Benzoxazole
Title | Journal |
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Direct C-H carboxylation with carbon dioxide using 1,2,3-triazol-5-ylidene copper(I) complexes. | Organic letters 20120803 |
Benzoheterocyclic amodiaquine analogues with potent antiplasmodial activity: synthesis and pharmacological evaluation. | Bioorganic & medicinal chemistry letters 20120801 |
Benzoxazole and benzothiazole amides as novel pharmacokinetic enhancers of HIV protease inhibitors. | Bioorganic & medicinal chemistry letters 20120801 |
Accessing the long-lived triplet excited states in bodipy-conjugated 2-(2-hydroxyphenyl) benzothiazole/benzoxazoles and applications as organic triplet photosensitizers for photooxidations. | The Journal of organic chemistry 20120720 |
Functionalized orthoesters as powerful building blocks for the efficient preparation of heteroaromatic bicycles. | Organic letters 20120706 |
Synthesis and structure-activity relationship of aminopyridines with substituted benzoxazoles as c-Met kinase inhibitors. | Bioorganic & medicinal chemistry letters 20120615 |
Identification of benzoxazole analogs as novel, S1P(3) sparing S1P(1) agonists. | Bioorganic & medicinal chemistry letters 20120615 |
Palladium-catalyzed C-H bond direct alkynylation of 5-membered heteroarenes: a well-defined synthetic route to azole derivatives containing two different alkynyl groups. | The Journal of organic chemistry 20120615 |
Nickel-catalyzed C-H direct amination of benzoxazoles with secondary amines. | Organic & biomolecular chemistry 20120514 |
A SAR study of novel antiproliferative ruthenium and osmium complexes with quinoxalinone ligands in human cancer cell lines. | Journal of medicinal chemistry 20120412 |
Evaluation of a multi-kinase inhibitor KRC-108 as an anti-tumor agent in vitro and in vivo. | Investigational new drugs 20120401 |
Antistaphylococcal activity of novel salicylanilide derivatives. | Current drug discovery technologies 20120301 |
Hit to lead SAR study on benzoxazole derivatives for an NPY Y5 antagonist. | Bioorganic & medicinal chemistry letters 20120301 |
Inhibitors of human histone deacetylase with potent activity against the African trypanosome Trypanosoma brucei. | Bioorganic & medicinal chemistry letters 20120301 |
Versatile chemical transformations of benzoxazole based ligands on complexation with 3d-metal ions. | Inorganic chemistry 20120220 |
Synthesis and antihormonal properties of novel 11β-benzoxazole-substituted steroids. | Bioorganic & medicinal chemistry letters 20120215 |
Novel benzothiazole, benzimidazole and benzoxazole derivatives as potential antitumor agents: synthesis and preliminary in vitro biological evaluation. | Molecules (Basel, Switzerland) 20120117 |
Synthesis and photo-physical characteristics of ESIPT inspired 2-substituted benzimidazole, benzoxazole and benzothiazole fluorescent derivatives. | Journal of fluorescence 20120101 |
A divergent and selective synthesis of isomeric benzoxazoles from a single N-Cl imine. | Organic letters 20111202 |
Synthesis, characterization, and spectroscopic investigation of benzoxazole conjugated Schiff bases. | The journal of physical chemistry. A 20111124 |
Palladium-catalyzed desulfitative C-arylation of a benzo[d]oxazole C-H bond with arene sulfonyl chlorides. | Chemical communications (Cambridge, England) 20111107 |
Photophysical, electrochemical and crystallographic investigations of the fluorophore 2,5-bis(5-tert-butyl-benzoxazol-2-yl)thiophene. | The journal of physical chemistry. B 20111103 |
2-(2-Hy-droxy-phen-yl)-1,3-benzothia-zole-6-carbaldehyde. | Acta crystallographica. Section E, Structure reports online 20111101 |
Paliperidone: 3-{2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]eth-yl}-9-hy-droxy-2-methyl-1,6,7,8,9,9a-hexa-hydro-pyrido[1,2-a]pyrimidin-4-one. | Acta crystallographica. Section E, Structure reports online 20111101 |
2-(1,3-Benzoxazol-2-yl)guanidinium chloride. | Acta crystallographica. Section E, Structure reports online 20111101 |
One-pot syntheses of pseudopteroxazoles from pseudopterosins: a rapid route to non-natural congeners with improved antimicrobial activity. | Journal of natural products 20111028 |
Iodine-catalyzed amination of benzoxazoles: a metal-free route to 2-aminobenzoxazoles under mild conditions. | The Journal of organic chemistry 20111007 |
2-(1,3-Benzoxazol-2-yl)-1-phenyl-ethenyl benzoate. | Acta crystallographica. Section E, Structure reports online 20111001 |
Bioinspired systems for metal-ion sensing: new emissive peptide probes based on benzo[d]oxazole derivatives and their gold and silica nanoparticles. | Inorganic chemistry 20110919 |
On orthogonal and selective activation of glycosyl thioimidates and thioglycosides: application to oligosaccharide assembly. | The Journal of organic chemistry 20110916 |
Benzoxazole-based heterometallic dodecanuclear complex [Dy(III)4Cu(II)8] with single-molecule-magnet behavior. | Inorganic chemistry 20110815 |
1,1,2,2-Tetra-kis(1,3-benzoxazol-2-yl)ethene. | Acta crystallographica. Section E, Structure reports online 20110801 |
Chlorination and ortho-acetoxylation of 2-arylbenzoxazoles. | Organic & biomolecular chemistry 20110721 |
The intrinsic redox reactions of polyamic acid derivatives and their application in hydrogen peroxide sensor. | Biomaterials 20110701 |
Ethyl 1-[2-(1,3-benzoxazol-2-ylsulfan-yl)acet-yl]-4-hy-droxy-2,6-diphenyl-1,2,5,6-tetra-hydro-pyridine-3-carboxyl-ate. | Acta crystallographica. Section E, Structure reports online 20110701 |
Ligand-free CuO nanospindle catalyzed arylation of heterocycle C-H bonds. | The Journal of organic chemistry 20110603 |
Design and synthesis of benzoxazole containing indole analogs as peroxisome proliferator-activated receptor-γ/δ dual agonists. | Bioorganic & medicinal chemistry letters 20110515 |
2-(4-Carbonylphenyl)benzoxazole inhibitors of CETP: attenuation of hERG binding and improved HDLc-raising efficacy. | Bioorganic & medicinal chemistry letters 20110501 |
Design and synthesis of antifungal benzoheterocyclic derivatives by scaffold hopping. | European journal of medicinal chemistry 20110501 |
2-Arylbenzothiazole, benzoxazole and benzimidazole derivatives as fluorogenic substrates for the detection of nitroreductase and aminopeptidase activity in clinically important bacteria. | Bioorganic & medicinal chemistry 20110501 |
Water attack umpolung aromatic systems to release hydrogen. | Inorganic chemistry 20110418 |
Photocatalytic degradation of the fungicide Fenhexamid in aqueous TiO(2) suspensions: identification of intermediates products and reaction pathways. | Chemosphere 20110401 |
Lewis acid catalyzed benzylic C-H bond functionalization of azaarenes: addition to enones. | Organic letters 20110401 |
Polymer supported synthesis of novel benzoxazole linked benzimidazoles under microwave conditions: in vitro evaluation of VEGFR-3 kinase inhibition activity. | Organic & biomolecular chemistry 20110321 |
2-(4-carbonylphenyl)benzoxazole inhibitors of CETP: scaffold design and advancement in HDLc-raising efficacy. | Bioorganic & medicinal chemistry letters 20110315 |
Discovery of potent inhibitors of soluble epoxide hydrolase by combinatorial library design and structure-based virtual screening. | Journal of medicinal chemistry 20110310 |
Pd- and Ni-catalyzed cross-coupling reactions of functionalized organozinc reagents with unsaturated thioethers. | Chemistry (Weinheim an der Bergstrasse, Germany) 20110301 |
Direct transition-metal-free intramolecular C-O bond formation: synthesis of benzoxazole derivatives. | Organic & biomolecular chemistry 20110221 |
Oxazoles revisited: On the nature of binding of benzoxazole and 2-methylbenzoxazole with the zinc and palladium halides. | Dalton transactions (Cambridge, England : 2003) 20110221 |
2-Methyl-1,3-benzoxazol-4-yl diphenyl-phosphinate. | Acta crystallographica. Section E, Structure reports online 20110201 |
Sesquiterpene benzoxazoles and sesquiterpene quinones from the marine sponge Dactylospongia elegans. | Journal of natural products 20110128 |
Spectroscopic studies of intramolecular proton transfer in 2-(4-fluorophenylamino)-5-(2,4-dihydroxybenzeno)-1,3,4-thiadiazole. | Journal of fluorescence 20110101 |
Effect of substitution on the antimycobacterial activity of 2-(substituted benzyl)sulfanyl benzimidazoles, benzoxazoles, and benzothiazoles--a quantitative structure-activity relationship study. | Chemical & pharmaceutical bulletin 20110101 |
Levantilides A and B, 20-membered macrolides from a Micromonospora strain isolated from the Mediterranean deep sea sediment. | Marine drugs 20110101 |
Integrin targeting for tumor optical imaging. | Theranostics 20110101 |
Variations in Mre11/Rad50/Nbs1 status and DNA damage-induced S-phase arrest in the cell lines of the NCI60 panel. | BMC cancer 20110101 |
Biomarkers in Alzheimer's disease. | Frontiers in neurology 20110101 |
Catecholthioether derivatives: preliminary study of in-vitro antimicrobial and antioxidant activities. | Chemical & pharmaceutical bulletin 20110101 |
High-throughput screen for identifying small molecules that target fungal zinc homeostasis. | PloS one 20110101 |
Cnidarians as a source of new marine bioactive compounds--an overview of the last decade and future steps for bioprospecting. | Marine drugs 20110101 |
Synthesis and evaluation of benzoxazole derivatives as 5-lipoxygenase inhibitors. | Bioorganic & medicinal chemistry 20101101 |
Light insensitive silver(I) cyanoximates as antimicrobial agents for indwelling medical devices. | Inorganic chemistry 20101101 |
1,3-Benzoxazole-4-carbonitrile as a novel antifungal scaffold of β-1,6-glucan synthesis inhibitors. | Bioorganic & medicinal chemistry 20101101 |
Design, synthesis and antifungal activity of isosteric analogues of benzoheterocyclic N-myristoyltransferase inhibitors. | European journal of medicinal chemistry 20100901 |
Oxidative cyclization of a phenolic Schiff base and synthesis of a cyclometalated ruthenium nitrosyl complex: photoinduced NO release by visible light. | Inorganic chemistry 20100816 |
Reactions of aromatic heterocycles with uranium alkyl complexes. | Inorganic chemistry 20100802 |
Discovery of aminopyridines substituted with benzoxazole as orally active c-Met kinase inhibitors. | Bioorganic & medicinal chemistry letters 20100715 |
Synthesis, DNA-binding ability and anticancer activity of benzothiazole/benzoxazole-pyrrolo[2,1-c][1,4]benzodiazepine conjugates. | Bioorganic & medicinal chemistry 20100701 |
Excited state intramolecular proton transfer and charge transfer dynamics of a 2-(2'-hydroxyphenyl)benzoxazole derivative in solution. | The journal of physical chemistry. A 20100513 |
Diversity-oriented synthesis of benzimidazole, benzoxazole, benzothiazole and quinazolin-4(3H)-one libraries via potassium persulfate-CuSO4-mediated oxidative coupling reactions of aldehydes in aqueous micelles. | Molecular diversity 20100501 |
Synthesis and characterization of the ligand based on benzoxazole and its transition metal complexes: DNA-binding and antitumor activity. | Journal of inorganic biochemistry 20100501 |
Highly specific substrates of proteinase 3 containing 3-(2-benzoxazol-5-yl)-l-alanine and their application for detection of this enzyme in human serum. | Analytical chemistry 20100501 |
Pd-catalyzed decarboxylative arylation of thiazole, benzoxazole, and polyfluorobenzene with substituted benzoic acids. | Organic letters 20100402 |
2-Amino-aryl-7-aryl-benzoxazoles as potent, selective and orally available JAK2 inhibitors. | Bioorganic & medicinal chemistry letters 20100301 |
Investigation of the photoisomerisation process in four p-benzoxazoyl-substituted stilbenes. | Photochemical & photobiological sciences : Official journal of the European Photochemistry Association and the European Society for Photobiology 20100301 |
Unexpected reactivity of o-nitrosophenol with RCH(2)Br: C-H bond cleavage and annulation to benzoxazoles and benzoxazines (R = Alkynyl). | Organic letters 20100219 |
Photo-controlled Zn(2+) release system with dual binding-sites and turn-on fluorescence. | Physical chemistry chemical physics : PCCP 20100207 |
2-Arylbenzoxazoles as CETP inhibitors: Substitution of the benzoxazole moiety. | Bioorganic & medicinal chemistry letters 20100101 |
(E)-4,4'-Bis(1,3-benzoxazol-2-yl)stilbene at 150 and 375 K. | Acta crystallographica. Section C, Crystal structure communications 20100101 |
Hypericins as potential leads for new therapeutics. | International journal of molecular sciences 20100101 |
In vivo imaging of zebrafish retinal cells using fluorescent coumarin derivatives. | BMC neuroscience 20100101 |
Metabotropic glutamate receptors: potential drug targets for psychiatric disorders. | The open medicinal chemistry journal 20100101 |
Cytotoxic terpene quinones from marine sponges. | Marine drugs 20100101 |
Antibacterial compounds from marine Vibrionaceae isolated on a global expedition. | Marine drugs 20100101 |
Methodology for detecting residual phosphoric acid in polybenzoxazole fibers. | Analytical chemistry 20091201 |
In situ generation and trapping of aryllithium and arylpotassium species by halogen, sulfur, and carbon electrophiles. | The Journal of organic chemistry 20091106 |
In vitro antifungal activity of 2-(2'-hydroxy-5'-aminophenyl)benzoxazole in Candida spp. strains. | Mycoses 20091101 |
Benzoxazole piperidines as selective and potent somatostatin receptor subtype 5 antagonists. | Bioorganic & medicinal chemistry letters 20091101 |
NHC-manganese(i) complexes as carbene transfer agents. | Dalton transactions (Cambridge, England : 2003) 20090921 |
In vitro characterisation of BF227 binding to alpha-synuclein/Lewy bodies. | European journal of pharmacology 20090901 |
2-(1,3-Benzoxazol-2-ylsulfan-yl)-1-phenyl-ethanone. | Acta crystallographica. Section E, Structure reports online 20090901 |
A ratiometric fluorescent sensor for zinc ions based on covalently immobilized derivative of benzoxazole. | Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20090815 |
Discovery of leukotriene A4 hydrolase inhibitors using metabolomics biased fragment crystallography. | Journal of medicinal chemistry 20090813 |
Classification of 5-HT(1A) receptor ligands on the basis of their binding affinities by using PSO-Adaboost-SVM. | International journal of molecular sciences 20090801 |
Antitumor compounds from marine actinomycetes. | Marine drugs 20090601 |
Preparation and in vitro evaluation of benzylsulfanyl benzoxazole derivatives as potential antituberculosis agents. | European journal of medicinal chemistry 20090501 |
The 'Corey's reagent,' 3,5-di-tert-butyl-1,2-benzoquinone, as a modifying agent in the synthesis of fluorescent and double-headed nucleosides. | Nucleosides, nucleotides & nucleic acids 20090501 |
Nickel-catalyzed biaryl coupling of heteroarenes and aryl halides/triflates. | Organic letters 20090416 |
Modulating the near-infrared luminescence of neodymium and ytterbium complexes with tridentate ligands based on benzoxazole-substituted 8-hydroxyquinolines. | Inorganic chemistry 20090406 |
Unexpected orthogonality of S-benzoxazolyl and S-thiazolinyl glycosides: application to expeditious oligosaccharide assembly. | Organic letters 20090219 |
Identification of a series of benzoxazoles as potent 5-HT6 ligands. | Bioorganic & medicinal chemistry letters 20090215 |
Caboxamycin, a new antibiotic of the benzoxazole family produced by the deep-sea strain Streptomyces sp. NTK 937. | The Journal of antibiotics 20090201 |
Trifluoromethoxy-benzylated ligands improve amyloid detection in the brain using (19)F magnetic resonance imaging. | Neuroscience research 20090101 |
Efficient synthesis of an alpha(2,9) trisialic acid by one-pot glycosylation and polymer-assisted deprotection. | Organic letters 20081218 |
5-tert-Butyl-2-[5-(5-tert-butyl-1,3-benzoxazol-2-yl)-2-thien-yl]-1,3-benzoxazole. | Acta crystallographica. Section E, Structure reports online 20081201 |
Focusing and stabilization of bis-intercalating dye-DNA complexes for high-sensitive CE-LIF DNA analysis. | Electrophoresis 20081101 |
Nataxazole, a new benzoxazole derivative with antitumor activity produced by Streptomyces sp. Tü 6176. | The Journal of antibiotics 20081101 |
Structure-activity relationships of novel heteroaryl-acrylonitriles as cytotoxic and antibacterial agents. | European journal of medicinal chemistry 20080901 |
Synthesis and biological properties of benzothiazole, benzoxazole, and chromen-4-one analogues of the potent antitumor agent 2-(3,4-dimethoxyphenyl)-5-fluorobenzothiazole (PMX 610, NSC 721648). | Journal of medicinal chemistry 20080828 |
Synthesis of new arylpiperazinylalkylthiobenzimidazole, benzothiazole, or benzoxazole derivatives as potent and selective 5-HT1A serotonin receptor ligands. | Journal of medicinal chemistry 20080814 |
Identification of a potent, selective, and orally active leukotriene a4 hydrolase inhibitor with anti-inflammatory activity. | Journal of medicinal chemistry 20080724 |
Toward prediction of alkane/water partition coefficients. | Journal of medicinal chemistry 20080710 |
Iron-catalyzed intramolecular o-arylation: synthesis of 2-aryl benzoxazoles. | Organic letters 20080703 |
Synthesis, potent anti-staphylococcal activity and QSARs of some novel 2-anilinobenzazoles. | European journal of medicinal chemistry 20080701 |
Synthesis of new carbon-11 labeled benzoxazole derivatives for PET imaging of 5-HT(3) receptor. | European journal of medicinal chemistry 20080701 |
2-(4-Amino-phen-yl)-1,3-benzoxazole. | Acta crystallographica. Section E, Structure reports online 20080701 |
Catalytic aza-Wittig cyclizations for heteroaromatic synthesis. | Organic letters 20080619 |
Gelation-induced fluorescence enhancement of benzoxazole-based organogel and its naked-eye fluoride detection. | Chemical communications (Cambridge, England) 20080528 |
Copper-catalyzed domino annulation approaches to the synthesis of benzoxazoles under microwave-accelerated and conventional thermal conditions. | The Journal of organic chemistry 20080502 |
Intramolecular exciplexes based on benzoxazole: photophysics and applications as fluorescent cation sensors. | Photochemical & photobiological sciences : Official journal of the European Photochemistry Association and the European Society for Photobiology 20080501 |
The dichotomy in the DNA-binding behaviour of ruthenium(II) complexes bearing benzoxazole and benzothiazole groups. | Journal of inorganic biochemistry 20080401 |
Application of glycosyl thioimidates in solid-phase oligosaccharide synthesis. | The Journal of organic chemistry 20080307 |
5-Fluorotryptamine is a partial agonist at 5-HT3 receptors, and reveals that size and electronegativity at the 5 position of tryptamine are critical for efficient receptor function. | European journal of pharmacology 20080212 |
Evaluation of metal-mediated DNA binding of benzoxazole ligands by electrospray ionization mass spectrometry. | Journal of the American Society for Mass Spectrometry 20080201 |
Deprotonative metalation of five-membered aromatic heterocycles using mixed lithium-zinc species. | The Journal of organic chemistry 20080104 |
Comparative in vitro and ex vivo activities of selected inhibitors of transthyretin aggregation: relevance in drug design. | The Biochemical journal 20071115 |
Rapid and efficient synthesis of 4-substituted pyrazol-5-one under microwave irradiation in solvent-free conditions. | Archiv der Pharmazie 20071101 |
Design, synthesis, and evaluation of orally active benzimidazoles and benzoxazoles as vascular endothelial growth factor-2 receptor tyrosine kinase inhibitors. | Journal of medicinal chemistry 20070906 |
Respiratory syncytial virus fusion inhibitors. Part 6: an examination of the effect of structural variation of the benzimidazol-2-one heterocycle moiety. | Bioorganic & medicinal chemistry letters 20070901 |
[Degradation mechanism and efficiency of organic pollutants of landfill leachate in different redox zones]. | Huan jing ke xue= Huanjing kexue 20070901 |
S-benzoxazolyl as a stable protecting moiety and a potent anomeric leaving group in oligosaccharide synthesis. | The Journal of organic chemistry 20070831 |
Design, synthesis, and in vitro evaluation of carbamate derivatives of 2-benzoxazolyl- and 2-benzothiazolyl-(3-hydroxyphenyl)-methanones as novel fatty acid amide hydrolase inhibitors. | Journal of medicinal chemistry 20070823 |
Design and synthesis of highly potent and selective human peroxisome proliferator-activated receptor alpha agonists. | Bioorganic & medicinal chemistry letters 20070815 |
Degenerate four-wave mixing in solution by cubic response theory and the polarizable continuum model. | The journal of physical chemistry. B 20070802 |
Regulatory molecules for the 5-HT3 receptor ion channel gating system. | Bioorganic & medicinal chemistry 20070515 |
Potential sialyltransferase inhibitors based on neuraminyl substitution by hetaryl rings. | Carbohydrate research 20070226 |
Synthesis and mass spectrometry of benzoxazoline, dimethyloxazoline and 4-phenyloxazoline derivatives of polyunsaturated fatty acids. | Rapid communications in mass spectrometry : RCM 20070101 |
Fluorescence characteristics and photostability of benzoxazole derived donor-acceptor dyes in constrained media. | Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20061001 |
Design of new benzoxazole-2-thione-derived inhibitors of Streptococcus pneumoniae hyaluronan lyase: structure of a complex with a 2-phenylindole. | Glycobiology 20060801 |
Computational studies of nucleophilic attack and protonation of electron-deficient benzoheterocycle triosmium clusters. | Inorganic chemistry 20060626 |
Synthesis, anti-inflammatory, analgesic and kinase (CDK-1, CDK-5 and GSK-3) inhibition activity evaluation of benzimidazole/benzoxazole derivatives and some Schiff's bases. | Bioorganic & medicinal chemistry 20060601 |
Thermal reactions of benzoxazole. Single pulse shock tube experiments and quantum chemical calculations. | The journal of physical chemistry. A 20060406 |
3D-QSAR study on heterocyclic topoisomerase II inhibitors using CoMSIA. | SAR and QSAR in environmental research 20060401 |
Parallel synthesis of a library of benzoxazoles and benzothiazoles using ligand-accelerated copper-catalyzed cyclizations of ortho-halobenzanilides. | The Journal of organic chemistry 20060303 |
Synthesis and biological evaluation of novel heterocyclic quinones as inhibitors of the dual specificity protein phosphatase CDC25C. | Bioorganic & medicinal chemistry letters 20060101 |
3D-QSAR analysis on benzazole derivatives as eukaryotic topoisomerase II inhibitors by using comparative molecular field analysis method. | Bioorganic & medicinal chemistry 20051201 |
Identification of the structural requirements of the receptor-binding affinity of diphenolic azoles to estrogen receptors alpha and beta by three-dimensional quantitative structure-activity relationship and structure-activity relationship analysis. | Journal of medicinal chemistry 20051201 |
Differential solvation and tautomer stability of a model base pair within the minor and major grooves of DNA. | Journal of the American Chemical Society 20051109 |
Orally active benzoxazole derivative as 5-HT3 receptor partial agonist for treatment of diarrhea-predominant irritable bowel syndrome. | Journal of medicinal chemistry 20051103 |
Synthesis of some novel benzoxazole derivatives as anticancer, anti-HIV-1 and antimicrobial agents. | European journal of medicinal chemistry 20050901 |
Deprotonation of benzoxazole and oxazole using lithium magnesates. | The Journal of organic chemistry 20050624 |
Anthryl-substituted heterocycles as acid-sensitive fluorescence probes. | The Journal of organic chemistry 20050513 |
Synthesis and characterisation of the first transition metal complex of zoxazolamine (2-amino-5-chlorobenzoxazole): the X-ray crystal structure determination of [ZnCl2(eta 1-Nbenzoxazole-2-amino-5-chlorobenzoxazole)2]. | Journal of inorganic biochemistry 20050201 |
Effects of positional and geometrical isomerism on the biological activity of some novel oxazolidinones. | Bioorganic & medicinal chemistry letters 20050117 |
[Toxicity of some benzothiazole and benzoxazole derivatives having an anthelminthic action]. | Meditsinskaia parazitologiia i parazitarnye bolezni 20050101 |
Evaluation of complexes of DNA duplexes and novel benzoxazoles or benzimidazoles by electrospray ionization mass spectrometry. | Journal of the American Society for Mass Spectrometry 20041101 |
Synthesis and biological activity of benzoxazole containing thiazolidinedione derivatives. | Archives of pharmacal research 20041101 |
Estrone formate: a novel type of irreversible inhibitor of human steroid sulfatase. | Bioorganic & medicinal chemistry letters 20041004 |
Determination of serotonin, noradrenaline, dopamine and their metabolites in rat brain extracts and microdialysis samples by column liquid chromatography with fluorescence detection following derivatization with benzylamine and 1,2-diphenylethylenediamine. | Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20040805 |
Study on photochromic diarylethene with phenolic Schiff base: preparation and photochromism of diarylethene with benzoxazole. | The Journal of organic chemistry 20040723 |
Synthesis and structure-activity relationship of novel benzoxazole derivatives as melatonin receptor agonists. | Bioorganic & medicinal chemistry letters 20040716 |
Bioisosteric replacement of anilide with benzoxazole: potent and orally bioavailable antagonists of VLA-4. | Bioorganic & medicinal chemistry letters 20040503 |
Syntheses and DNA-binding studies of a series of unsymmetrical cyanine dyes: structural influence on the degree of minor groove binding to natural DNA. | Bioorganic & medicinal chemistry 20040501 |
Some fused heterocyclic compounds as eukaryotic topoisomerase II inhibitors. | Biochemical and biophysical research communications 20040430 |
Aminopyridine-benzoxanthene enantioselective receptor for sulfonylamino acids. | Organic letters 20040401 |
Design and synthesis of benzoxazole derivatives as novel melatoninergic ligands. | Bioorganic & medicinal chemistry letters 20040308 |
Vibrational analysis of structure activity relationships (SAR) in molecular binding. | Applied spectroscopy 20040301 |
Emission ratiometric imaging of intracellular zinc: design of a benzoxazole fluorescent sensor and its application in two-photon microscopy. | Journal of the American Chemical Society 20040128 |
Discovery of novel modulators of metabotropic glutamate receptor subtype-5. | Bioorganic & medicinal chemistry 20040102 |
[Investigation of the trichinellocidal activity of the agents from a series of benzthiazole and benzoxazole]. | Meditsinskaia parazitologiia i parazitarnye bolezni 20040101 |
[Biologically active benzoxazoles]. | Ceska a Slovenska farmacie : casopis Ceske farmaceuticke spolecnosti a Slovenske farmaceuticke spolecnosti 20031101 |
A new approach to the synthesis of benzothiazole, benzoxazole, and pyridine nucleosides as potential antitumor agents. | Nucleosides, nucleotides & nucleic acids 20031101 |
Cobalt-catalyzed arylation of azole heteroarenes via direct C-H bond functionalization. | Organic letters 20031002 |
Simultaneous determination of 5-hydroxyindoles and catechols by high-performance liquid chromatography with fluorescence detection following derivatization with benzylamine and 1,2-diphenylethylenediamine. | Journal of chromatography. A 20030919 |
Synthesis and activity of novel benzoxazole derivatives of mannopeptimycin glycopeptide antibiotics. | Bioorganic & medicinal chemistry letters 20030804 |
Synthesis and pharmacological characterization of a new benzoxazole derivative as a potent 5-HT3 receptor agonist. | Bioorganic & medicinal chemistry 20030703 |
A procedure for preparing oxazolines of highly unsaturated fatty acids to determine double bond positions by mass spectrometry. | Journal of lipid research 20030501 |
Scope and mechanism of palladium-catalyzed amination of five-membered heterocyclic halides. | The Journal of organic chemistry 20030404 |
Design, synthesis and biological evaluation of benzimidazole/benzothiazole and benzoxazole derivatives as cyclooxygenase inhibitors. | Bioorganic & medicinal chemistry letters 20030224 |
Simultaneous determination of norepinephrine, serotonin, and 5-hydroxyindole-3-acetic acid in microdialysis samples from rat brain by microbore column liquid chromatography with fluorescence detection following derivatization with benzylamine. | Analytical biochemistry 20030115 |
Photophysics and spectroscopic properties of 3-benzoxazol-2-yl-chromen-2-one. | Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20030115 |
Synthesis and insecticidal activity of benzoheterocyclic analogues of N'-benzoyl-N-(tert-butyl)benzohydrazide: Part 1. Design of benzoheterocyclic analogues. | Pest management science 20030101 |
Synthesis and evaluation of anticancer benzoxazoles and benzimidazoles related to UK-1. | Bioorganic & medicinal chemistry 20021201 |
Heterocyclic benzazole derivatives with antimycobacterial in vitro activity. | Bioorganic & medicinal chemistry letters 20021118 |
Metal chelation aptitudes of bis(o-azaheteroaryl)methanes as tuned by heterocycle charge demands. | The Journal of organic chemistry 20020809 |
Synthesis of macrocyclic, potential protease inhibitors using a generic scaffold. | The Journal of organic chemistry 20020712 |
II. Synthesis and biological evaluation of some bioisosteres and congeners of the antitumor agent, 2-(4-[(7-chloro-2-quinoxalinyl)oxy]phenoxy)propionic acid (XK469). | Journal of medicinal chemistry 20020704 |
Synthesis and microbiological activity of some N-(2-hydroxy-4-substitutedphenyl)benzamides, phenylacetamides and furamides as the possible metabolites of antimicrobial active benzoxazoles. | Farmaco (Societa chimica italiana : 1989) 20020601 |
Synthesis and antimicrobial activity of some novel 2-(p-substituted-phenyl)-5-substituted-carbonylaminobenzoxazoles. | Farmaco (Societa chimica italiana : 1989) 20020301 |
Silacyclic derivatives of heteroaromatic sulfides as selective cholesterol level lowering and vasodilating agents. | Metal-based drugs 20020101 |
Application of 2-(3,5,6-trifluoro-2-hydroxy-4-methoxyphenyl)benzoxazole and -benzothiazole to fluorescent probes sensing pH and metal cations. | The Journal of organic chemistry 20011102 |
Iminocoumarin-based low affinity fluorescent Ca2+ indicators excited with visible light. | Cell calcium 20011101 |
Catalytic asymmetric cyclopropanation of heteroaryldiazoacetates. | The Journal of organic chemistry 20011005 |
Catalytic turnover of benzylamine by a model for the lysine tyrosylquinone (LTQ) cofactor of lysyl oxidase. | Journal of the American Chemical Society 20011003 |
2-benzoxazolyl and 2-benzimidazolyl hydrazones derived from 2-acetylpyridine: a novel class of antitumor agents. | International journal of cancer 20011001 |
Design, synthesis, and evaluation of alpha-ketoheterocycles as class C beta-lactamase inhibitors. | Bioorganic & medicinal chemistry 20010801 |
Synthesis, structure-activity relationships, and pharmacokinetic profiles of nonpeptidic alpha-keto heterocycles as novel inhibitors of human chymase. | Journal of medicinal chemistry 20010412 |
Catalytic turnover of substrate benzylamines by the quinone-dependent plasma amine oxidase leads to H2O2-dependent inactivation: evidence for generation of a cofactor-derived benzoxazole. | Biochemistry 20010123 |
AJI9561, a new cytotoxic benzoxazole derivative produced by Streptomyces sp. | The Journal of antibiotics 20010101 |
Interaction of cyanine dyes with nucleic acids. XXI. Arguments for half-intercalation model of interaction. | Biopolymers 20010101 |
Solid-phase synthesis of benzoxazoles from 3-nitrotyrosine. | Journal of combinatorial chemistry 20010101 |