Benzenesulfonamide
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Synthesis of some new benzisothiazolone and benzenesulfonamide derivatives of biological interest starting from saccharin sodium. | Archiv der Pharmazie 20131001 |
Amide derivatives of benzene-sulfonanilide, pharmaceutical composition thereof and method for cancer treatment using the same (US20120095092). | Expert opinion on therapeutic patents 20121001 |
Eight isostructural 4,4'-disubstituted N-phenylbenzenesulfonamides. | Acta crystallographica. Section C, Crystal structure communications 20121001 |
Benzenesulfonamide attenuates monocrotaline-induced pulmonary arterial hypertension in a rat model. | European journal of pharmacology 20120905 |
Virtual screening leads to the discovery of novel non-nucleotide P2Y₁ receptor antagonists. | Bioorganic & medicinal chemistry 20120901 |
Placing supercritical fluid chromatography one step ahead of reversed-phase high performance liquid chromatography in the achiral purification arena: a hydrophilic interaction chromatography cross-linked diol chemistry as a new generic stationary phase. | Journal of chromatography. A 20120810 |
Magnetic levitation as a platform for competitive protein-ligand binding assays. | Analytical chemistry 20120717 |
FT-IR, FT-Raman and computational study of (E)-N-carbamimidoyl-4-((4-methoxybenzylidene)amino)benzenesulfonamide. | Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20120615 |
Sulfonamide bearing oligonucleotides: simple synthesis and efficient RNA recognition. | Bioorganic & medicinal chemistry 20120615 |
The novel endocrine disruptor tolylfluanid impairs insulin signaling in primary rodent and human adipocytes through a reduction in insulin receptor substrate-1 levels. | Biochimica et biophysica acta 20120601 |
Research on the structure-surface adsorptive activity relationships of triazolyl glycolipid derivatives for mild steel in HCl. | Carbohydrate research 20120601 |
Design of [(2-pyrimidinylthio)acetyl]benzenesulfonamides as inhibitors of human carbonic anhydrases. | European journal of medicinal chemistry 20120501 |
N-(3-Methyl-benzo-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20120501 |
N-(3-Nitro-benzo-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20120501 |
Molecular cloning, characterization, and inhibition studies of a β-carbonic anhydrase from Malassezia globosa, a potential antidandruff target. | Journal of medicinal chemistry 20120412 |
Discovery of novel 2-N-aryl-substituted benzenesulfonamidoacetamides: orally bioavailable tubulin polymerization inhibitors with marked antitumor activities. | ChemMedChem 20120401 |
(3aR*,6S*,7aR*)-7a-Chloro-6-methyl-2-(4-methyl-phenyl-sulfon-yl)-2,3,3a,6,7,7a-hexa-hydro-3a,6-ep-oxy-1H-isoindole. | Acta crystallographica. Section E, Structure reports online 20120401 |
Identification of novel kynurenine production-inhibiting benzenesulfonamide derivatives in cancer cells. | Biochemical and biophysical research communications 20120316 |
Inhibitory effects of azole-type fungicides on interleukin-17 gene expression via retinoic acid receptor-related orphan receptors α and γ. | Toxicology and applied pharmacology 20120315 |
Synthesis and evaluation of anticancer activity of some novel 6-aryl-2-(p-sulfamylphenyl)-pyridazin-3(2H)-ones. | European journal of medicinal chemistry 20120301 |
4-{(4Z)-4-[(2Z)-3-(4-Fluoro-anilino)-1-hy-droxy-but-2-en-1-yl-idene]-3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-1-yl}-benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20120301 |
Selective precipitation and purification of monovalent proteins using oligovalent ligands and ammonium sulfate. | Bioconjugate chemistry 20120215 |
Synthesis and carbonic anhydrase inhibitory properties of novel cyclohexanonyl bromophenol derivatives. | Bioorganic & medicinal chemistry letters 20120201 |
N-Ethyl-N-(4-methyl-phen-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20120201 |
2-(N-Cyclo-hexyl-carbamo-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20120201 |
Dependence of avidity on linker length for a bivalent ligand-bivalent receptor model system. | Journal of the American Chemical Society 20120111 |
5-HT₂c receptor selectivity and structure-activity relationship of N-methyl-N-(1-methylpiperidin-4-yl)benzenesulfonamide analogs. | Bioorganic & medicinal chemistry letters 20120101 |
Hydroxybenzothiazoles as new nonsteroidal inhibitors of 17β-hydroxysteroid dehydrogenase type 1 (17β-HSD1). | PloS one 20120101 |
Novel 4-(4-substituted-thiazol-2-ylamino)-N-(pyridin-2-yl)-benzenesulfonamides as cytotoxic and radiosensitizing agents. | Archives of pharmacal research 20120101 |
Synthesis, in-vitro anticancer screening and radiosensitizing evaluation of some new N-(quinoxalin-2-yl)benzenesulfonamide derivatives. | Arzneimittel-Forschung 20120101 |
Regulation of expression of citrate synthase by the retinoic acid receptor-related orphan receptor α (RORα). | PloS one 20120101 |
FH535 potentiation of cigarette smoke condensate cytotoxicity is associated with changes in β-catenin and EGR-1 signaling. | International journal of toxicology 20120101 |
Label-free detection of protein binding with multisine SPR microchips. | Lab on a chip 20111221 |
Estimation of analyte concentration by surface plasmon resonance-based biosensing using parameter identification techniques. | Analytical biochemistry 20111215 |
FT-IR, FT-Raman and quantum chemical calculations of (E)-N-carbamimidoyl-4-((3,4-dimethoxybenzylidene) amino) benzenesulfonamide. | Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20111215 |
Radiosynthesis of three [11C]ureido-substituted benzenesulfonamides as PET probes for carbonic anhydrase IX in tumors. | Bioorganic & medicinal chemistry letters 20111201 |
Synthesis and biological evaluation of some new 2-pyrazolines bearing benzene sulfonamide moiety as potential anti-inflammatory and anti-cancer agents. | European journal of medicinal chemistry 20111201 |
Synthesis, in vitro anticancer screening and radiosensitizing evaluation of some new 4-[3-(substituted)thioureido]-N-(quinoxalin-2-yl)-benzenesulfonamide derivatives. | Acta pharmaceutica (Zagreb, Croatia) 20111201 |
Synthesis and acrosin inhibitory activity of substituted 4-amino-N-(diaminomethylene) benzenesulfonamide derivatives. | Bioorganic & medicinal chemistry letters 20111115 |
A double prodrug system for colon targeting of benzenesulfonamide COX-2 inhibitors. | Bioorganic & medicinal chemistry letters 20111115 |
Rhodium-catalyzed annulation of N-benzoylsulfonamide with isocyanide through C-H activation. | Chemistry (Weinheim an der Bergstrasse, Germany) 20111104 |
Substituted phenyl 4-(2-oxoimidazolidin-1-yl)benzenesulfonamides as antimitotics. Antiproliferative, antiangiogenic and antitumoral activity, and quantitative structure-activity relationships. | European journal of medicinal chemistry 20111101 |
2,4-Dichloro-N-(3,5-dimethyl-phen-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20111101 |
4-Chloro-N-(3,4-dichloro-phen-yl)-2-methyl-benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20111101 |
Identification of novel small molecule inhibitors of 4-diphosphocytidyl-2-C-methyl-D-erythritol (CDP-ME) kinase of Gram-negative bacteria. | Bioorganic & medicinal chemistry 20111001 |
Design and synthesis of new N-(5-trifluoromethyl)-1H-1,2,4-triazol-3-yl benzenesulfonamides as possible antimalarial prototypes. | Molecules (Basel, Switzerland) 20110920 |
Synthesis of rhodamine B-benzenesulfonamide conjugates and their inhibitory activity against human α- and bacterial/fungal β-carbonic anhydrases. | Bioorganic & medicinal chemistry letters 20110915 |
Fluoroalkyl and alkyl chains have similar hydrophobicities in binding to the 'hydrophobic wall' of carbonic anhydrase. | Journal of the American Chemical Society 20110907 |
Synthesis and in vivo evaluation of [O-methyl-11C] N-[3,5-dichloro-2-(methoxy)phenyl]-4-(methoxy)-3-(1-piperazinyl)benzenesulfonamide as an imaging probe for 5-HT6 receptors. | Bioorganic & medicinal chemistry 20110901 |
N-(2,6-Dimethyl-phen-yl)-2,4-dimethyl-benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20110901 |
1-Benzyl-2,5-diphenyl-3-tosylimidazol-idin-4-one. | Acta crystallographica. Section E, Structure reports online 20110901 |
4-(3-Methyl-5-phenyl-1H-pyrazol-1-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20110901 |
4-(3,7-Dimethyl-4-oxo-4,5-dihydro-isoxazolo[4,5-d]pyridazin-5-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20110901 |
4-(5-Oxo-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20110901 |
4-(3-Methyl-4,5-dihydro-1H-benzo[g]indazol-1-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20110901 |
Using covalent dimers of human carbonic anhydrase II to model bivalency in immunoglobulins. | Journal of the American Chemical Society 20110803 |
Potassium N-bromo-2-methyl-benzene-sulfonamidate sesquihydrate. | Acta crystallographica. Section E, Structure reports online 20110801 |
2-(4-Chloro-phen-yl)-5-(cyclo-hex-1-en-1-yl)-3-(4-methyl-phenyl-sulfon-yl)-1-phenyl-imidazolidin-4-one. | Acta crystallographica. Section E, Structure reports online 20110801 |
4-Chloro-N-(3,5-dimethyl-phen-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20110801 |
Systematic errors in isothermal titration calorimetry: concentrations and baselines. | Analytical biochemistry 20110715 |
Synthesis of some new 1,3,5-trisubstituted pyrazolines bearing benzene sulfonamide as anticancer and anti-inflammatory agents. | Bioorganic & medicinal chemistry letters 20110715 |
Potassium N,2-dichloro-benzene-sulfonamidate sesquihydrate. | Acta crystallographica. Section E, Structure reports online 20110701 |
Potassium N,4-dichloro-benzene-sulfonamidate monohydrate. | Acta crystallographica. Section E, Structure reports online 20110701 |
Potassium N-bromo-4-chloro-benzene-sulfonamidate monohydrate. | Acta crystallographica. Section E, Structure reports online 20110701 |
Amino-caprolactam γ-secretase inhibitors showing potential for the treatment of Alzheimer's disease. | Bioorganic & medicinal chemistry letters 20110615 |
Conformational variability of different sulfonamide inhibitors with thienyl-acetamido moieties attributes to differential binding in the active site of cytosolic human carbonic anhydrase isoforms. | Bioorganic & medicinal chemistry 20110615 |
Crossing borders to bind proteins--a new concept in protein recognition based on the conjugation of small organic molecules or short peptides to polypeptides from a designed set. | Analytical and bioanalytical chemistry 20110601 |
Ethyl 3-[2-(3,4-dimeth-oxy-benz-yl)-1-phenyl-sulfonyl-1H-indol-3-yl]acrylate chloro-form hemisolvate. | Acta crystallographica. Section E, Structure reports online 20110601 |
A novel COX-2 inhibitor pyrazole derivative proven effective as an anti-inflammatory and analgesic drug. | Basic & clinical pharmacology & toxicology 20110401 |
Synthesis and biological evaluation of some 4-functionalized-pyrazoles as antimicrobial agents. | European journal of medicinal chemistry 20110401 |
2-(4-Chloro-phen-yl)-1,5-diphenyl-3-tosyl-imidazolidin-4-one. | Acta crystallographica. Section E, Structure reports online 20110401 |
4-Chloro-N-(4-nitro-benzo-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20110401 |
2-Methyl-N-(4-nitro-benzo-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20110401 |
2-Chloro-N-(4-nitro-benzo-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20110401 |
Studies of tricyclic piperazine/piperidine furnished molecules as novel integrin αvβ3/αIIbβ3 dual antagonists using 3D-QSAR and molecular docking. | Journal of molecular graphics & modelling 20110201 |
N-(4-Meth-oxy-phen-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20110201 |
Molecular structure and vibrational investigation of benzenesulfonic acid methyl ester using DFT (LSDA, B3LYP, B3PW91 and MPW1PW91) theory calculations. | Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20110101 |
Synthesis and in vitro anticancer evaluation of some novel hexahydroquinoline derivatives having a benzenesulfonamide moiety. | European journal of medicinal chemistry 20110101 |
Correlation analyses on binding affinity of substituted benzenesulfonamides with carbonic anhydrase using ab initio MO calculations on their complex structures (II). | Bioorganic & medicinal chemistry letters 20110101 |
Inhibition of β-carbonic anhydrases with ureido-substituted benzenesulfonamides. | Bioorganic & medicinal chemistry letters 20110101 |
4-Chloro-N-(2,3-dichloro-phen-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20110101 |
N-(2,5-Dichloro-phen-yl)-4-methyl-benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20110101 |
2,4-Dimethyl-N-(4-methyl-phen-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20110101 |
Induction of SCEs and DNA fragmentation in bovine peripheral lymphocytes by in vitro exposure to tolylfluanid-based fungicide. | Genetics and molecular biology 20110101 |
Copper and its complexes in medicine: a biochemical approach. | Molecular biology international 20110101 |
Virtual screening of 2,3-disubstituted-4(3H)-quinazolinones possessing benzenesulfonamide moiety for COX-2 inhibitor. | Bioinformation 20110101 |
Inhibition of influenza A virus (H1N1) fusion by benzenesulfonamide derivatives targeting viral hemagglutinin. | PloS one 20110101 |
Selective elution of target protein from affinity resins by a simple reductant with a thiol group. | Bioorganic & medicinal chemistry letters 20101215 |
4- and 6-(p-Sulphamoylphenyl)androstenediones: Studies of aromatase inhibitor-based oestrone sulphatase inhibition. | Steroids 20101201 |
Design and synthesis of an androgen receptor pure antagonist (CH5137291) for the treatment of castration-resistant prostate cancer. | Bioorganic & medicinal chemistry 20101201 |
N-(2,3-Dichloro-phen-yl)-2,4-dimethyl-benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20101201 |
N-(2,6-Dichloro-phen-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20101201 |
N-(2,3-Dichloro-phen-yl)-4-methyl-benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20101201 |
N-(2,3-Dimethyl-phen-yl)-4-methyl-benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20101201 |
5,6,7,8-Tetrahydropyrido[4,3-d]pyrimidines as novel class of potent and highly selective CaMKII inhibitors. | Bioorganic & medicinal chemistry letters 20101115 |
A diverse series of substituted benzenesulfonamides as aldose reductase inhibitors with antioxidant activity: design, synthesis, and in vitro activity. | Journal of medicinal chemistry 20101111 |
4-[N-(substituted 4-pyrimidinyl)amino]benzenesulfonamides as inhibitors of carbonic anhydrase isozymes I, II, VII, and XIII. | Bioorganic & medicinal chemistry 20101101 |
Indapamide-like benzenesulfonamides as inhibitors of carbonic anhydrases I, II, VII, and XIII. | Bioorganic & medicinal chemistry 20101101 |
Free-solution interaction assay of carbonic anhydrase to its inhibitors using back-scattering interferometry. | Electrophoresis 20101101 |
N-(5-Chloro-2-meth-oxy-phen-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20101101 |
4-[(2-Hy-droxy-benzyl-idene)amino]-N-(5-methyl-isoxazol-3-yl)benzene-sulfonamide: a monoclinic polymorph. | Acta crystallographica. Section E, Structure reports online 20101001 |
Synthesis of anti-microtubule N-(2-Arylindol-7-yl)benzenesulfonamide derivatives and their antitumor mechanisms. | ChemMedChem 20100903 |
Discovery of pyrrole-indoline-2-ones as Aurora kinase inhibitors with a different inhibition profile. | Journal of medicinal chemistry 20100826 |
Identification of N-(2-(azepan-1-yl)-2-phenylethyl)-benzenesulfonamides as novel inhibitors of GlyT1. | Bioorganic & medicinal chemistry letters 20100815 |
2-Methyl-N-(2-methyl-benzo-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20100801 |
N-(4-Chloro-benzo-yl)-2-methyl-benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20100801 |
Cell adhesion to unnatural ligands mediated by a bifunctional protein. | Journal of the American Chemical Society 20100721 |
Pteridine-sulfonamide conjugates as dual inhibitors of carbonic anhydrases and dihydrofolate reductase with potential antitumor activity. | Bioorganic & medicinal chemistry 20100715 |
Coumarinyl-substituted sulfonamides strongly inhibit several human carbonic anhydrase isoforms: solution and crystallographic investigations. | Bioorganic & medicinal chemistry 20100715 |
Synthesis of quinazolines from N-(2-nitrophenylsulfonyl)iminodiacetate and alpha-(2-nitrophenylsulfonyl)amino ketones via 2H-indazole 1-oxides. | The Journal of organic chemistry 20100702 |
Synthesis and in vitro anticancer screening of some novel 4-[2-amino-3-cyano-4-substituted-5,6,7,8-tetrahydroquinolin-1-(4H)-yl]benzenesulfonamides. | European journal of medicinal chemistry 20100701 |
2,4-Dichloro-N-(3-methyl-phen-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20100701 |
2,4-Dichloro-N-(3-chloro-phen-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20100701 |
N-(4-Methyl-benzo-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20100701 |
New hydroxypyrimidinone-containing sulfonamides as carbonic anhydrase inhibitors also acting as MMP inhibitors. | Bioorganic & medicinal chemistry letters 20100615 |
A rationale for the activity profile of benzenesulfonamide derivatives as cyclooxygenase (COX) inhibitors. | European journal of medicinal chemistry 20100601 |
4-Chloro-N-(3,4-dimethyl-phen-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20100601 |
N-(Phenyl-sulfon-yl)acetamide. | Acta crystallographica. Section E, Structure reports online 20100601 |
2-Chloro-N-(3-chloro-benzo-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20100601 |
2-Chloro-N-(4-methyl-benzo-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20100601 |
Correlation analyses on binding affinity of substituted benzenesulfonamides with carbonic anhydrase using ab initio MO calculations on their complex structures. | Journal of chemical information and modeling 20100524 |
3D-QSAR study of benzene sulfonamide analogs as carbonic anhydrase II inhibitors. | Bioorganic & medicinal chemistry letters 20100515 |
Thioether benzenesulfonamide inhibitors of carbonic anhydrases II and IV: structure-based drug design, synthesis, and biological evaluation. | Bioorganic & medicinal chemistry 20100501 |
17,18-Dibromo-8-methyl-4,12-ditosyl-3,4,5,6,7,8,9,10,11,12,13,14-dodeca-hydro-2H-benzo[b][1,4,7,11,15]dioxatriaza-cyclo-hepta-decine. | Acta crystallographica. Section E, Structure reports online 20100501 |
N-Phenyl-N-(prop-2-en-1-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20100501 |
N-(4-Hydroxy-phen-yl)benzene-sulfon-amide. | Acta crystallographica. Section E, Structure reports online 20100501 |
N-(3,5-Dichloro-phen-yl)-2,4-dimethyl-benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20100501 |
N-(2,6-Dimethyl-phen-yl)-4-methyl-benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20100501 |
catena-Poly[neodymium(III)-bis-[μ-N-(dimorpholinophosphor-yl)benzene-sulfonamidato]-sodium(I)-bis-[μ-N-(dimorpholinophosphor-yl)benzene-sulfonamidato]]. | Acta crystallographica. Section E, Structure reports online 20100401 |
N-Cyclo-hexyl-4-meth-yl-N-propyl-benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20100401 |
2-Methyl-N-(4-methyl-benzo-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20100401 |
2,4-Dimethyl-N-(3-methyl-phen-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20100401 |
Recognition and binding of a helix-loop-helix peptide to carbonic anhydrase occurs via partly folded intermediate structures. | Biophysical journal 20100203 |
N-(2-Chloro-benzo-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20100201 |
N-(4-Chloro-benzo-yl)-4-methyl-benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20100201 |
2-Methyl-N-(3-methyl-benzo-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20100201 |
cis-N-(2-Hydroxy-cyclo-hexyl)-p-toluene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20100201 |
Computational study of the interactions between guanine derivatives and cyclin-dependent kinase 2 (CDK2) by CoMFA and QM/MM. | Journal of chemical information and modeling 20100101 |
Synthesis and biological activities of some novel triazoloquinazolines and triazinoquinazolines containing benzenesulfonamide moieties. | Arzneimittel-Forschung 20100101 |
Tamsulosin-induced severe hypotension during general anesthesia: a case report. | Journal of medical case reports 20100101 |
Pharmacophore elucidation and molecular docking studies on 5-phenyl-1-(3-pyridyl)-1h-1,2,4-triazole-3-carboxylic acid derivatives as COX-2 inhibitors. | Scientia pharmaceutica 20100101 |
[Synthesis and investigation on antidiabetic activity of 4-(1-aryl-3-oxo-5-phenylpentylamino) benzenesulfonamide]. | Yao xue xue bao = Acta pharmaceutica Sinica 20100101 |
N-Cyclo-hexyl-N-ethyl-4-methyl-benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20100101 |
N,N'-Bis(phenyl-sulfon-yl)succinamide. | Acta crystallographica. Section E, Structure reports online 20100101 |
N,N'-Bis(phenyl-sulfon-yl)maleamide. | Acta crystallographica. Section E, Structure reports online 20100101 |
Environmentally sensitive fluorescent sensors based on synthetic peptides. | Sensors (Basel, Switzerland) 20100101 |
Radiolabelling of proteins with fluorine-18 via click chemistry. | Chemical communications (Cambridge, England) 20091228 |
Thermodynamic optimisation in drug discovery: a case study using carbonic anhydrase inhibitors. | ChemMedChem 20091201 |
N-Benzyl-N-cyclo-hexyl-benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20091201 |
4-Benzene-sulfonamido-benzoic acid. | Acta crystallographica. Section E, Structure reports online 20091201 |
N-Cyclo-hexyl-N-(prop-2-en-1-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20091201 |
N-Benzyl-N-cyclo-hexyl-4-methyl-benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20091201 |
N-(4-Chloro-benzo-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20091201 |
N-Cyclo-hexyl-N-propyl-benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20091201 |
4-Methyl-N-(2-methyl-phen-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20091201 |
Discovery and optimization of novel 4-[(aminocarbonyl)amino]-N-[4-(2-aminoethyl)phenyl]benzenesulfonamide ghrelin receptor antagonists. | Bioorganic & medicinal chemistry letters 20091101 |
In vivo and in vitro anti-leishmanial activities of 4-nitro-N-pyrimidin- and N-pyrazin-2-ylbenzenesulfonamides, and N2-(4-nitrophenyl)-N1-propylglycinamide. | Bioorganic & medicinal chemistry 20091101 |
2,2-Dimethyl-N-(phenyl-sulfon-yl)acetamide. | Acta crystallographica. Section E, Structure reports online 20091101 |
N-(3-Chloro-benzo-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20091101 |
N-(2,5-Dimethyl-phen-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20091101 |
N-Cyclohexyl-N-methylbenzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20091101 |
Theoretical characterization of substrate access/exit channels in the human cytochrome P450 3A4 enzyme: involvement of phenylalanine residues in the gating mechanism. | The journal of physical chemistry. B 20091001 |
N-Benzo-ylbenzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20091001 |
Carbonic anhydrase inhibitors. Inhibition of the Rv1284 and Rv3273 beta-carbonic anhydrases from Mycobacterium tuberculosis with diazenylbenzenesulfonamides. | Bioorganic & medicinal chemistry letters 20090901 |
2-Chloro-benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20090901 |
N-(2-Formyl-phen-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20090901 |
N-(2-Acetyl-phen-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20090901 |
o-Toluene-sulfonamide: a redetermination. | Acta crystallographica. Section E, Structure reports online 20090901 |
4-[(Z)-(2-Eth-oxy-4-oxochroman-3-yl-idene)methyl-amino]benzene-sulfonamide monohydrate. | Acta crystallographica. Section E, Structure reports online 20090801 |
2,4-Dichloro-N-(3,4-dichloro-phen-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20090801 |
In vitro pharmacological characterization of a novel allosteric modulator of alpha 7 neuronal acetylcholine receptor, 4-(5-(4-chlorophenyl)-2-methyl-3-propionyl-1H-pyrrol-1-yl)benzenesulfonamide (A-867744), exhibiting unique pharmacological profile. | The Journal of pharmacology and experimental therapeutics 20090701 |
Hybrid molecules between benzenesulfonamides and active antimicrobial benzo[d]isothiazol-3-ones. | European journal of medicinal chemistry 20090601 |
Toward the development of metal-based synthetic nucleases: DNA binding and oxidative DNA cleavage of a mixed copper(II) complex with N-(9H-purin-6-yl)benzenesulfonamide and 1,10-phenantroline. Antitumor activity in human Caco-2 cells and Jurkat T lymphocytes. Evaluation of p53 and Bcl-2 proteins in the apoptotic mechanism. | Journal of inorganic biochemistry 20090601 |
Sodium N-chloro-2-methyl-benzene-sulfonamidate sesquihydrate. | Acta crystallographica. Section E, Structure reports online 20090601 |
4-Methyl-N-phenyl-benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20090601 |
Discovery of 4-(5-(4-chlorophenyl)-2-methyl-3-propionyl-1H-pyrrol-1-yl)benzenesulfonamide (A-867744) as a novel positive allosteric modulator of the alpha7 nicotinic acetylcholine receptor. | Journal of medicinal chemistry 20090528 |
Investigation of the fate of sulfonamides downgradient of a decommissioned sewage farm near Berlin, Germany. | Journal of contaminant hydrology 20090512 |
Ligand-directed tosyl chemistry for protein labeling in vivo. | Nature chemical biology 20090501 |
Synthesis and biological evaluation of novel pyrazoles and pyrazolo[3,4-d]pyrimidines incorporating a benzenesulfonamide moiety. | Archiv der Pharmazie 20090401 |
N-(3,4-Dimethyl-phen-yl)-4-methyl-benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20090401 |
Addition reactions of chloro- or iodomethyllithium to imines. Synthesis of enantiopure aziridines and beta-chloroamines. | The Journal of organic chemistry 20090320 |
Synthesis and biological evaluation of sulfonylurea and thiourea derivatives substituted with benzenesulfonamide groups as potential hypoglycemic agents. | Bioorganic & medicinal chemistry letters 20090315 |
Improvement of monolithic solid material by utilization of spacer for identification of the target using affinity resins. | Bioorganic & medicinal chemistry letters 20090301 |
Carbonic anhydrase inhibitors: two-prong versus mono-prong inhibitors of isoforms I, II, IX, and XII exemplified by photochromic cis-1,2-alpha-dithienylethene derivatives. | Bioorganic & medicinal chemistry letters 20090301 |
Ethyl 2-[N-(2-Formyl-phen-yl)benzene-sulfonamido]acetate. | Acta crystallographica. Section E, Structure reports online 20090301 |
A novel class of allosteric modulators of AMPA/Kainate receptors. | Bioorganic & medicinal chemistry letters 20090215 |
Synthesis and biological evaluation of benzenesulfonamide-substituted 4-(6-alkylpyridin-2-yl)-5-(quinoxalin-6-yl)imidazoles as transforming growth factor-beta type 1 receptor kinase inhibitors. | European journal of medicinal chemistry 20090201 |
Synthesis of some pyrazolyl benzenesulfonamide derivatives as dual anti-inflammatory antimicrobial agents. | Journal of enzyme inhibition and medicinal chemistry 20090201 |
N-(2,3-Dimethyl-phen-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20090201 |
Cryptophane xenon-129 nuclear magnetic resonance biosensors targeting human carbonic anhydrase. | Journal of the American Chemical Society 20090121 |
Synthesis and antiinflammatory activity of some new 1,3,5-trisubstituted pyrazolines bearing benzene sulfonamide. | Bioorganic & medicinal chemistry letters 20090101 |
Label-free determination of protein-ligand binding constants using mass spectrometry and validation using surface plasmon resonance and isothermal titration calorimetry. | Journal of molecular recognition : JMR 20090101 |
Synthesis and Antiviral Studies of Novel N-Sulphonamidomethyl piperazinyl Fluoroquinolones. | Indian journal of pharmaceutical sciences 20090101 |
Dual inhibitors of matrix metalloproteinases and carbonic anhydrases: iminodiacetyl-based hydroxamate-benzenesulfonamide conjugates. | Journal of medicinal chemistry 20081225 |
Synthesis of biologically active N-methyl derivatives of amidines and cyclized five-membered products of amidines with oxalyl chloride. | European journal of medicinal chemistry 20081201 |
Recent improvements in the development of A(2B) adenosine receptor agonists. | Purinergic signalling 20081201 |
Effect of the oral absorption of benzenesulfonanilide-type cyclooxygenase-1 inhibitors on analgesic action and gastric ulcer formation. | Journal of pharmaceutical sciences 20081201 |
N-(3,5-Dichloro-phen-yl)benzene-sulfonamide. | Acta crystallographica. Section E, Structure reports online 20081101 |
External pH influences the transcriptional profile of the carbonic anhydrase, CAH-4b in Caenorhabditis elegans. | Molecular and biochemical parasitology 20081001 |
Tetra-aquabis-(2-sulfamoylbenzoato)manganese(II). | Acta crystallographica. Section E, Structure reports online 20081001 |
Residual ligand entropy in the binding of p-substituted benzenesulfonamide ligands to bovine carbonic anhydrase II. | Journal of the American Chemical Society 20080917 |
Chromofluorescent indicator for intracellular Zn2+/Hg2+ dynamic exchange. | Organic letters 20080904 |
Photophysical and complexation properties of benzenesulfonamide derivatives with different donor and acceptor moieties. | Journal of fluorescence 20080901 |
Tetramethylcyclopropyl analogue of the leading antiepileptic drug, valproic acid: evaluation of the teratogenic effects of its amide derivatives in NMRI mice. | Birth defects research. Part A, Clinical and molecular teratology 20080901 |
Chemometrical examination of active parameters and interactions in flow injection-capillary electrophoresis. | Electrophoresis 20080901 |
Inhibition of human mitochondrial carbonic anhydrases VA and VB with para-(4-phenyltriazole-1-yl)-benzenesulfonamide derivatives. | Bioorganic & medicinal chemistry letters 20080815 |
2,2,2-Trimethyl-N-(phenyl-sulfon-yl)-acetamide. | Acta crystallographica. Section E, Structure reports online 20080801 |
2,2-Dichloro-N-(phenyl-sulfon-yl)-acetamide. | Acta crystallographica. Section E, Structure reports online 20080801 |
Affinity-labeling-based introduction of a reactive handle for natural protein modification. | Chemistry, an Asian journal 20080707 |
Carbonic anhydrase inhibitors: design of spin-labeled sulfonamides incorporating TEMPO moieties as probes for cytosolic or transmembrane isozymes. | Bioorganic & medicinal chemistry letters 20080615 |
Exploration of physicochemical properties and molecular modelling studies of 2-sulfonyl-phenyl-3-phenyl-indole analogs as cyclooxygenase-2 inhibitors. | European journal of medicinal chemistry 20080601 |
Similar sulfonamides with different crystal structures: sulfasymazine and sulfatriazine. | Acta crystallographica. Section C, Crystal structure communications 20080601 |
Antidiabetic activity of N-(6-substituted-1,3-benzothiazol-2-yl)benzenesulfonamides. | Bioorganic & medicinal chemistry letters 20080501 |
2-[N-(X-chlorophenyl)carbamoyl]benzenesulfonamide (with X = 2 and 4). | Acta crystallographica. Section C, Crystal structure communications 20080501 |
Functional human 5-HT6 receptor assay for high throughput screening of chemical ligands and binding proteins. | Combinatorial chemistry & high throughput screening 20080501 |
Behaviour and biodegradation of sulfonamides (p-TSA, o-TSA, BSA) during drinking water treatment. | Chemosphere 20080401 |
Carbonic anhydrase inhibitors: inhibition of human cytosolic isozymes I and II and tumor-associated isozymes IX and XII with S-substituted 4-chloro-2-mercapto-5-methyl-benzenesulfonamides. | Bioorganic & medicinal chemistry 20080401 |
Design and synthesis of N-(3,5-difluoro-4-hydroxyphenyl)benzenesulfonamides as aldose reductase inhibitors. | Bioorganic & medicinal chemistry 20080401 |
Electrophysiological characterization of a novel Kv channel blocker N,N'-[oxybis(2,1-ethanediyloxy-2,1-ethanediyl) ]bis(4-methyl)-benzenesulfonamide found in virtual screening. | Acta pharmacologica Sinica 20080401 |
Ethyl 2-(bromo-meth-yl)-5-meth-oxy-1-phenyl-sulfonyl-1H-indole-3-carboxyl-ate. | Acta crystallographica. Section E, Structure reports online 20080401 |
Identification and significance of sulphonamides (p-TSA, o-TSA, BSA) in an urban water cycle (Berlin, Germany). | Water research 20080301 |
Selective COX-2 inhibitors. Part 2: synthesis and biological evaluation of 4-benzylideneamino- and 4-phenyliminomethyl-benzenesulfonamides. | Bioorganic & medicinal chemistry 20080301 |
Pyrazolo-triazolo-pyrimidines as adenosine receptor antagonists: Effect of the N-5 bond type on the affinity and selectivity at the four adenosine receptor subtypes. | Purinergic signalling 20080301 |
Synthesis and cyclooxygenase inhibitory activities of linear 1-(methanesulfonylphenyl or benzenesulfonamido)-2-(pyridyl)acetylene regioisomers. | Bioorganic & medicinal chemistry 20080215 |
Benzenesulfonamide indole inhibitors of cytosolic phospholipase A2alpha: optimization of in vitro potency and rat pharmacokinetics for oral efficacy. | Bioorganic & medicinal chemistry 20080201 |
Metal-based sulfonamides: their preparation, characterization and in-vitro antibacterial, antifungal & cytotoxic properties. X-ray structure of 4-[(2-hydroxybenzylidene) amino] benzenesulfonamide. | Journal of enzyme inhibition and medicinal chemistry 20080201 |
Ethyl 2-[(phenyl-sulfan-yl)meth-yl]-1-(phenyl-sulfon-yl)-1H-indole-3-carboxyl-ate. | Acta crystallographica. Section E, Structure reports online 20080201 |
(2-Methyl-1-phenyl-sulfonyl-1H-indol-3-yl)methanol. | Acta crystallographica. Section E, Structure reports online 20080201 |
Carbonic anhydrase inhibitors: copper(II) complexes of polyamino-polycarboxylamido aromatic/heterocyclic sulfonamides are very potent inhibitors of the tumor-associated isoforms IX and XII. | Bioorganic & medicinal chemistry letters 20080115 |
New celecoxib derivatives as anti-inflammatory agents. | Journal of medicinal chemistry 20080110 |
Identification of N-(quinolin-8-yl)benzenesulfonamides as agents capable of down-regulating NFkappaB activity within two separate high-throughput screens of NFkappaB activation. | Bioorganic & medicinal chemistry letters 20080101 |
An efficient solvent-free synthesis of benzoxanthenes catalyzed by BSA or O-TSA. | Preparative biochemistry & biotechnology 20080101 |
Antimicrobial activity of some sulfonamide derivatives on clinical isolates of Staphylococus aureus. | Annals of clinical microbiology and antimicrobials 20080101 |
Binding modes of two novel non-nucleoside reverse transcriptase inhibitors, YM-215389 and YM-228855, to HIV type-1 reverse transcriptase. | Antiviral chemistry & chemotherapy 20080101 |
Small molecule inhibitors of integrin alpha2beta1. | Journal of medicinal chemistry 20071101 |
A remarkable accelerating effect of Ag-salt on intramolecular cyclization of o-(1-alkynyl)benzenesulfonamides. | The Journal of organic chemistry 20071026 |
A strategy for designing 'multi-prong' enzyme inhibitors by incorporating selective ligands to the liposomal surface. | Chemical communications (Cambridge, England) 20070828 |
Design, synthesis and pharmacological evaluation of 4-[2-alkylthio-5(4)-(4-substitutedphenyl)imidazole-4(5)yl]benzenesulfonamides as selective COX-2 inhibitors. | Acta pharmacologica Sinica 20070801 |
Quantitative determination of three sulfonamides in environmental water samples using liquid chromatography coupled to electrospray tandem mass spectrometry. | Journal of chromatography. A 20070720 |
Structure-based design of 2-arylamino-4-cyclohexylmethoxy-5-nitroso-6-aminopyrimidine inhibitors of cyclin-dependent kinase 2. | Organic & biomolecular chemistry 20070521 |
Structural analysis of charge discrimination in the binding of inhibitors to human carbonic anhydrases I and II. | Journal of the American Chemical Society 20070502 |
Pharmacophoric 2-hydroxyalkyl benzenesulfonamide: a single-step synthesis from benzenesulfonamide via hemiaminal. | European journal of medicinal chemistry 20070401 |
Carbonic anhydrase inhibitors: inhibition of cytosolic/tumor-associated isoforms I, II, and IX with iminodiacetic carboxylates/hydroxamates also incorporating benzenesulfonamide moieties. | Bioorganic & medicinal chemistry letters 20070315 |
Synthesis and in vivo evaluation of [18F]-4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-yl]benzenesulfonamide as a PET imaging probe for COX-2 expression. | Bioorganic & medicinal chemistry 20070215 |
Dependence of effective molarity on linker length for an intramolecular protein-ligand system. | Journal of the American Chemical Society 20070207 |
Thermodynamic parameters for the association of fluorinated benzenesulfonamides with bovine carbonic anhydrase II. | Chemistry, an Asian journal 20070108 |
Strategies for controlled placement of nanoscale building blocks. | Nanoscale research letters 20070101 |
Discovery of HIV-1 protease inhibitors with picomolar affinities incorporating N-aryl-oxazolidinone-5-carboxamides as novel P2 ligands. | Journal of medicinal chemistry 20061214 |
Thiol-mediated anchoring of ligands to self-assembled monolayers for studies of biospecific interactions. | Langmuir : the ACS journal of surfaces and colloids 20061121 |
Synthesis and in vitro antitumor evaluation of some indeno[1,2-c]pyrazol(in)es substituted with sulfonamide, sulfonylurea(-thiourea) pharmacophores, and some derived thiazole ring systems. | Bioorganic & medicinal chemistry 20061001 |
Intracellular inhibition of carboxylesterases by benzil: modulation of CPT-11 cytotoxicity. | Molecular cancer therapeutics 20060901 |
Binding of sulfonyl-containing arylalkylamines at human 5-HT6 serotonin receptors. | Journal of medicinal chemistry 20060824 |
Urotensin-II blockade with SB-611812 attenuates cardiac dysfunction in a rat model of coronary artery ligation. | Journal of molecular and cellular cardiology 20060801 |
Sorption-desorption of flucarbazone and propoxycarbazone and their benzenesulfonamide and triazolinone metabolites in two soils. | Pest management science 20060701 |
Carbonic anhydrase inhibitors: cloning and sulfonamide inhibition studies of a carboxyterminal truncated alpha-carbonic anhydrase from Helicobacter pylori. | Bioorganic & medicinal chemistry letters 20060415 |
Molecular structure and conformations of benzenesulfonamide: gas electron diffraction and quantum chemical calculations. | The Journal of organic chemistry 20060414 |
Benzoxazole benzenesulfonamides are novel allosteric inhibitors of fructose-1,6-bisphosphatase with a distinct binding mode. | Bioorganic & medicinal chemistry letters 20060401 |
Carbonic anhydrase inhibitors: DNA cloning and inhibition studies of the alpha-carbonic anhydrase from Helicobacter pylori, a new target for developing sulfonamide and sulfamate gastric drugs. | Journal of medicinal chemistry 20060323 |
Ultrahigh resolution crystal structures of human carbonic anhydrases I and II complexed with 'two-prong' inhibitors reveal the molecular basis of high affinity. | Journal of the American Chemical Society 20060308 |
Carbonic anhydrase inhibitors: Valdecoxib binds to a different active site region of the human isoform II as compared to the structurally related cyclooxygenase II 'selective' inhibitor celecoxib. | Bioorganic & medicinal chemistry letters 20060115 |
Downregulation of survivin expression and concomitant induction of apoptosis by celecoxib and its non-cyclooxygenase-2-inhibitory analog, dimethyl-celecoxib (DMC), in tumor cells in vitro and in vivo. | Molecular cancer 20060101 |
Short communication inhibitory activity of 4-[(1,2-dihydro-2-oxo-3H-indol-3-ylidene)amino]-N-(4,6-dimethylpyrimidin-2-yl) benzenesulphonamide and its derivatives against orthopoxvirus replication in vitro. | Antiviral chemistry & chemotherapy 20060101 |
CC 05, a novel anti-inflammatory compound, exerts its effect by inhibition of cyclooxygenase-2 activity. | European journal of pharmacology 20050927 |
QSAR analysis of thiazole benzenesulfonamide substituted 3-pyridylethanolamines as beta3-adrenergic receptor agonist. | Bioorganic & medicinal chemistry letters 20050615 |
Carbonic anhydrase inhibitors. Inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, IX, and XII with Schiff's bases incorporating chromone and aromatic sulfonamide moieties, and their zinc complexes. | Bioorganic & medicinal chemistry letters 20050615 |
Synthesis and biological evaluation of 3,4-diphenyl-1,2,5-oxadiazole-2-oxides and 3,4-diphenyl-1,2,5-oxadiazoles as potential hybrid COX-2 inhibitor/nitric oxide donor agents. | Bioorganic & medicinal chemistry 20050415 |
Design, synthesis, and biological evaluation of N-acetyl-2-carboxybenzenesulfonamides: a novel class of cyclooxygenase-2 (COX-2) inhibitors. | Bioorganic & medicinal chemistry 20050401 |
Carbonic anhydrase inhibitors: X-ray crystal structure of a benzenesulfonamide strong CA II and CA IX inhibitor bearing a pentafluorophenylaminothioureido tail in complex with isozyme II. | Bioorganic & medicinal chemistry letters 20050401 |
Benzenesulfonamide analogs of fluoroquinolones. Antibacterial activity and QSAR studies. | European journal of medicinal chemistry 20050401 |
Discovery and selection of TMC114, a next generation HIV-1 protease inhibitor. | Journal of medicinal chemistry 20050324 |
Spacer-based selectivity in the binding of 'two-prong' ligands to recombinant human carbonic anhydrase I. | Biochemistry 20050308 |
Studies of non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 2: synthesis and structure-activity relationships of 2-cyano and 2-hydroxy thiazolidenebenzenesulfonamide derivatives. | Bioorganic & medicinal chemistry 20050215 |
QSAR studies on benzene sulfonamide carbonic anhydrase inhibitors: need of hydrophobic parameter for topological modeling of binding constants of sulfonamides to human CA-II. | Bioorganic & medicinal chemistry letters 20050215 |
Novel use of chemical shift in NMR as molecular descriptor: a first report on modeling carbonic anhydrase inhibitory activity and related parameters. | Bioorganic & medicinal chemistry letters 20050215 |
Characterization of beta3-adrenergic receptor: determination of pharmacophore and 3D QSAR model for beta3 adrenergic receptor agonism. | Journal of computer-aided molecular design 20050201 |
Predictive flip regression: a technique for QSAR of derivatives of symmetric molecules. | Journal of chemical information and modeling 20050101 |
In situ click chemistry: enzyme-generated inhibitors of carbonic anhydrase II. | Angewandte Chemie (International ed. in English) 20041217 |
Studies of nonnucleoside HIV-1 reverse transcriptase inhibitors. Part 1: Design and synthesis of thiazolidenebenzenesulfonamides. | Bioorganic & medicinal chemistry 20041201 |
Pharmacomodulation of a sulfamide 5-HT6 receptor ligand. | Journal of enzyme inhibition and medicinal chemistry 20041201 |
Topological modeling of lipophilicity, diuretic activity, and carbonic inhibition activity of benzene sulfonamides: a molecular connectivity approach. | Bioorganic & medicinal chemistry letters 20041115 |
Carbonic anhydrase inhibitors: inhibition of human cytosolic isozyme II and mitochondrial isozyme V with a series of benzene sulfonamide derivatives. | Bioorganic & medicinal chemistry letters 20041115 |
Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating 1,2,4-triazine moieties. | Bioorganic & medicinal chemistry letters 20041101 |
Two-prong inhibitors for human carbonic anhydrase II. | Journal of the American Chemical Society 20041020 |
Novel synthesis of 3,4-diarylisoxazole analogues of valdecoxib: reversal cyclooxygenase-2 selectivity by sulfonamide group removal. | Journal of medicinal chemistry 20040923 |
Protein surface-assisted enhancement in the binding affinity of an inhibitor for recombinant human carbonic anhydrase-II. | Journal of the American Chemical Society 20040908 |
Synthesis and antiviral activity of P1' arylsulfonamide azacyclic urea HIV protease inhibitors. | Bioorganic & medicinal chemistry letters 20040802 |
Synthesis, antiviral, and anti-HIV-1 integrase activities of 3-aroyl-1,1-dioxo-1,4,2-benzodithiazines. | Bioorganic & medicinal chemistry 20040701 |
Rewiring cell adhesion. | Journal of the American Chemical Society 20040602 |
A versatile polypeptide platform for integrated recognition and reporting: affinity arrays for protein-ligand interaction analysis. | Chemistry (Weinheim an der Bergstrasse, Germany) 20040517 |
New heteroarylbenzenesulphonamides as matrix metalloproteinase inhibitors. | Bioorganic & medicinal chemistry letters 20040308 |
Abeta aggregation inhibitors. Part 1: Synthesis and biological activity of phenylazo benzenesulfonamides. | Bioorganic & medicinal chemistry letters 20040308 |
QSAR study on benzenesulphonamide carbonic anhydrase inhibitors: topological approach using Balaban index. | Bioorganic & medicinal chemistry 20040215 |
Polar substitutions in the benzenesulfonamide ring of celecoxib afford a potent 1,5-diarylpyrazole class of COX-2 inhibitors. | Bioorganic & medicinal chemistry letters 20040119 |
Application of CoMFA and CoMSIA 3D-QSAR and docking studies in optimization of mercaptobenzenesulfonamides as HIV-1 integrase inhibitors. | Journal of medicinal chemistry 20040115 |
QSAR study using topological indices for inhibition of carbonic anhydrase II by sulfanilamides and Schiff bases. | Molecular diversity 20040101 |
Synthesis and cyclooxygenase-2 inhibiting property of 1,5-diarylpyrazoles with substituted benzenesulfonamide moiety as pharmacophore: Preparation of sodium salt for injectable formulation. | Journal of medicinal chemistry 20030911 |
Sorption-desorption of two 'aged' sulfonylaminocarbonyltriazolinone herbicide metabolites in soil. | Journal of agricultural and food chemistry 20030604 |
Synthesis of 1-(6-chloro-1,1-dioxo-1,4,2-benzodithiazin-3-yl)semi-carbazides and their transformation into 4-chloro-2-mercapto-N-(4,5-dihydro-5-oxo-4-phenyl-1H-1,2,4-triazol-3-yl)benzenesulfonamides as potential anticancer and anti-HIV agents. | Farmaco (Societa chimica italiana : 1989) 20030601 |
Valdecoxib-induced toxic epidermal necrolysis in a patient allergic to sulfa drugs. | Pharmacotherapy 20030401 |
Tripodal ligand incorporating dual fluorescent ionophore: a coordinative control of photoinduced electron transfer. | Photochemical & photobiological sciences : Official journal of the European Photochemistry Association and the European Society for Photobiology 20030301 |
Synthesis of heteroaromatic analogues of (2-aryl-1-cyclopentenyl-1-alkylidene)-(arylmethyloxy)amine COX-2 inhibitors: effects on the inhibitory activity of the replacement of the cyclopentene central core with pyrazole, thiophene or isoxazole ring. | European journal of medicinal chemistry 20030201 |
Using cyclooxygenase-2 inhibitors as molecular platforms to develop a new class of apoptosis-inducing agents. | Journal of the National Cancer Institute 20021204 |
Diversity in the oxidation of substrates by cytochrome P450 2D6: lack of an obligatory role of aspartate 301-substrate electrostatic bonding. | Biochemistry 20020910 |
An excretion balance and pharmacokinetic study of the novel anticancer agent E7070 in cancer patients. | Anti-cancer drugs 20020901 |
The pharmacokinetics of a thiazole benzenesulfonamide beta 3-adrenergic receptor agonist and its analogs in rats, dogs, and monkeys: improving oral bioavailability. | Drug metabolism and disposition: the biological fate of chemicals 20020701 |
Metabolism of a thiazole benzenesulfonamide derivative, a potent and elective agonist of the human beta3-adrenergic receptor, in rats: identification of a novel isethionic acid conjugate. | Drug metabolism and disposition: the biological fate of chemicals 20020701 |
Effects of soil pH and soil water content on prosulfuron dissipation. | Journal of agricultural and food chemistry 20020522 |
Enantiomeric separation of a thiazolbenzenesulfonamide compound using packed-column subcritical fluid chromatography. | Chirality 20020515 |
Synthesis of unsymmetrical aroyl acyl imides by aminocarbonylation of aryl bromides. | The Journal of organic chemistry 20020125 |
Rational determination of transfer free energies of small drugs across the water-oil interface. | Journal of medicinal chemistry 20020103 |
Synthesis, characterization and antifungal activities of some benzenesulphonylamino acid derivatives. | Bollettino chimico farmaceutico 20020101 |
Synthesis and anti-HIV activity of 4-[(1,2-dihydro-2-oxo-3H-indol-3-ylidene) amino]-N(4,6-dimethyl-2-pyrimidinyl)-benzene sulfonamide and its derivatives. | European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20011201 |
Comparative study of new benzenesulphonamide fluoroquinolones structurally related to ciprofloxacin against selected ciprofloxacin-susceptible and -resistant Gram-positive cocci. | The Journal of antimicrobial chemotherapy 20011101 |
Subtle differences in dissociation rates of interactions between destabilized human carbonic anhydrase II mutants and immobilized benzenesulfonamide inhibitors probed by a surface plasmon resonance biosensor. | Analytical biochemistry 20010915 |
Two isomorphous benzenesulfonamide crystal structures determined by intermolecular C-H...O, C-H...pi and C-H...Cl interactions. | Acta crystallographica. Section C, Crystal structure communications 20010901 |
Synthesis of optically active N-(2-pyridyloxiran-2-ylmethyl) benzenesulfonamide derivatives and their herbicidal activity. | Bioscience, biotechnology, and biochemistry 20010701 |
Ethenesulfonamide derivatives, a novel class of orally active endothelin-A receptor antagonists. | Chemical & pharmaceutical bulletin 20010501 |
QSAR of antineoplastics IV: Hansch analysis of N-(7-indolyl)benzenesulfonamides against KB human nasopharynx carcinoma, colon 38 murine adenocarcinoma and P388 murine leukemia cell lines. | Drug design and discovery 20010101 |
QSAR of antineoplastics V: Exploration of receptor interaction sites of antitumor N-(7-indolyl)benzenesulfonamides targeting GI phase using electrotopological state atom index. | Drug design and discovery 20010101 |
Design and synthesis of benzoic acid derivatives as influenza neuraminidase inhibitors using structure-based drug design. | Journal of medicinal chemistry 19971205 |