Ru 58841
Title | Journal |
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Development of an in silico model for human skin permeation based on a Franz cell skin permeability assay. | Bioorganic & medicinal chemistry letters 20100101 |
Diphenyl ethers as androgen receptor antagonists for the topical suppression of sebum production. | Bioorganic & medicinal chemistry letters 20090415 |
4-(Alkylthio)- and 4-(arylthio)-benzonitrile derivatives as androgen receptor antagonists for the topical suppression of sebum production. | Bioorganic & medicinal chemistry letters 20090301 |
Rational design and synthesis of 4-((1R,2R)-2-hydroxycyclohexyl)-2(trifluoromethyl)benzonitrile (PF-998425), a novel, nonsteroidal androgen receptor antagonist devoid of phototoxicity for dermatological indications. | Journal of medicinal chemistry 20081113 |
Novel vesicular and particulate drug delivery systems for topical treatment of acne. | Expert opinion on drug delivery 20080601 |
(1R,2S)-4-(2-cyano-cyclohexyl-oxy)-2-trifluoromethyl-benzonitrile, a potent androgen receptor antagonist for stimulating hair growth and reducing sebum production. | Bioorganic & medicinal chemistry letters 20071101 |
Preparation of 4-aryl-2-trifluoromethylbenzonitrile derivatives as androgen receptor antagonists for topical suppression of sebum production. | Bioorganic & medicinal chemistry letters 20071015 |
Synthesis and biological evaluation of amino-pyridines as androgen receptor antagonists for stimulating hair growth and reducing sebum production. | Bioorganic & medicinal chemistry letters 20071015 |
Cyproterone acetate loading to lipid nanoparticles for topical acne treatment: particle characterisation and skin uptake. | Pharmaceutical research 20070501 |
Three-dimensional structure-activity relationships of nonsteroidal ligands in complex with androgen receptor ligand-binding domain. | Journal of medicinal chemistry 20050224 |
Synthesis and structure-activity investigation of iodinated arylhydantoins and arylthiohydantoins for development as androgen receptor radioligands. | Bioorganic & medicinal chemistry letters 20041101 |
Synthesis and structure-activity studies of side-chain derivatized arylhydantoins for investigation as androgen receptor radioligands. | Bioorganic & medicinal chemistry letters 20010423 |