4-(2-Keto-1-benzimidazolinyl)piperidine
| Title | Journal |
|---|---|
| Discovery of a Chemical Tool Inhibitor Targeting the Bromodomains of TRIM24 and BRPF. | Journal of medicinal chemistry 20160225 |
| Synthesis and antibacterial activities of 1-alkyl-3-methacryloyl (acryloyl) of benzimidazolone (thione) derivatives. | International journal of molecular sciences 20120101 |
| Effect of nitro groups on the photo physical properties of benzimidazolone: a solvatochromic study. | Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20111215 |
| Benzimidazolone as potent chymase inhibitor: modulation of reactive metabolite formation in the hydrophobic (P1) region. | Bioorganic & medicinal chemistry letters 20110801 |
| N-aryl-benzimidazolones as novel small molecule HSP90 inhibitors. | Bioorganic & medicinal chemistry letters 20101215 |
| Design, synthesis, and structure-activity relationships of 1,3-dihydrobenzimidazol-2-one analogues as anti-HIV agents. | Bioorganic & medicinal chemistry 20090815 |
| Design and synthesis of isoform-selective phospholipase D (PLD) inhibitors. Part I: Impact of alternative halogenated privileged structures for PLD1 specificity. | Bioorganic & medicinal chemistry letters 20090401 |
| Structures of six industrial benzimidazolone pigments from laboratory powder diffraction data. | Acta crystallographica. Section B, Structural science 20090401 |
| Benzimidazolone-based serotonin 5-HT1A or 5-HT7R ligands: synthesis and biological evaluation. | Bioorganic & medicinal chemistry letters 20090315 |
| Potent benzimidazolone-based CGRP receptor antagonists. | Bioorganic & medicinal chemistry letters 20081201 |
| The SAR studies of novel CB2 selective agonists, benzimidazolone derivatives. | Bioorganic & medicinal chemistry letters 20080601 |
| Towards the synthesis of new benzimidazolone derivatives with surfactant properties. | Carbohydrate research 20080225 |
| Structural elucidation of rabeprazole sodium photodegradation products. | Journal of pharmaceutical and biomedical analysis 20080107 |
| New 'chemical probes' to examine the role of the hFPRL1 (or ALXR) receptor in inflammation. | Bioorganic & medicinal chemistry letters 20071201 |
| Potent benzimidazolone based human beta(3)-adrenergic receptor agonists. | Bioorganic & medicinal chemistry letters 20061101 |
| The SAR of 4-substituted (6,6-bicyclic) piperidine cathepsin S inhibitors. | Bioorganic & medicinal chemistry letters 20060415 |
| Recent advances in the solid-phase combinatorial synthetic strategies for the quinoxaline, quinazoline and benzimidazole based privileged structures. | Mini reviews in medicinal chemistry 20060101 |
| Theoretical and experimental design of atypical kinase inhibitors: application to p38 MAP kinase. | Journal of medicinal chemistry 20050908 |
| SAR studies of 6-aryl-1,3-dihydrobenzimidazol-2-ones as progesterone receptor antagonists. | Bioorganic & medicinal chemistry letters 20050801 |
| Benzimidazolones and indoles as non-thiol farnesyltransferase inhibitors based on tipifarnib scaffold: synthesis and activity. | Bioorganic & medicinal chemistry letters 20050602 |
| Discovery and SAR studies of a novel series of noncovalent cathepsin S inhibitors. | Bioorganic & medicinal chemistry letters 20050315 |
| Multiple tandem mass spectrometry-based investigation of the behaviour of some thiazol-benzimidazolones and 2-benzimidazolylsulfanyl ethanones. | European journal of mass spectrometry (Chichester, England) 20050101 |
| Natural modulators of large-conductance calcium-activated potassium channels. | Planta medica 20031001 |
| CFTR activation in human bronchial epithelial cells by novel benzoflavone and benzimidazolone compounds. | American journal of physiology. Lung cellular and molecular physiology 20030701 |
| In vitro inhibition of pimozide N-dealkylation by selective serotonin reuptake inhibitors and azithromycin. | Journal of clinical psychopharmacology 20020401 |
| Rapid liquid-phase combinatorial synthesis of heterocyclic libraries. | Methods in molecular biology (Clifton, N.J.) 20020101 |
| Synthesis and progesterone receptor antagonist activities of 6-aryl benzimidazolones and benzothiazolones. | Bioorganic & medicinal chemistry letters 20011022 |
| N-acylated alpha-(3-pyridylmethyl)-beta-aminotetralin antagoinists of the human neuropeptide Y Y5 receptor. | Bioorganic & medicinal chemistry letters 20000807 |