4-(2-Aminoethyl)benzenesulfonyl fluoride, HCl
| Title | Journal |
|---|---|
| Amyloid β induces NLRP3 inflammasome activation in retinal pigment epithelial cells via NADPH oxidase- and mitochondria-dependent ROS production. | Journal of biochemical and molecular toxicology 20170601 |
| Crystal structures of BapA complexes with β-lactam-derived inhibitors illustrate substrate specificity and enantioselectivity of β-aminopeptidases. | Chembiochem : a European journal of chemical biology 20120924 |
| Synthesis and evaluation of silanediols as highly selective uncompetitive inhibitors of human neutrophil elastase. | Journal of medicinal chemistry 20120913 |
| Deficiency of αB crystallin augments ER stress-induced apoptosis by enhancing mitochondrial dysfunction. | Free radical biology & medicine 20120901 |
| Androgen deprivation causes truncation of the C-terminal region of androgen receptor in human prostate cancer LNCaP cells. | Cancer science 20120601 |
| Doxycycline indirectly inhibits proteolytic activation of tryptic kallikrein-related peptidases and activation of cathelicidin. | The Journal of investigative dermatology 20120501 |
| Pitfalls in the determination of human acylated ghrelin plasma concentrations using a double antibody enzyme immunometric assay. | Clinical biochemistry 20120101 |
| A model to evaluate toxic factors influencing islets during collagenase digestion: the role of serine protease inhibitor in the protection of islets. | Cell transplantation 20120101 |
| Serine protease inhibitor attenuates ovalbumin induced inflammation in mouse model of allergic airway disease. | PloS one 20120101 |
| Serine protease inhibitor, 4-(2-aminoethyl)-benzene sulfonyl fluoride, impairs IL-12-induced activation of pSTAT4β, NFκB, and select pro-inflammatory mediators from estrogen-treated mice. | Immunobiology 20111201 |
| Serine protease inhibitor 4-(2-aminoethyl)benzenesulfonyl fluoride hydrochloride (AEBSF) inhibits the rat embryo implantation in vivo and interferes with cell adhesion in vitro. | Contraception 20111201 |
| Development of a fluorescence resonance energy transfer peptide library technology for detection of protease contaminants in protein-based raw materials used in diagnostic assays. | Assay and drug development technologies 20111001 |
| Fluoride does not inhibit enamel protease activity. | Journal of dental research 20110401 |
| A practical guide for the stabilization of acylghrelin in human blood collections. | Clinical endocrinology 20110301 |
| Inhibition of proprotein convertase SKI-1 blocks transcription of key extracellular matrix genes regulating osteoblastic mineralization. | The Journal of biological chemistry 20110121 |
| A trypsin-like serine protease is involved in pseudorabies virus invasion through the basement membrane barrier of porcine nasal respiratory mucosa. | Veterinary research 20110101 |
| Peptidases of pinworms Syphacia muris and Passalurus ambiguus. | Experimental parasitology 20101001 |
| Comparative pharmacology of chemically distinct NADPH oxidase inhibitors. | British journal of pharmacology 20101001 |
| Serine proteases in histone deacetylase inhibitor-induced apoptosis. | Molecular cancer therapeutics 20100801 |
| Multiple protective functions of catalase against intercellular apoptosis-inducing ROS signaling of human tumor cells. | Biological chemistry 20100601 |
| Ontogeny of acylated ghrelin degradation in the rat. | Peptides 20100201 |
| Carboxymethyl-starch excipients for gastrointestinal stable oral protein formulations containing protease inhibitors. | Journal of pharmacy & pharmaceutical sciences : a publication of the Canadian Society for Pharmaceutical Sciences, Societe canadienne des sciences pharmaceutiques 20100101 |
| Serine protease inhibitors suppress pancreatic endogenous proteases and modulate bacterial neutral proteases. | Islets 20100101 |
| HIV-1 integrase-hydrolyzing antibodies from sera of HIV-infected patients. | Biochimie 20090901 |
| Astragalus polysaccharides decreased the expression of PTP1B through relieving ER stress induced activation of ATF6 in a rat model of type 2 diabetes. | Molecular and cellular endocrinology 20090813 |
| Tumour necrosis factor-alpha processing in interstitial lung disease: a potential role for exogenous proteinase-3. | Clinical and experimental immunology 20090501 |
| Shedding of gACE from residual body membrane of rat sperm. | Legal medicine (Tokyo, Japan) 20090401 |
| The effect of bafilomycin A1 and protease inhibitors on the degradation and recycling of a Class 5-mutant LDLR. | Acta biochimica et biophysica Sinica 20090301 |
| Comparison of trypsin inhibitors in preservation solution for islet isolation. | Cell transplantation 20090101 |
| Potential role of proprotein convertase SKI-1 in the mineralization of primary bone. | Cells, tissues, organs 20081201 |
| Modification of amyloid-beta(1-40) by a protease inhibitor creates risk of error in mass spectrometric quantitation of amyloid-beta(1-42). | Analytical biochemistry 20081115 |
| Zinc chelation induces rapid depletion of the X-linked inhibitor of apoptosis and sensitizes prostate cancer cells to TRAIL-mediated apoptosis. | Cell death and differentiation 20081101 |
| A method for quantifying melanosome transfer efficacy from melanocytes to keratinocytes in vitro. | Pigment cell & melanoma research 20081001 |
| Treatment of cells with n-alpha-tosyl-L-phenylalanine-chloromethyl ketone induces the proteolytic loss of STAT6 transcription factor. | Molecular immunology 20080901 |
| Novel phospholipolytic activities associated with electronegative low-density lipoprotein are involved in increased self-aggregation. | Biochemistry 20080805 |
| Human laminin-332 degradation by Candida proteinases. | Journal of oral pathology & medicine : official publication of the International Association of Oral Pathologists and the American Academy of Oral Pathology 20080701 |
| GRP78 and Raf-1 cooperatively confer resistance to endoplasmic reticulum stress-induced apoptosis. | Journal of cellular physiology 20080601 |
| Sulphur and nitrogen regulation of the protease-encoding ACP1 gene in the fungus Botrytis cinerea: correlation with a phospholipase D activity. | Microbiology (Reading, England) 20080501 |
| Protease activity of allergenic pollen of cedar, cypress, juniper, birch and ragweed. | Allergology international : official journal of the Japanese Society of Allergology 20080301 |
| Endogenous pancreatic protease activity and methods for impeding their function. | Transplantation proceedings 20080301 |
| Relationship between carbachol hyperstimulation-induced pancreatic intracellular trypsinogen and NF-kappa B activation in rats in vitro. | Journal of Huazhong University of Science and Technology. Medical sciences = Hua zhong ke ji da xue xue bao. Yi xue Ying De wen ban = Huazhong keji daxue xuebao. Yixue Yingdewen ban 20080201 |
| Proinflammatory impact of Staphylococcus epidermidis on the nasal epithelium quantified by IL-8 and GRO-alpha responses in primary human nasal epithelial cells. | International archives of allergy and immunology 20080101 |
| Reactive oxygen species generation by the ethylene-bis-dithiocarbamate (EBDC) fungicide mancozeb and its contribution to neuronal toxicity in mesencephalic cells. | Neurotoxicology 20071101 |
| Intracellular PAF catabolism by PAF acetylhydrolase counteracts continual PAF synthesis. | Journal of lipid research 20071101 |
| The role of fungal proteinases in pathophysiology of Stachybotrys chartarum. | Mycopathologia 20071001 |
| Association of specific proteolytic processing of bone sialoprotein and bone acidic glycoprotein-75 with mineralization within biomineralization foci. | The Journal of biological chemistry 20070907 |
| A single intrauterine injection of the serine protease inhibitor 4-(2-aminoethyl)benzenesulfonyl fluoride hydrochloride reversibly inhibits embryo implantation in mice. | Contraception 20070901 |
| A novel 51-kDa fragment of the large subunit of ribulose-1,5-bisphosphate carboxylase/oxygenase formed in the stroma of chloroplasts in dark-induced senescing wheat leaves. | Physiologia plantarum 20070901 |
| PAR-2 activation regulates IL-8 and GRO-alpha synthesis by NF-kappaB, but not RANTES, IL-6, eotaxin or TARC expression in nasal epithelium. | Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology 20070701 |
| Potential effects of PKC or protease inhibitors on acute pancreatitis-induced tissue injury in rats. | Vascular pharmacology 20070601 |
| Endoplasmic reticulum stress-induced cell death mediated by the proteasome. | Cell death and differentiation 20070601 |
| A Bax/Bak-independent mechanism of cytochrome c release. | The Journal of biological chemistry 20070601 |
| Geldanamycin induces CHOP expression through a 4-(2-aminoethyl)-benzenesulfonyl fluoride-responsive serine protease. | Cell research 20070201 |
| Adjustment of digestion enzyme composition improves islet isolation outcome from marginal grade human donor pancreata. | Cell and tissue banking 20070101 |
| Endoplasmic reticulum stress causes the activation of sterol regulatory element binding protein-2. | The international journal of biochemistry & cell biology 20070101 |
| Characterization of the de novo biosynthetic enzyme of platelet activating factor, DDT-insensitive cholinephosphotransferase, of human mesangial cells. | Mediators of inflammation 20070101 |
| Cleavage of misfolded nuclear receptor corepressor confers resistance to unfolded protein response-induced apoptosis. | Cancer research 20061015 |
| Nitric oxide-induced down-regulation of beta-catenin in colon cancer cells by a proteasome-independent specific pathway. | Gastroenterology 20061001 |
| Induction of CXC chemokines in A549 airway epithelial cells by trypsin and staphylococcal proteases - a possible route for neutrophilic inflammation in chronic rhinosinusitis. | Clinical and experimental immunology 20060601 |
| Microsphere-based protease assays and screening application for lethal factor and factor Xa. | Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501 |
| The influence of fibrin polymerization and platelet-mediated contractile forces on citrated whole blood thromboelastography profile. | Thrombosis and haemostasis 20060501 |
| Platelet-activating factor-acetylhydrolase can monodeacylate and inactivate lipoteichoic acid. | Clinical and vaccine immunology : CVI 20060401 |
| Cleavage of epidermal growth factor receptor by caspase during apoptosis is independent of its internalization. | Oncogene 20060309 |
| Rigidity and flexibility of dipeptidyl peptidase IV: crystal structures of and docking experiments with DPIV. | Journal of molecular biology 20060127 |
| Coronary microvascular endothelial cell growth regulates expression of the gene encoding p22-phox. | Free radical biology & medicine 20051115 |
| Shedding of the germinal angiotensin I-converting enzyme (gACE) involves a serine protease and is activated by epididymal fluid. | Biology of reproduction 20051101 |
| Abrogation of IFN-gamma mediated epithelial barrier disruption by serine protease inhibition. | Clinical and experimental immunology 20051101 |
| Cleavage of p21/WAF1/CIP1 by proteinase 3 modulates differentiation of a monocytic cell line. Molecular analysis of the cleavage site. | The Journal of biological chemistry 20050826 |
| Reactive oxygen species-linked regulation of the multidrug resistance transporter P-glycoprotein in Nox-1 overexpressing prostate tumor spheroids. | FEBS letters 20050815 |
| Coupling of size-exclusion chromatography to a continuous assay for subtilisin using a fluorescence resonance energy transfer peptide substrate: testing of two standard inhibitors. | Journal of chromatography. A 20050722 |
| Heme oxygenase-1 gene activation by the NAD(P)H oxidase inhibitor 4-(2-aminoethyl) benzenesulfonyl fluoride via a protein kinase B, p38-dependent signaling pathway in monocytes. | The Journal of biological chemistry 20050610 |
| The interaction of human tryptase-beta with small molecule inhibitors provides new insights into the unusual functional instability and quaternary structure of the protease. | Biochemistry 20050308 |
| Antioxidants inhibit human endothelial cell functions through down-regulation of endothelial nitric oxide synthase activity. | European journal of pharmacology 20050307 |
| c-Src and hydrogen peroxide mediate transforming growth factor-beta1-induced smooth muscle cell-gene expression in 10T1/2 cells. | Arteriosclerosis, thrombosis, and vascular biology 20050201 |
| Pro- and anti-apoptotic effects of an inhibitor of chymotrypsin-like serine proteases. | Cell cycle (Georgetown, Tex.) 20041201 |
| Proteasome proteolytic activity in hematopoietic cells from patients with chronic myeloid leukemia and multiple myeloma. | Haematologica 20041201 |
| The N-terminal extension of plant mitochondrial carrier proteins is removed by two-step processing: the first cleavage is by the mitochondrial processing peptidase. | Journal of molecular biology 20041119 |
| NADPH oxidase-dependent acid production in airway epithelial cells. | The Journal of biological chemistry 20040827 |
| Aminoethyl benzenesulfonyl fluoride and its hexapeptide (Ac-VFRSLK) conjugate are both in vitro inhibitors of subtilisin kexin isozyme-1. | FEBS letters 20040827 |
| Antioxidants inhibit angiogenesis in vivo through down-regulation of nitric oxide synthase expression and activity. | Free radical research 20040501 |
| Potent bivalent inhibition of human tryptase-beta by a synthetic inhibitor. | Biological chemistry 20031201 |
| Serine proteases mediate apoptosis-like cell death and phagocytosis under caspase-inhibiting conditions. | Cell death and differentiation 20031001 |
| A serine protease is involved in the initiation of DNA damage-induced apoptosis. | Cell death and differentiation 20031001 |
| A serine protease inhibitor prevents endoplasmic reticulum stress-induced cleavage but not transport of the membrane-bound transcription factor ATF6. | The Journal of biological chemistry 20030815 |
| Reelin promotes peripheral synapse elimination and maturation. | Science (New York, N.Y.) 20030801 |
| Identification and partial characterization of two inducible gelatin-cleavage activities localized to the sea urchin extraembryonic matrix, the hyaline layer. | Biochimica et biophysica acta 20030407 |
| Characterization of a serine protease activity in Sarcocystis neurona merozoites. | The Journal of parasitology 20030401 |
| Evaluation of Pefabloc as a serine protease inhibitor during human-islet isolation. | Transplantation 20030227 |
| CIAP1 and the serine protease HTRA2 are involved in a novel p53-dependent apoptosis pathway in mammals. | Genes & development 20030201 |
| Inhibition of telomerase increases resistance of melanoma cells to temozolomide, but not to temozolomide combined with poly (adp-ribose) polymerase inhibitor. | Molecular pharmacology 20030101 |
| Improved islet yields from Macaca nemestrina and marginal human pancreata after two-layer method preservation and endogenous trypsin inhibition. | American journal of transplantation : official journal of the American Society of Transplantation and the American Society of Transplant Surgeons 20030101 |
| Gibberellin-mediated proteasome-dependent degradation of the barley DELLA protein SLN1 repressor. | The Plant cell 20021201 |
| Effect of pefabloc on islet isolation from cold preserved rat pancreas. | Transplantation proceedings 20021101 |
| Platelet phagocytosis and processing of beta-amyloid precursor protein as a mechanism of macrophage activation in atherosclerosis. | Circulation research 20020614 |
| Evaluation of two inhibitors of invasion: LY311727 [3-(3-acetamide-1-benzyl-2-ethyl-indolyl-5-oxy)propane phosphonic acid] and AEBSF [4-(2-aminoethyl)-benzenesulphonyl fluoride] in acute murine toxoplasmosis. | The Journal of antimicrobial chemotherapy 20020501 |
| Oxidative stress increased respiration and generation of reactive oxygen species, resulting in ATP depletion, opening of mitochondrial permeability transition, and programmed cell death. | Plant physiology 20020401 |
| Phospholipase D contributes to transmural pressure control of prorenin processing in juxtaglomerular cell. | Hypertension (Dallas, Tex. : 1979) 20020201 |
| Inhibition of NADH/NADPH oxidase affects signal transduction by growth factor receptors in normal fibroblasts. | Archives of biochemistry and biophysics 20020115 |
| The central role of thromboxane and platelet activating factor receptors in ex vivo regulation of endotoxin-induced monocyte tissue factor activity in human whole blood. | Journal of endotoxin research 20020101 |
| Induction of IkappaB-kinase by cholecystokinin is mediated by trypsinogen activation in rat pancreatic lobules. | Digestion 20020101 |
| Inhibition of lipoprotein-associated phospholipase A2 diminishes the death-inducing effects of oxidised LDL on human monocyte-macrophages. | FEBS letters 20010921 |
| Islet isolation: simple modifications can still yield big improvements. | Transplantation 20010827 |
| Serine-protease inhibition during islet isolation increases islet yield from human pancreases with prolonged ischemia. | Transplantation 20010827 |
| Tumor necrosis factor-related apoptosis inducing ligand (TRAIL)-induced apoptosis is dependent on activation of cysteine and serine proteases. | Cytokine 20010807 |
| Unique pathway of thrombin-induced platelet aggregation mediated by glycoprotein Ib. | The Journal of biological chemistry 20010615 |
| Soluble CD44 inhibits melanoma tumor growth by blocking cell surface CD44 binding to hyaluronic acid. | Oncogene 20010607 |
| Serine protease inhibitor causes F-actin redistribution and inhibition of calcium-mediated secretion in pancreatic acini. | Gastroenterology 20010601 |
| Protein kinase C activation by PMA rapidly induces apoptosis through caspase-3/CPP32 and serine protease(s) in a gastric cancer cell line. | International journal of oncology 20010501 |
| Characterization of a protease responsible for truncated actin increase in neutrophils of patients with Behçet's disease. | Biological & pharmaceutical bulletin 20010201 |
| Studies on digestive proteases from midgut glands of a shrimp, Penaeus indicus, and a lobster, Nephrops norvegicus: Part 1. Proteolytic activity. | Applied biochemistry and biotechnology 20010201 |
| Inhibitors of trypsin-like serine proteases prevent DNA damage-induced neuronal death by acting upstream of the mitochondrial checkpoint and of p53 induction. | Neuroscience 20010101 |
| A role for serine proteases in mediating phorbol ester-induced differentiation of HL-60 cells. | Experimental cell research 20000410 |