4-Quinolinecarboxamide, N-[(2R,4S)-1-[3,5-bis(trifluoromethyl)benzoyl]-2-[(4-chlorophenyl)methyl]-4-piperidinyl]-
Title | Journal |
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Non-peptide NK1 receptor ligands based on the 4-phenylpyridine moiety. | Bioorganic & medicinal chemistry 20110401 |
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors. | Journal of medicinal chemistry 20081113 |
The NK1 receptor antagonist NKP608 lacks anxiolytic-like activity in Swiss-Webster mice exposed to the elevated plus-maze. | Behavioural brain research 20040923 |
Expression of functional neurokinin-1 receptors in regenerative glands during gastric wound healing in rodents. | Gastroenterology 20040301 |
Effect of a novel NK1 receptor selective antagonist (NKP608) on citric acid induced cough and airway obstruction. | Pulmonary pharmacology & therapeutics 20040101 |
Comparison of the functional blockade of rat substance P (NK1) receptors by GR205171, RP67580, SR140333 and NKP-608. | Neuropharmacology 20030801 |
Anxiolytic effect of NKP608, a NK1-receptor antagonist, in the social investigation test in gerbils. | Behavioural brain research 20020718 |
Antagonism by NKP608 of substance P-induced plasma protein exudation in a novel preparation of perfused trachea in rats and guinea-pigs in vivo. | Inflammation research : official journal of the European Histamine Research Society ... [et al.] 20020701 |
Pharmacological and endocrinological characterisation of stress-induced hyperthermia in singly housed mice using classical and candidate anxiolytics (LY314582, MPEP and NKP608). | European journal of pharmacology 20020125 |