Piperidine-1-carboxamide
| Title | Journal |
|---|---|
| Behavioral and neurochemical profile of some novel phenacyl based isonipecotamide derivatives. | Pakistan journal of pharmaceutical sciences 20121001 |
| Anti-AIDS agents 90. novel C-28 modified bevirimat analogues as potent HIV maturation inhibitors. | Journal of medicinal chemistry 20120927 |
| A β-tryptase inhibitor with a tropanylamide scaffold to improve in vitro stability and to lower hERG channel binding affinity. | Bioorganic & medicinal chemistry letters 20120215 |
| Development of Metarhizium anisopliae and Beauveria bassiana formulations for control of malaria mosquito larvae. | Parasites & vectors 20110101 |
| New classes of alanine racemase inhibitors identified by high-throughput screening show antimicrobial activity against Mycobacterium tuberculosis. | PloS one 20110101 |
| A conformationally constrained inhibitor with an enhanced potency for β-tryptase and stability against semicarbazide-sensitive amine oxidase (SSAO). | Bioorganic & medicinal chemistry letters 20101115 |
| Non-peptidic antagonists of the CGRP receptor, BIBN4096BS and MK-0974, interact with the calcitonin receptor-like receptor via methionine-42 and RAMP1 via tryptophan-74. | Biochemical and biophysical research communications 20100101 |
| Discovery of 4-morpholino-6-aryl-1H-pyrazolo[3,4-d]pyrimidines as highly potent and selective ATP-competitive inhibitors of the mammalian target of rapamycin (mTOR): optimization of the 6-aryl substituent. | Journal of medicinal chemistry 20091224 |
| Optimization of 2-piperidin-4-yl-acetamides as melanin-concentrating hormone receptor 1 (MCH-R1) antagonists: Designing out hERG inhibition. | Bioorganic & medicinal chemistry letters 20090801 |
| Optimization of piperidin-4-yl-urea-containing melanin-concentrating hormone receptor 1 (MCH-R1) antagonists: Reducing hERG-associated liabilities. | Bioorganic & medicinal chemistry letters 20090801 |
| Synthesis and structure-activity relationship of novel diarylpyrazole imide analogues as CB1 cannabinoid receptor ligands. | Bioorganic & medicinal chemistry 20090415 |
| The design and discovery of novel amide CCR5 antagonists. | Bioorganic & medicinal chemistry letters 20090215 |
| Casopitant: a novel NK(1)-receptor antagonist in the prevention of chemotherapy-induced nausea and vomiting. | Therapeutics and clinical risk management 20090101 |
| 1-, 3- and 8-substituted-9-deazaxanthines as potent and selective antagonists at the human A2B adenosine receptor. | Bioorganic & medicinal chemistry 20080315 |
| Functional antagonism between endogenous neuropeptide Y and calcitonin gene-related peptide in mesenteric resistance arteries. | The Journal of pharmacology and experimental therapeutics 20080301 |
| Methoxy- and fluorine-substituted analogs of O-1302: synthesis and in vitro binding affinity for the CB1 cannabinoid receptor. | Chemical & pharmaceutical bulletin 20070801 |
| Piperidine amides as 11beta-hydroxysteroid dehydrogenase type 1 inhibitors. | Bioorganic & medicinal chemistry letters 20070615 |
| Pharmacological characterisation of capsaicin-induced relaxations in human and porcine isolated arteries. | Naunyn-Schmiedeberg's archives of pharmacology 20070301 |
| Enantioselective strecker reaction of phosphinoyl ketoimines catalyzed by in situ prepared chiral N,N'-dioxides. | The Journal of organic chemistry 20070105 |
| Determinants of 1-piperidinecarboxamide, N-[2-[[5-amino-l-[[4-(4-pyridinyl)-l-piperazinyl]carbonyl]pentyl]amino]-1-[(3,5-dibromo-4-hydroxyphenyl)methyl]-2-oxoethyl]-4-(1,4-dihydro-2-oxo-3(2H)-quinazolinyl) (BIBN4096BS) affinity for calcitonin gene-related peptide and amylin receptors--the role of receptor activity modifying protein 1. | Molecular pharmacology 20061201 |
| A key role for transmembrane prolines in calcitonin receptor-like receptor agonist binding and signalling: implications for family B G-protein-coupled receptors. | Molecular pharmacology 20050101 |
| Noncompetitive antagonism of BIBN4096BS on CGRP-induced responses in human subcutaneous arteries. | British journal of pharmacology 20041201 |
| Structure activity relationship by NMR and by computer: a comparative study. | Journal of the American Chemical Society 20020918 |
| GC/MS investigations of the minor constituents of Piper guineense stem. | Die Pharmazie 20020901 |
| A piperidine amide extracted from Piper longum L. fruit shows activity against Aedes aegypti mosquito larvae. | Journal of agricultural and food chemistry 20020619 |
| Tandem mass spectrum of a growth hormone secretagogue: amide bond cleavage and resultant gas-phase rearrangement. | Journal of the American Society for Mass Spectrometry 20020401 |