Cyclopentaneacetamide, N-[(1S)-4-[(aminoiminomethyl)amino]-1-[[[2-(3,5-dioxo-1,2-diphenyl-1,2,4-triazolidin-4-yl)ethyl]amino]carbonyl]butyl]-1-[2-[4-(6,11-dihydro-6-oxo-5H-dibenz[b,e]azepin-11-yl)-1-piperazinyl]-2-oxoethyl]-
| Title | Journal |
|---|---|
| Anorexia induction by the trichothecene deoxynivalenol (vomitoxin) is mediated by the release of the gut satiety hormone peptide YY. | Toxicological sciences : an official journal of the Society of Toxicology 20121201 |
| A role for neuropeptide Y in the gender-specific gastrointestinal, corticosterone and feeding responses to stress. | British journal of pharmacology 20120801 |
| Role of Y(2) receptors in the regulation of gastric tone in rats. | American journal of physiology. Gastrointestinal and liver physiology 20120401 |
| Role of neuropeptide Y Y₁ and Y₂ receptors on behavioral despair in a rat model of depression with co-morbid anxiety. | Neuropharmacology 20120101 |
| Distinct effects of NPY13-36, a specific NPY Y2 agonist, in a model of rodent endotoxemia on leukocyte subsets and cytokine levels. | Annals of anatomy = Anatomischer Anzeiger : official organ of the Anatomische Gesellschaft 20111220 |
| Attenuation of pain-related behavior evoked by injury through blockade of neuropeptide Y Y2 receptor. | Pain 20110501 |
| High expression of NPY receptors in the human testis. | Molecular and cellular endocrinology 20110430 |
| Neuropeptide Y and its Y2 receptor: potential targets in neuroblastoma therapy. | Oncogene 20101014 |
| Mutagenesis of human neuropeptide Y/peptide YY receptor Y2 reveals additional differences to Y1 in interactions with highly conserved ligand positions. | Regulatory peptides 20100809 |
| Selective and brain penetrant neuropeptide y y2 receptor antagonists discovered by whole-cell high-throughput screening. | Molecular pharmacology 20100101 |
| Peripheral peptide YY inhibits propulsive colonic motor function through Y2 receptor in conscious mice. | American journal of physiology. Gastrointestinal and liver physiology 20100101 |
| Effect of pharmacological manipulations of neuropeptide Y and corticotropin-releasing factor neurotransmission on incubation of conditioned fear. | Neuroscience 20091229 |
| The identification and optimisation of novel and selective diamide neuropeptide Y Y2 receptor antagonists. | Bioorganic & medicinal chemistry letters 20090801 |
| Neuropeptide Y fragments derived from neprilysin processing are neuroprotective in a transgenic model of Alzheimer's disease. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20090128 |
| Different regulation of atrial ANP release through neuropeptide Y2 and Y4 receptors. | Journal of Korean medical science 20081201 |
| Activity-dependent volume transmission by transgene NPY attenuates glutamate release and LTP in the subiculum. | Molecular and cellular neurosciences 20081001 |
| Endogenous PYY and NPY mediate tonic Y1- and Y2-mediated absorption in human and mouse colon. | Nutrition (Burbank, Los Angeles County, Calif.) 20080901 |
| Neuropeptide Y receptors in primary human brain tumors: overexpression in high-grade tumors. | Journal of neuropathology and experimental neurology 20080801 |
| Neuropeptide Y reduces acetylcholine release and vagal bradycardia via a Y2 receptor-mediated, protein kinase C-dependent pathway. | Journal of molecular and cellular cardiology 20080301 |
| Role of CCK1 and Y2 receptors in activation of hindbrain neurons induced by intragastric administration of bitter taste receptor ligands. | American journal of physiology. Regulatory, integrative and comparative physiology 20080101 |
| NPY gene transfer in the hippocampus attenuates synaptic plasticity and learning. | Hippocampus 20080101 |
| Oligomerization of neuropeptide Y (NPY) Y2 receptors in CHO cells depends on functional pertussis toxin-sensitive G-proteins. | Regulatory peptides 20071204 |
| Sigma 1 receptor-mediated increase in hippocampal extracellular dopamine contributes to the mechanism of the anticonvulsant action of neuropeptide Y. | The European journal of neuroscience 20071201 |
| A novel long-acting selective neuropeptide Y2 receptor polyethylene glycol-conjugated peptide agonist reduces food intake and body weight and improves glucose metabolism in rodents. | The Journal of pharmacology and experimental therapeutics 20071101 |
| Selective role of neuropeptide Y receptor subtype Y2 in the control of gonadotropin secretion in the rat. | American journal of physiology. Endocrinology and metabolism 20071101 |
| Neuropeptide Y-induced enhancement of the evoked release of newly synthesized dopamine in rat striatum: mediation by Y2 receptors. | Neuropharmacology 20070501 |
| Infusion of neuropeptide Y into CA3 region of hippocampus produces antidepressant-like effect via Y1 receptor. | Hippocampus 20070101 |
| Neuropeptide Y regulates recurrent mossy fiber synaptic transmission less effectively in mice than in rats: Correlation with Y2 receptor plasticity. | Neuroscience 20061228 |
| Fluorescence- and luminescence-based methods for the determination of affinity and activity of neuropeptide Y2 receptor ligands. | European journal of pharmacology 20061203 |
| Anxiolytic-like effect of the selective neuropeptide Y Y2 receptor antagonist BIIE0246 in the elevated plus-maze. | Peptides 20061201 |
| Ventricular fibrillation induced by ischemia-reperfusion is not prevented by the NPY Y2 receptor antagonist BIIE0246. | Journal of cardiovascular pharmacology and therapeutics 20060901 |
| Neuropeptide Y2 receptors are involved in enhanced neurogenic vasoconstriction in spontaneously hypertensive rats. | British journal of pharmacology 20060701 |
| Irreversible binding kinetics of neuropeptide Y ligands to Y2 but not to Y1 and Y5 receptors. | Pharmacology 20051201 |
| Neuropeptide Y bioavailability is suppressed in the hindlimb of female Sprague-Dawley rats. | The Journal of physiology 20051015 |
| Influence of endogenous neuropeptide Y (NPY) on the sympathetic-parasympathetic interaction in the canine heart. | Journal of cardiovascular pharmacology 20051001 |
| The anti-epileptic actions of neuropeptide Y in the hippocampus are mediated by Y and not Y receptors. | The European journal of neuroscience 20050901 |
| Intravenous peptide YY3-36 and Y2 receptor antagonism in the rat: effects on feeding behaviour. | Journal of neuroendocrinology 20050701 |
| Blockade of the neuropeptide Y Y2 receptor with the specific antagonist BIIE0246 attenuates the effect of endogenous and exogenous peptide YY(3-36) on food intake. | Brain research 20050510 |
| Suppression of ethanol self-administration by the neuropeptide Y (NPY) Y2 receptor antagonist BIIE0246: evidence for sensitization in rats with a history of dependence. | Neuroscience letters 20050227 |
| Spontaneous release of neuropeptide Y tonically inhibits recurrent mossy fiber synaptic transmission in epileptic brain. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20050216 |
| Differential expression of Y receptors and signaling pathways in intestinal circular and longitudinal smooth muscle. | Regulatory peptides 20050215 |
| Endogenous neuropeptide Y depresses the afferent signaling of gastric acid challenge to the mouse brainstem via neuropeptide Y type Y2 and Y4 receptors. | Neuroscience 20050101 |
| Neuropeptide Y inhibits acetylcholine release in human heart atrium by activation of Y2-receptors. | Naunyn-Schmiedeberg's archives of pharmacology 20040501 |
| Involvement of peripheral neuropeptide Y receptors in sympathetic modulation of acute cutaneous flare induced by intradermal capsaicin. | Neuroscience 20040101 |
| Stimulation of neurons in rat ARC inhibits gastric acid secretion via hypothalamic CRF1/2- and NPY-Y1 receptors. | American journal of physiology. Gastrointestinal and liver physiology 20031201 |
| Development and characterization of a highly selective neuropeptide Y Y5 receptor agonist radioligand: [125I][hPP1-17, Ala31, Aib32]NPY. | British journal of pharmacology 20030801 |
| Functional consequences of neuropeptide Y Y 2 receptor knockout and Y2 antagonism in mouse and human colonic tissues. | British journal of pharmacology 20030601 |
| Functional interaction between neuropeptide Y receptors and modulation of calcium channels in the rat hippocampus. | Neuropharmacology 20030201 |
| Selective mediation of nerve injury-induced tactile hypersensitivity by neuropeptide Y. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20021115 |
| Blockade of central neuropeptide Y (NPY) Y2 receptors reduces ethanol self-administration in rats. | Neuroscience letters 20021025 |
| Blockade of neuropeptide Y(2) receptors and suppression of NPY's anti-epileptic actions in the rat hippocampal slice by BIIE0246. | British journal of pharmacology 20020601 |
| Antagonistic interaction between BIIE 0246, a neuropeptide Y Y2-receptor antagonist, and omega-conotoxin GVIA, a Ca2+ channel antagonist, in presynaptic transmitter releases in dog splenic arteries. | Japanese journal of pharmacology 20020601 |
| Reciprocal mutations of neuropeptide Y receptor Y2 in human and chicken identify amino acids important for antagonist binding. | FEBS letters 20020508 |
| The neuropeptide Y (NPY) Y1 receptor subtype mediates NPY-induced antidepressant-like activity in the mouse forced swimming test. | Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20020501 |
| Neuropeptide Y inhibits double peaked vasoconstrictor responses to periarterial nerve stimulation primarily through prejunctional Y2 receptor subtype in canine splenic arteries. | Autonomic & autacoid pharmacology 20020401 |
| Autoinhibitory function of the sympathetic prejunctional neuropeptide Y Y(2) receptor evidenced by BIIE0246. | European journal of pharmacology 20020329 |
| Role of neuropeptide Y Y(2) receptors in modulation of cardiac parasympathetic neurotransmission. | Regulatory peptides 20020215 |
| Effects of the neuropeptide Y Y2 receptor antagonist BIIE0246 on sympathetic transmitter release in the pig in vivo. | Naunyn-Schmiedeberg's archives of pharmacology 20020201 |
| Brain neuropeptide Y (NPY) in stress and alcohol dependence. | Reviews in the neurosciences 20020101 |
| Involvement of NPY Y2 receptor subtype in the control of the spontaneous NO/GnRH release at the rat median eminence. | Neuroreport 20011029 |
| Existence of both neuropeptide Y, Y1 and Y2 receptors in pig spleen: evidence using subtype-selective antagonists in vivo. | Life sciences 20010914 |
| Vascular pharmacology of BIIE0246, the first selective non-peptide neuropeptide Y Y(2) receptor antagonist, in vivo. | British journal of pharmacology 20010801 |
| The peptide YY-preferring receptor mediating inhibition of small intestinal secretion is a peripheral Y(2) receptor: pharmacological evidence and molecular cloning. | Molecular pharmacology 20010701 |
| Effects of a selective neuropeptide Y Y2 receptor antagonist, BIIE0246, on Y2 receptors at peripheral neuroeffector junctions. | British journal of pharmacology 20010201 |
| BIIE0246: a selective and high affinity neuropeptide Y Y(2) receptor antagonist. | European journal of pharmacology 19991119 |