4-(1H-Indol-3-yl)pyrimidin-2-amine
Title | Journal |
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Inhibiting NF-κB-inducing kinase (NIK): discovery, structure-based design, synthesis, structure-activity relationship, and co-crystal structures. | Bioorganic & medicinal chemistry letters 20130301 |
Synthesis, protein kinase inhibitory potencies, and in vitro antiproliferative activities of meridianin derivatives. | Journal of medicinal chemistry 20110714 |
Rapid synthesis of bis(hetero)aryls by one-pot Masuda borylation-Suzuki coupling sequence and its application to concise total syntheses of meridianins A and G. | Organic & biomolecular chemistry 20110507 |
Fragment and knowledge-based design of selective GSK-3beta inhibitors using virtual screening models. | European journal of medicinal chemistry 20090601 |
In-vitro antiproliferative activities and kinase inhibitory potencies of meridianin derivatives. | Anti-cancer drugs 20080901 |
Identification of two meridianins from the crude extract of the tunicate Aplidium meridianum by tandem mass spectrometry. | Natural product research 20070520 |
Synthesis and antitumor activity of indolylpyrimidines: marine natural product meridianin D analogues. | Bioorganic & medicinal chemistry 20070201 |
Meridianins, a new family of protein kinase inhibitors isolated from the ascidian Aplidium meridianum. | Bioorganic & medicinal chemistry letters 20040405 |