1-cyclohexyl-3-({4-[2-(7-methoxy-4,4-dimethyl-1,3-dioxo-1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]benzene}sulfonyl)urea
| Title | Journal |
|---|---|
| In vitro inhibition of AKR1Cs by sulphonylureas and the structural basis. | Chemico-biological interactions 20151005 |
| A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development. | Toxicological sciences : an official journal of the Society of Toxicology 20131101 |
| Towards therapeutic applications of arthropod venom k(+)-channel blockers in CNS neurologic diseases involving memory acquisition and storage. | Journal of toxicology 20120101 |
| Effects of Sulfonylureas on Peroxisome Proliferator-Activated Receptor γ Activity and on Glucose Uptake by Thiazolidinediones. | Diabetes & metabolism journal 20110801 |
| Gliquidone. | Acta crystallographica. Section E, Structure reports online 20110601 |
| Impact of clinical factors and CYP2C9 variants for the risk of severe sulfonylurea-induced hypoglycemia. | European journal of clinical pharmacology 20110501 |
| Simultaneous identification and validated quantification of 11 oral hypoglycaemic drugs in plasma by electrospray ionisation liquid chromatography-mass spectrometry. | Analytical and bioanalytical chemistry 20110401 |
| Simultaneous determination of gliquidone, pioglitazone hydrochloride, and verapamil in formulation and human serum by RP-HPLC. | Journal of chromatographic science 20110201 |
| Effect of glibenclamide on antinociceptive effects of antidepressants of different classes. | Clinics (Sao Paulo, Brazil) 20110201 |
| Smoking and risk for diabetes incidence and mortality in Korean men and women. | Diabetes care 20101201 |
| Synthesis and SAR studies of 1,4-benzoxazine MenB inhibitors: novel antibacterial agents against Mycobacterium tuberculosis. | Bioorganic & medicinal chemistry letters 20101101 |
| Efficacy of anti-wrinkle products in skin surface appearance: a comparative study using non-invasive methods. | Skin research and technology : official journal of International Society for Bioengineering and the Skin (ISBS) [and] International Society for Digital Imaging of Skin (ISDIS) [and] International Society for Skin Imaging (ISSI) 20101101 |
| Severe sulfonylurea-induced hypoglycemia: a problem of uncritical prescription and deficiencies of diabetes care in geriatric patients. | Expert opinion on drug safety 20100901 |
| Drug therapy in patients with chronic renal failure. | Deutsches Arzteblatt international 20100901 |
| Simultaneous determination of gliquidone, fexofenadine, buclizine, and levocetirizine in dosage formulation and human serum by RP-HPLC. | Journal of chromatographic science 20100101 |
| Determination of glycyrrhizin in dog plasma by liquid chromatography-mass spectrometry and its application in pharmacokinetic studies. | European journal of mass spectrometry (Chichester, England) 20100101 |
| Twice daily fractionated dose administration of prednisolone compared to standard once daily administration to patients with glomerulonephritis or with kidney transplants. | Medizinische Klinik (Munich, Germany : 1983) 20090615 |
| Glucose and pharmacological modulators of ATP-sensitive K+ channels control [Ca2+]c by different mechanisms in isolated mouse alpha-cells. | Diabetes 20090201 |
| Sulfonylurea-induced hypoglycaemia: use of octreotide. | Acta clinica Belgica 20090101 |
| Risk of cardiovascular disease and all cause mortality among patients with type 2 diabetes prescribed oral antidiabetes drugs: retrospective cohort study using UK general practice research database. | BMJ (Clinical research ed.) 20090101 |
| Metformin, sulfonylureas, or other antidiabetes drugs and the risk of lactic acidosis or hypoglycemia: a nested case-control analysis. | Diabetes care 20081101 |
| Rapid simultaneous quantification of five active constituents in rat plasma by high-performance liquid chromatography/tandem mass spectrometry after oral administration of Da-Cheng-Qi decoction. | Journal of pharmaceutical and biomedical analysis 20080715 |
| Gliquidone therapy of new-onset diabetes mellitus after kidney transplantation. | Clinical nephrology 20080701 |
| Bioavailability of the amino acid-attached prodrug as a new anti-HIV agent in rats. | Journal of veterinary science 20070901 |
| Simultaneous assay of metformin and glibenclamide in human plasma based on extraction-less sample preparation procedure and LC/(APCI)MS. | Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20070701 |
| Development of a RP-HPLC method for screening potentially counterfeit anti-diabetic drugs. | Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20070615 |
| Determination of glibenclamide in human plasma by liquid chromatography and atmospheric pressure chemical ionization/MS-MS detection. | Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20070201 |
| Sulfonylureas and glinides exhibit peroxisome proliferator-activated receptor gamma activity: a combined virtual screening and biological assay approach. | Molecular pharmacology 20070201 |
| Spectrophotometric method for quantitative determination of gliquidone in bulk drug, pharmaceutical formulations and human serum. | Pakistan journal of pharmaceutical sciences 20060701 |
| Microsphere-based protease assays and screening application for lethal factor and factor Xa. | Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501 |
| Synthesis and antihyperglycemic evaluation of various protoberberine derivatives. | Bioorganic & medicinal chemistry letters 20060301 |
| Gliquidone contributes to improvement of type 2 diabetes mellitus management: a review of pharmacokinetic and clinical trial data. | Drugs in R&D 20060101 |
| Effect of glurenorm on immunohistochemical changes in pancreatic beta cells of rats in experimental diabetes. | Indian journal of experimental biology 20050301 |
| Protective effects of glurenorm (gliquidone) treatment on the liver injury of experimental diabetes. | Drug and chemical toxicology 20050101 |
| [Effect of liuwei dihuang pill on erythrocyte aldose reductase activity in early diabetic nephropathy patients]. | Zhongguo Zhong xi yi jie he za zhi Zhongguo Zhongxiyi jiehe zazhi = Chinese journal of integrated traditional and Western medicine 20041201 |
| Improvement of gliquidone hypoglycaemic effect in rats by cyclodextrin formulations. | European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20040901 |
| [Gliquidon induced-desensitization of pancreatic beta cells and the partial reversion of responsiveness after the desensitization of exposure to drug in normal and STZ type 2 diabetic rats]. | Sichuan da xue xue bao. Yi xue ban = Journal of Sichuan University. Medical science edition 20040501 |
| Enhancement of dissolution and oral bioavailability of gliquidone with hydroxy propyl-beta-cyclodextrin. | Die Pharmazie 20031101 |
| Hydroxyl-substituted sulfonylureas as potent inhibitors of specific [3H]glyburide binding to rat brain synaptosomes. | Bioorganic & medicinal chemistry 20030501 |
| [Severe hypoglycemia in diabetics with impaired renal function]. | Deutsche medizinische Wochenschrift (1946) 20030207 |
| Effect of pH and complexation on transdermal permeation of gliquidone. | Die Pharmazie 20020901 |
| Antiaggregatory activity of hypoglycaemic sulphonylureas. | Diabetologia 20020701 |
| Screening, library-assisted identification and validated quantification of oral antidiabetics of the sulfonylurea-type in plasma by atmospheric pressure chemical ionization liquid chromatography-mass spectrometry. | Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20020615 |
| The effect of Glurenorm (gliquidone) on lenses and skin in experimental diabetes. | Free radical biology & medicine 20011101 |
| Methylamine and benzylamine induced hypophagia in mice: modulation by semicarbazide-sensitive benzylamine oxidase inhibitors and aODN towards Kv1.1 channels. | British journal of pharmacology 20011001 |
| Role of K+ -channels in homotaurine-induced analgesia. | Fundamental & clinical pharmacology 20010601 |