3-Pyrroline
Title | Journal |
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Synthesis of sulfur containing dihydro-pyrrolo derivatives and their biological evaluation as antioxidants. | Bioorganic & medicinal chemistry 20120901 |
Synthesis of 1,2-disubstituted cyclopentenes by palladium-catalyzed reaction of homopropargyl-substituted dicarbonyl compounds with organic halides via 5-endo-dig cyclization. | Organic letters 20120601 |
A highly enantioselective approach towards 2-substituted 3-bromopyrrolidines. | Organic & biomolecular chemistry 20120521 |
3D-QSAR studies of dihydropyrazole and dihydropyrrole derivatives as inhibitors of human mitotic kinesin Eg5 based on molecular docking. | Molecules (Basel, Switzerland) 20120217 |
Exploiting the ring strain in bicyclo[2.2.1]heptane systems for the stereoselective preparation of highly functionalized cyclopentene, dihydrofuran, pyrroline, and pyrrolidine scaffolds. | Organic letters 20111202 |
A computational reinvestigation of the formation of N-alkylpyrroles via intermolecular redox amination. | Organic letters 20111118 |
The catalytic asymmetric 1,3-dipolar cycloaddition of ynones with azomethine ylides. | Organic letters 20110902 |
Silver-catalyzed intramolecular chloroamination of allenes: easy access to functionalized 3-pyrroline and pyrrole derivatives. | Organic letters 20110902 |
A straightforward route to enantiopure 2-substituted-3,4-dehydro-β-proline via ring closing metathesis. | Amino acids 20110801 |
Tungsten(0)- and rhenium(I)-catalyzed tandem cyclization of acetylenic dienol silyl ethers based on geminal carbo-functionalization of alkynes. | Chemistry (Weinheim an der Bergstrasse, Germany) 20110418 |
Gold(I)-catalyzed cycloisomerization of 1,6-diynes: synthesis of 2,3-disubstituted 3-pyrroline derivatives. | Angewandte Chemie (International ed. in English) 20110307 |
(5S)-3-Chloro-4-(2,5-dihydro-1H-pyrrol-1-yl)-5-[(1R,2S,5R)-2-isopropyl-5-methyl-cyclo-hex-yloxy]furan-2(5H)-one. | Acta crystallographica. Section E, Structure reports online 20110101 |
Identification and characterization of mechanism of action of P61-E7, a novel phosphine catalysis-based inhibitor of geranylgeranyltransferase-I. | PloS one 20110101 |
The ultraviolet photodissociation of axial and equatorial conformers of 3-pyrroline. | The Journal of chemical physics 20101121 |
Ruthenium-catalyzed tandem ring-opening/ring-closing/cross-metathesis of 1,6-cyclopropene-ynes and olefins for the construction of the 3-pyrroline skeleton. | Organic letters 20101015 |
Biodegradation of the major color containing compounds in distillery wastewater by an aerobic bacterial culture and characterization of their metabolites. | Biodegradation 20100901 |
Asymmetric one-pot sequential organo- and gold catalysis for the enantioselective synthesis of dihydropyrrole derivatives. | Chemistry (Weinheim an der Bergstrasse, Germany) 20100816 |
Asymmetric synthesis of 2-alkyl-substituted 2,5-dihydropyrroles from optically active aza-Baylis-Hillman adducts. Formal synthesis of (-)-trachelanthamidine. | The Journal of organic chemistry 20100604 |
8a-Methyl-5,6,8,8a,9,10-hexa-hydro-10,12a-epoxy-isoindolo[1,2-a]isoquinolinium iodide. | Acta crystallographica. Section E, Structure reports online 20100601 |
Mechanism study of the gold-catalyzed cycloisomerization of alpha-aminoallenes: oxidation state of active species and influence of counterion. | The journal of physical chemistry. A 20100408 |
Stereoselective synthesis of an active metabolite of the potent PI3 kinase inhibitor PKI-179. | The Journal of organic chemistry 20100305 |
Total synthesis of uniflorine A, casuarine, australine, 3-epi-australine, and 3,7-di-epi-australine from a common precursor. | The Journal of organic chemistry 20100205 |
Formation of N-alkylpyrroles via intermolecular redox amination. | Journal of the American Chemical Society 20091125 |
An efficient synthetic approach to polycyclic 2,5-dihydropyrroles from alpha-silyloxy ketones. | The Journal of organic chemistry 20091106 |
Zn and Fe complexes containing a redox active macrocyclic biquinazoline ligand. | Inorganic chemistry 20090406 |
Annulations of enantioenriched allenylsilanes with in situ generated iminium ions: stereoselective synthesis of diverse heterocycles. | Organic letters 20090115 |
Knorr-Rabe partial reduction of pyrroles: application to the synthesis of indolizidine alkaloids. | Beilstein journal of organic chemistry 20080101 |
Identification of novel chemical inhibitors for ubiquitin C-terminal hydrolase-L3 by virtual screening. | Bioorganic & medicinal chemistry 20071101 |
Microwave-assisted preparations of dihydropyrroles from alkenone O-phenyl oximes. | Chemical communications (Cambridge, England) 20071021 |
TD-DFT investigation of diarylethene dyes with cyclopentene, dihydrothiophene, and dihydropyrrole bridges. | The journal of physical chemistry. A 20070628 |
The double reduction of cyclic sulfonamides for the synthesis of (4S-Phenylpyrrolidin-2R-yl)methanol and 2S-methyl-4S-phenylpyrrolidine. | The Journal of organic chemistry 20070302 |
Highly potent 3-pyrroline mechanism-based inhibitors of bovine plasma amine oxidase and mass spectrometric confirmation of cofactor derivatization. | Bioorganic & medicinal chemistry 20070215 |
Total synthesis, molecular editing and evaluation of a tripyrrolic natural product: the case of 'butylcycloheptylprodigiosin'. | Chemistry (Weinheim an der Bergstrasse, Germany) 20070101 |
Design and synthesis of a 3,4-dehydroproline amide discovery library. | Journal of combinatorial chemistry 20070101 |
Efficient approach to the Azaspirane core of FR 901483. | Organic letters 20061012 |
Study on photochromism of diarylethenes with a 2,5-dihydropyrrole bridging unit: a convenient preparation of 3,4-diarylpyrroles from 3,4-diaryl-2,5-dihydropyrroles. | The Journal of organic chemistry 20050624 |
Molecular structure of 2,5-dihydropyrrole (C4NH7), obtained by gas-phase electron diffraction and theoretical calculations. | The journal of physical chemistry. A 20050609 |
In vitro antifungal activity of 2-(3,4-dimethyl-2,5-dihydro-1H-pyrrol-2-yl)-1-methylethyl pentanoate, a dihydropyrrole derivative. | Journal of medical microbiology 20050601 |
Chiral oxime ethers in asymmetric synthesis. O-(1-Phenylbutyl)benzyloxyacetaldoxime, a versatile reagent for the asymmetric synthesis of protected 1,2-aminoalcohols, alpha-amino acid derivatives, and 2-hydroxymethyl nitrogen heterocycles including iminosugars. | Organic & biomolecular chemistry 20050407 |
Synthesis of 4-aryl-2-pyrrolidones and beta-aryl-gamma-amino-butyric acid (GABA) analogues by Heck arylation of 3-pyrrolines with arenediazonium tetrafluoroborates. Synthesis of (+/-)-rolipram on a multigram scale and chromatographic resolution by semipreparative chiral simulated moving bed chromatography. | The Journal of organic chemistry 20050204 |
SM-216601, a novel parenteral 1beta-methylcarbapenem: structure-activity relationships of antibacterial activity and neurotoxicity in mice. | The Journal of antibiotics 20050201 |
Characterization of human liver cytochrome P450 enzymes involved in the metabolism of a new H+/K+-ATPase inhibitor KR-60436. | Toxicology letters 20050115 |
Solvent-dependent chemoselectivities in additions of beta-carbonyl imines to allyltrimethylsilane with CTAN. | The Journal of organic chemistry 20040917 |
Adsorption of 3-pyrroline on Si(100) from first principles. | The Journal of chemical physics 20040522 |
Fragmentation patterns of novel dispirocyclopiperazinium dibromides with strong analgesic activity under electrospray ionization tandem mass spectrometry conditions. | Rapid communications in mass spectrometry : RCM 20040101 |
Synthesis and insecticidal activity of novel N-oxydihydropyrrole derivatives with a substituted spirocyclohexyl group. | Bioscience, biotechnology, and biochemistry 20030601 |
A stereoselective and short total synthesis of the polyhydroxylated gamma-amino acid (-)-detoxinine, based on stereoselective preparation of dihydropyrrole derivatives from lithiated alkoxyallenes. | Chemistry (Weinheim an der Bergstrasse, Germany) 20030317 |
Synthesis and insecticidal activity of novel dihydropyrrole derivatives with N-sulfanyl, sulfinyl, and sulfonyl moieties. | Bioorganic & medicinal chemistry 20030220 |
Synthesis and insecticidal activity of N-oxydihydropyrroles: 4-hydroxy-3-mesityl-5,5-dimethyl derivatives with various substituents at the 1-position. | Bioscience, biotechnology, and biochemistry 20021101 |
3-pyrrolines are mechanism-based inactivators of the quinone-dependent amine oxidases but only substrates of the flavin-dependent amine oxidases. | Journal of the American Chemical Society 20021016 |
3-Pyrroline containing arylacetamides: a novel series of remarkably selective kappa-agonists. | Bioorganic & medicinal chemistry letters 20020902 |
Enantioselective total syntheses of manzamine a and related alkaloids. | Journal of the American Chemical Society 20020724 |
LC-MS/MS identification of in vitro metabolites of a new H+/K+ ATPase inhibitor, KR-60436 produced by rat and human liver microsomes. | Journal of pharmaceutical and biomedical analysis 20020601 |
A convenient method for 3-pyrroline synthesis. | Organic letters 20011018 |
[Development of aziridination and azetizination reactions of amino allenes using a palladium catalyst]. | Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan 20011001 |
Stereoselective synthesis of 2-alkenylaziridines and 2-alkenylazetidines by palladium-catalyzed intramolecular amination of alpha- and beta-amino allenes. | The Journal of organic chemistry 20010713 |