The antioxidant behaviour of melatonin and structural analogues during lipid peroxidation depends not only on their functional groups but also on the assay system.

Biochemical and biophysical research communications 20120713

Total synthesis of Akuammiline alkaloid (-)-vincorine via intramolecular oxidative coupling.

Journal of the American Chemical Society 20120606

Prospective acetylcholinesterase inhibitory activity of indole and its analogs.

Bioorganic & medicinal chemistry letters 20120415

Inotropic effects of prokinetic agents with 5-HT(4) receptor agonist actions on human isolated myocardial trabeculae.

Life sciences 20120409

5-HT receptors as novel targets for optimizing pigmentary responses in dorsal skin melanophores of frog, Hoplobatrachus tigerinus.

British journal of pharmacology 20120301

Developmental exposure to a serotonin agonist produces subsequent behavioral and neurochemical changes in the adult male prairie vole.

Physiology & behavior 20120118

Principles of psychoneuroendocrinoimmunotherapy of cancer.

Immunotherapy 20120101

Effects of power frequency electromagnetic fields on melatonin and sleep in the rat.

Emerging health threats journal 20120101

A reinterpretation of the pathogenesis and cure of cancer according to the psychoneuroimmunological discoveries.

Methods in molecular biology (Clifton, N.J.) 20120101

Inhibition of itch-related responses at spinal level in rats.

Acta physiologica Hungarica 20111201

A quantitative method for simultaneous determination of 5-methoxy-N,N-diisopropyltryptamine and its metabolites in urine using liquid chromatography-electrospray ionization-tandem mass spectrometry.

Journal of forensic sciences 20110701

Measurement of melatonin in body fluids: standards, protocols and procedures.

Child's nervous system : ChNS : official journal of the International Society for Pediatric Neurosurgery 20110601

5-methoxy-N,N-di(iso)propyltryptamine hydrochloride (Foxy)-induced cognitive deficits in rat after exposure in adolescence.

Physiology & behavior 20110503

Preliminary analgesic properties of deltorphin-5-methoxytryptamine chimeric opioid peptides.

Peptides 20110501

Melatonin as an antioxidant and its semi-lunar rhythm in green macroalga Ulva sp.

Journal of experimental botany 20110301

Drug-induced psychosis: how to avoid star gazing in schizophrenia research by looking at more obvious sources of light.

Frontiers in behavioral neuroscience 20110101

The impact of serotonergic stimulation on reelin and glutamate decarboxylase gene expression in adult female rats.

Bratislavske lekarske listy 20110101

[Radioprotective properties of indralin combined with cystamine and mexamine].

Radiatsionnaia biologiia, radioecologiia 20110101

Evaluation of nootropic and neuroprotective effects of low dose aspirin in rats.

Journal of pharmacology & pharmacotherapeutics 20110101

Current state of type 1 diabetes immunotherapy: incremental advances, huge leaps, or more of the same?

Clinical & developmental immunology 20110101

Subjective food hypersensitivity: assessment of enterochromaffin cell markers in blood and gut lavage fluid.

International journal of general medicine 20110101

Serotonin-induced contraction in isolated intestine from a teleost fish (Carassius auratus): characterization and interactions with melatonin.

Neurogastroenterology and motility : the official journal of the European Gastrointestinal Motility Society 20101201

5-benzyloxytryptamine as an antagonist of TRPM8.

Bioorganic & medicinal chemistry letters 20101201

Synthesis and SAR studies of 1,4-benzoxazine MenB inhibitors: novel antibacterial agents against Mycobacterium tuberculosis.

Bioorganic & medicinal chemistry letters 20101101

Melatonin metabolism in the central nervous system.

Current neuropharmacology 20100901

Development and validation of a high throughput direct radioimmunoassay for the quantitative determination of serum and plasma melatonin (N-acetyl-5-methoxytryptamine) in mice.

Journal of immunological methods 20100630

Tandem intramolecular photocycloaddition-retro-Mannich fragmentation as a route to spiro[pyrrolidine-3,3'-oxindoles]. Total synthesis of (+/-)-coerulescine, (+/-)-horsfiline, (+/-)-elacomine, and (+/-)-6-deoxyelacomine.

The Journal of organic chemistry 20100604

Brain chemistry: how does P450 catalyze the O-demethylation reaction of 5-methoxytryptamine to yield serotonin?

The journal of physical chemistry. B 20100527

Biogenic amines modulate pulse rate in the dorsal blood vessel of Lumbriculus variegatus.

Comparative biochemistry and physiology. Toxicology & pharmacology : CBP 20100501

MT1 melatonin receptors mediate somatic, behavioral, and reproductive neuroendocrine responses to photoperiod and melatonin in Siberian hamsters (Phodopus sungorus).

Endocrinology 20100201

Glucose and corticosterone changes in developing and adult rats following exposure to (+/-)-3,4-methylendioxymethamphetamine or 5-methoxydiisopropyltryptamine.

Neurotoxicology and teratology 20100101

Cytosine methylation dysregulation in neonates following intrauterine growth restriction.

PloS one 20100101

Melatonin and structurally-related compounds protect synaptosomal membranes from free radical damage.

International journal of molecular sciences 20100101

Synthesis and preliminary screening of novel tryptamines as 5-HT4 receptor ligands.

Current medicinal chemistry 20100101

Circulating Antibodies to IDO/THO Pathway Metabolites in Alzheimer's Disease.

International journal of Alzheimer's disease 20100101

Human and mouse trace amine-associated receptor 1 have distinct pharmacology towards endogenous monoamines and imidazoline receptor ligands.

The Biochemical journal 20091023

N-[(Dihydroxyphenyl)acyl]serotonins as potent inhibitors of tyrosinase from mouse and human melanoma cells.

Bioorganic & medicinal chemistry letters 20090801

Synthesis and preliminary screening of novel indole-3-methanamines as 5-HT4 receptor ligands.

European journal of medicinal chemistry 20090701

The serotonergic system: its role in pathogenesis and early developmental treatment of autism.

Current neuropharmacology 20090601

The conformational landscape of 5-methoxytryptamine studied by rotationally resolved fluorescence spectroscopy and resonant ionization spectroscopy.

Physical chemistry chemical physics : PCCP 20090414

Effects of naphthalene, beta-naphthoflavone and benzo(a)pyrene on the diurnal and nocturnal indoleamine metabolism and melatonin content in the pineal organ of rainbow trout, Oncorhynchus mykiss.

Aquatic toxicology (Amsterdam, Netherlands) 20090402

New approaches in the management of insomnia: weighing the advantages of prolonged-release melatonin and synthetic melatoninergic agonists.

Neuropsychiatric disease and treatment 20090101

The use of tripeptides for lead discovery of 5-HT4 receptor ligands.

Protein and peptide letters 20090101

Melatonin, hormone of darkness and more: occurrence, control mechanisms, actions and bioactive metabolites.

Cellular and molecular life sciences : CMLS 20080701

Contribution of active and inactive states of the human 5-HT4d receptor to the functional activities of 5-HT4-receptor agonists.

Journal of pharmacological sciences 20080701

Intraocular microinjections repair experimental Parkinson's disease.

Brain research 20080627

Indolealkylamines: biotransformations and potential drug-drug interactions.

The AAPS journal 20080601

Functional human 5-HT6 receptor assay for high throughput screening of chemical ligands and binding proteins.

Combinatorial chemistry & high throughput screening 20080501

Direct determination of serotonin in gut lavage fluid by liquid chromatographic ion trap tandem mass spectrometry.

Talanta 20080415

The roles of amino acid residues at positions 216 and 219 in the structural stability and metabolic functions of rat cytochrome P450 2D1 and 2D2.

Chemico-biological interactions 20080310

Solubilization of 5-methoxy tryptamine molecular probes in CTAB and SDS micelles: a cmc and binding constant study.

Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20080301

5-Fluorotryptamine is a partial agonist at 5-HT3 receptors, and reveals that size and electronegativity at the 5 position of tryptamine are critical for efficient receptor function.

European journal of pharmacology 20080212

Oxidation of 5-methoxy-N,N-diisopropyltryptamine in rat liver microsomes and recombinant cytochrome P450 enzymes.

Biochemical pharmacology 20080201

Problems in three Japanese drug users with Human Immunodeficiency Virus infection.

The journal of medical investigation : JMI 20080201

Further studies in the developmental hyperserotonemia model (DHS) of autism: social, behavioral and peptide changes.

Brain research 20080116

Perinatal exposure to 5-methoxytryptamine, behavioural-stress reactivity and functional response of 5-HT1A receptors in the adolescent rat.

Behavioural brain research 20080110

Neuropsychotoxicity of abused drugs: molecular and neural mechanisms of neuropsychotoxicity induced by methamphetamine, 3,4-methylenedioxymethamphetamine (ecstasy), and 5-methoxy-N,N-diisopropyltryptamine (foxy).

Journal of pharmacological sciences 20080101

Evaluation of the effects of a new drug candidate (GEMSP) in a chronic EAE model.

International journal of biological sciences 20080101

[Protective action of radioprotectors and shielding against high-energy protons in experiments with rats].

Aviakosmicheskaia i ekologicheskaia meditsina = Aerospace and environmental medicine 20080101

Antioxidant systems and oxidative stress in the testes.

Oxidative medicine and cellular longevity 20080101

Effect of CTAB and SDS micelles on the excited state equilibria of some indole probes.

Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20071101

Effects of pre- and postnatal exposure to 5-methoxytryptamine and early handling on an object-place association learning task in adolescent rat offspring.

Neuroscience research 20070901

Pharmacology of serotonin-induced salivary secretion in Periplaneta americana.

Journal of insect physiology 20070801

The effect of melatonin and structural analogues on the lipid peroxidation of triglycerides enriched in omega-3 polyunsaturated fatty acids.

Life sciences 20070704

Alterations in body temperature, corticosterone, and behavior following the administration of 5-methoxy-diisopropyltryptamine ('foxy') to adult rats: a new drug of abuse.

Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20070601

CYP2D6 genotype in relation to perphenazine concentration and pituitary pharmacodynamic tissue sensitivity in Asians: CYP2D6-serotonin-dopamine crosstalk revisited.

Pharmacogenetics and genomics 20070501

5-Methoxy-N,N-diisopropyltryptamine (Foxy), a selective and high affinity inhibitor of serotonin transporter.

Toxicology letters 20070405

Acute confusional state after designer tryptamine abuse.

Psychiatry and clinical neurosciences 20070401

Dimethyl sulfoxide: an antagonist in scintillation proximity assay [(35)S]-GTPgammaS binding to rat 5-HT(6) receptor cloned in HEK-293 cells?

Journal of neuroscience methods 20070315

Nitration of specific tyrosine residues of cytochrome C is associated with caspase-cascade inactivation.

Biological & pharmaceutical bulletin 20070101

Indorenate improves motor function in rats with chronic spinal cord injury.

Basic & clinical pharmacology & toxicology 20070101

Biochemotherapy with immunomodulating pineal hormones other than melatonin: 5-methoxytryptamine as a new oncostatic pineal agent.

Pathologie-biologie 20070101

[Comparative protective action of radiorotectors and shielding in gamma-irradiated mice].

Aviakosmicheskaia i ekologicheskaia meditsina = Aerospace and environmental medicine 20070101

[5-hydroxytryptamine and 5-methoxytryptamine increase tolerance to global cerebral ischemia].

Eksperimental'naia i klinicheskaia farmakologiia 20070101

Cholesterol depletion reduces serotonin binding and signaling via human 5-HT(7(a)) receptors.

European journal of pharmacology 20061215

Could endogenous substrates of drug-metabolizing enzymes influence constitutive physiology and drug target responsiveness?

Pharmacogenomics 20061201

Functional activity of 5-HT4 receptors in children with congenital heart disease.

Bulletin of experimental biology and medicine 20061201

A fatal poisoning with 5-methoxy-N,N-diisopropyltryptamine, Foxy.

Forensic science international 20061110

Tryptamine induces cell death with ultrastructural features of autophagy in neurons and glia: Possible relevance for neurodegenerative disorders.

The anatomical record. Part A, Discoveries in molecular, cellular, and evolutionary biology 20060901

Human trabecular meshwork cells express functional serotonin-2A (5HT2A) receptors: role in IOP reduction.

Investigative ophthalmology & visual science 20060901

Indorenate modifies a1-adrenergic and benzodiazepine receptor binding in the rat brain: an autoradiography study.

The Journal of pharmacy and pharmacology 20060901

Functional roles of 5-hydroxytryptamine 3/4 receptors in neurons of rat dorsal motor nucleus of the vagus.

Neuroscience 20060825

1H- and 13C-NMR, FTIR, UV-VIS, ESI-MS, and PM5 studies as well as emission properties of a new Schiff base of gossypol with 5-methoxytryptamine and a new hydrazone of gossypol with dansylhydrazine.

Biopolymers 20060805

An examination of the effects of 5-Methoxy-n, n-di(ISO)propyltryptamine hydrochloride (Foxy) on cognitive development in rats.

Psychological reports 20060601

Microsphere-based protease assays and screening application for lethal factor and factor Xa.

Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501

Preparation and identification of anti-melatonin monoclonal antibodies.

Journal of pineal research 20060501

Oxidative metabolism of 5-methoxy-N,N-diisopropyltryptamine (Foxy) by human liver microsomes and recombinant cytochrome P450 enzymes.

Biochemical pharmacology 20060428

Pharmacological characterization of 5-hydroxytryptamine-induced contraction in the chicken gastrointestinal tract.

Autonomic & autacoid pharmacology 20060401

Rhabdomyolysis after ingestion of 'foxy,' a hallucinogenic tryptamine derivative.

Mayo Clinic proceedings 20060401

A 3-synapse positive feedback loop regulates the excitability of an interneuron critical for sensitization in the leech.

The Journal of neuroscience : the official journal of the Society for Neuroscience 20060329

Solvent effects in the preparation of molecularly imprinted polymers for melatonin using N-propionyl-5-methoxytryptamine as the pseudo template.

Analytical and bioanalytical chemistry 20060301

On-line preconcentration techniques in determination of melatonin and its precursors/metabolites using micellar electrokinetic chromatography.

Journal of chromatography. A 20060203

Metabolism of the psychotomimetic tryptamine derivative 5-methoxy-N,N-diisopropyltryptamine in humans: identification and quantification of its urinary metabolites.

Drug metabolism and disposition: the biological fate of chemicals 20060201

Simultaneous liquid chromatographic measurement of melatonin and related indoles through post-column electrochemical demethylation and fluorescence derivatization.

Analytical sciences : the international journal of the Japan Society for Analytical Chemistry 20060201

Hallucinogen-like actions of 5-methoxy-N,N-diisopropyltryptamine in mice and rats.

Pharmacology, biochemistry, and behavior 20060101

Functional and molecular identification of 5-hydroxytryptamine receptors in rabbit pulmonary artery: involvement in complex regulation of noradrenaline release.

Pharmacological reports : PR 20060101

Substance use and sexual behaviours of Japanese men who have sex with men: a nationwide internet survey conducted in Japan.

BMC public health 20060101

Foxy methoxy: a new drug of abuse.

Journal of medical toxicology : official journal of the American College of Medical Toxicology 20051201

[Melatoninergic receptor agonists and antagonists: pharmacological aspects and therapeutic perspective].

Annales pharmaceutiques francaises 20051101

Determination of melatonin and its precursors and metabolites using capillary electrophoresis with UV and fluorometric detection.

Journal of separation science 20051101

Indoleamines and 5-methoxyindoles in trout pineal organ in vivo: daily changes and influence of photoperiod.

General and comparative endocrinology 20051001

5-HT1A receptor agonists modify epileptic seizures in three experimental models in rats.

Neuropharmacology 20050901

The role of ML-23 and other melatonin analogues in the treatment and management of Parkinson's disease.

Drug news & perspectives 20050901

Sensitive determination of alpha-methyltryptamine (AMT) and 5-methoxy-N,N-diisopropyltryptamine (5MeO-DIPT) in whole blood and urine using gas chromatography-mass spectrometry.

Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20050825

Impact of the CYP2D6 ultra-rapid metabolizer genotype on doxepin pharmacokinetics and serotonin in platelets.

Pharmacogenetics and genomics 20050801

Serotonin 5-HT7 receptors coupled to induction of interleukin-6 in human microglial MC-3 cells.

Neuropharmacology 20050701

Clozapine attenuates the locomotor sensitisation and the prepulse inhibition deficit induced by a repeated oral administration of Catha edulis extract and cathinone in rats.

Behavioural brain research 20050528

Medicinal chemistry driven approaches toward novel and selective serotonin 5-HT6 receptor ligands.

Journal of medicinal chemistry 20050324

A foxy intoxication.

Forensic science international 20050210

Voltage-dependent inhibition of recombinant NMDA receptor-mediated currents by 5-hydroxytryptamine.

British journal of pharmacology 20050201

Behavioral and cellular consequences of increasing serotonergic activity during brain development: a role in autism?

International journal of developmental neuroscience : the official journal of the International Society for Developmental Neuroscience 20050201

Effect of the postsynaptic 5-HT1A receptor antagonist MM-77 on stressed mice treated with 5-HT1A receptor agents.

European journal of pharmacology 20050131

Recovery from experimental Parkinson's disease in the 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine hydrochloride treated marmoset with the melatonin analogue ML-23.

Pharmacology, biochemistry, and behavior 20050101

Evidence for 5-HT2B and 5-HT7 receptor-mediated relaxation in pulmonary arteries of weaned pigs.

Naunyn-Schmiedeberg's archives of pharmacology 20050101

Statistical distribution of blood serotonin as a predictor of early autistic brain abnormalities.

Theoretical biology & medical modelling 20050101

Melatonin, a potent agent in antioxidative defense: actions as a natural food constituent, gastrointestinal factor, drug and prodrug.

Nutrition & metabolism 20050101

Rapid, accurate and precise quantitative drug analysis: comparing liquid chromatography tandem mass spectrometry and chip-based nanoelectrospray ionisation mass spectrometry.

European journal of mass spectrometry (Chichester, England) 20050101

The actions of a charged melatonin receptor ligand, TMEPI, and an irreversible MT2 receptor agonist, BMNEP, on mouse hippocampal evoked potentials in vitro.

Life sciences 20041112

Analytical chemistry of synthetic routes to psychoactive tryptamines. Part I. Characterisation of the Speeter and Anthony synthetic route to 5-methoxy-N,N-diisopropyltryptamine using ESI-MS-MS and ESI-TOF-MS.

The Analyst 20041101

Recovery of experimental Parkinson's disease with the melatonin analogues ML-23 and S-20928 in a chronic, bilateral 6-OHDA model: a new mechanism involving antagonism of the melatonin receptor.

Pharmacology, biochemistry, and behavior 20041101

Functional expression of the serotonin 5-HT7 receptor in human glioblastoma cell lines.

British journal of pharmacology 20041001

New drugs of abuse update: Foxy Methoxy.

Journal of emergency nursing: JEN : official publication of the Emergency Department Nurses Association 20041001

A general screening and confirmation approach to the analysis of designer tryptamines and phenethylamines in blood and urine using GC-EI-MS and HPLC-electrospray-MS.

Journal of analytical toxicology 20040901

Opposing electrophysiological actions of 5-HT on noncholinergic and cholinergic neurons in the rat ventral pallidum in vitro.

Journal of neurophysiology 20040701

[Latest cases of acute poisoning in clinical practice--5MeO-DIPT and GHB precursor].

Chudoku kenkyu : Chudoku Kenkyukai jun kikanshi = The Japanese journal of toxicology 20040701

Binding of tryptamine analogs at h5-HT1E receptors: a structure-affinity investigation.

Bioorganic & medicinal chemistry 20040515

Inhibition of p38 mitogen-activated protein kinase enhances adrenergic-stimulated arylalkylamine N-acetyltransferase activity in rat pinealocytes.

Endocrinology 20040301

Endogenous and dietary indoles: a class of antioxidants and radical scavengers in the ABTS assay.

Free radical research 20040301

Early serotonergic projections to Cajal-Retzius cells: relevance for cortical development.

The Journal of neuroscience : the official journal of the Society for Neuroscience 20040218

Involvement of melatonin metabolites in the long-term inhibitory effect of the hormone on rat spinal nociceptive transmission.

Pharmacology, biochemistry, and behavior 20040201

Molecular cloning and pharmacological characterization of the guinea pig 5-HT1E receptor.

European journal of pharmacology 20040126

Autoradiographic distribution of 5-HT7 receptors in the human brain using [3H]mesulergine: comparison to other mammalian species.

British journal of pharmacology 20040101

Synthesis of internal labeled standards of melatonin and its metabolite N1-acetyl-N2-formyl-5-methoxykynuramine for their quantification using an on-line liquid chromatography-electrospray tandem mass spectrometry system.

Journal of pineal research 20040101

Selective scavenging property of the indole moiety for the nitrating species of peroxynitrite.

Chemical & pharmaceutical bulletin 20040101

The implementation of acute versus chronic animal models for treatment discovery in Parkinson's disease.

Reviews in the neurosciences 20040101

Peroxynitrite scavenging activity of indole derivatives: interaction of indoles with peroxynitrite.

Journal of medicinal food 20040101

Characterization of the 5-HT(7) receptor. Determination of the pharmacophore for 5-HT(7) receptor agonism and CoMFA-based modeling of the agonist binding site.

Journal of medicinal chemistry 20031204

Expression of human organic anion transporters in the choroid plexus and their interactions with neurotransmitter metabolites.

Journal of pharmacological sciences 20031201

Pharmacological characterization of a serotonin receptor (5-HT7) stimulating cAMP production in human corneal epithelial cells.

Investigative ophthalmology & visual science 20031101

Interaction of singlet molecular oxygen with melatonin and related indoles.

Photochemistry and photobiology 20031101

Depression of mGluR-mediated IPSCs by 5-HT in dopamine neurons of the rat substantia nigra pars compacta.

The European journal of neuroscience 20031101

Circadian rhythms, oxidative stress, and antioxidative defense mechanisms.

Chronobiology international 20031101

Relative reactivities of histamine and indoleamines with acetaldehyde.

Biological & pharmaceutical bulletin 20030801

Characterization of the 5-HT6 receptor coupled to Ca2+ signaling using an enabling chimeric G-protein.

European journal of pharmacology 20030704

Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7).

Journal of medicinal chemistry 20030703

Functional activity of serotoninergic and melatoninergic systems expressed in the skin.

Journal of cellular physiology 20030701

[Levels of psilocybin and psilocin in various types of mushrooms].

Soudni lekarstvi 20030701

In search of endogenous CYP2D6 substrates.

Pharmacogenetics 20030601

Screening for endogenous substrates reveals that CYP2D6 is a 5-methoxyindolethylamine O-demethylase.

Pharmacogenetics 20030601

Fourier transform infrared spectra and molecular structure of 5-methoxytryptamine, N-acetyl-5-methoxytryptamine and N-phenylsulfonamide-5-methoxytryptamine.

Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20030401

Melatonin preserves arachidonic and docosapentaenoic acids during ascorbate-Fe2+ peroxidation of rat testis microsomes and mitochondria.

The international journal of biochemistry & cell biology 20030301

Regeneration of serotonin from 5-methoxytryptamine by polymorphic human CYP2D6.

Pharmacogenetics 20030301

5-HT7 receptor-mediated relaxation of the oviduct in nonpregnant proestrus pigs.

European journal of pharmacology 20030214

Photoperiod affects amplitude but not duration of in vitro melatonin production in the ruin lizard (Podarcis sicula).

Journal of biological rhythms 20030201

Further evidence that the discriminative stimulus properties of indorenate are mediated by 5-HT 1A/1B/2C receptors.

Pharmacology, biochemistry, and behavior 20030101

Reduction of cisplatin-induced anemia by the pineal indole 5-methoxytryptamine in metastatic lung cancer patients.

Neuro endocrinology letters 20030101

Foxy, a designer tryptamine hallucinogen.

Journal of analytical toxicology 20030101

Total pineal endocrine substitution therapy (TPEST) as a new neuroendocrine palliative treatment of untreatable metastatic solid tumor patients: a phase II study.

Neuro endocrinology letters 20030101

Photochemical properties of kynurenine pathway metabolites and indoleamines.

Advances in experimental medicine and biology 20030101

Indorenate produces antidepressant-like actions in the rat forced swimming test via 5-HT1A receptors.

Psychopharmacology 20021201

Role of melatonin in the induction and maintenance of sleep.

Dialogues in clinical neuroscience 20021201

Melatonin's unique radical scavenging properties - roles of its functional substituents as revealed by a comparison with its structural analogs.

Journal of pineal research 20020801

Characterization and regulation of a CHO cell line stably expressing human serotonin N-acetyltransferase (EC 2.3.1.87).

Cellular and molecular life sciences : CMLS 20020801

The effects of treatment with melatonin on the ultrastructure of mouse Leydig cells: a quantitative study.

Brazilian journal of biology = Revista brasleira de biologia 20020801

Influence of forced swimming-induced stress on the anxiolytic-like effect of 5HT(1A) agents in mice.

Psychopharmacology 20020701

Full substitution of the discriminative cue of a 5-HT(1A/1B/2C) agonist with the combined administration of a 5-HT(1B/2C) and a 5-HT(1A) agonist.

Behavioural pharmacology 20020701

Demonstration of antifungal and anti-human immunodeficiency virus reverse transcriptase activities of 6-methoxy-2-benzoxazolinone and antibacterial activity of the pineal indole 5-methoxyindole-3-acetic acid.

Comparative biochemistry and physiology. Toxicology & pharmacology : CBP 20020601

Modulation of 5-HT4 receptor function in the rat isolated ileum by fluoxetine: the involvement of endogenous 5-hydroxytryptamine.

British journal of pharmacology 20020501

Activity-dependent bidirectional regulation of GABA(A) receptor channels by the 5-HT(4) receptor-mediated signalling in rat prefrontal cortical pyramidal neurons.

The Journal of physiology 20020501

Desensitization of pigment granule aggregation in Xenopus leavis melanophores: melatonin degradation rather than receptor down-regulation is responsible.

Journal of neurochemistry 20020501

Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells.

The Journal of biological chemistry 20020419

Generalized loss of inhibitory innervation reverses serotonergic inhibition into excitation in a rabbit model of TNBS-colitis.

British journal of pharmacology 20020401

The neuroprotective activities of melatonin against the Alzheimer beta-protein are not mediated by melatonin membrane receptors.

Journal of pineal research 20020401

DARPP-32 mediates serotonergic neurotransmission in the forebrain.

Proceedings of the National Academy of Sciences of the United States of America 20020305

Behavioral and magnetic resonance spectroscopic studies in the rat hyperserotonemic model of autism.

Physiology & behavior 20020301

Modulation by serotonin 5-HT(4) receptors of long-term potentiation and depotentiation in the dentate gyrus of freely moving rats.

Cerebral cortex (New York, N.Y. : 1991) 20020201

Conversion of L-tryptophan to serotonin and melatonin in human melanoma cells.

FEBS letters 20020130

Differences in signal transduction of two 5-HT4 receptor splice variants: compound specificity and dual coupling with Galphas- and Galphai/o-proteins.

Molecular pharmacology 20020101

Clinical safety and effectiveness of indorenate in essential hypertension.

Proceedings of the Western Pharmacology Society 20020101

[Study of the antiradical and radioprotective properties of S-containing compounds using the complex of in vitro test-systems].

Radiatsionnaia biologiia, radioecologiia 20020101

Functional modification of cytochrome c by peroxynitrite in an electron transfer reaction.

Chemical & pharmaceutical bulletin 20011201

[Morphofunctional changes in the pineal gland during adaptation to hypothermia].

Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova 20011201

Examination of pineal indoles and 6-methoxy-2-benzoxazolinone for antioxidant and antimicrobial effects.

Comparative biochemistry and physiology. Toxicology & pharmacology : CBP 20011101

Guest-to-host proton transfer in melatonin-beta-cyclodextrin inclusion complex by ionspray, fast atom bombardment and tandem mass spectrometry.

Journal of mass spectrometry : JMS 20011101

Effect of carrier excipient and processing on stability of indorenate hydrochloride/excipient mixtures.

Pharmaceutical development and technology 20011101

Synthesis of valproic acid amides of a melatonin derivative, a piracetam and amantadine for biological tests.

Neurochemical research 20011001

[Presynaptic 5-hydroxytryptamine receptors enhance cholinergic neurosecretion in the human iris-ciliary body].

[Zhonghua yan ke za zhi] Chinese journal of ophthalmology 20010901

Putative regulatory molecules in plants: evaluating melatonin.

Journal of pineal research 20010801

The effects of acute melatonin and ethanol treatment on antioxidant enzyme activities in rat testes.

Pharmacological research 20010801

[(3)H]-serotonin release from bovine iris-ciliary body: pharmacology of prejunctional serotonin (5-HT(7)) autoreceptors.

Experimental eye research 20010701

The cloned human 5-HT7 receptor splice variants: a comparative characterization of their pharmacology, function and distribution.

Naunyn-Schmiedeberg's archives of pharmacology 20010601

A 5-HT(7) receptor-mediated depolarization in the anterodorsal thalamus. I. Pharmacological characterization.

The Journal of pharmacology and experimental therapeutics 20010401

Thrombopoietic properties of 5-methoxytryptamine plus melatonin versus melatonin alone in the treatment of cancer-related thrombocytopenia.

Journal of pineal research 20010301

Discriminative stimulus properties of indorenate, a 5-HT1A, 5-HT1B and 5-HT2C agonist: a study in rats.

Journal of psychopharmacology (Oxford, England) 20010301

Discriminative stimulus properties of indorenate in a conditioned taste aversion paradigm.

Pharmacology, biochemistry, and behavior 20010301

Endogenous indoles as novel polyamine site ligands at the N-methyl-D-aspartate receptor complex.

Brain research 20010202

5HT4(a) and 5-HT4(b) receptors have nearly identical pharmacology and are both expressed in human atrium and ventricle.

Naunyn-Schmiedeberg's archives of pharmacology 20010201

Unravelling the pharmacological profile of the canine external carotid vasodilator '5-HT1-like' receptors: coexistence of sympatho-inhibitory 5-HT1B and postjunctional 5-HT7 receptors.

Naunyn-Schmiedeberg's archives of pharmacology 20010101

High-performance liquid chromatography assay for indorenate in pharmaceutical powders.

Drug development and industrial pharmacy 20010101

Pineal indoles stimulate the gene expression of immunomodulating cytokines.

Journal of neural transmission (Vienna, Austria : 1996) 20010101

Pharmacological characterization of the human 5-HT(4(d)) receptor splice variant stably expressed in Chinese hamster ovary cells.

British journal of pharmacology 20001001

2-Substituted tryptamines: agents with selectivity for 5-HT(6) serotonin receptors.

Journal of medicinal chemistry 20000309

Agonist high and low affinity state ratios predict drug intrinsic activity and a revised ternary complex mechanism at serotonin 5-HT(2A) and 5-HT(2C) receptors.

Synapse (New York, N.Y.) 20000201

Structure of the human serotonin 5-HT4 receptor gene and cloning of a novel 5-HT4 splice variant.

Journal of neurochemistry 20000201

Isolation of the serotoninergic 5-HT4(e) receptor from human heart and comparative analysis of its pharmacological profile in C6-glial and CHO cell lines.

British journal of pharmacology 20000201

Identification of residues in transmembrane regions III and VI that contribute to the ligand binding site of the serotonin 5-HT6 receptor.

Journal of neurochemistry 19981101

Cloning, expression, and pharmacology of four human 5-hydroxytryptamine 4 receptor isoforms produced by alternative splicing in the carboxyl terminus.

Journal of neurochemistry 19980601

Cloning and expression of a human serotonin 5-HT4 receptor cDNA.

Journal of neurochemistry 19971101

Activating mutations of the serotonin 5-HT2C receptor.

Journal of neurochemistry 19970901

Cloning, expression and pharmacology of a truncated splice variant of the human 5-HT7 receptor (h5-HT7b).

British journal of pharmacology 19970901

[3H]RS 57639, a high affinity, selective 5-HT4 receptor partial agonist, specifically labels guinea-pig striatal and rat cloned (5-HT4S and 5-HT4L) receptors.

Neuropharmacology 19970101

Functional and radioligand binding characterization of rat 5-HT6 receptors stably expressed in HEK293 cells.

Neuropharmacology 19970101

Alniditan, a new 5-hydroxytryptamine1D agonist and migraine-abortive agent: ligand-binding properties of human 5-hydroxytryptamine1D alpha, human 5-hydroxytryptamine1D beta, and calf 5-hydroxytryptamine1D receptors investigated with [3H]5-hydroxytryptamine and [3H]alniditan.

Molecular pharmacology 19961201

Cloning, expression and pharmacology of the mouse 5-HT(4L) receptor.

FEBS letters 19961125

Two amino acid differences in the sixth transmembrane domain are partially responsible for the pharmacological differences between the 5-HT1D beta and 5-HT1E 5-hydroxytryptamine receptors.

Journal of neurochemistry 19961101

[3H]5-hydroxytryptamine labels the agonist high affinity state of the cloned rat 5-HT4 receptor.

European journal of pharmacology 19960523

Cloning, characterization, and chromosomal localization of a human 5-HT6 serotonin receptor.

Journal of neurochemistry 19960101

The 5-HT4 receptor: molecular cloning and pharmacological characterization of two splice variants.

The EMBO journal 19950615

Species variations in transmembrane region V of the 5-hydroxytryptamine type 2A receptor alter the structure-activity relationship of certain ergolines and tryptamines.

Molecular pharmacology 19940201

Cloning of a novel human serotonin receptor (5-HT7) positively linked to adenylate cyclase.

The Journal of biological chemistry 19931105

Molecular cloning, characterization, and localization of a high-affinity serotonin receptor (5-HT7) activating cAMP formation.

Proceedings of the National Academy of Sciences of the United States of America 19930915

Molecular cloning and expression of a 5-hydroxytryptamine7 serotonin receptor subtype.

The Journal of biological chemistry 19930825

Molecular cloning of a mammalian serotonin receptor that activates adenylate cyclase.

Molecular pharmacology 19930801

The role of receptor binding in drug discovery.

Journal of natural products 19930401

Cloning and expression of a novel serotonin receptor with high affinity for tricyclic psychotropic drugs.

Molecular pharmacology 19930301

Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor.

Molecular pharmacology 19930301

Cloning of another human serotonin receptor (5-HT1F): a fifth 5-HT1 receptor subtype coupled to the inhibition of adenylate cyclase.

Proceedings of the National Academy of Sciences of the United States of America 19930115

Human serotonin 1D receptor is encoded by a subfamily of two distinct genes: 5-HT1D alpha and 5-HT1D beta.

Proceedings of the National Academy of Sciences of the United States of America 19920415

Primary structure and functional characterization of a human 5-HT1D-type serotonin receptor.

Molecular pharmacology 19910801