Methanesulfonamide
| Title | Journal |
|---|---|
| A novel carbohydrate derived compound FCP5 causes DNA strand breaks and oxidative modifications of DNA bases in cancer cells. | Chemico-biological interactions 20150205 |
| Pyrrolo[2,3-b]quinoxalines as inhibitors of firefly luciferase: their Cu-mediated synthesis and evaluation as false positives in a reporter gene assay. | Bioorganic & medicinal chemistry letters 20121015 |
| Amide derivatives of benzene-sulfonanilide, pharmaceutical composition thereof and method for cancer treatment using the same (US20120095092). | Expert opinion on therapeutic patents 20121001 |
| RCAI-84, 91, and 105-108, ureido and thioureido analogs of KRN7000: their synthesis and bioactivity for mouse lymphocytes to produce Th1-biased cytokines. | Bioorganic & medicinal chemistry 20120715 |
| Conformational analysis, vibrational and NMR spectroscopic study of the methanesulfonamide-N,N'-1,2-ethanediylbis. | Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20120601 |
| Total synthesis of a marine alkaloid--rigidin E. | Marine drugs 20120601 |
| Synthesis, evaluation and docking studies on 3-alkoxy-4-methanesulfonamido acetophenone derivatives as non ulcerogenic anti-inflammatory agents. | European journal of medicinal chemistry 20120301 |
| Rosuvastatin blocks hERG current and prolongs cardiac repolarization. | Journal of pharmaceutical sciences 20120201 |
| Managing atrial fibrillation in the elderly: critical appraisal of dronedarone. | Clinical interventions in aging 20120101 |
| Rosuvastatin: a review of the pharmacology and clinical effectiveness in cardiovascular disease. | Clinical Medicine Insights. Cardiology 20120101 |
| N-[4-(4-Fluoro-phen-yl)-5-hy-droxy-methyl-6-isopropyl-pyrimidin-2-yl]-N-methyl-methane-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20111201 |
| The structure of NS-398 bound to cyclooxygenase-2. | Journal of structural biology 20111101 |
| Methanesulfonamido-cyclohexylamine derivatives of 2,4-diaminopyrimidine as potent ALK inhibitors. | Bioorganic & medicinal chemistry letters 20110701 |
| Synthesis and antibacterial activity of pentacyclines: a novel class of tetracycline analogs. | Journal of medicinal chemistry 20110609 |
| Discovery of new chromone containing sulfonamides as potent inhibitors of bovine cytosolic carbonic anhydrase. | Bioorganic & medicinal chemistry 20110601 |
| N,N'-Dibenzyl-N,N'-dimethyl-N''-(methyl-sulfon-yl)phospho-ric triamide. | Acta crystallographica. Section E, Structure reports online 20110601 |
| Mild Pd-catalyzed N-arylation of methanesulfonamide and related nucleophiles: avoiding potentially genotoxic reagents and byproducts. | Organic letters 20110520 |
| 2-(N-Phenyl-methane-sulfonamido)-ethyl 1H-pyrrole-2-carboxyl-ate. | Acta crystallographica. Section E, Structure reports online 20110501 |
| Clinical utility of rosuvastatin and other statins for cardiovascular risk reduction among the elderly. | Clinical interventions in aging 20110101 |
| Application of molecular topology for the prediction of reaction yields and anti-inflammatory activity of heterocyclic amidine derivatives. | International journal of molecular sciences 20110101 |
| Optimization of Benzoisothiazole dioxide inhibitory activity of the NS5B polymerase of HCV genotype 4 using ligand-steered homological modeling, reaction-driven scaffold-hopping and Enovo workflow. | Bioinformation 20110101 |
| A diverse series of substituted benzenesulfonamides as aldose reductase inhibitors with antioxidant activity: design, synthesis, and in vitro activity. | Journal of medicinal chemistry 20101111 |
| Expanding the diversity of allosteric bcr-abl inhibitors. | Journal of medicinal chemistry 20101014 |
| Impact of dronedarone in atrial fibrillation and flutter on stroke reduction. | Clinical interventions in aging 20100101 |
| Studies of benzothiadiazine derivatives as hepatitis C virus NS5B polymerase inhibitors using 3D-QSAR, molecular docking and molecular dynamics. | Current medicinal chemistry 20100101 |
| Non-nucleoside inhibitors of HCV polymerase NS5B. Part 4: structure-based design, synthesis, and biological evaluation of benzo[d]isothiazole-1,1-dioxides. | Bioorganic & medicinal chemistry letters 20091001 |
| Bis(tetra-phenyl-phospho-nium) tris-[N-(methyl-sulfon-yl)dithio-carbimato(2-)-κS,S']stannate(IV). | Acta crystallographica. Section E, Structure reports online 20091001 |
| Synthesis, antiviral and anticancer activity of some novel thioureas derived from N-(4-nitro-2-phenoxyphenyl)-methanesulfonamide. | European journal of medicinal chemistry 20090901 |
| Novel indoline-based acyl-CoA: cholesterol acyltransferase inhibitor: Effects of introducing a methanesulfonamide group on physicochemical properties and biological activities. | Bioorganic & medicinal chemistry 20090815 |
| Regulation of the apoptosis-inducing kinase DRAK2 by cyclooxygenase-2 in colorectal cancer. | British journal of cancer 20090804 |
| Synthesis, anticancer, and anti-inflammatory activity evaluation of methanesulfonamide and amidine derivatives of 3,4-diaryl-2-imino-4-thiazolines. | Molecular diversity 20090801 |
| Development and validation of an LC-MS/MS method for determination of methanesulfonamide in human urine. | Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20090715 |
| Non-nucleoside inhibitors of HCV polymerase NS5B. Part 2: Synthesis and structure-activity relationships of benzothiazine-substituted quinolinediones. | Bioorganic & medicinal chemistry letters 20090701 |
| Methanesulfonamide: a cosolvent and a general acid catalyst in sharpless asymmetric dihydroxylations. | The Journal of organic chemistry 20090417 |
| Cytotoxic activity of platinum(II) and palladium(II) complexes of N-3-pyridinylmethanesulfonamide: the influence of electroporation. | Zeitschrift fur Naturforschung. C, Journal of biosciences 20090101 |
| Novel transthyretin amyloid fibril formation inhibitors: synthesis, biological evaluation, and X-ray structural analysis. | PloS one 20090101 |
| Long-term use of rosuvastatin: a critical risk benefit appraisal and comparison with other antihyperlipidemics. | Drug, healthcare and patient safety 20090101 |
| An experimental and theoretical study of dipole moments of N-[4-(9-acridinylamino)-3-methoxyphenyl]methanesulfonamide. | Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20080901 |
| (4R)-4-[(1R)-1,2-Dihydroxy-ethyl]-1-[(1R)-1-phenyl-ethyl]pyrrolidin-2-one. | Acta crystallographica. Section E, Structure reports online 20080901 |
| Clinical efficacy and safety of statins in managing cardiovascular risk. | Vascular health and risk management 20080401 |
| beta-N-Biaryl ether sulfonamide hydroxamates as potent gelatinase inhibitors: part 1. Design, synthesis, and lead identification. | Bioorganic & medicinal chemistry letters 20080201 |
| Methyl 2-(N-ethyl-methane-sulfonamido)benzoate. | Acta crystallographica. Section E, Structure reports online 20080201 |
| Synthesis and biological evaluation of novel sulfonanilide compounds as antiproliferative agents for breast cancer. | Journal of combinatorial chemistry 20080101 |
| A new strategy for the synthesis of benzylic sulfonamides: palladium-catalyzed arylation and sulfonamide metathesis. | The Journal of organic chemistry 20071012 |
| Discovery of a highly active ligand of human pregnane x receptor: a case study from pharmacophore modeling and virtual screening to 'in vivo' biological activity. | Molecular pharmacology 20070901 |
| Optimization of triaryl bis-sulfones as cannabinoid-2 receptor ligands. | Bioorganic & medicinal chemistry letters 20070701 |
| A single component ratiometric pH probe with long wavelength excitation of europium emission. | Chemical communications (Cambridge, England) 20070207 |
| Synthesis and biological evaluation of methanesulfonamide analogues of rofecoxib: Replacement of methanesulfonyl by methanesulfonamido decreases cyclooxygenase-2 selectivity. | Bioorganic & medicinal chemistry 20070115 |
| Inhibition of human phenol and estrogen sulfotransferase by certain non-steroidal anti-inflammatory agents. | Current drug metabolism 20061001 |
| Carbonic anhydrase inhibitors: inhibition of the human isozymes I, II, VA, and IX with a library of substituted difluoromethanesulfonamides. | Bioorganic & medicinal chemistry letters 20051201 |
| Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, IX, and XII with N-hydroxysulfamides--a new zinc-binding function in the design of inhibitors. | Bioorganic & medicinal chemistry letters 20050502 |
| Structural determinants of HERG channel block by clofilium and ibutilide. | Molecular pharmacology 20040801 |
| [Synthesis and anti-inflammatory activity of N-(4-arylamidophenyl) methanesulfonamide derivatives]. | Yao xue xue bao = Acta pharmaceutica Sinica 20040701 |
| Methanesulfonamide group at position-4 of the C-5-phenyl ring of 1,5-diarylpyrazole affords a potent class of cyclooxygenase-2 (COX-2) inhibitors. | Bioorganic & medicinal chemistry letters 20040405 |
| N-4-Substituted-benzyl-N'-tert-butylbenzyl thioureas as vanilloid receptor ligands: investigation on the role of methanesulfonamido group in antagonistic activity. | Bioorganic & medicinal chemistry letters 20040209 |
| Differential recovery of action potential duration and HERG currents from the effects of two methanesulfonamide class III antiarrhythmic agents, KCB-328 and dofetilide. | Journal of cardiovascular pharmacology 20031101 |
| Variations of acidic functions at position 2 and substituents at positions 4, 5 and 6 of the indole moiety and their effect on NMDA-glycine site affinity. | European journal of medicinal chemistry 20031001 |
| Synthesis and prostaglandin synthase inhibitory activity of new aromatic O-alkyloxime ethers substituted with methylsulfonamido or methylsulfonyl groups on their aliphatic portion. | Farmaco (Societa chimica italiana : 1989) 20030901 |
| Acetic acid-derived prostaglandin-dependent colonic adaptive cytoprotection is preserved in chronic colitis: role of cyclo-oxygenase. | International journal of colorectal disease 20030501 |
| [Anti-arrhythmic action of N-(aminoalkylene) derivatives of indoline-2,3-diones and 1,2-benzene-dicarboxiamides]. | Medicina (Kaunas, Lithuania) 20020101 |
| Substituted indole-5-carboxamides and -acetamides as potent nonpeptide GnRH receptor antagonists. | Bioorganic & medicinal chemistry letters 20010709 |