4H-Pyrido[1,2-a]pyrimidin-4-one
| Title | Journal |
|---|---|
| Fused bicycles as arylketone bioisosteres leading to potent, orally active thiadiazole H3 antagonists. | Bioorganic & medicinal chemistry letters 20120501 |
| Suzuki-Miyaura cross-coupling reactions of halo derivatives of 4H-pyrido[1,2-a]pyrimidin-4-ones. | Organic & biomolecular chemistry 20111007 |
| Synthesis and antiproliferative activity of novel diaryl ureas possessing a 4H-pyrido[1,2-a]pyrimidin-4-one group. | Archiv der Pharmazie 20100101 |
| Anti-ischaemic activity of an antioxidant aldose reductase inhibitor on diabetic and non-diabetic rat hearts. | The Journal of pharmacy and pharmacology 20100101 |
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidate. | Bioorganic & medicinal chemistry 20071115 |
| Pyrido[1,2-a]pyrimidin-4-one derivatives as a novel class of selective aldose reductase inhibitors exhibiting antioxidant activity. | Journal of medicinal chemistry 20071004 |
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 6: exploration of aromatic substituents. | Bioorganic & medicinal chemistry 20061215 |
| MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 5: Carbon-substituted analogues at the C-2 position. | Bioorganic & medicinal chemistry 20060315 |
| Isocyanate acting as a carbonyl precursor: pyridyl group-assisted formation of 4H-pyrido[1,2-a]pyrimidin-4-ones from ketimines and isocyanates. | Organic & biomolecular chemistry 20060121 |
| Synthesis and biological activities of flavonoid derivatives as A3 adenosine receptor antagonists. | Journal of medicinal chemistry 19960607 |