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| Title | Journal |
|---|---|
| Raf-1/CK2 and RhoA/ROCK signaling promote TNF-α-mediated endothelial apoptosis via regulating vimentin cytoskeleton. | Toxicology 20170815 |
| CK2 activity is required for the interaction of FGF14 with voltage-gated sodium channels and neuronal excitability. | FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20160601 |
| BET protein Brd4 activates transcription in neurons and BET inhibitor Jq1 blocks memory in mice. | Nature neuroscience 20151001 |
| Synthesis and physico-chemical properties in aqueous medium of all possible isomeric bromo analogues of benzo-1H-triazole, potential inhibitors of protein kinases. | The journal of physical chemistry. B 20120621 |
| Protein kinase CK2 mediates peroxynitrite-induced heme oxygenase-1 expression in articular chondrocytes. | International journal of molecular medicine 20120601 |
| Indeno[1,2-b]indole derivatives as a novel class of potent human protein kinase CK2 inhibitors. | Bioorganic & medicinal chemistry 20120401 |
| Protein kinase CK2 triggers cytosolic zinc signaling pathways by phosphorylation of zinc channel ZIP7. | Science signaling 20120207 |
| A pharmacologically-based array to identify targets of cyclosporine A-induced toxicity in cultured renal proximal tubule cells. | Toxicology and applied pharmacology 20120115 |
| Time schedule-dependent effect of the CK2 inhibitor TBB on PC-3 human prostate cancer cell viability. | Oncology reports 20120101 |
| Influence of five potential anticancer drugs on wnt pathway and cell survival in human biliary tract cancer cells. | International journal of biological sciences 20120101 |
| Phosphorylation of CRN2 by CK2 regulates F-actin and Arp2/3 interaction and inhibits cell migration. | Scientific reports 20120101 |
| Inhibition of casein kinase 2 modulates XBP1-GRP78 arm of unfolded protein responses in cultured glial cells. | PloS one 20120101 |
| GPCRs regulate the assembly of a multienzyme complex for purine biosynthesis. | Nature chemical biology 20111201 |
| Multisite-directed inhibitors of protein kinase CK2: new challenges. | Molecular and cellular biochemistry 20111001 |
| Design and synthesis of CK2 inhibitors. | Molecular and cellular biochemistry 20111001 |
| Down-regulation of CK2 activity results in a decrease in the level of cdc25C phosphatase in different prostate cancer cell lines. | Molecular and cellular biochemistry 20111001 |
| The kinase DYRKIA regulates pre-mRNA splicing in spermatogonia and proliferation of spermatogonia and Sertoli cells by phosphorylating a spliceosomal component, SAP155, in postnatal murine testes. | Molecular and cellular biochemistry 20110901 |
| The protein kinase CK2 inhibitor TBB mediates up-regulation of MEK3/6 and p38δ activities, down-regulation of ERK1/2 activity and induction of G1/S arrest in normal human epidermal autocrine proliferating keratinocytes. | Journal of dermatological science 20110801 |
| The cytosolic protein kinase CK2 phosphorylates cardiac calsequestrin in intact cells. | Molecular and cellular biochemistry 20110701 |
| CK2 phosphorylates AP-2α and increases its transcriptional activity. | BMB reports 20110701 |
| Protein kinase CK2 increases glutamatergic input in the hypothalamus and sympathetic vasomotor tone in hypertension. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20110601 |
| Brain-derived neurotrophic factor enhances Bcl-xL expression through protein kinase casein kinase 2-activated and nuclear factor kappa B-mediated pathway in rat hippocampus. | Brain pathology (Zurich, Switzerland) 20110301 |
| Treatment of cultured human astrocytes and vascular endothelial cells with protein kinase CK2 inhibitors induces early changes in cell shape and cytoskeleton. | Molecular and cellular biochemistry 20110301 |
| CK2 inhibition induces apoptosis via the ER stress response. | Cellular signalling 20110101 |
| A specific inhibitor of protein kinase CK2 delays gamma-H2Ax foci removal and reduces clonogenic survival of irradiated mammalian cells. | Radiation oncology (London, England) 20110101 |
| CK2 is acting upstream of MEK3/6 as a part of the signal control of ERK1/2 and p38 MAPK during keratinocytes autocrine differentiation. | Zeitschrift fur Naturforschung. C, Journal of biosciences 20110101 |
| IL-6 stabilizes Twist and enhances tumor cell motility in head and neck cancer cells through activation of casein kinase 2. | PloS one 20110101 |
| Downregulation of protein kinase CK2 activity facilitates tumor necrosis factor-α-mediated chondrocyte death through apoptosis and autophagy. | PloS one 20110101 |
| Bromophenols in marine algae and their bioactivities. | Marine drugs 20110101 |
| Apigenin inhibits proliferation and induces apoptosis in human multiple myeloma cells through targeting the trinity of CK2, Cdc37 and Hsp90. | Molecular cancer 20110101 |
| CK2 phosphorylation of Schistosoma mansoni HMGB1 protein regulates its cellular traffic and secretion but not its DNA transactions. | PloS one 20110101 |
| Label-free integrative pharmacology on-target of drugs at the β(2)-adrenergic receptor. | Scientific reports 20110101 |
| Facilitation of long-term potentiation by muscarinic M(1) receptors is mediated by inhibition of SK channels. | Neuron 20101209 |
| Reconstitution of PTEN activity by CK2 inhibitors and interference with the PI3-K/Akt cascade counteract the antiapoptotic effect of human stromal cells in chronic lymphocytic leukemia. | Blood 20101007 |
| Phosphorylation of the von Hippel-Lindau protein (VHL) by protein kinase CK2 reduces its protein stability and affects p53 and HIF-1alpha mediated transcription. | The international journal of biochemistry & cell biology 20101001 |
| The inhibitory effect of acrylamide on NCAM expression in human neuroblastoma cells: involvement of CK2/Ikaros signaling pathway. | Toxicology in vitro : an international journal published in association with BIBRA 20101001 |
| Relative role of halogen bonds and hydrophobic interactions in inhibition of human protein kinase CK2α by tetrabromobenzotriazole and some C5-substituted analogues. | The journal of physical chemistry. B 20100819 |
| A medicinal chemist's guide to molecular interactions. | Journal of medicinal chemistry 20100722 |
| Genome-wide screen in Saccharomyces cerevisiae identifies vacuolar protein sorting, autophagy, biosynthetic, and tRNA methylation genes involved in life span regulation. | PLoS genetics 20100701 |
| Casein kinase 2 inhibition differentially modulates apoptotic effect of trichostatin A against epithelial ovarian carcinoma cell lines. | Molecular and cellular biochemistry 20100501 |
| Dynamic regulation of a metabolic multi-enzyme complex by protein kinase CK2. | The Journal of biological chemistry 20100409 |
| A FRET-based microplate assay for human protein kinase CK2, a target in neoplastic disease. | Journal of enzyme inhibition and medicinal chemistry 20100401 |
| Regulation of PTEN by CK2 and Notch1 in primary T-cell acute lymphoblastic leukemia: rationale for combined use of CK2- and gamma-secretase inhibitors. | Haematologica 20100401 |
| p53 is dispensable for the induction of apoptosis after inhibition of protein kinase CK2. | The Prostate 20100201 |
| Halogenated imidazole derivatives block RNA polymerase II elongation along mitogen inducible genes. | BMC molecular biology 20100101 |
| A CE-based assay for human protein kinase CK2 activity measurement and inhibitor screening. | Electrophoresis 20100101 |
| Conserved and distinct modes of CREB/ATF transcription factor regulation by PP2A/B56gamma and genotoxic stress. | PloS one 20100101 |
| Kinome profiling of myxoid liposarcoma reveals NF-kappaB-pathway kinase activity and casein kinase II inhibition as a potential treatment option. | Molecular cancer 20100101 |
| The 14-3-3ζ protein binds to the cell adhesion molecule L1, promotes L1 phosphorylation by CKII and influences L1-dependent neurite outgrowth. | PloS one 20100101 |
| Protein kinase C and rho activated coiled coil protein kinase 2 (ROCK2) modulate Alzheimer's APP metabolism and phosphorylation of the Vps10-domain protein, SorL1. | Molecular neurodegeneration 20100101 |
| Efficacy and mechanism of anti-tumor action of new potential CK2 inhibitors toward glioblastoma cells. | International journal of oncology 20091101 |
| Selectivity analysis of protein kinase CK2 inhibitors DMAT, TBB and resorufin in cisplatin-induced stress responses. | International journal of oncology 20091101 |
| Protein kinase CK2 regulates cytoskeletal reorganization during ionizing radiation-induced senescence of human mesenchymal stem cells. | Cancer research 20091015 |
| PACS-1 mediates phosphorylation-dependent ciliary trafficking of the cyclic-nucleotide-gated channel in olfactory sensory neurons. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20090826 |
| Inhibition of protein kinase CK2 induces E2F1 nuclear export, formation of p21/E2F1 complexes and suppression of DNA synthesis in normal human epidermal keratinocytes. | Journal of dermatological science 20090801 |
| Involvement of reactive oxygen species in apoptosis induced by pharmacological inhibition of protein kinase CK2. | Annals of the New York Academy of Sciences 20090801 |
| Structural insight into human CK2alpha in complex with the potent inhibitor ellagic acid. | Bioorganic & medicinal chemistry letters 20090601 |
| DMAT, an inhibitor of protein kinase CK2 induces reactive oxygen species and DNA double strand breaks. | Oncology reports 20090601 |
| Synthesis of new analogs of benzotriazole, benzimidazole and phthalimide--potential inhibitors of human protein kinase CK2. | Bioorganic & medicinal chemistry 20090215 |
| Phosphorylation of the HuR ligand APRIL by casein kinase 2 regulates CD83 expression. | European journal of immunology 20090101 |
| Identification of hematein as a novel inhibitor of protein kinase CK2 from a natural product library. | BMC cancer 20090101 |
| The selectivity of inhibitors of protein kinase CK2: an update. | The Biochemical journal 20081101 |
| Protein kinase CK2 catalyzes tyrosine phosphorylation in mammalian cells. | Cellular signalling 20081101 |
| New inhibitors of protein kinase CK2, analogues of benzimidazole and benzotriazole. | Molecular and cellular biochemistry 20080901 |
| Evaluating CK2 activity with the antibody specific for the CK2-phosphorylated form of a kinase-targeting cochaperone Cdc37. | Molecular and cellular biochemistry 20080901 |
| Impact of protein kinase CK2 on inhibitor of apoptosis proteins in prostate cancer cells. | Molecular and cellular biochemistry 20080901 |
| Role of heme oxygenase-2 in pial arteriolar response to acetylcholine in mice with and without transfusion of cell-free hemoglobin polymers. | American journal of physiology. Regulatory, integrative and comparative physiology 20080801 |
| Hemoglobin neurotoxicity is attenuated by inhibitors of the protein kinase CK2 independent of heme oxygenase activity. | Current neurovascular research 20080801 |
| Protein kinase CK2 modulates synaptic plasticity by modification of synaptic NMDA receptors in the hippocampus. | The Journal of physiology 20080701 |
| An unbiased evaluation of CK2 inhibitors by chemoproteomics: characterization of inhibitor effects on CK2 and identification of novel inhibitor targets. | Molecular & cellular proteomics : MCP 20080601 |
| Regulation of the epithelial Na+ channel by the protein kinase CK2. | The Journal of biological chemistry 20080509 |
| Inhibition of casein kinase 2 enhances the death ligand- and natural kiler cell-induced hepatocellular carcinoma cell death. | Clinical and experimental immunology 20080501 |
| A role for CK2 upon interkinetic nuclear migration in the cell cycle of retinal progenitor cells. | Developmental neurobiology 20080401 |
| CK2beta gene silencing increases cell susceptibility to influenza A virus infection resulting in accelerated virus entry and higher viral protein content. | Journal of molecular signaling 20080101 |
| Ecto-phosphorylation of CD98 regulates cell-cell interactions. | PloS one 20080101 |
| A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases. | Proceedings of the National Academy of Sciences of the United States of America 20071218 |
| Inhibition of HCV replicon cell growth by 2-arylbenzofuran derivatives isolated from Mori Cortex Radicis. | Planta medica 20071101 |
| The reverse in-gel kinase assay to profile physiological kinase substrates. | Nature methods 20071101 |
| Organization and regulation of small conductance Ca2+-activated K+ channel multiprotein complexes. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20070227 |
| Protein kinase CK2alpha as an unfavorable prognostic marker and novel therapeutic target in acute myeloid leukemia. | Clinical cancer research : an official journal of the American Association for Cancer Research 20070201 |
| Tetrabromocinnamic acid (TBCA) and related compounds represent a new class of specific protein kinase CK2 inhibitors. | Chembiochem : a European journal of chemical biology 20070102 |
| CK2 phosphorylation of SAG at Thr10 regulates SAG stability, but not its E3 ligase activity. | Molecular and cellular biochemistry 20070101 |
| Differential regulation of mouse equilibrative nucleoside transporter 1 (mENT1) splice variants by protein kinase CK2. | Molecular membrane biology 20070101 |
| A CK2-dependent mechanism for degradation of the PML tumor suppressor. | Cell 20060728 |
| Expression of protein kinase CK2 in astroglial cells of normal and neovascularized retina. | The American journal of pathology 20060501 |
| Intracellular hydrogen peroxide production is an upstream event in apoptosis induced by down-regulation of casein kinase 2 in prostate cancer cells. | Molecular cancer research : MCR 20060501 |
| Role of protein kinase CK2 in the regulation of tumor necrosis factor-related apoptosis inducing ligand-induced apoptosis in prostate cancer cells. | Cancer research 20060215 |
| Adaptor heat shock protein complex formation regulates trafficking of the asialoglycoprotein receptor. | American journal of physiology. Gastrointestinal and liver physiology 20060201 |
| Transcriptional analysis of calcium-dependent and calcium-independent signalling pathways induced by oligogalacturonides. | Journal of experimental botany 20060101 |
| Tetrabromobenzotriazole (TBBt) and tetrabromobenzimidazole (TBBz) as selective inhibitors of protein kinase CK2: evaluation of their effects on cells and different molecular forms of human CK2. | Biochimica et biophysica acta 20051230 |
| CDK phosphorylation inhibits the DNA-binding and ATP-hydrolysis activities of the Drosophila origin recognition complex. | The Journal of biological chemistry 20051202 |
| A protein kinase CK2 site flanking the nuclear targeting signal enhances nuclear transport of human cytomegalovirus ppUL44. | Traffic (Copenhagen, Denmark) 20051101 |
| Development and exploitation of CK2 inhibitors. | Molecular and cellular biochemistry 20050601 |
| Phosphorylation of the acidic domain of Mdm2 by protein kinase CK2. | Molecular and cellular biochemistry 20050601 |
| Spinal CK2 regulates nociceptive signaling in models of inflammatory pain. | Pain 20050501 |
| Control of hepatitis C: a medicinal chemistry perspective. | Journal of medicinal chemistry 20050113 |
| Synthesis and biological activity of 1H-benzotriazole and 1H-benzimidazole analogues--inhibitors of the NTpase/helicase of HCV and of some related Flaviviridae. | Antiviral chemistry & chemotherapy 20050101 |
| Optimization of protein kinase CK2 inhibitors derived from 4,5,6,7-tetrabromobenzimidazole. | Journal of medicinal chemistry 20041202 |
| Inhibitors of the NTPase/helicases of hepatitis C and related Flaviviridae viruses. | Acta poloniae pharmaceutica 20041201 |
| Flow-dependent regulation of endothelial Toll-like receptor 2 expression through inhibition of SP1 activity. | Circulation research 20041001 |
| 2-Dimethylamino-4,5,6,7-tetrabromo-1H-benzimidazole: a novel powerful and selective inhibitor of protein kinase CK2. | Biochemical and biophysical research communications 20040903 |
| Expression of the Stp1 LMW-PTP and inhibition of protein CK2 display a cooperative effect on immunophilin Fpr3 tyrosine phosphorylation and Saccharomyces cerevisiae growth. | Cellular and molecular life sciences : CMLS 20040501 |
| Protein kinase CK2 phosphorylates the cell cycle regulatory protein Geminin. | Biochemical and biophysical research communications 20040319 |
| TBBz but not TBBt discriminates between two molecular forms of CK2 in vivo and its implications. | Biochemical and biophysical research communications 20031219 |
| Biochemical and three-dimensional-structural study of the specific inhibition of protein kinase CK2 by [5-oxo-5,6-dihydroindolo-(1,2-a)quinazolin-7-yl]acetic acid (IQA). | The Biochemical journal 20030915 |
| Alternative binding modes of an inhibitor to two different kinases. | European journal of biochemistry 20030801 |
| Selectivity of 4,5,6,7-tetrabromobenzimidazole as an ATP-competitive potent inhibitor of protein kinase CK2 from various sources. | Biochemical and biophysical research communications 20030620 |
| Halogenated benzimidazoles and benzotriazoles as inhibitors of the NTPase/helicase activities of hepatitis C and related viruses. | European journal of biochemistry 20030401 |
| The role of calcium in oligogalacturonide-activated signalling in soybean cells. | Planta 20020801 |
| Identification of protein kinase CK2 as a potent kinase of Epstein-Barr virus latent membrane protein 1. | Biochemical and biophysical research communications 20020614 |
| Protein kinase CK2 inhibitor 4,5,6,7-tetrabromobenzotriazole (TBB) induces apoptosis and caspase-dependent degradation of haematopoietic lineage cell-specific protein 1 (HS1) in Jurkat cells. | The Biochemical journal 20020515 |
| Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells. | The Journal of biological chemistry 20020419 |
| Toward the rational design of protein kinase casein kinase-2 inhibitors. | Pharmacology & therapeutics 20020101 |
| Structural features underlying selective inhibition of protein kinase CK2 by ATP site-directed tetrabromo-2-benzotriazole. | Protein science : a publication of the Protein Society 20011101 |
| Selectivity of 4,5,6,7-tetrabromobenzotriazole, an ATP site-directed inhibitor of protein kinase CK2 ('casein kinase-2'). | FEBS letters 20010504 |