamydia trachomatis infections. BMC microbiology 20080101
Cell culture-based analysis of postsynaptic membrane assembly in muscle cells. Biological procedures online 20080101
Homogenous fluorescent assays for characterizing small-molecule activators of AMP-activated protein kinase (AMPK). Current chemical genomics 20080101
N,N'-dihydroxyamidines: a new prodrug principle to improve the oral bioavailability of amidines. Journal of medicinal chemistry 20071227
Small-scale, semi-automated purification of eukaryotic proteins for structure determination. Journal of structural and functional genomics 20071201
Edema toxin impairs anthracidal phospholipase A2 expression by alveolar macrophages. PLoS pathogens 20071201
Apicoplast lipoic acid protein ligase B is not essential for Plasmodium falciparum. PLoS pathogens 20071201
Identification of aberrant forms of alkaline sphingomyelinase (NPP7) associated with human liver tumorigenesis. British journal of cancer 20071119
Effects of serine protease inhibitors on viability and morphology of Leishmania (Leishmania) amazonensis promastigotes. Parasitology research 20071101
Development of an open-tubular trypsin reactor for on-line digestion of proteins. Analytical and bioanalytical chemistry 20071101
Three-dimensional analysis of a viral RNA replication complex reveals a virus-induced mini-organelle. PLoS biology 20070901
Change of the expression of human telomerase reverse transcriptase mRNA and human telomerase RNA after cisplatin and 5-fluorouracil exposure in head and neck squamous cell carcinoma cell lines. Journal of Korean medical science 20070901
Structural basis of PP2A inhibition by small t antigen. PLoS biology 20070801
Cancer-associated retinopathy in patients with breast carcinoma. Archivum immunologiae et therapiae experimentalis 20070801
Co-localization and functional cross-talk between A1 and P2Y1 purine receptors in rat hippocampus. The European journal of neuroscience 20070801
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Computation of entropy contribution to protein-ligand binding free energy. Biochemistry. Biokhimiia 20070701
Quantification of growth factors in allogenic bone grafts extracted with three different methods. Cell and tissue banking 20070601
Dual lipolytic control of body fat storage and mobilization in Drosophila. PLoS biology 20070601
Sensitivity of yeast strains with long G-tails to levels of telomere-bound telomerase. PLoS genetics 20070601
Lipid-bound factor Xa regulates tissue factor activity. Biochemistry 20070522
Solution behaviour and biological activity of bisamidine complexes of platinum(II). Journal of biological inorganic chemistry : JBIC : a publication of the Society of Biological Inorganic Chemistry 20070501
Palmitoylation of the TPbeta isoform of the human thromboxane A2 receptor. Modulation of G protein: effector coupling and modes of receptor internalization. Cellular signalling 20070501
Centrosomal latency of incoming foamy viruses in resting cells. PLoS pathogens 20070501
Purification and properties of a coagulant thrombin-like enzyme from the venom of Bothrops leucurus. Comparative biochemistry and physiology. Part A, Molecular & integrative physiology 20070401
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Crystal structure of the catalytic domain of DESC1, a new member of the type II transmembrane serine proteinase family. The FEBS journal 20070401
Antibody to aquaporin 4 in the diagnosis of neuromyelitis optica. PLoS medicine 20070401
Design, synthesis and molecular modelling of 1-amidinopiperidine thrombin inhibitors. Die Pharmazie 20070401
Activation of trypsinogen in large endocytic vacuoles of pancreatic acinar cells. Proceedings of the National Academy of Sciences of the United States of America 20070327
Purification and biological activity of the thrombin-like substance isolated from Bothrops insularis venom. Toxicon : official journal of the International Society on Toxinology 20070301
Understanding binding selectivity toward trypsin and factor Xa: the role of aromatic interactions. ChemMedChem 20070301
The gene vitellogenin has multiple coordinating effects on social organization. PLoS biology 20070301
Impact of trivalent arsenicals on selenoprotein synthesis. Environmental health perspectives 20070301
Aging-associated reductions in AMP-activated protein kinase activity and mitochondrial biogenesis. Cell metabolism 20070207
Method for stabilizing protein-ligand complexes in nanoelectrospray ionization mass spectrometry. Analytical chemistry 20070115
A novel fibrinolytic serine protease from the polychaete Nereis (Neanthes) virens (Sars): purification and characterization. Biochimie 20070101
A comparative study of the expression of serine proteinases in quiescent seeds and in developing Canavalia ensiformis plants. Journal of experimental botany 20070101
Distinct glucose-dependent stress responses revealed by translational profiling in pancreatic beta-cells. The Journal of endocrinology 20070101
pRb-mediated control of epithelial cell proliferation and Indian hedgehog expression in mouse intestinal development. BMC developmental biology 20070101
Isolation and characterization of a novel acid proteinase, tropiase, from Candida tropicalis IFO 0589. Nihon Ishinkin Gakkai zasshi = Japanese journal of medical mycology 20070101
Glycogen synthase kinase 3, circadian rhythms, and bipolar disorder: a molecular link in the therapeutic action of lithium. Journal of circadian rhythms 20070101
Temporal dynamics of gene expression in the lung in a baboon model of E. coli sepsis. BMC genomics 20070101
Identification of a human TFPI-2 splice variant that is upregulated in human tumor tissues. Molecular cancer 20070101
Subfertility in mice harboring a mutation in betaB2-crystallin. Molecular vision 20070101
Repressor element-1 silencing transcription factor/neuronal restrictive silencer factor (REST/NRSF) can regulate HSV-1 immediate-early transcription via histone modification. Virology journal 20070101
Differential expression and role of p21cip/waf1 and p27kip1 in TNF-alpha-induced inhibition of proliferation in human glioma cells. Molecular cancer 20070101
The Sas3p and Gcn5p histone acetyltransferases are recruited to similar genes. Genome biology 20070101
Crystal structure of vaccinia virus uracil-DNA glycosylase reveals dimeric assembly. BMC structural biology 20070101
Neuronal conduction of excitation without action potentials based on ceramide production. PloS one 20070101
Developmental expression of three small GTPases in the mouse eye. Molecular vision 20070101
Analysis of the Rana catesbeiana tadpole tail fin proteome and phosphoproteome during T3-induced apoptosis: identification of a novel type I keratin. BMC developmental biology 20070101
De novo protein sequence analysis of Macaca mulatta. BMC genomics 20070101
C-terminal processing of yeast Spt7 occurs in the absence of functional SAGA complex. BMC biochemistry 20070101
Identification of serine proteases from Leishmania braziliensis. Zeitschrift fur Naturforschung. C, Journal of biosciences 20070101
p21 is decreased in polycystic kidney disease and leads to increased epithelial cell cycle progression: roscovitine augments p21 levels. BMC nephrology 20070101
Arterial response to shear stress critically depends on endothelial TRPV4 expression. PloS one 20070101
A new method to precipitate myosin V from rat brain soluble fraction. Acta biochimica Polonica 20070101
Deletion of PKBalpha/Akt1 affects thymic development. PloS one 20070101
Procollagen triple helix assembly: an unconventional chaperone-assisted folding paradigm. PloS one 20070101
The p11/S100A10 light chain of annexin A2 is dispensable for annexin A2 association to endosomes and functions in endosomal transport. PloS one 20070101
The redox sensor TXNL1 plays a regulatory role in fluid phase endocytosis. PloS one 20070101
Diversity and evolution of phycobilisomes in marine Synechococcus spp.: a comparative genomics study. Genome biology 20070101
Asn 362 in gp120 contributes to enhanced fusogenicity by CCR5-restricted HIV-1 envelope glycoprotein variants from patients with AIDS. Retrovirology 20070101
A large-scale proteomic analysis of human embryonic stem cells. BMC genomics 20070101
Expression of junctional proteins in choroid plexus epithelial cell lines: a comparative study. Cerebrospinal fluid research 20070101
Paradoxical role of an Egr transcription factor family member, Egr2/Krox20, in learning and memory. Frontiers in behavioral neuroscience 20070101
Canine plasminogen: spectral responses to changes in 6-aminohexanoate and temperature. Analytical chemistry insights 20070101
Potent and selective TF/FVIIa inhibitors containing a neutral P1 ligand. Bioorganic & medicinal chemistry 20061201
Genotoxic activity of halogenated phenylglycine derivatives. Bioorganic & medicinal chemistry letters 20061201
Enhancement of transfection activity of lipoplexes by complexation with transferrin-bearing fusogenic polymer-modified liposomes. International journal of pharmaceutics 20061115
Inhibitory effect of carboxylic acid group on hERG binding. Bioorganic & medicinal chemistry letters 20061101
Proteolytic processing of a sea urchin, ECM-localized protein into lower mol mass species possessing collagen-cleavage activity. Journal of cellular biochemistry 20061015
Structure of Staphylococcus aureus guanylate monophosphate kinase. Acta crystallographica. Section F, Structural biology and crystallization communications 20061001
The structural basis for promoter -35 element recognition by the group IV sigma factors. PLoS biology 20060901
Degradation of extracellular matrix proteins (fibronectin, vitronectin and laminin) by serine-proteinases isolated from Lonomia achelous caterpillar hemolymph. Blood coagulation & fibrinolysis : an international journal in haemostasis and thrombosis 20060901
Crystallization and X-ray data analysis of the 10 kDa C-terminal lid subdomain from Caenorhabditis elegans Hsp70. Acta crystallographica. Section F, Structural biology and crystallization communications 20060901
High resolution structures of p-aminobenzamidine- and benzamidine-VIIa/soluble tissue factor: unpredicted conformation of the 192-193 peptide bond and mapping of Ca2+, Mg2+, Na+, and Zn2+ sites in factor VIIa. The Journal of biological chemistry 20060825
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Structure of Staphylococcus aureus cytidine monophosphate kinase in complex with cytidine 5'-monophosphate. Acta crystallographica. Section F, Structural biology and crystallization communications 20060801
Crystallization and preliminary X-ray diffraction analysis of BipD, a virulence factor from Burkholderia pseudomallei. Acta crystallographica. Section F, Structural biology and crystallization communications 20060801
Arsenic exposure is associated with decreased DNA repair in vitro and in individuals exposed to drinking water arsenic. Environmental health perspectives 20060801
Binding characteristics of the Lactobacillus brevis ATCC 8287 surface layer to extracellular matrix proteins. FEMS microbiology letters 20060701
Investigating the basis of substrate recognition in the pC221 relaxosome. Molecular microbiology 20060601
Morphology and preliminary enzyme characterization of the salivary glands from the predatory bug Podisus nigrispinus (Heteroptera: Pentatomidae). Bulletin of entomological research 20060601
Microsphere-based protease assays and screening application for lethal factor and factor Xa. Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501
Isolation and characterization of a trypsin fraction from the pyloric ceca of chinook salmon (Oncorhynchus tshawytscha). Comparative biochemistry and physiology. Part B, Biochemistry & molecular biology 20060401
SAR and inhibitor complex structure determination of a novel class of potent and specific Aurora kinase inhibitors. Bioorganic & medicinal chemistry letters 20060301
The crystal structure of TrpD, a metabolic enzyme essential for lung colonization by Mycobacterium tuberculosis, in complex with its substrate phosphoribosylpyrophosphate. Journal of molecular biology 20060127
Upregulated but insufficient generation of activated protein C is associated with development of multiorgan failure in severe acute pancreatitis. Critical care (London, England) 20060101
Direct interaction between the catalytic subunit of Protein Phosphatase 1 and pRb. Cancer cell international 20060101
Levels of protein C and activated protein C: what do they mean? Critical care (London, England) 20060101
Cartilage oligomeric matrix protein is involved in human limb development and in the pathogenesis of osteoarthritis. Arthritis research & therapy 20060101
The quest for bioisosteric replacements. Journal of chemical information and modeling 20060101
Functional characterisation of the regulation of CAAT enhancer binding protein alpha by GSK-3 phosphorylation of Threonines 222/226. BMC molecular biology 20060101
Differences in MAP kinase phosphorylation in response to mechanical strain in asthmatic fibroblasts. Respiratory research 20060101
Induction of release and up-regulated gene expression of interleukin (IL)-8 in A549 cells by serine proteinases. BMC cell biology 20060101
Large-scale and high-confidence proteomic analysis of human seminal plasma. Genome biology 20060101
Synthetic protein-protein interaction domains created by shuffling Cys2His2 zinc-fingers. Molecular systems biology 20060101
Identification of specific calcitonin-like receptor residues important for calcitonin gene-related peptide high affinity binding. BMC pharmacology 20060101
Alteration of serotonin transporter density and activity in fibromyalgia. Arthritis research & therapy 20060101
Histone deacetylase enzymes as potential drug targets in cancer and parasitic diseases. Journal of biomedicine & biotechnology 20060101
Integration of metabolite with transcript and enzyme activity profiling during diurnal cycles in Arabidopsis rosettes. Genome biology 20060101
Isolation and characterization of a novel elastase inhibitor, AFLEI from Aspergillus flavus. Nihon Ishinkin Gakkai zasshi = Japanese journal of medical mycology 20060101
Glycogen synthase kinase 3 has a limited role in cell cycle regulation of cyclin D1 levels. BMC cell biology 20060101
New insight into the role of phosphodiesterase 3A in porcine oocyte maturation. BMC developmental biology 20060101
The effects of continuous venovenous hemofiltration on coagulation activation. Critical care (London, England) 20060101
Implantation Serine Proteinases heterodimerize and are critical in hatching and implantation. BMC developmental biology 20060101
Amino terminal tyrosine phosphorylation of human MIXL1. Journal of molecular signaling 20060101
Agonist mediated internalization of M2 mAChR is beta-arrestin-dependent. Journal of molecular signaling 20060101
[Plasminogen activator from Agkistrodon halys halys venom]. Ukrains'kyi biokhimichnyi zhurnal (1999 ) 20060101
Specific conformational changes of plasminogen induced by chloride ions, 6-aminohexanoic acid and benzamidine, but not the overall openness of plasminogen regulate, production of biologically active angiostatins. The Biochemical journal 20051215
Ankyrin-B coordinates the Na/K ATPase, Na/Ca exchanger, and InsP3 receptor in a cardiac T-tubule/SR microdomain. PLoS biology 20051201
Tryptase increases proliferative activity of human conjunctival fibroblasts through protease-activated receptor-2. Investigative ophthalmology & visual science 20051201
Investigation of early protein changes in the urinary bladder following partial bladder outlet obstruction by proteomic approach. Journal of Korean medical science 20051201
A capillary electrophoresis method for the characterization of ecto-nucleoside triphosphate diphosphohydrolases (NTPDases) and the analysis of inhibitors by in-capillary enzymatic microreaction. Purinergic signalling 20051201
Thrombomodulin-independent activation of protein C and specificity of hemostatically active snake venom serine proteinases: crystal structures of native and inhibited Agkistrodon contortrix contortrix protein C activator. The Journal of biological chemistry 20051125
Out-of-shape DNA minor groove binders: induced fit interactions of heterocyclic dications with the DNA minor groove. Biochemistry 20051115
Hepatic, extrahepatic, microsomal, and mitochondrial activation of the N-hydroxylated prodrugs benzamidoxime, guanoxabenz, and Ro 48-3656 ([[1-[(2s)-2-[[4-[(hydroxyamino)iminomethyl]benzoyl]amino]-1-oxopropyl]-4-piperidinyl]oxy]-acetic acid). Drug metabolism and disposition: the biological fate of chemicals 20051101
Thermodynamic evaluation and modeling of proton and water exchange associated with benzamidine and berenil binding to beta-trypsin. Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas 20051101
Perspectives of digestive pest control with proteinase inhibitors that mainly affect the trypsin-like activity of Anticarsia gemmatalis Hübner (Lepidoptera: Noctuidae). Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas 20051101
Proteolytic, edematogenic and myotoxic activities of a hemorrhagic metalloproteinase isolated from Bothrops alternatus venom. Toxicon : official journal of the International Society on Toxinology 20051001
Mutation of surface residues to promote crystallization of activated factor XI as a complex with benzamidine: an essential step for the iterative structure-based design of factor XI inhibitors. Acta crystallographica. Section D, Biological crystallography 20051001
Cloning and characterization of the ecto-nucleotidase NTPDase3 from rat brain: Predicted secondary structure and relation to other members of the E-NTPDase family and actin. Purinergic signalling 20050901
Development of a Mammalian suspension culture for expression of active recombinant human urokinase-type plasminogen activator. Cytotechnology 20050901
Release of IL-1beta via IL-1beta-converting enzyme in a skin dendritic cell line exposed to 2,4-dinitrofluorobenzene. Mediators of inflammation 20050814
Biochemical and molecular modeling analysis of the ability of two p-aminobenzamidine-based sorbents to selectively purify serine proteases (fibrinogenases) from snake venoms. Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20050805
Hydrolysis of myelin basic protein by IgM and IgA antibodies from the sera of patients with multiple sclerosis. Medical science monitor : international medical journal of experimental and clinical research 20050801
Purification and characterization of a serine protease (CPM-2) with fibrinolytic activity from the dung beetles. Archives of pharmacal research 20050701
Immobilization of an anticoagulant benzamidine derivative: effect of spacer arms and carrier hydrophobicity on thrombin binding. Acta biomaterialia 20050701
Structure-based design and synthesis of pyrazinones containing novel P1 'side pocket' moieties as inhibitors of TF/VIIa. Bioorganic & medicinal chemistry letters 20050615
A novel type of myofibril-bound serine protease from white croaker (Argyrosomus argentatus). Comparative biochemistry and physiology. Part B, Biochemistry & molecular biology 20050601
Protein/ligand binding free energies calculated with quantum mechanics/molecular mechanics. The journal of physical chemistry. B 20050526
Altered expression of topoisomerase IIalpha contributes to cross-resistant to etoposide K562/MX2 cell line by aberrant methylation. British journal of cancer 20050425
Structure based design of 4-(3-aminomethylphenyl)piperidinyl-1-amides: novel, potent, selective, and orally bioavailable inhibitors of betaII tryptase. Bioorganic & medicinal chemistry 20050415
Trypsin crystallization by membrane-based techniques. Journal of structural biology 20050401
Purification and characterization of a hemorrhagic metalloproteinase from Bothrops lanceolatus (Fer-de-lance) snake venom. Toxicon : official journal of the International Society on Toxinology 20050315
Duvernoy's gland secretion of Philodryas patagoniensis from the northeast of Argentina: its effects on blood coagulation. Toxicon : official journal of the International Society on Toxinology 20050315
Flexible docking in solution using metadynamics. Journal of the American Chemical Society 20050302
Partial purification and characterization of digestive trypsin-like proteases from the velvet bean caterpillar, Anticarsia gemmatalis. Comparative biochemistry and physiology. Part B, Biochemistry & molecular biology 20050301
Increasing the intracellular availability of all-trans retinoic acid in neuroblastoma cells. British journal of cancer 20050227
Synthesis and biological activity of novel 1,2-disubstituted benzene derivatives as factor Xa inhibitors. Bioorganic & medicinal chemistry 20050215
Receptor rigidity and ligand mobility in trypsin-ligand complexes. Proteins 20050201
Isolation and characterization of trypsin from pyloric caeca of Monterey sardine Sardinops sagax caerulea. Comparative biochemistry and physiology. Part B, Biochemistry & molecular biology 20050101
A critical role for Gly25 in the B chain of human thrombin. Journal of thrombosis and haemostasis : JTH 20050101
The p53-dependent apoptotic pathway of breast cancer cells (BC-M1) induced by the bis-type bioreductive compound aziridinylnaphthoquinone. Breast cancer research : BCR 20050101
Cyclic nucleotide binding proteins in the Arabidopsis thaliana and Oryza sativa genomes. BMC bioinformatics 20050101
Induction of chondro-, osteo- and adipogenesis in embryonic stem cells by bone morphogenetic protein-2: effect of cofactors on differentiating lineages. BMC developmental biology 20050101
Signalling crosstalk in FGF2-mediated protection of endothelial cells from HIV-gp120. BMC neuroscience 20050101
A2B adenosine receptor activity is reduced in neutrophils from patients with systemic sclerosis. Arthritis research & therapy 20050101
Chronic ethanol exposure increases microtubule content in PC12 cells. BMC neuroscience 20050101
Metabolism of benzamidoxime (N-hydroxyamidine) in human hepatocytes and role of UDP-glucuronosyltransferases. Xenobiotica; the fate of foreign compounds in biological systems 20050101
Airway epithelial cell tolerance to Pseudomonas aeruginosa. Respiratory research 20050101
Alterations of prolyl endopeptidase activity in the plasma of children with autistic spectrum disorders. BMC psychiatry 20050101
Computer simulation of protein-ligand interactions: challenges and applications. Methods in molecular biology (Clifton, N.J.) 20050101
Beta-adrenergic receptor activation in immortalized human urothelial cells stimulates inflammatory responses by PKA-independent mechanisms. Cell communication and signaling : CCS 20050101
Protective action of a hexane crude extract of Pterodon emarginatus fruits against oxidative and nitrosative stress induced by acute exercise in rats. BMC complementary and alternative medicine 20050101
Easy detection of chromatin binding proteins by the Histone Association Assay. Biological procedures online 20050101
The use of cystatin C to inhibit epithelial-mesenchymal transition and morphological transformation stimulated by transforming growth factor-beta. Breast cancer research : BCR 20050101
5-aminoimidazole-4-carboxamide-1-beta-4-ribofuranoside (AICAR) attenuates the expression of LPS- and Abeta peptide-induced inflammatory mediators in astroglia. Journal of neuroinflammation 20050101
Purification and kinetic studies of recombinant gibberellin dioxygenases. BMC plant biology 20050101
Distinct effects of glucose and glucosamine on vascular endothelial and smooth muscle cells: evidence for a protective role for glucosamine in atherosclerosis. Cardiovascular diabetology 20050101
Respiratory epithelial cells require Toll-like receptor 4 for induction of human beta-defensin 2 by lipopolysaccharide. Respiratory research 20050101
Exotic diseases of dogs and cats at risk of importation to Ireland. Irish veterinary journal 20050101
Determination of ligand-protein dissociation constants by electrospray mass spectrometry-based diffusion measurements. Analytical chemistry 20041201
A novel serine protease complexed with alpha2-macroglobulin from skeletal muscle of lizard fish (Saurida undosquamis). Comparative biochemistry and physiology. Part B, Biochemistry & molecular biology 20041201
Purification and characterization of jararassin-I, A thrombin-like enzyme from Bothrops jararaca snake venom. Acta biochimica et biophysica Sinica 20041201
Kinetic analysis of zymogen autoactivation in the presence of a reversible inhibitor. European journal of biochemistry 20041201
Design, synthesis, and evaluation of oxyanion-hole selective inhibitor substituents for the S1 subsite of factor Xa. Bioorganic & medicinal chemistry letters 20041018
No topoisomerase I alteration in a neuroblastoma model with in vivo acquired resistance to irinotecan. British journal of cancer 20040913
On the modeling of snake venom serine proteinase interactions with benzamidine-based thrombin inhibitors. Protein science : a publication of the Protein Society 20040901
Novel non-covalent azaphenylalanine thrombin inhibitors with an aminomethyl or amino group at the P1 position. Die Pharmazie 20040901
Phenyl substitution of furamidine markedly potentiates its anti-parasitic activity against Trypanosoma cruzi and Leishmania amazonensis. Biochemical pharmacology 20040815
In vitro blood compatibility of polymeric biomaterials through covalent immobilization of an amidine derivative. Biomaterials 20040801
The telomeric protein TRF2 binds the ATM kinase and can inhibit the ATM-dependent DNA damage response. PLoS biology 20040801
Sample displacement chromatography of Atlantic Salmon (Salmo salar) thrombin. Journal of biochemical and biophysical methods 20040730
Proteolytic conversion of STAT3alpha to STAT3gamma in human neutrophils: role of granule-derived serine proteases. The Journal of biological chemistry 20040723
Benzamides and benzamidines as specific inhibitors of epidermal growth factor receptor and v-Src protein tyrosine kinases. Bioorganic & medicinal chemistry 20040701
Crystal structures of QacR-diamidine complexes reveal additional multidrug-binding modes and a novel mechanism of drug charge neutralization. The Journal of biological chemistry 20040402
Regulation of glomerular endothelial cell proteoglycans by glucose. Journal of Korean medical science 20040401
Thrombin inhibitors built on an azaphenylalanine scaffold. Bioorganic & medicinal chemistry letters 20040322
Collagen degradation by host-derived enzymes during aging. Journal of dental research 20040301
Site-directed mutagenesis at the human B2 receptor and molecular modelling to define the pharmacophore of non-peptide bradykinin receptor antagonists. Biochemical pharmacology 20040215
Thrombin generation: phenotypic quantitation. Journal of thrombosis and haemostasis : JTH 20040201
Ala226 to Gly and Ser189 to Asp mutations convert rat chymotrypsin B to a trypsin-like protease. Protein engineering, design & selection : PEDS 20040201
Understanding protein-ligand interactions: the price of protein flexibility. Journal of molecular biology 20040130
Protein interaction networks by proteome peptide scanning. PLoS biology 20040101
IL-17 induces production of IL-6 and IL-8 in rheumatoid arthritis synovial fibroblasts via NF-kappaB- and PI3-kinase/Akt-dependent pathways. Arthritis research & therapy 20040101
Arterial heparan sulfate is negatively associated with hyperglycemia and atherosclerosis in diabetic monkeys. Cardiovascular diabetology 20040101
Resistance to gemcitabine in a human follicular lymphoma cell line is due to partial deletion of the deoxycytidine kinase gene. BMC pharmacology 20040101
The role of cyclin D2 and p21/waf1 in human T-cell leukemia virus type 1 infected cells. Retrovirology 20040101
Xenopus Cdc14 alpha/beta are localized to the nucleolus and centrosome and are required for embryonic cell division. BMC cell biology 20040101
The p68 and p72 DEAD box RNA helicases interact with HDAC1 and repress transcription in a promoter-specific manner. BMC molecular biology 20040101
Flagellin acting via TLR5 is the major activator of key signaling pathways leading to NF-kappa B and proinflammatory gene program activation in intestinal epithelial cells. BMC microbiology 20040101
Combined analysis of expression data and transcription factor binding sites in the yeast genome. BMC genomics 20040101
Glycogen synthase kinase-3 regulates IGFBP-1 gene transcription through the thymine-rich insulin response element. BMC molecular biology 20040101
Hydrolysis of myelin basic protein by polyclonal catalytic IgGs from the sera of patients with multiple sclerosis. Journal of cellular and molecular medicine 20040101
Traceless solid-phase synthesis of nitrogen-containing heterocycles and their biological evaluations as inhibitors of neuronal sodium channels. Journal of combinatorial chemistry 20040101
Leptin and insulin stimulation of signalling pathways in arcuate nucleus neurones: PI3K dependent actin reorganization and KATP channel activation. BMC neuroscience 20040101
A serine protease from a detergent-soluble extract of Leishmania (Leishmania) amazonensis. Zeitschrift fur Naturforschung. C, Journal of biosciences 20040101
[Isolation and characteristics of the protein C activator from Agkistrodon halys halys snake venom]. Ukrains'kyi biokhimichnyi zhurnal (1999 ) 20040101
Characterization of a trypsin-like serine protease of activated B cells mediating the cleavage of surface proteins. Biochimica et biophysica acta 20031205
Multinuclear magnetic resonance and theoretical calculations in the study of structure and tautomerism of some 2-amino-N'-(aryl)-benzamidines. Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20031101
[Preparation of high-purity and safe autologous plasmin and its clinical application]. Nippon Ganka Gakkai zasshi 20031101
Structure-based design of novel guanidine/benzamidine mimics: potent and orally bioavailable factor Xa inhibitors as novel anticoagulants. Journal of medicinal chemistry 20031009
CD26/dipeptidyl peptidase IV enhances expression of topoisomerase II alpha and sensitivity to apoptosis induced by topoisomerase II inhibitors. British journal of cancer 20031006
Molecular cloning of trypsin-like cDNAs and comparison of proteinase activities in the salivary glands and gut of the tarnished plant bug Lygus lineolaris (Heteroptera: Miridae). Insect biochemistry and molecular biology 20030901
Lactate dehydrogenase-5 (LDH-5) overexpression in non-small-cell lung cancer tissues is linked to tumour hypoxia, angiogenic factor production and poor prognosis. British journal of cancer 20030901
Modulation of enzymatic activity of human mast cell tryptase and chymase by protease inhibitors. Acta pharmacologica Sinica 20030901
Efficacious and orally bioavailable thrombin inhibitors based on a 2,5-thienylamidine at the P1 position: discovery of N-carboxymethyl-d-diphenylalanyl-l-prolyl[(5-amidino-2-thienyl)methyl]amide. Journal of medicinal chemistry 20030814
Novel oxidative alpha-tosyloxylation of alcohols with iodosylbenzene and p-toluenesulfonic acid and its synthetic use for direct preparation of heteroaromatics. The Journal of organic chemistry 20030808
Design and synthesis of highly constrained factor Xa inhibitors: amidine-substituted bis(benzoyl)--diazepan-2-ones and bis(benzylidene)-bis(gem-dimethyl)cycloketones. Bioorganic & medicinal chemistry 20030805
Engineering the primary substrate specificity of Streptomyces griseus trypsin. Biochemistry 20030805
Zoledronic acid induces antiproliferative and apoptotic effects in human pancreatic cancer cells in vitro. British journal of cancer 20030616
Characterisation of integrin-linked kinase signalling in sporadic human colon cancer. British journal of cancer 20030602
Inhibition of purified factor Xa amidolytic activity may not be predictive of inhibition of in vivo thrombosis: implications for identification of therapeutically active inhibitors. Arteriosclerosis, thrombosis, and vascular biology 20030601
Discovery of 3-amino-4-chlorophenyl P1 as a novel and potent benzamidine mimic via solid-phase synthesis of an isoxazoline library. Bioorganic & medicinal chemistry letters 20030519
Rational design, synthesis, and structure-activity relationships of novel factor Xa inhibitors: (2-substituted-4-amidinophenyl)pyruvic and -propionic acids. Journal of medicinal chemistry 20030508
A role for BRCA1 in sporadic breast cancer. British journal of cancer 20030422
Identification and partial characterization of two inducible gelatin-cleavage activities localized to the sea urchin extraembryonic matrix, the hyaline layer. Biochimica et biophysica acta 20030407
Purification, properties and substrate specificity of a digestive trypsin from Periplaneta americana (Dictyoptera) adults. Insect biochemistry and molecular biology 20030401
Nonbenzamidine isoxazoline derivatives as factor Xa inhibitors. Bioorganic & medicinal chemistry letters 20030324
Molecular structures of human factor Xa complexed with ketopiperazine inhibitors: preference for a neutral group in the S1 pocket. Journal of medicinal chemistry 20030227
Nonbenzamidine tetrazole derivatives as factor Xa inhibitors. Bioorganic & medicinal chemistry letters 20030210
Effect of CD26/dipeptidyl peptidase IV on Jurkat sensitivity to G2/M arrest induced by topoisomerase II inhibitors. British journal of cancer 20030210
A novel influenza A virus activating enzyme from porcine lung: purification and characterization. Biological chemistry 20030201
Structure and activity of human pancreasin, a novel tryptic serine peptidase expressed primarily by the pancreas. The Journal of biological chemistry 20030131
Reconstructing the binding site of factor Xa in trypsin reveals ligand-induced structural plasticity. Journal of molecular biology 20030131
Purification and partial characterization of feline classical pancreatic lipase. Comparative biochemistry and physiology. Part B, Biochemistry & molecular biology 20030101
Disruption of vitellogenin gene function in adult honeybees by intra-abdominal injection of double-stranded RNA. BMC biotechnology 20030101
Steroid-induced polycystic ovaries in rats: effect of electro-acupuncture on concentrations of endothelin-1 and nerve growth factor (NGF), and expression of NGF mRNA in the ovaries, the adrenal glands, and the central nervous system. Reproductive biology and endocrinology : RB&E 20030101
Complexes between the LKB1 tumor suppressor, STRAD alpha/beta and MO25 alpha/beta are upstream kinases in the AMP-activated protein kinase cascade. Journal of biology 20030101
Inhibitors of benzamidine type influence the virulence properties of Porphyromonas gingivalis strains. Acta biochimica Polonica 20030101
Type III secretion proteins PcrV and PcrG from Pseudomonas aeruginosa form a 1:1 complex through high affinity interactions. BMC microbiology 20030101
Synthesis of L-ascorbic acid in the phloem. BMC plant biology 20030101
Cloning and characterization of a transmembrane-type serine protease from rat kidney, a new sodium channel activator. Biological chemistry 20030101
Purification and characterization of a serine protease with fibrinolytic activity from the dung beetles, Catharsius molossus. Thrombosis research 20030101
[Isolation and properties of the protein C activator from Agkistrodon halys halys venom]. Biomeditsinskaia khimiia 20030101
Pattern recognition and massively distributed computing. Journal of computational chemistry 20021201
Thrombin inhibition by novel benzamidine derivatives: a free-energy perturbation study. Journal of medicinal chemistry 20021107
Identification, characterization, and cloning of an immunoglobulin degrading enzyme in the cat flea, Ctenocephalides felis. Archives of insect biochemistry and physiology 20021101
Mutant K-ras oncogene regulates steroidogenesis of normal human adrenocortical cells by the RAF-MEK-MAPK pathway. British journal of cancer 20021021
Evaluation of 2-deoxy-D-glucose as a chemotherapeutic agent: mechanism of cell death. British journal of cancer 20020923
Crystal structures of uninhibited factor VIIa link its cofactor and substrate-assisted activation to specific interactions. Journal of molecular biology 20020920
Purification, characterization and crystallization of Jararacussin-I, a fibrinogen-clotting enzyme isolated from the venom of Bothrops jararacussu. Toxicon : official journal of the International Society on Toxinology 20020901
Substituted acrylamides as factor Xa inhibitors: improving bioavailability by P1 modification. Bioorganic & medicinal chemistry letters 20020805
High-gradient magnetic affinity separation of trypsin from porcine pancreatin. Biotechnology and bioengineering 20020805
Identification of prolylcarboxypeptidase as the cell matrix-associated prekallikrein activator. FEBS letters 20020717
Crystallization and preliminary X-ray crystallographic studies of monoacylglycerol lipase of the moderately thermophilic Bacillus sp. H-257. Acta crystallographica. Section D, Biological crystallography 20020701
Simultaneous analysis of monosaccharides and oligosaccharides by high-performance liquid chromatography with postcolumn fluorescence derivatization. Journal of chromatography. A 20020628
The first synthetic receptor for the RGD sequence. Organic letters 20020627
Design, synthesis and biological activity of novel non-amidine factor Xa inhibitors. Part 1: P(1) structure-activity relationships of the substituted 1-(2-Naphthyl)-1H-pyrazole-5-carboxylamides. Bioorganic & medicinal chemistry letters 20020617
Simple, intuitive calculations of free energy of binding for protein-ligand complexes. 1. Models without explicit constrained water. Journal of medicinal chemistry 20020606
[Single-chain urokinase-type plasminogen activator (scu-PA) purification by immuno-affinity chromatography]. Sheng wu gong cheng xue bao = Chinese journal of biotechnology 20020501
Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells. The Journal of biological chemistry 20020419
Noncovalent tripeptidic thrombin inhibitors incorporating amidrazone, amine and amidine functions at P1. Bioorganic & medicinal chemistry letters 20020408
Linear mixed irreversible inhibition of the autocatalytic activation of zymogens. Kinetic analysis checked by simulated progress curves. The international journal of biochemistry & cell biology 20020401
PRO_SELECT: combining structure-based drug design and array-based chemistry for rapid lead discovery. 2. The development of a series of highly potent and selective factor Xa inhibitors. Journal of medicinal chemistry 20020314
Purification and characterization of a prothrombin-activating protease from Nephila clavata. Toxicon : official journal of the International Society on Toxinology 20020301
Evaluation of the proacrosin/acrosin system and its mechanism of activation in human sperm extracts. Journal of reproductive immunology 20020301
Crystal structure reveals basis for the inhibitor resistance of human brain trypsin. Journal of molecular biology 20020201
DPC-423 Bristol-Myers Squibb. Current opinion in investigational drugs (London, England : 2000) 20020201
Catalytic domain structures of MT-SP1/matriptase, a matrix-degrading transmembrane serine proteinase. The Journal of biological chemistry 20020118
Development and validation of a capillary electrophoresis method for ximelagatran assay and related substance determination in drug substance and tablets. Journal of pharmaceutical and biomedical analysis 20020115
An oxyanion-hole selective serine protease inhibitor in complex with trypsin. Bioorganic & medicinal chemistry 20020101
Amidolytic activity of prostatic acid phosphatase on human semenogelins and semenogelin-derived synthetic substrates. European journal of biochemistry 20020101
Design and synthesis of a series of indole glycoprotein IIb/IIIa inhibitors. European journal of medicinal chemistry 20020101
Expression of interleukin-18 receptor in fibroblast-like synoviocytes. Arthritis research 20020101
Ca2+-mediated activation of ERK in hepatocytes by norepinephrine and prostaglandin F2 alpha: role of calmodulin and Src kinases. BMC cell biology 20020101
Ecdysteroids and oocyte development in the black fly Simulium vittatum. BMC developmental biology 20020101
The regulation of protein synthesis and translation factors by CD3 and CD28 in human primary T lymphocytes. BMC biochemistry 20020101
Probing the importance and potential roles of the binding of the PH-domain protein Boi1 to acidic phospholipids. BMC cell biology 20020101
Interaction of neuronal nitric oxide synthase with alpha1-adrenergic receptor subtypes in transfected HEK-293 cells. BMC pharmacology 20020101
The PEST sequence does not contribute to the stability of the cystic fibrosis transmembrane conductance regulator. BMC biochemistry 20020101
Aggregation and retention of human urokinase type plasminogen activator in the yeast endoplasmic reticulum. BMC molecular biology 20020101
Inhibition of arginine gingipains (RgpB and HRgpA) with benzamidine inhibitors: zinc increases inhibitory potency. Biological chemistry 20020101
The effect of Puerariae radix on lipoprotein metabolism in liver and intestinal cells. BMC complementary and alternative medicine 20020101
[Purification and characterization of the fibrinolytic enzyme from Agkistrodon halys halys venom]. Ukrains'kyi biokhimichnyi zhurnal (1999 ) 20020101
Triacylglycerol-rich lipophorins are found in the dipteran infraorder Culicomorpha, not just in mosquitoes. Journal of insect science (Online) 20020101
Acrosin activity in turkey spermatozoa: assay by clinical method and effect of zinc and benzamidine on the activity. Theriogenology 20010915
Monocharged inhibitors of mast cell tryptase derived from potent and selective dibasic inhibitors. Bioorganic & medicinal chemistry letters 20010903
Tryptase and agonists of PAR-2 induce the proliferation of human airway smooth muscle cells. Journal of applied physiology (Bethesda, Md. : 1985) 20010901
Synthesis and pharmacology of modified amidine isoxazoline glycoprotein IIb/IIIa receptor antagonists. Bioorganic & medicinal chemistry letters 20010820
Selected contribution: tryptase-induced PAR-2-mediated Ca(2+) signaling in human airway smooth muscle cells. Journal of applied physiology (Bethesda, Md. : 1985) 20010801
Role of mast cell tryptase in renal interstitial fibrosis. Journal of the American Society of Nephrology : JASN 20010801
Aromatic polyamidines inhibiting the Tat-induced HIV-1 transcription recognize structured TAR-RNA. Antisense & nucleic acid drug development 20010801
Dibasic inhibitors of human mast cell tryptase. Part 3: identification of a series of potent and selective inhibitors containing the benzamidine functionality. Bioorganic & medicinal chemistry letters 20010709
Electrostatic effects play a central role in cold adaptation of trypsin. FEBS letters 20010615
Proteolytic action of Bothrops jararaca venom upon its own constituents. Toxicon : official journal of the International Society on Toxinology 20010601
Discovery of the factor Xa inhibitor, ZK 807834 (CI-1031). Current topics in medicinal chemistry 20010601
The design and synthesis of noncovalent factor Xa inhibitors. Current topics in medicinal chemistry 20010601
The design of competitive, small-molecule inhibitors of coagulation factor Xa. Current topics in medicinal chemistry 20010601
Purification and characterization of a plasmin-like protease from Tenodera sinensis (Chinese mantis). Insect biochemistry and molecular biology 20010427
2-Acylimino-3H-thiazoline derivatives: a novel template for platelet GPIIb/IIIa receptor antagonists. Bioorganic & medicinal chemistry letters 20010423
Synthesis and SAR of benzamidine factor Xa inhibitors containing a vicinally-substituted heterocyclic core. Bioorganic & medicinal chemistry letters 20010312
Phase 2 metabolites of N-hydroxylated amidines (amidoximes): synthesis, in vitro formation by pig hepatocytes, and mutagenicity testing. Chemical research in toxicology 20010301
Discovery of 1-[3-(aminomethyl)phenyl]-N-3-fluoro-2'-(methylsulfonyl)-[1,1'-biphenyl]-4-yl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide (DPC423), a highly potent, selective, and orally bioavailable inhibitor of blood coagulation factor Xa. Journal of medicinal chemistry 20010215
X-ray crystallographic analyses of complexes between bovine beta-trypsin and Schiff base copper(II) or iron(III) chelates. Journal of molecular biology 20010119
Linear competitive inhibition of human tissue kallikrein by 4-aminobenzamidine and benzamidine and linear mixed inhibition by 4-nitroaniline and aniline. Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas 20010101
Evidence for the involvement of Gi2 in activation of extracellular signal-regulated kinases in hepatocytes. BMC cell biology 20010101
Processing of the insulin-like growth factor-II-mannose 6-phosphate receptor in isolated liver subcellular fractions. Biochemistry and cell biology = Biochimie et biologie cellulaire 20010101
Chum salmon trypsin-catalyzed preferential formation of peptides containing D-amino acid. Amino acids 20010101
Pentamidine is a potent inhibitor of [3H]idazoxan binding to imidazoline I2 receptors. Annals of the New York Academy of Sciences 19990621
Structural and functional analyses of benzamidine-based inhibitors in complex with trypsin: implications for the inhibition of factor Xa, tPA, and urokinase. Journal of medicinal chemistry 19981231
1,5-Bis(4-amidinophenoxy)pentane (pentamidine) is a potent inhibitor of [3H]idazoxan binding to imidazoline I2 binding sites. European journal of pharmacology 19980717
Identification and characterization of an endo/exonuclease in Pneumocystis carinii that is inhibited by dicationic diarylfurans with efficacy against Pneumocystis pneumonia. The Journal of eukaryotic microbiology 19980101
Characterization of an insulin-like growth factor binding protein-5 protease produced by rat articular chondrocytes and a neuroblastoma cell line. Growth regulation 19960901
A trypsin-like serine protease activity on activated human B cells and various B cell lines. European journal of immunology 19921001
Chymotrypsinogen: an activating enzyme in the mitochondrial membrane of rat submaxillary gland. Biochemistry international 19911201
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