1-(2-methoxyphenyl)piperazine
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Structure-dependent inhibition of the human α1β2γ2 GABAA receptor by piperazine derivatives: A novel mode of action. | Neurotoxicology 20151201 |
Molecular determinants of selectivity and efficacy at the dopamine D3 receptor. | Journal of medicinal chemistry 20120809 |
A straightforward approach for engineering efficacy and selectivity at GPCRs. | Journal of medicinal chemistry 20120809 |
Investigations on the 1-(2-biphenyl)piperazine motif: identification of new potent and selective ligands for the serotonin(7) (5-HT(7)) receptor with agonist or antagonist action in vitro or ex vivo. | Journal of medicinal chemistry 20120726 |
Synthesis, characterization and biological evaluation of novel neutral fac-M(CO)3(SNO) complexes (M=Re, 99mTc) bearing the o-methoxyphenylpiperazine moiety. | Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine 20120601 |
MDHS 25 revisited: part 2, modified sampling and analytical procedures applied to HDI-based isocyanates. | The Annals of occupational hygiene 20120501 |
Amine-alkyl derivatives of hydantoin: new tool to combat resistant bacteria. | European journal of medicinal chemistry 20111201 |
Synthesis, alpha-adrenoceptors affinity and alpha 1-adrenoceptor antagonistic properties of some 1,4-substituted piperazine derivatives. | Die Pharmazie 20111001 |
Synthesis and in vivo evaluation of [O-methyl-11C] N-[3,5-dichloro-2-(methoxy)phenyl]-4-(methoxy)-3-(1-piperazinyl)benzenesulfonamide as an imaging probe for 5-HT6 receptors. | Bioorganic & medicinal chemistry 20110901 |
Effect of cyclosporin A on the uptake of D3-selective PET radiotracers in rat brain. | Nuclear medicine and biology 20110701 |
Synthesis and biological evaluation of new [Tc(N)(PS)]-based mixed-ligand compounds useful in the design of target-specific radiopharmaceuticals: the 2-methoxyphenylpiperazine dithiocarbamate derivatives as an example. | Journal of biological inorganic chemistry : JBIC : a publication of the Society of Biological Inorganic Chemistry 20110101 |
Antidepressant potential of nitrogen-containing heterocyclic moieties: An updated review. | Journal of pharmacy & bioallied sciences 20110101 |
3-(1-Adamant-yl)-1-{[4-(2-meth-oxy-phen-yl)piperazin-1-yl]meth-yl}-4-methyl-1H-1,2,4-triazole-5(4H)-thione. | Acta crystallographica. Section E, Structure reports online 20100701 |
Synthesis and characterization of environment-sensitive fluorescent ligands for human 5-HT1A receptors with 1-arylpiperazine structure. | Journal of medicinal chemistry 20091210 |
[(18)F]-labeled 2-methoxyphenylpiperazine derivative as a potential brain positron emission tomography imaging agent. | Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine 20091101 |
'Click' D(1) receptor agonists with a 5-HT(1A) receptor pharmacophore producing D(2) receptor activity. | Bioorganic & medicinal chemistry 20090715 |
Aniline in hydrolyzed urine and plasma--possible biomarkers for phenylisocyanate exposure. | Journal of occupational and environmental hygiene 20081001 |
Structural modifications of N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinehexanamides: influence on lipophilicity and 5-HT7 receptor activity. Part III. | Journal of medicinal chemistry 20080925 |
Underestimation of toluene diisocyanate concentration using long-term sampling with 1-(2-methoxyphenyl) piperazine impregnated filters. | International journal of hygiene and environmental health 20080701 |
Synthesis, alpha 1-adrenoceptor antagonist activity, and SAR study of novel arylpiperazine derivatives of phenytoin. | Bioorganic & medicinal chemistry 20080601 |
Quantitative monitoring of dermal and inhalation exposure to 1,6-hexamethylene diisocyanate monomer and oligomers. | Journal of environmental monitoring : JEM 20080401 |
Sampling and analytical methodology development for the determination of primary and secondary low molecular weight amines in ambient air. | Journal of environmental monitoring : JEM 20080301 |
Abstracts of papers presented at the 2007 pittsburgh conference. | Journal of automated methods & management in chemistry 20070101 |
Validation of a diffusive sampling method for airborne low-molecular isocyanates using 4-nitro-7-piperazinobenzo-2-oxa-1,3-diazole-impregnated filters and liquid chromatography-tandem mass spectrometry. | Journal of chromatography. A 20061117 |
The synthesis of L-carvone and limonene derivatives with increased antiproliferative effect and activation of ERK pathway in prostate cancer cells. | Bioorganic & medicinal chemistry 20061001 |
Effects of humidity and filter material on diffusive sampling of isocyanates using reagent-coated filters. | Journal of environmental monitoring : JEM 20061001 |
Synthesis and characterization of novel '3 + 2' oxorhenium complexes, ReO[SNO][NN]. | Inorganic chemistry 20060710 |
Determination of airborne isocyanates generated during the thermal degradation of car paint in body repair shops. | The Annals of occupational hygiene 20060601 |
Tape-strip sampling for measuring dermal exposure to 1,6-hexamethylene diisocyanate. | Scandinavian journal of work, environment & health 20060601 |
Selective antagonist at D3 receptors, but not non-selective partial agonists, influences the expression of cocaine-induced conditioned place preference in free-feeding rats. | Pharmacology, biochemistry, and behavior 20051201 |
Validation of a solvent-free sampler for the determination of low molecular weight aliphatic isocyanates under thermal degradation conditions. | Journal of occupational and environmental hygiene 20050901 |
1-(1-Naphthyl)piperazine as a novel template for 5-HT6 serotonin receptor ligands. | Bioorganic & medicinal chemistry letters 20050315 |
Synthesis and in vitro binding of N-phenyl piperazine analogs as potential dopamine D3 receptor ligands. | Bioorganic & medicinal chemistry 20050103 |
Characterisation of derivatised monomeric and prepolymeric isocyanates by matrix-assisted laser desorption/ionisation time-of-flight mass spectrometry and structural elucidation by tandem mass spectrometry. | European journal of mass spectrometry (Chichester, England) 20050101 |
Synthesis and evaluation of in vivo activity of diphenylhydantoin basic derivatives. | European journal of medicinal chemistry 20041201 |
A study on application of impregnated synthetic peptide TLC stationary phases for the screening of 5-HT1A ligands. Part 2. | Biomedical chromatography : BMC 20041001 |
Biological monitoring of exposure to toluene diisocyanate. | Scandinavian journal of work, environment & health 20041001 |
A survey of airborne isocyanate exposure in 13 Swedish polyurethane industries. | The Annals of occupational hygiene 20040701 |
Determination of isocyanates in air using 1-(2-methoxyphenyl)piperazine-impregnated filters: long-term sampling performance and field comparison with impingers with dibutylamine. | The Annals of occupational hygiene 20040701 |
New imide 5-HT1A receptor ligands - modification of terminal fragment geometry. | Molecules (Basel, Switzerland) 20040227 |
Serotonergic and dopaminergic influence of the duration of embryogenesis and intracapsular locomotion of Lymnaea stagnalis L. | Acta biologica Hungarica 20040101 |
Toxicological detection of the new designer drug 1-(4-methoxyphenyl)piperazine and its metabolites in urine and differentiation from an intake of structurally related medicaments using gas chromatography-mass spectrometry. | Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20031225 |
Characterization of the 5-HT(7) receptor. Determination of the pharmacophore for 5-HT(7) receptor agonism and CoMFA-based modeling of the agonist binding site. | Journal of medicinal chemistry 20031204 |
Evaluation of some aroxyethylamine derivatives for hypotensive properties and their affinities for adrenergic receptors. | Die Pharmazie 20031201 |
Investigation of the competitive rate of derivatization of several secondary amines with phenylisocyanate (PHI), hexamethylene-1,6-diisocyanate (HDI), 4,4'-methylenebis(phenyl isocyanate) (MDI) and toluene diisocyanate (TDI) in liquid medium. | The Analyst 20030201 |
Novel oxorhenium and oxotechnetium MO(NS)(S)2 complexes in the development of 5-HT1A receptor imaging agents. | Journal of inorganic biochemistry 20030115 |
Workplace monitoring of isocyanates using ion trap liquid chromatography/tandem mass spectrometry. | Rapid communications in mass spectrometry : RCM 20030101 |
Synthesis, in vitro and in vivo 5-HT1A/5-HT2A serotonin receptor activity of new hybrid 1,2,3,4-tetrahydro-gamma-carbolines with 1-(2-methoxyphenyl)piperazine moiety. | Polish journal of pharmacology 20030101 |
Oxotechnetium 99mTcO[SN(R)S][S] complexes as potential 5-HT1A receptor imaging agents. | Nuclear medicine and biology 20021101 |
Development of a diffusive sampling method for determination of methyl isocyanate in air. | Journal of environmental monitoring : JEM 20021001 |
Exposure to airborne isocyanates and other thermal degradation products at polyurethane-processing workplaces. | Journal of environmental monitoring : JEM 20021001 |
Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells. | The Journal of biological chemistry 20020419 |
Comparison of sampling methods for 1,6-hexamethylene diisocyanate, (HDI) in a commercial spray box. | The Analyst 20020101 |
Two routes to [11C-carbonyl]organo-isocyanates utilizing [11C]phosgene ([11C]organo-isocyanates from [11C]phosgene). | Nuclear medicine and biology 20011101 |
Substituted phenoxyalkylpiperazines as dopamine D3 receptor ligands. | Die Pharmazie 20010401 |
Development of novel mixed-ligand oxotechnetium [SNS/S] complexes as potential 5-HT1A receptor imaging agents. | Journal of biological inorganic chemistry : JBIC : a publication of the Society of Biological Inorganic Chemistry 20010301 |
A comparison of solid sampler methods for the determination of hexamethylene-based isocyanates in spray-painting operations. | AIHAJ : a journal for the science of occupational and environmental health and safety 20010101 |
2-H- and 2-acyl-9- [omega-[4-(2-methoxyphenyl)piperazinyl]-alkyl]-1,2,3,4-tetrahydro-beta-carbolines as ligands of 5-HT1A and 5-HT2A receptors. | Polish journal of pharmacology 20010101 |
Molecular cloning and expression of a 5-hydroxytryptamine7 serotonin receptor subtype. | The Journal of biological chemistry 19930825 |