Low-temperature loading of Cu+ species over porous metal-organic frameworks (MOFs) and adsorptive desulfurization with Cu+-loaded MOFs.

Journal of hazardous materials 20121030

Toluene dioxygenase-catalyzed cis-dihydroxylation of benzo[b]thiophenes and benzo[b]furans: synthesis of benzo[b]thiophene 2,3-oxide.

Organic & biomolecular chemistry 20120928

Synthesis and Anti-hyperlipidemic Activity of 3H-benzo [4, 5] thieno [2, 3-d] [1, 2, 3] triazin-4-ones: Possible Mechanism of Altered Lipid Metabolism.

Oman medical journal 20120901

C3-heteroaroyl cannabinoids as photolabeling ligands for the CB2 cannabinoid receptor.

Bioorganic & medicinal chemistry letters 20120815

Efficient synthesis and 5-LOX/COX-inhibitory activity of some 3-hydroxybenzo[b]thiophene-2-carboxylic acid derivatives.

Bioorganic & medicinal chemistry letters 20120801

Symmetrical approach of spiro-pyrazolidinediones as acetyl-CoA carboxylase inhibitors.

Bioorganic & medicinal chemistry letters 20120715

Management of singlet and triplet excitons in a single emission layer: a simple approach for a high-efficiency fluorescence/phosphorescence hybrid white organic light-emitting device.

Advanced materials (Deerfield Beach, Fla.) 20120703

Novel substituted benzothiophene and thienothiophene carboxanilides and quinolones: synthesis, photochemical synthesis, DNA-binding properties, antitumor evaluation and 3D-derived QSAR analysis.

Journal of medicinal chemistry 20120614

Design, synthesis, and structure-activity relationships of novel spiro-piperidines as acetyl-CoA carboxylase inhibitors.

Bioorganic & medicinal chemistry letters 20120601

Preliminary antifungal and cytotoxic evaluation of synthetic cycloalkyl[b]thiophene derivatives with PLS-DA analysis.

Acta pharmaceutica (Zagreb, Croatia) 20120601

Discovery of Ipragliflozin (ASP1941): a novel C-glucoside with benzothiophene structure as a potent and selective sodium glucose co-transporter 2 (SGLT2) inhibitor for the treatment of type 2 diabetes mellitus.

Bioorganic & medicinal chemistry 20120515

Modulation of proteasome machinery by natural and synthetic analogues of the marine bioactive compound petrosaspongiolide M.

Chembiochem : a European journal of chemical biology 20120507

Protein tyrosine phosphatase 1B inhibitors: a molecular level legitimate approach for the management of diabetes mellitus.

Medicinal research reviews 20120501

Synthesis and structure-activity relationship studies of 3-biaryl-8-oxabicyclo[3.2.1]octane-2-carboxylic acid methyl esters.

Bioorganic & medicinal chemistry 20120415

Synthesis and biological evaluation of novel small non-peptidic HIV-1 PIs: the benzothiophene ring as an effective moiety.

Bioorganic & medicinal chemistry letters 20120415

Highly efficient extraction and oxidative desulfurization system using Na7H2LaW10O36⋅32 H2O in [bmim]BF4 at room temperature.

Chemistry (Weinheim an der Bergstrasse, Germany) 20120410

Binding affinity prediction for ligands and receptors forming tautomers and ionization species: inhibition of mitogen-activated protein kinase-activated protein kinase 2 (MK2).

Journal of medicinal chemistry 20120308

Toward the accurate analysis of C1-C4 polycyclic aromatic sulfur heterocycles.

Analytical chemistry 20120306

(E)-N-(1-Benzothio-phen-3-yl-methyl-idene)-2,6-dimethyl-aniline.

Acta crystallographica. Section E, Structure reports online 20120301

(Z)-3-(1H-Indol-3-yl)-2-(3,4,5-tri-methoxy-phen-yl)acrylonitrile.

Acta crystallographica. Section E, Structure reports online 20120301

(Z)-3-(1-Benzofuran-2-yl)-2-(3,4,5-tri-meth-oxy-phen-yl)acrylonitrile.

Acta crystallographica. Section E, Structure reports online 20120301

Oxidative desulfurization of benzothiophene and thiophene with WOx/ZrO2 catalysts: effect of calcination temperature of catalysts.

Journal of hazardous materials 20120227

Synthesis, docking studies and biological evaluation of benzo[b]thiophen-2-yl-3-(4-arylpiperazin-1-yl)-propan-1-one derivatives on 5-HT1A serotonin receptors.

Molecules (Basel, Switzerland) 20120203

(E)-3-[(2-Methyl-4-nitro-phen-yl)imino-meth-yl]-1-benzothio-phene.

Acta crystallographica. Section E, Structure reports online 20120201

Bacterial dioxygenase- and monooxygenase-catalysed sulfoxidation of benzo[b]thiophenes.

Organic & biomolecular chemistry 20120128

Remarkable adsorption capacity of CuCl2-loaded porous vanadium benzenedicarboxylate for benzothiophene.

Angewandte Chemie (International ed. in English) 20120127

Synthesis and characterization of nonsymmetric cyclopentene-based dithienylethenes.

The Journal of organic chemistry 20120106

Argentation chromatography for the separation of polycyclic aromatic compounds according to ring number.

Journal of chromatography. A 20120106

Gynecologic effects of arzoxifene in postmenopausal women with osteoporosis or low bone mass.

Menopause (New York, N.Y.) 20120101

Comparative modeling of DszC, an enzyme in biodesulfurization, and performing in silico point mutation for increasing tendency to oil.

Bioinformation 20120101

Detection of horizontal gene transfers from phylogenetic comparisons.

International journal of evolutionary biology 20120101

Carotenoids play a positive role in the degradation of heterocycles by Sphingobium yanoikuyae.

PloS one 20120101

Investigation on the binding mode of benzothiophene analogues as potent factor IXa (FIXa) inhibitors in thrombosis by CoMFA, docking and molecular dynamic studies.

Journal of enzyme inhibition and medicinal chemistry 20111201

Benzothiophene carboxamide derivatives as inhibitors of Plasmodium falciparum enoyl-ACP reductase.

IUBMB life 20111201

Benzothiophene carboxamide derivatives as novel antimalarials.

IUBMB life 20111201

Pharmacophore-based discovery of FXR-agonists. Part II: identification of bioactive triterpenes from Ganoderma lucidum.

Bioorganic & medicinal chemistry 20111115

Importance of heterocylic aromatic compounds in monitored natural attenuation for coal tar contaminated aquifers: A review.

Journal of contaminant hydrology 20111101

Synthesis of benzothiophene derivatives by Pd-catalyzed or radical-promoted heterocyclodehydration of 1-(2-mercaptophenyl)-2-yn-1-ols.

The Journal of organic chemistry 20111021

Conformationally constrained farnesoid X receptor (FXR) agonists: alternative replacements of the stilbene.

Bioorganic & medicinal chemistry letters 20111015

A practical, one-pot synthesis of highly substituted thiophenes and benzo[b]thiophenes from bromoenynes and o-alkynylbromobenzenes.

Organic letters 20111007

Breast cancer medications and vision: effects of treatments for early-stage disease.

Current eye research 20111001

(E)-2-[1-(1-Benzothio-phen-2-yl)ethyl-idene]-N-phenyl-hydrazinecarboxamide.

Acta crystallographica. Section E, Structure reports online 20111001

Design and synthesis of 1,3-biarylsulfanyl derivatives as new anti-breast cancer agents.

Bioorganic & medicinal chemistry 20110915

Novel cyclopalladated imino-thiophenes: synthesis and reactivity toward alkynes and carbon monoxide.

Inorganic chemistry 20110905

Structural features determining the intestinal epithelial permeability and efflux of novel HIV-1 protease inhibitors.

Journal of pharmaceutical sciences 20110901

Reprint of 'effect of carbohydrate amino group modifications on the cytotoxicity of glycosylated 2-phenyl-benzo[b]thiophenes and 2-phenyl-benzo[b]furans' [Bioorg. Med. Chem. Lett. 21 (2011) 2591-2596].

Bioorganic & medicinal chemistry letters 20110901

Synthesis, structure and cytotoxicity of 3-C, N, S, Se substituted benzo[b]selenophene derivatives.

European journal of medicinal chemistry 20110801

Benzimidazolone as potent chymase inhibitor: modulation of reactive metabolite formation in the hydrophobic (P1) region.

Bioorganic & medicinal chemistry letters 20110801

Palladium-catalyzed three-component domino reaction for the preparation of benzo[b]thiophene and related compounds.

Organic & biomolecular chemistry 20110721

Multimetal Fischer carbene complexes of Group VI transition metals: synthesis, structure and substituent effect investigation.

Dalton transactions (Cambridge, England : 2003) 20110707

7-Methyl-5,6,7,8-tetra-hydro-1-benzo-thieno[2,3-d]pyrimidin-4-amine.

Acta crystallographica. Section E, Structure reports online 20110701

3'-(4-Meth-oxy-phen-yl)-4'-phenyl-3H,4'H-spiro-[1-benzothio-phene-2,5'-isoxazol]-3-one.

Acta crystallographica. Section E, Structure reports online 20110701

Effect of carbohydrate amino group modifications on the cytotoxicity of glycosylated 2-phenyl-benzo[b]thiophenes and 2-phenyl-benzo[b]furans.

Bioorganic & medicinal chemistry letters 20110501

5-Methyl-phenanthro[2,3-b]thio-phene.

Acta crystallographica. Section E, Structure reports online 20110501

Novel benzo[b]thiophene derivatives as new potential antidepressants with rapid onset of action.

Journal of medicinal chemistry 20110428

Ring-closure reactions of 1,2-diaza-4,5-benzoheptatrienyl metal compounds: experiment and theory.

The Journal of organic chemistry 20110401

Synthesis, evaluation and structural studies of antiproliferative tubulin-targeting azetidin-2-ones.

Bioorganic & medicinal chemistry 20110401

2-Phenyl-8,9,10,11-tetra-hydro-1-benzo-thieno[3,2-e][1,2,4]triazolo[1,5-c]pyrimidine.

Acta crystallographica. Section E, Structure reports online 20110401

Carbon-sulfur bond cleavage and hydrodesulfurization of thiophenes by tungsten.

Journal of the American Chemical Society 20110323

Oxidative desulfurization of fuels catalyzed by Fenton-like ionic liquids at room temperature.

ChemSusChem 20110321

Synthesis, photophysical characterization, and enzymatic incorporation of a microenvironment-sensitive fluorescent uridine analog.

Organic letters 20110304

2-Amino-6-methyl-4,5,6,7-tetra-hydro-1-benzothio-phene-3-carbonitrile.

Acta crystallographica. Section E, Structure reports online 20110301

Ruthenium-catalyzed oxidative vinylation of heteroarene carboxylic acids with alkenes via regioselective C-H bond cleavage.

Organic letters 20110218

Photon-quantitative reaction of a dithiazolylarylene in solution.

Angewandte Chemie (International ed. in English) 20110211

Tetrahydrobenzothiophene derivatives: conformationally restricted inhibitors of type II dehydroquinase.

ChemMedChem 20110207

Remarkable adsorptive performance of a metal-organic framework, vanadium-benzenedicarboxylate (MIL-47), for benzothiophene.

Chemical communications (Cambridge, England) 20110128

Solution-processable organic single crystals with bandlike transport in field-effect transistors.

Advanced materials (Deerfield Beach, Fla.) 20110125

The identification of substituted benzothiophene derivatives as PGE(2) subtype 4 receptor antagonists: From acid to non-acid.

Bioorganic & medicinal chemistry letters 20110115

Benzothieno[3,2-b]quinolinium and 3-(phenylthio)quinolinium compounds: Synthesis and evaluation against opportunistic fungal pathogens.

Bioorganic & medicinal chemistry 20110101

Synthesis of benzothiophene carboxamide derivatives and their pharmacological evaluation as potent antihypertriglyceridemic agents in rats.

Zeitschrift fur Naturforschung. C, Journal of biosciences 20110101

Desulfurization of dibenzothiophene (DBT) by a novel strain Lysinibacillus sphaericus DMT-7 isolated from diesel contaminated soil.

Journal of environmental sciences (China) 20110101

Conformational toggling of yeast iso-1-cytochrome C in the oxidized and reduced states.

PloS one 20110101

Raloxifene and desmethylarzoxifene block estrogen-induced malignant transformation of human breast epithelial cells.

PloS one 20110101

Potent and selective 5-LO inhibitor bearing benzothiophene pharmacophore: discovery of MK-5286.

Bioorganic & medicinal chemistry letters 20101215

Crystal structure prediction and isostructurality of three small molecules.

Chemistry (Weinheim an der Bergstrasse, Germany) 20101108

Synthesis of regioselectively functionalized benzo[b]thiophenes by combined ortho-lithiation-halocyclization strategies.

The Journal of organic chemistry 20101105

Indole- and benzothiophene-based histamine H3 antagonists.

Bioorganic & medicinal chemistry letters 20101101

Synthesis of benzofuran, benzothiophene, and benzothiazole-based thioamides and their evaluation as K(ATP) channel openers.

ChemMedChem 20101004

Pharmacophore mapping of arylamino-substituted benzo[b]thiophenes as free radical scavengers.

Journal of molecular modeling 20101001

Electrochromic thin films from a redox active diarylethene by electrochemical polymerization.

Journal of nanoscience and nanotechnology 20101001

2-Amino-7-oxo-4,5,6,7-tetra-hydro-1-benzothio-phene-3-carbonitrile.

Acta crystallographica. Section E, Structure reports online 20101001

Synthesis, electrochemical, and optical properties of new fluorescent, substituted thieno[3,2-b][1]benzothiophenes.

Journal of fluorescence 20100901

Rotary molecular motors: a large increase in speed through a small change in design.

The Journal of organic chemistry 20100806

Ladder-type pi-conjugated 4-hetero-1,4-dihydrophosphinines: a structure-property study.

Chemistry, an Asian journal 20100802

Benzo[b]thiophene-6-carboxamide 1,1-dioxides: inhibitors of human cancer cell growth at nanomolar concentrations.

Bioorganic & medicinal chemistry 20100801

Di(hetero)arylamines in the benzo[b]thiophene series as novel potent antioxidants.

Drug discoveries & therapeutics 20100801

Polymer-bound oxidovanadium(IV) and dioxidovanadium(V) complexes as catalysts for the oxidative desulfurization of model fuel diesel.

Inorganic chemistry 20100719

QSAR analysis of antitumor active amides and quinolones from thiophene series.

International journal of pharmaceutics 20100715

Synthesis and characterization of selective dopamine D2 receptor antagonists. 2. Azaindole, benzofuran, and benzothiophene analogs of L-741,626.

Bioorganic & medicinal chemistry 20100715

Substituted 2-(3',4',5'-trimethoxybenzoyl)-benzo[b]thiophene derivatives as potent tubulin polymerization inhibitors.

Bioorganic & medicinal chemistry 20100715

Toward the discovery of new agents able to inhibit the expression of microsomal prostaglandin E synthase-1 enzyme as promising tools in drug development.

Chemical biology & drug design 20100701

New cyclopalladated benzothiophenes: a catalyst precursor for the Suzuki coupling of deactivated aryl chlorides.

Organic & biomolecular chemistry 20100628

Solution-processable flower-shaped hierarchical structures: self-assembly, formation, and state transition of biomimetic superhydrophobic surfaces.

Chemistry (Weinheim an der Bergstrasse, Germany) 20100625

Ester-directed regioselective borylation of heteroarenes catalyzed by a silica-supported iridium complex.

The Journal of organic chemistry 20100604

A benzothiophene inhibitor of mitogen-activated protein kinase-activated protein kinase 2 inhibits tumor necrosis factor alpha production and has oral anti-inflammatory efficacy in acute and chronic models of inflammation.

The Journal of pharmacology and experimental therapeutics 20100601

Benzothiophene containing Rho kinase inhibitors: Efficacy in an animal model of glaucoma.

Bioorganic & medicinal chemistry letters 20100601

3-(4-Methoxy-benz-yl)-1-benzothio-phene.

Acta crystallographica. Section E, Structure reports online 20100601

One-pot synthesis of amine-substituted aryl sulfides and benzo[b]thiophene derivatives.

Organic letters 20100521

Photochromism of diarylethene molecules and crystals.

Proceedings of the Japan Academy. Series B, Physical and biological sciences 20100511

Facile oxidation of electron-poor benzo[b]thiophenes to the corresponding sulfones with an aqueous solution of H2O2 and P2O5.

Chemical communications (Cambridge, England) 20100407

The effect of substituted thiophene and benzothiophene derivates on PPARgamma expression and glucose metabolism.

Journal of enzyme inhibition and medicinal chemistry 20100401

Synthesis and study of some new 1,3-isoindoledione derivatives as potential antibacterial agents.

European journal of medicinal chemistry 20100401

Novel benzothiophene H1-antihistamines for the treatment of insomnia.

Bioorganic & medicinal chemistry letters 20100401

1-(Phenyl-sulfon-yl)benzo[1,2:2',3']thieno[5',4'-b]carbazole.

Acta crystallographica. Section E, Structure reports online 20100401

Diverse methyl sulfone-containing benzo[b]thiophene library via iodocyclization and palladium-catalyzed coupling.

Journal of combinatorial chemistry 20100308

Dopamine D3 receptor selective ligands with varying intrinsic efficacies at adenylyl cyclase inhibition and mitogenic signaling pathways.

Synapse (New York, N.Y.) 20100301

Fragment-based screen against HIV protease.

Chemical biology & drug design 20100301

Substituted benzothiophene or benzofuran derivatives as a novel class of bone morphogenetic protein-2 up-regulators: synthesis, structure-activity relationships, and preventive bone loss efficacies in senescence accelerated mice (SAMP6) and ovariectomized rats.

Journal of medicinal chemistry 20100225

Structure based drug design: development of potent and selective factor IXa (FIXa) inhibitors.

Journal of medicinal chemistry 20100225

Studies of benzothiophene template as potent factor IXa (FIXa) inhibitors in thrombosis.

Journal of medicinal chemistry 20100225

Synthesis, characterization and biological activities of some new benzo[b]thiophene derivatives.

European journal of medicinal chemistry 20100201

Raloxifene inhibits bone loss and improves bone strength through an Opg-independent mechanism.

Endocrine 20100201

Modulation on C- and N-terminal moieties of a series of potent and selective linear tachykinin NK(2) receptor antagonists.

ChemMedChem 20100101

Immunogenetics and the Pathological Mechanisms of Human T-Cell Leukemia VirusType 1- (HTLV-1-)Associated Myelopathy/Tropical Spastic Paraparesis (HAM/TSP).

Interdisciplinary perspectives on infectious diseases 20100101

Novel protein kinase D inhibitors cause potent arrest in prostate cancer cell growth and motility.

BMC chemical biology 20100101

QSAR studies of benzofuran/benzothiophene biphenyl derivatives as inhibitors of PTPase-1B.

Journal of pharmacy & bioallied sciences 20100101

As many as six tandem reactions in one step! Unprecedented formation of highly functionalized benzothiophenes.

Chemical communications (Cambridge, England) 20091214

Ethyl 2-(3,3-dibutyl-thio-ureido)-4,5,6,7-tetra-hydro-benzo[b]thio-phene-3-carboxyl-ate.

Acta crystallographica. Section E, Structure reports online 20091201

Domino palladium-catalyzed Heck-intermolecular direct arylation reactions.

Organic letters 20091015

Synthesis and evaluation of benzo[b]thiophene derivatives as inhibitors of alkaline phosphatases.

Bioorganic & medicinal chemistry 20091015

Intramolecular cross-coupling of gem-dibromoolefins: a mild approach to 2-bromo benzofused heterocycles.

Chemical communications (Cambridge, England) 20090921

Facile C-S, S-H, and S-S bond cleavage using a nickel(0) NHC complex.

Dalton transactions (Cambridge, England : 2003) 20090921

Characterization of novel selective H1-antihistamines for clinical evaluation in the treatment of insomnia.

Journal of medicinal chemistry 20090910

Novel reactivity of dibenzothiophene monooxygenase from Bacillus subtilis WU-S2B.

Bioscience, biotechnology, and biochemistry 20090901

Biodegradation of thiodiglycol, a hydrolyzate of the chemical weapon Yperite, by benzothiophene-desulfurizing bacteria.

Journal of hazardous materials 20090815

FXR agonist activity of conformationally constrained analogs of GW 4064.

Bioorganic & medicinal chemistry letters 20090815

Benzothiophene inhibitors of MK2. Part 2: improvements in kinase selectivity and cell potency.

Bioorganic & medicinal chemistry letters 20090815

Benzothiophene inhibitors of MK2. Part 1: structure-activity relationships, assessments of selectivity and cellular potency.

Bioorganic & medicinal chemistry letters 20090815

Novel Route to 2,3-Substituted Benzo[b]thiophenes via Intramolecular Radical Cyclization.

The Journal of organic chemistry 20090807

Synthesis and properties of symmetric and unsymmetric dibenzothienopyrroles.

Organic letters 20090806

Synthesis and evaluation of 1-(1-(Benzo[b]thiophen-2-yl)cyclohexyl)piperidine (BTCP) analogues as inhibitors of trypanothione reductase.

ChemMedChem 20090803

Potent agonists of the Hedgehog signaling pathway.

Bioorganic & medicinal chemistry letters 20090801

Effects of arzoxifene on bone mineral density and endometrium in postmenopausal women with normal or low bone mass.

The Journal of clinical endocrinology and metabolism 20090701

One-pot synthesis of benzo[b]thiophenes and benzo[b]selenophenes from o-halo-substituted ethynylbenzenes: convenient approach to mono-, bis-, and tris-chalcogenophene-annulated benzenes.

Organic letters 20090604

Mutagenicity of an aged gasworks soil during bioslurry treatment.

Environmental and molecular mutagenesis 20090601

Investigation of various N-heterocyclic substituted piperazine versions of 5/7-{[2-(4-aryl-piperazin-1-yl)-ethyl]-propyl-amino}-5,6,7,8-tetrahydro-naphthalen-2-ol: effect on affinity and selectivity for dopamine D3 receptor.

Bioorganic & medicinal chemistry 20090601

Benzothiophene piperazine and piperidine urea inhibitors of fatty acid amide hydrolase (FAAH).

Bioorganic & medicinal chemistry letters 20090515

Binding in thiophene and benzothiophene dimers investigated by density functional theory with dispersion-correcting potentials.

The journal of physical chemistry. A 20090507

Synthesis of novel 3-(aryl)benzothieno[2,3-c]pyran-1-ones from Sonogashira products and intramolecular cyclization: Antitumoral activity evaluation.

European journal of medicinal chemistry 20090501

QSAR model for predicting radical scavenging activity of di(hetero)arylamines derivatives of benzo[b]thiophenes.

European journal of medicinal chemistry 20090501

Synthesis and pharmacological evaluation of 2-substituted benzo[b]thiophenes as anti-inflammatory and analgesic agents.

European journal of medicinal chemistry 20090401

Density functional study of the adsorption and van der Waals binding of aromatic and conjugated compounds on the basal plane of MoS(2).

The Journal of chemical physics 20090314

Fragmentation pathways of some benzothiophene radical cations formed by atmospheric pressure chemical ionisation.

Rapid communications in mass spectrometry : RCM 20090301

Application of a rhodium-catalyzed addition/cyclization sequence toward the synthesis of polycyclic heteroaromatics.

The Journal of organic chemistry 20090220

Efficient second harmonic generation from thin films of V-shaped benzo[b]thiophene based molecules.

Optics express 20090216

Molecular mechanism of thioflavin-T binding to the surface of beta-rich peptide self-assemblies.

Journal of molecular biology 20090130

In situ growing and patterning of aligned organic nanowire arrays via dip coating.

Langmuir : the ACS journal of surfaces and colloids 20090120

Effect of periodic replacement of the heteroatom on the spectroscopic properties of indole and benzofuran derivatives.

The journal of physical chemistry. A 20090115

Structural modulation of oxidative metabolism in design of improved benzothiophene selective estrogen receptor modulators.

Drug metabolism and disposition: the biological fate of chemicals 20090101

Bacterial degradation of aromatic compounds.

International journal of environmental research and public health 20090101

Raloxifene: mechanism of action, effects on bone tissue, and applicability in clinical traumatology practice.

The open orthopaedics journal 20090101

Solution-phase parallel synthesis of a multi-substituted benzo[b]thiophene library.

Journal of combinatorial chemistry 20090101

Efficient synthesis of benzothiophenes by an unusual palladium-catalyzed vinylic C-S coupling.

Angewandte Chemie (International ed. in English) 20090101

Novel inhibitors of the calcineurin/NFATc hub - alternatives to CsA and FK506?

Cell communication and signaling : CCS 20090101

Lasofoxifene for the prevention and treatment of postmenopausal osteoporosis.

Therapeutics and clinical risk management 20090101

1-Benzothio-phene-2-carbaldehyde 4-ethyl-thio-semicarbazone.

Acta crystallographica. Section E, Structure reports online 20090101

C-H bond activation of heteroarenes mediated by a half-sandwich iron complex of N-heterocyclic carbene.

Journal of the American Chemical Society 20081217

Synthesis and properties of the anti and syn isomers of dibenzothieno[b,d]pyrrole.

Chemical communications (Cambridge, England) 20081214

Reactivity of Mo(PMe3)6 towards benzothiophene and selenophenes: new pathways relevant to hydrodesulfurization.

Journal of the American Chemical Society 20081203

Microbial transformation of benzothiophenes, with carbazole as the auxiliary substrate, by Sphingomonas sp. strain XLDN2-5.

Microbiology (Reading, England) 20081201

Managing the risk of invasive breast cancer in women at risk for breast cancer and osteoporosis: the role of raloxifene.

Clinical interventions in aging 20081201

5-n-Butyl-4-[2-(2-ethyl-1-benzothio-phen-3-yl)-3,3,4,4,5,5-hexa-fluoro-cyclo-pent-1-en-1-yl]thio-phene-2-carbaldehyde.

Acta crystallographica. Section E, Structure reports online 20081201

Palladium-catalysed direct synthesis of benzo[b]thiophenes from thioenols.

Chemical communications (Cambridge, England) 20081121

[Functional correlation of dibenzothiophene and benzothiophene desulfurization enzymes].

Huan jing ke xue= Huanjing kexue 20081101

Novel A-ring and B-ring modified combretastatin A-4 (CA-4) analogues endowed with interesting cytotoxic activity.

Journal of medicinal chemistry 20081009

Antifungal activity of synthetic di(hetero)arylamines based on the benzo[b]thiophene moiety.

Bioorganic & medicinal chemistry 20080901

Raloxifene, a selective estrogen receptor modulator, induces mitochondria-mediated apoptosis in human endometrial carcinoma cells.

Medical molecular morphology 20080901

alpha,alpha-Cyclopentaneglycine dipeptides capped with biaryls as tachykinin NK(2) receptor antagonists.

ChemMedChem 20080701

Liquid phase adsorption by microporous coordination polymers: removal of organosulfur compounds.

Journal of the American Chemical Society 20080604

Desulfurization of various organic sulfur compounds and the mixture of DBT + 4,6-DMDBT by Mycobacterium sp. ZD-19.

Bioresource technology 20080601

5,7-Bis(1-benzothio-phen-2-yl)-2,3-dihydro-thieno[3,4-b][1,4]dioxine.

Acta crystallographica. Section E, Structure reports online 20080601

(11R,11aS)-11-Hydr-oxy-1,5,11,11a-tetra-hydro-1-benzothieno[2,3-f]indolizin-3(2H)-one.

Acta crystallographica. Section E, Structure reports online 20080601

New thermally irreversible and fluorescent photochromic diarylethenes.

The journal of physical chemistry. A 20080529

Raloxifene in breast cancer prevention.

Expert opinion on drug safety 20080501

Preventing breast cancer in high-risk women, 2008.

Oncology (Williston Park, N.Y.) 20080501

Screening for antidepressant, sedative and analgesic activities of novel fused thiophene derivatives.

Acta pharmaceutica (Zagreb, Croatia) 20080301

Comparison of effects of alendronate and raloxifene on lumbar bone mineral density, bone turnover, and lipid metabolism in elderly women with osteoporosis.

Yonsei medical journal 20080227

Deprotonative metalation of five-membered aromatic heterocycles using mixed lithium-zinc species.

The Journal of organic chemistry 20080104

Amino acid derivatives as histone deacetylase inhibitors.

Bioorganic & medicinal chemistry letters 20080101

Carbonic anhydrase IX in oligodendroglial brain tumors.

BMC cancer 20080101

S35225 is a direct inhibitor of Plasminogen Activator Inhibitor type-1 activity in the blood.

Thrombosis research 20080101

[Synthetic estrogens: some new pharmacological actions and mechanisms].

Nihon rinsho. Japanese journal of clinical medicine 20080101

Efficacy of tibolone and raloxifene for the maintenance of skeletal muscle strength, bone mineral density, balance, body composition, cognitive function, mood/depression, anxiety and quality of life/well-being in late postmenopausal women >/= 70 years: study design of a randomized, double-blind, double-dummy, placebo-controlled, single-center trial.

Trials 20080101

Human genetics branches out in Barcelona.

Genome biology 20080101

Synthesis of thienyl analogues of PCBM and investigation of morphology of mixtures in P3HT.

Beilstein journal of organic chemistry 20080101

Development of a groundwater biobarrier for the removal of polycyclic aromatic hydrocarbons, BTEX, and heterocyclic hydrocarbons.

Water science and technology : a journal of the International Association on Water Pollution Research 20080101

S,C-sulfonium ylides from thiophenes: potential carbene precursors.

Journal of the American Chemical Society 20071226

Synthesis of benzo[b]thiophenes by cyclization of arylketene dithioacetal monoxides under pummerer-like conditions.

Organic letters 20071220

(Z)-3-(Benzo[b]thiophen-2-yl)-2-(3,4,5-trimethoxyphenyl)acrylonitrile and (E)-3-(benzo[b]thiophen-2-yl)-2-(3,4-dimethoxyphenyl)acrylonitrile. [corrected].

Acta crystallographica. Section C, Crystal structure communications 20071201

Zipper-mode double C-H activation: palladium-catalyzed direct construction of highly-fused heterocyclic systems.

Organic letters 20071108

Discovery of a new series of potent and selective linear tachykinin NK2 receptor antagonists.

Journal of medicinal chemistry 20071004

Sulfur from benzothiophene and alkylbenzothiophenes supports growth of Rhodococcus sp. strain JVH1.

Biodegradation 20071001

Structure-activity relationships for a family of benzothiophene selective estrogen receptor modulators including raloxifene and arzoxifene.

ChemMedChem 20071001

Synthesis and evaluation of dual wavelength fluorescent benzo[b]thiophene boronic acid derivatives for sugar sensing.

Chemical biology & drug design 20071001

Structural modulation of reactivity/activity in design of improved benzothiophene selective estrogen receptor modulators: induction of chemopreventive mechanisms.

Molecular cancer therapeutics 20070901

Effect of estrogens on skin aging and the potential role of SERMs.

Clinical interventions in aging 20070901

Update on bazedoxifene: a novel selective estrogen receptor modulator.

Clinical interventions in aging 20070901

Benzo[b]thiophene-based histone deacetylase inhibitors.

Bioorganic & medicinal chemistry letters 20070815

Chromatographic methods applied in the monitoring of biodesulfurization processes--state of the art.

Talanta 20070815

Selectivity among organic sulfur compounds in one- and two-liquid-phase cultures of Rhodococcus sp. strain JVH1.

Biodegradation 20070801

Nonconjugated dendritic iridium(III) complexes with tunable pyridine-based ligands: synthesis, photophysical, electrochemical, and electroluminescent properties.

Inorganic chemistry 20070709

Synthesis and SAR of selective benzothiophene, benzofuran, and indole-based peroxisome proliferator-activated receptor delta agonists.

Bioorganic & medicinal chemistry letters 20070701

Benzothiophene selective estrogen receptor modulators with modulated oxidative activity and receptor affinity.

Journal of medicinal chemistry 20070531

Environmental factors influencing sorption of heterocyclic aromatic compounds to soil.

Environmental science & technology 20070501

[Determination and distribution of sulfur compounds in coked gasoline by gas chromatography-sulfur chemiluminescence detection].

Se pu = Chinese journal of chromatography 20070501

Raloxifene blocks estradiol induction of the serotonin transporter and 5-hydroxytryptamine2A receptor in female rat brain.

Neuroscience letters 20070424

Desulfurization of liquid fuels by adsorption on carbon-based sorbents and ultrasound-assisted sorbent regeneration.

Langmuir : the ACS journal of surfaces and colloids 20070327

Does aromaticity in a reaction product increase or decrease the intrinsic barrier? Kinetics of the reversible deprotonation of benzofuran-3(2H)-one and benzothiophene-3(2H)-one.

Journal of the American Chemical Society 20070307

Chiral helicenoid diarylethene with large change in specific optical rotation by photochromism.

The Journal of organic chemistry 20070302

The differential effects of bisphosphonates, SERMS (selective estrogen receptor modulators), and parathyroid hormone on bone remodeling in osteoporosis.

Clinical interventions in aging 20070301

Potential sialyltransferase inhibitors based on neuraminyl substitution by hetaryl rings.

Carbohydrate research 20070226

Medicinal chemistry and emerging strategies applied to the development of selective estrogen receptor modulators (SERMs).

Current medicinal chemistry 20070101

Interactions of the human cytosolic sulfotransferases and steroid sulfatase in the metabolism of tibolone and raloxifene.

The Journal of steroid biochemistry and molecular biology 20070101

Estrogenic or antiestrogenic therapies for multiple myeloma?

Molecular cancer 20070101

Transition-metal/Lewis acid free synthesis of acyl benzothiophenes via C-C bond forming reaction.

Beilstein journal of organic chemistry 20070101

GABA A/Bz receptor subtypes as targets for selective drugs.

Current medicinal chemistry 20070101

Arzoxifene: the evidence for its development in the management of breast cancer.

Core evidence 20070101

The cardiovascular effects of selective estrogen receptor modulators.

Annals of the New York Academy of Sciences 20061201

A systematic resolution of sulfur in reticulated vitreous carbon using X-ray absorption spectroscopy.

Inorganic chemistry 20061127

Syntheses and structures of novel heteroarene-fused coplanar pi-conjugated chromophores.

Organic letters 20061026

Solid-phase synthesis of tetrahydro-beta-carbolines and tetrahydroisoquinolines by stereoselective intramolecular N-carbamyliminium Pictet-Spengler reactions.

Chemistry (Weinheim an der Bergstrasse, Germany) 20061025

Synthesis and antimicrobial activity studies of ortho-chlorodiarylamines and heteroaromatic tetracyclic systems in the benzo[b]thiophene series.

Bioorganic & medicinal chemistry 20061015

Sorption of heterocyclic organic compounds to reference soils: column studies for process identification.

Environmental science & technology 20061001

Effect of ormeloxifene on ovariectomy-induced bone resorption, osteoclast differentiation and apoptosis and TGF beta-3 expression.

The Journal of steroid biochemistry and molecular biology 20060801

Synthesis and evaluation of benzothiophene derivatives as ligands for imaging beta-amyloid plaques in Alzheimer's disease.

Nuclear medicine and biology 20060801

The reaction of o-alkynylarene and heteroarene carboxaldehyde derivatives with iodonium ions and nucleophiles: a versatile and regioselective synthesis of 1H-isochromene, naphthalene, indole, benzofuran, and benzothiophene compounds.

Chemistry (Weinheim an der Bergstrasse, Germany) 20060724

Gold-catalyzed intramolecular carbothiolation of alkynes: synthesis of 2,3-disubstituted benzothiophenes from (alpha-alkoxy alkyl) (ortho-alkynyl phenyl) sulfides.

Angewandte Chemie (International ed. in English) 20060703

New HIV-1 reverse transcriptase inhibitors based on a tricyclic benzothiophene scaffold: synthesis, resolution, and inhibitory activity.

Bioorganic & medicinal chemistry letters 20060601

Novel combretastatin analogues endowed with antitumor activity.

Journal of medicinal chemistry 20060601

Chemical modification modulates estrogenic activity, oxidative reactivity, and metabolic stability in 4'F-DMA, a new benzothiophene selective estrogen receptor modulator.

Chemical research in toxicology 20060601

[Isolation and characterization of a benzothiophene-desulfurizing bacterium].

Huan jing ke xue= Huanjing kexue 20060601

Biodesulfurization of alkylated forms of dibenzothiophene and benzothiophene by Sphingomonas subarctica T7b.

Journal of bioscience and bioengineering 20060401

Liquid-phase adsorption of multi-ring thiophenic sulfur compounds on carbon materials with different surface properties.

The journal of physical chemistry. B 20060316

Evaluation of the antioxidant properties of diarylamines in the benzo[b]thiophene series by free radical scavenging activity and reducing power.

Bioorganic & medicinal chemistry letters 20060301

Raloxifene: a selective estrogen-receptor modulator for postmenopausal osteoporosis - a clinical update on efficacy and safety.

Women's health (London, England) 20060301

Characteristics of sulfur response in a micro-flame photometric detector.

Journal of chromatography. A 20060210

Induction of apoptosis by photoexcited tetracyclic compounds derivatives of benzo[b]thiophenes and pyridines.

Journal of photochemistry and photobiology. B, Biology 20060201

CFTR chloride channel drug discovery--inhibitors as antidiarrheals and activators for therapy of cystic fibrosis.

Current pharmaceutical design 20060101

Benzothieno and benzofurano annelated estranes.

Steroids 20051201

One-electron reduction potential for oxygen- and sulfur-centered organic radicals in protic and aprotic solvents.

Journal of the American Chemical Society 20051116

Synthesis, characterization, and structure of cyclopenta[c]thiophenes and their manganese complexes.

Journal of the American Chemical Society 20051102

Synthesis and biological activity of alpha-bromoacryloyl lexitropsin conjugates.

European journal of medicinal chemistry 20051101

Carbonic anhydrase inhibitors: inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with benzo[b]thiophene 1,1-dioxide sulfonamides.

Bioorganic & medicinal chemistry letters 20051101

Synthesis of oxadiazoles, thiadiazoles and triazoles derived from benzo[b]thiophene.

Molecules (Basel, Switzerland) 20050930

Decoys for docking.

Journal of medicinal chemistry 20050602

Hydroxylation activity of P450 BM-3 mutant F87V towards aromatic compounds and its application to the synthesis of hydroquinone derivatives from phenolic compounds.

Applied microbiology and biotechnology 20050601

Biodesulfurization of dibenzothiophene and other organic sulfur compounds by a newly isolated Microbacterium strain ZD-M2.

FEMS microbiology letters 20050601

Prediction of genotoxicity of chemical compounds by statistical learning methods.

Chemical research in toxicology 20050601

Triplet-triplet energy transfer controlled by the donor-acceptor distance in rigidly held palladium-containing cofacial bisporphyrins.

Chemistry (Weinheim an der Bergstrasse, Germany) 20050520

Selective adsorption of thiophene and 1-benzothiophene on metal-ion-exchanged zeolites in organic medium.

Journal of colloid and interface science 20050515

Efficient access to 2-aryl-3-substituted benzo[b]thiophenes.

The Journal of organic chemistry 20050429

Synthesis and binding affinities of novel SRIF-mimicking beta-D-glucosides satisfying the requirement for a pi-cloud at C1.

Organic letters 20050317

Poly(thiaheterohelicene): a stiff conjugated helical polymer comprised of fused benzothiophene rings.

Organic letters 20050303

Benzothiophenes containing a piperazine side chain as selective ligands for the estrogen receptor alpha and their bioactivities in vivo.

Bioorganic & medicinal chemistry letters 20050301

Desulfurization of dibenzothiophene, benzothiophene, and other thiophene analogs by a newly isolated bacterium, Gordonia alkanivorans strain 1B.

Applied biochemistry and biotechnology 20050301

Benzo[b]thiophenesulphonamide 1,1-dioxide derivatives inhibit tNOX activity in a redox state-dependent manner.

British journal of cancer 20050227

In vitro metabolic fate of a novel structural class: evidence for the formation of a reactive intermediate on a benzothiophene moiety.

Chemico-biological interactions 20050227

Design, synthesis, and biological evaluation of novel potent and selective alphavbeta3/alphavbeta5 integrin dual inhibitors with improved bioavailability. Selection of the molecular core.

Journal of medicinal chemistry 20050224

Simultaneous determination of NSO-heterocycles, homocycles and their metabolites in groundwater of tar oil contaminated sites using LC with diode array UV and fluorescence detection.

Journal of chromatography. A 20050218

Organoboron compounds with an 8-hydroxyquinolato chelate and its derivatives: substituent effects on structures and luminescence.

Inorganic chemistry 20050207

Thermophilic biodesulfurization of various heterocyclic sulfur compounds and crude straight-run light gas oil fraction by a newly isolated strain Mycobacterium phlei WU-0103.

Current microbiology 20050201

Endocrinology and hormone therapy in breast cancer: selective oestrogen receptor modulators and downregulators for breast cancer - have they lost their way?

Breast cancer research : BCR 20050101

Benefit-risk assessment of raloxifene in postmenopausal osteoporosis.

Drug safety 20050101

Adsorption, desorption, and conversion of thiophene on H-ZSM5.

Langmuir : the ACS journal of surfaces and colloids 20041207

Screening of antimicrobial activity of diarylamines in the 2,3,5-trimethylbenzo[b]thiophene series: a structure-activity evaluation study.

Bioorganic & medicinal chemistry letters 20041206

Synthesis and NMR spectroscopic studies of allylsulfanyl-N1-alkyl-N4-phenyl-1,4-phenylenediamines and their cyclization products, 2,3-dihydro-1-benzothiophenes and thiochromans.

Magnetic resonance in chemistry : MRC 20041201

Palladium-catalyzed tandem reaction of yne-propargylic carbonates with boronic acids: a simple method for the synthesis of fused aromatic rings through allene-mediated electrocyclization.

Chemistry (Weinheim an der Bergstrasse, Germany) 20041025

Benzothiophene and naphthalene derived constrained SERMs.

Bioorganic & medicinal chemistry letters 20041018

Phenylpiperazinylmethylheterocycle derivatives: synthesis and dopamine receptor binding profiles.

Archiv der Pharmazie 20040701

New 3-[4-(2,3-dihydro-14-benzodioxin-5-yl)piperazin-1-yl]-1-(5-substituted benzo[b]thiophen-3-yl)propanol derivatives with dual action at 5-HT(1A) serotonin receptors and serotonin transporter as a new class of antidepressants.

Die Pharmazie 20040701

C17,20-lyase inhibitors I. Structure-based de novo design and SAR study of C17,20-lyase inhibitors.

Bioorganic & medicinal chemistry 20040501

[Determination of sulfur compounds in fluid catalytic cracking gasoline by gas chromatography with a sulfur chemiluminescence detector].

Se pu = Chinese journal of chromatography 20040501

Synthesis and serotonergic activity of variously substituted (3-amido)phenylpiperazine derivatives and benzothiophene-4-piperazine derivatives: novel antagonists for the vascular 5-HT1B receptor.

European journal of medicinal chemistry 20040401

Discovery of novel heteroaryl-substituted chalcones as inhibitors of TNF-alpha-induced VCAM-1 expression.

Bioorganic & medicinal chemistry letters 20040322

Design, synthesis and structure-activity relationship of novel RXR-selective modulators.

Bioorganic & medicinal chemistry letters 20040322

Efficient isomer-pure synthesis of a benzo[b]thiophene analogue of pentacene.

The Journal of organic chemistry 20040319

Synthesis and cytotoxic activity of lipophilic sulphonamide derivatives of the benzo[b]thiophene 1,1-dioxide.

Bioorganic & medicinal chemistry 20040301

Synthesis of new thiophene and benzo[b]thiophene hydrazide derivatives as human NPY Y(5) antagonists.

Bioorganic & medicinal chemistry letters 20040209

A synthesis of heteroaromatic analogues of 1-methyl-1,2,3,4-tetrahydroisoquinoline using the Pummerer-type cyclization reaction: observation of tandem cyclization reaction.

Chemical & pharmaceutical bulletin 20040201

Elimination of sulfur from aromatic heterocycles by a water-soluble arene ruthenium cluster: synthesis and molecular structure of [H2S2Ru4(C6H6)4]Cl2.

Chemical communications (Cambridge, England) 20040121

Modulation of selective serotonin reuptake inhibitor and 5-HT1A antagonist activity in 8-aza-bicyclo[3.2.1]octane derivatives of 2,3-dihydro-1,4-benzodioxane.

Bioorganic & medicinal chemistry letters 20040119

Combined application of stable carbon isotope analysis and specific metabolites determination for assessing in situ degradation of aromatic hydrocarbons in a tar oil-contaminated aquifer.

Environmental science & technology 20040115

Advances in estrogen receptor biology: prospects for improvements in targeted breast cancer therapy.

Breast cancer research : BCR 20040101

Potent inhibition of human liver aldehyde oxidase by raloxifene.

Drug metabolism and disposition: the biological fate of chemicals 20040101

NH2-SEP-PAK cartridges for enrichment of Aromatic Sulfur Compounds from sea water: determination by GC-FID and GC-MS.

Annali di chimica 20040101

Monitoring toxicity of industrial wastewater and specific chemicals to a green alga, nitrifying bacteria and an aquatic bacterium.

Water science and technology : a journal of the International Association on Water Pollution Research 20040101

Structure-activity relationship of benzo[b]thiophene-2-sulfonamide derivatives as novel human chymase inhibitors.

Bioorganic & medicinal chemistry letters 20031117

Reactions that generate aromatic molecules: is aromatic stabilization less or more advanced than bond changes at the transition state? Kinetic and thermodynamic acidities of rhenium carbene complexes.

Journal of the American Chemical Society 20031008

Nitrosation, nitration, and autoxidation of the selective estrogen receptor modulator raloxifene by nitric oxide, peroxynitrite, and reactive nitrogen/oxygen species.

Chemical research in toxicology 20031001

2,6-disubstituted pyran-4-one and thiopyran-4-one inhibitors of DNA-Dependent protein kinase (DNA-PK).

Bioorganic & medicinal chemistry letters 20030915

2-(2'-Hydroxyphenyl)benzene sulfinate desulfinase from the thermophilic desulfurizing bacterium Paenibacillus sp. strain A11-2: purification and characterization.

Applied microbiology and biotechnology 20030901

Synthesis and binding affinities of fluoroalkylated raloxifenes.

Bioorganic & medicinal chemistry 20030815

Target specificity of selective estrogen receptor modulators within human endometrial cancer cells.

The Journal of steroid biochemistry and molecular biology 20030701

Diastereoselective photochromism of a bisbenzothienylethene governed by steric as well as electronic interactions.

Journal of the American Chemical Society 20030618

Preparation and characterization of organotin-oxomolybdate coordination polymers and their use in sulfoxidation catalysis.

Chemistry (Weinheim an der Bergstrasse, Germany) 20030616

New benzo(b)thiophenesulphonamide 1,1-dioxide derivatives induce a reactive oxygen species-mediated process of apoptosis in tumour cells.

Oncogene 20030612

Anaerobic desulphurisation of thiophenes by mixed microbial communities from oilfields.

Biodegradation 20030601

The effect of minor-groove hydrogen-bond acceptors and donors on the stability and replication of four unnatural base pairs.

Journal of the American Chemical Society 20030521

New fibrinolytic agents: benzothiophene derivatives as inhibitors of the t-PA-PAI-1 complex formation.

Bioorganic & medicinal chemistry letters 20030519

Discovery and characterization of a potent and selective non-amidine inhibitor of human factor Xa.

Biochemical pharmacology 20030501

Selective estrogen receptor modulators.

Southern medical journal 20030501

Hydrogenation and carbon-sulfur bond hydrogenolysis of benzothiophene promoted by Re2(CO)10 and H4Re4(CO)12.

Inorganic chemistry 20030407

Effect of treatment with the selective oestrogen receptor modulator LY117018-HCl on pituitary sensitivity to GnRH and subsequent ovulation.

Reproduction (Cambridge, England) 20030401

Design, synthesis and in vitro evaluation of novel benzo[b]thiophene derivatives as serotonin N-acetyltransferase (AANAT) inhibitors.

Journal of enzyme inhibition and medicinal chemistry 20030401

Photochemistry and photophysics of thienocarbazoles.

Photochemistry and photobiology 20030201

Advances in breast cancer treatment and prevention: preclinical studies on aromatase inhibitors and new selective estrogen receptor modulators (SERMs).

Breast cancer research : BCR 20030101

Crystal structures of two potent nonamidine inhibitors bound to factor Xa.

Biochemistry 20021231

[Determination of sulfur compounds in catalytic diesel oil by gas chromatography with atomic emission detector and its applications].

Se pu = Chinese journal of chromatography 20021101

Recombinant Rhodococcus sp. strain T09 can desulfurize DBT in the presence of inorganic sulfate.

Current microbiology 20021001

Purification and characterization of the monooxygenase catalyzing sulfur-atom specific oxidation of dibenzothiophene and benzothiophene from the thermophilic bacterium Paenibacillus sp. strain A11-2.

Applied microbiology and biotechnology 20021001

4-Substituted D-glutamic acid analogues: the first potent inhibitors of glutamate racemase (MurI) enzyme with antibacterial activity.

Journal of medicinal chemistry 20020926

Synthesis and molecular modeling of new 1-aryl-3-[4-arylpiperazin-1-yl]-1-propane derivatives with high affinity at the serotonin transporter and at 5-HT(1A) receptors.

Journal of medicinal chemistry 20020912

Isolation and characterization of a moderate thermophile, Mycobacterium phlei GTIS10, capable of dibenzothiophene desulfurization.

Applied microbiology and biotechnology 20020901

Synthesis of fluoren-9-ones by the palladium-catalyzed cyclocarbonylation of o-halobiaryls.

The Journal of organic chemistry 20020809

Geochemical and physiological evidence for mixed aerobic and anaerobic field biodegradation of coal tar waste by subsurface microbial communities.

Microbial ecology 20020801

Biodesulfurization of naphthothiophene and benzothiophene through selective cleavage of carbon-sulfur bonds by Rhodococcus sp. strain WU-K2R.

Applied and environmental microbiology 20020801

Analysis of aromatic sulfur compounds in gas oils using GC with sulfur chemiluminescence detection and high-resolution MS.

Analytical chemistry 20020801

Biodesulfurization of benzothiophene and dibenzothiophene by a newly isolated Rhodococcus strain.

Applied microbiology and biotechnology 20020701

Cytochrome P450 3A4-mediated bioactivation of raloxifene: irreversible enzyme inhibition and thiol adduct formation.

Chemical research in toxicology 20020701

One-pot synthesis of benzo[b]furan and indole inhibitors of tubulin polymerization.

Journal of medicinal chemistry 20020606

New 3-[4-(aryl)piperazin-1-yl]-1-(benzo[b]thiophen-2-yl)propane derivatives with dual action at 5-HT1A serotonin receptors and serotonin transporter as a new class of antidepressants.

Die Pharmazie 20020601

Benzoyl and cinnamoyl nitrogen mustard derivatives of benzoheterocyclic analogues of the tallimustine: synthesis and antitumour activity.

Bioorganic & medicinal chemistry 20020501

Macrophage inducible nitric oxide synthase gene expression is blocked by a benzothiophene derivative with anti-HIV properties.

Molecular genetics and metabolism 20020401

Toward selective ERbeta agonists for central nervous system disorders: synthesis and characterization of aryl benzthiophenes.

Journal of medicinal chemistry 20020328

Metabolic response against sulfur-containing heterocyclic compounds by the lignin-degrading basidiomycete Coriolus versicolor.

Applied microbiology and biotechnology 20020301

Re(2)(CO)(10)-promoted S-binding, C-S bond cleavage, and hydrogenation of benzothiophenes: organometallic models for the hydrodesulfurization of thiophenes.

Journal of the American Chemical Society 20020227

Aerobic co-metabolism of sulfur, nitrogen and oxygen heterocycles by three marine bacterial consortia.

Journal of basic microbiology 20020101

Isolation and characterization of thermophilic benzothiophene-degrading Mycobacterium sp.

Applied biochemistry and biotechnology 20020101

Physical organic chemistry of transition metal carbene complexes. 23. Kinetic and thermodynamic acidities of cationic benzothienyl- and selenylcarbene complexes of rhenium in aqueous acetonitrile.

Journal of the American Chemical Society 20011205

Raloxifene.

Current drug targets 20011201

Effects of the new selective estrogen receptor modulator LY353381.HCl (Arzoxifene) on human endometrial cancer growth in athymic mice.

Clinical cancer research : an official journal of the American Association for Cancer Research 20011201

Synthesis and studies on spectroscopic as well as electron donating properties of the two alkoxy benzo[b]thiophenes.

Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20011201

Selective estrogen receptor modulator effects on serum lipoproteins and vascular function in postmenopausal women and in hypercholesterolemic men.

Annals of the New York Academy of Sciences 20011201

New cytotoxic benzo(b)thiophenilsulfonamide 1,1-dioxide derivatives inhibit a NADH oxidase located in plasma membranes of tumour cells.

British journal of cancer 20011101

Benzo[b]thiophene desulfurization by Gordonia rubropertinctus strain T08.

Applied microbiology and biotechnology 20011001

Desulfurization of benzothiophene by the Gram-negative bacterium, Sinorhizobium sp. KT55.

Current microbiology 20010901

1-(2-[4-[6-Hydroxy-2-(4-hydroxyphenyl)benzo[b]thiol-3-ylcarbonyl]phenoxy]ethyl)piperidinium chloride.

Acta crystallographica. Section C, Crystal structure communications 20010901

Effect of raloxifene on serum triglycerides in postmenopausal women: influence of predisposing factors for hypertriglyceridemia.

Clinical therapeutics 20010901

Identification and characterization of a benzothiophene inhibitor of herpes simplex virus type 1 replication which acts at the immediate early stage of infection.

Antiviral research 20010801

Analysis of cross-resistance of the selective estrogen receptor modulators arzoxifene (LY353381) and LY117018 in tamoxifen-stimulated breast cancer xenografts.

Clinical cancer research : an official journal of the American Association for Cancer Research 20010801

Microbial desulfurization of alkylated dibenzothiophene and alkylated benzothiophene by recombinant Rhodococcus sp. strain T09.

Applied microbiology and biotechnology 20010701

Phase I study of a third-generation selective estrogen receptor modulator, LY353381.HCL, in metastatic breast cancer.

Journal of clinical oncology : official journal of the American Society of Clinical Oncology 20010401

A novel palladium-mediated coupling approach to 2,3-disubstituted benzo(b)thiophenes and its application to the synthesis of tubulin binding agents.

Organic letters 20010308

Electron transfer compatible molecular design of benzothiophene-acetophenone bichromophores: a theoretical approach.

Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20010301

Update on endocrine aspects of breast cancer: report from the 23rd San Antonio Breast Cancer Symposium, San Antonio, Texas, USA, 6-9 December 2000.

Breast cancer research : BCR 20010101

Selective estrogen receptor modulators: mechanism of action and clinical experience. Focus on raloxifene.

Reproduction, fertility, and development 20010101

Raloxifene: another selective estrogen modulator.

In vivo (Athens, Greece) 20010101

Isolation of a unique benzothiophene-desulphurizing bacterium, Gordona sp. strain 213E (NCIMB 40816), and characterization of the desulphurization pathway.

Microbiology (Reading, England) 19980901

Synthesis and in vitro LTD4 antagonist activity of bicyclic and monocyclic cyclopentylurethane and cyclopentylacetamide N-arylsulfonyl amides.

Journal of medicinal chemistry 19900901