1H-1,2,3-Triazole-tethered isatin-7-chloroquinoline and 3-hydroxy-indole-7-chloroquinoline conjugates: synthesis and antimalarial evaluation.

Bioorganic & medicinal chemistry letters 20140201

Optimization of potency and pharmacokinetics of tricyclic indole derived inhibitors of HCV NS5B polymerase. Identification of ester prodrugs with improved oral pharmacokinetics.

Bioorganic & medicinal chemistry 20140101

Discovery of MK-8742: an HCV NS5A inhibitor with broad genotype activity.

ChemMedChem 20131201

Investigations on the metabolic stability of cytosolic phospholipase A2α inhibitors with 1-indolylpropan-2-one structure.

Chemico-biological interactions 20131125

Synthesis and biological activity of benzo-fused 7-deazaadenosine analogues. 5- and 6-substituted 4-amino- or 4-alkylpyrimido[4,5-b]indole ribonucleosides.

Bioorganic & medicinal chemistry 20130901

Unique and potent effects of acute ibogaine on zebrafish: the developing utility of novel aquatic models for hallucinogenic drug research.

Behavioural brain research 20130101

Inhibitors of HIV-1 attachment. Part 8: the effect of C7-heteroaryl substitution on the potency, and in vitro and in vivo profiles of indole-based inhibitors.

Bioorganic & medicinal chemistry letters 20130101

Inhibitors of HIV-1 attachment. Part 7: indole-7-carboxamides as potent and orally bioavailable antiviral agents.

Bioorganic & medicinal chemistry letters 20130101

Small molecules inhibit growth, viability and ergosterol biosynthesis in Candida albicans.

SpringerPlus 20130101

Quantitative determination of the boar taint compounds androstenone, skatole, indole, 3α-androstenol and 3β-androstenol in wild boars (Sus scrofa) reveals extremely low levels of the tryptophan-related degradation products.

Food chemistry 20121215

A spirooxazine derivative as a highly sensitive cyanide sensor by means of UV-visible difference spectroscopy.

The Analyst 20121207

Photophysics of indole, tryptophan and N-acetyl-L-tryptophanamide (NATA): heavy atom effect.

Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20121201

Synthesis and biological evaluation of novel heterocyclic derivatives of combretastatin A-4.

Bioorganic & medicinal chemistry letters 20121201

2C-Methyl- D- erythritol 2,4-cyclodiphosphate synthase from Stevia rebaudiana Bertoni is a functional gene.

Molecular biology reports 20121201

Synthesis of functionalized 2-aryl-4-(indol-3-yl)-4H-chromenes via iodine-catalyzed domino Michael addition-intramolecular cyclization reaction.

Organic & biomolecular chemistry 20121128

Transition metal-free direct C-H bond thiolation of 1,3,4-oxadiazoles and related heteroarenes.

Chemical communications (Cambridge, England) 20121128

A domino synthetic strategy leading to two-carbon-tethered fused acridine/indole pairs and fused acridine derivatives.

Organic & biomolecular chemistry 20121114

3-Alkenylation or 3-alkylation of indole with propargylic alcohols: construction of 3,4-dihydrocyclopenta[b]indole and 1,4-dihydrocyclopenta[b]indole in the presence of different catalysts.

The Journal of organic chemistry 20121102

Otariodibacter oris gen. nov., sp. nov., a member of the family Pasteurellaceae isolated from the oral cavity of pinnipeds.

International journal of systematic and evolutionary microbiology 20121101

Isolates belonging to CDC group II-i belong predominantly to Sphingobacterium mizutaii Yabuuchi et al. 1983: emended descriptions of S. mizutaii and of the genus Sphingobacterium.

International journal of systematic and evolutionary microbiology 20121101

Indole-3-acetaldehyde from Rhodococcus sp. BFI 332 inhibits Escherichia coli O157:H7 biofilm formation.

Applied microbiology and biotechnology 20121101

Tryptophan tryptophylquinone biosynthesis: a radical approach to posttranslational modification.

Biochimica et biophysica acta 20121101

Reduced diversity and imbalance of fecal microbiota in patients with ulcerative colitis.

Digestive diseases and sciences 20121101

Evaluation of various boar taint detection methods.

Animal : an international journal of animal bioscience 20121101

Molecular model of the ring-opening and ring-closure reaction of a fluorinated indolylfulgide.

The journal of physical chemistry. A 20121101

Formulation and characterization of polyester/polycarbonate nanoparticles for delivery of a novel microtubule destabilizing agent.

Pharmaceutical research 20121101

[Pityriasis versicolor : new aspects of an old disease].

Der Hautarzt; Zeitschrift fur Dermatologie, Venerologie, und verwandte Gebiete 20121101

Microfractionation bioactivity-based ultra performance liquid chromatography/quadrupole time-of-flight mass spectrometry for the identification of nuclear factor-κB inhibitors and β2 adrenergic receptor agonists in an alkaloidal extract of the folk herb Alstonia scholaris.

Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20121101

CO2 on a tightrope: stabilization, room-temperature decarboxylation, and sodium-induced carboxylate migration.

Chemistry (Weinheim an der Bergstrasse, Germany) 20121029

AlCl3 mediated unexpected migration of sulfonyl groups: regioselective synthesis of 7-sulfonyl indoles of potential pharmacological interest.

Chemical communications (Cambridge, England) 20121028

Ir(I)-catalyzed C-H bond alkylation of C2-position of indole with alkenes: selective synthesis of linear or branched 2-alkylindoles.

Journal of the American Chemical Society 20121024

Precise RNAi-mediated silencing of metabolically active proteins in the defence secretions of juvenile leaf beetles.

Proceedings. Biological sciences 20121022

Acute toxicity and gastroprotective effect of the Schiff base ligand ¹H-indole-3-ethylene-5-nitrosalicylaldimine and its nickel (II) complex on ethanol induced gastric lesions in rats.

Molecules (Basel, Switzerland) 20121022

Palladium(II)-catalyzed oxidative C-H/C-H coupling and eliminative S(N)(H) reactions in direct functionalization of imidazole oxides with indoles.

The Journal of organic chemistry 20121019

Synthesis of the pentacyclic skeleton of the indole alkaloid arboflorine.

Organic letters 20121019

Synthesis of π-extended porphyrins via intramolecular oxidative coupling.

Chemical communications (Cambridge, England) 20121018

Studies on 2-arylhydrazononitriles: synthesis of 3-aryl-2-arylhydrazopropanenitriles and their utility as precursors to 2-substituted indoles, 2-substituted-1,2,3-triazoles, and 1-substituted pyrazolo[4,3-d]pyrimidines.

Molecules (Basel, Switzerland) 20121018

Enantioselective synthesis of tetrahydrocarbazoles through a Michael addition/Ciamician-Plancher rearrangement sequence: asymmetric synthesis of a potent constrained analogue of MS-245.

Chemistry (Weinheim an der Bergstrasse, Germany) 20121015

Synthesis and antiviral activity of 4,6-disubstituted pyrimido[4,5-b]indole ribonucleosides.

Bioorganic & medicinal chemistry 20121015

Synthesis of hexahydroindoles by intramolecular C(sp3)-H alkenylation: application to the synthesis of the core of aeruginosins.

Angewandte Chemie (International ed. in English) 20121008

Bacterial synthesis of diverse indole terpene alkaloids by an unparalleled cyclization sequence.

Angewandte Chemie (International ed. in English) 20121008

Gallium(III)-catalyzed three-component (4+3) cycloaddition reactions.

Angewandte Chemie (International ed. in English) 20121008

A BODIPY derivative as a highly selective 'Off-On' fluorescent chemosensor for hydrogen sulfate anion.

The Analyst 20121007

Aerobic palladium(II)-catalyzed dehydrogenation of cyclohexene-1-carbonyl indole amides: an indole-directed aromatization.

The Journal of organic chemistry 20121005

Comprehensive synthesis of photoreactive (3-trifluoromethyl)diazirinyl indole derivatives from 5- and 6- trifluoroacetylindoles for photoaffinity labeling.

The Journal of organic chemistry 20121005

Enantioselective cyclopropanation of indoles: construction of all-carbon quaternary stereocenters.

Organic letters 20121005

Direct amidation of carboxylic acids catalyzed by ortho-iodo arylboronic acids: catalyst optimization, scope, and preliminary mechanistic study supporting a peculiar halogen acceleration effect.

The Journal of organic chemistry 20121005

Mechanistic studies on CymD: a tryptophan reverse N-prenyltransferase.

Biochemistry 20121002

Pharmacokinetics and effect of food after oral administration of prolonged-release tablets of ropinirole hydrochloride in Japanese patients with Parkinson's disease.

Journal of clinical pharmacy and therapeutics 20121001

Volatile organic compounds at swine facilities: a critical review.

Chemosphere 20121001

Methyl jasmonate and yeast extract stimulate mitragynine production in Mitragyna speciosa (Roxb.) Korth. shoot culture.

Biotechnology letters 20121001

Aerobic degradation of phenolics and aromatic hydrocarbons in presence of cyanide.

Bioresource technology 20121001

Non-genetic mechanisms communicating antibiotic resistance: rethinking strategies for antimicrobial drug design.

Expert opinion on drug discovery 20121001

Indole derivative production by the root endophyte Piriformospora indica is not required for growth promotion but for biotrophic colonization of barley roots.

The New phytologist 20121001

Threshold detection of boar taint chemicals using parasitic wasps.

Journal of food science 20121001

Synthesis and evaluation of indole-containing 3,5-diarylisoxazoles as potential pro-apoptotic antitumour agents.

European journal of medicinal chemistry 20121001

Synthesis and biological activity of obatoclax derivatives as novel and potent SHP-1 agonists.

European journal of medicinal chemistry 20121001

Thiourea-catalysed ring opening of episulfonium ions with indole derivatives by means of stabilizing non-covalent interactions.

Nature chemistry 20121001

3-(2-Acetamido-eth-yl)-1H-indol-5-yl 4-nitro-phenyl carbonate.

Acta crystallographica. Section E, Structure reports online 20121001

Electrospray ionization tandem mass spectrometry of chaetoglobosins.

Rapid communications in mass spectrometry : RCM 20120930

16,17-Dihydro-17b-hydroxy isomitraphylline alkaloid as an inhibitor of DPP-IV, and its effect on incretin hormone and β-cell proliferation in diabetic rat.

European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20120929

Acute toxicity, antinociceptive activity and indole alkaloids of aqueous extract from bark of Aspidosperma cuspa (Kunth) Blake.

Journal of ethnopharmacology 20120928

Caffeine and sugars interact in aqueous solutions: a simulation and NMR study.

The journal of physical chemistry. B 20120927

Molecular dynamics of β-hairpin models of epigenetic recognition motifs.

Journal of the American Chemical Society 20120926

Volatiles from apple trees infested with light brown apple moth larvae attract the parasitoid Dolichogenidia tasmanica.

Journal of agricultural and food chemistry 20120926

Rhodium acetate/base-catalyzed N-silylation of indole derivatives with hydrosilanes.

Chemical communications (Cambridge, England) 20120925

Highly enantioselective Friedel-Crafts alkylation of indoles and pyrrole with β,γ-unsaturated α-ketoesters catalyzed by heteroarylidene-tethered bis(oxazoline) copper complexes.

Chemical communications (Cambridge, England) 20120925

Catalytic coupling of arene C-H bonds and alkynes for the synthesis of coumarins: substrate scope and application to the development of neuroimaging agents.

The Journal of organic chemistry 20120921

A cascade reaction of azolopyrimidines. Synthesis of unusual indole and azaindole derivatives.

Chemical communications (Cambridge, England) 20120921

Copper-catalyzed tandem synthesis of indolo-, pyrrolo[2,1-a]isoquinolines, naphthyridines and bisindolo/pyrrolo[2,1-a]isoquinolines via hydroamination of ortho-haloarylalkynes followed by C-2 arylation.

The Journal of organic chemistry 20120921

FeCl3·6H2O-catalyzed alkenylation of indoles with aldehydes.

The Journal of organic chemistry 20120921

Synthesis of pyrrolo[2,3-b]indole via iodine(III)-mediated intramolecular annulation.

Organic letters 20120921

Small-molecule-based affinity chromatography method for antibody purification via nucleotide binding site targeting.

Analytical chemistry 20120918

Mechanistic aspects of nitrogen-heterocyclic compound adsorption on bamboo charcoal.

Journal of colloid and interface science 20120915

Zero kinetic energy photoelectron spectroscopy of tryptamine and the dissociation pathway of the singly hydrated cation cluster.

The Journal of chemical physics 20120914

Structure and catalytic mechanism of a cyclic dipeptide prenyltransferase with broad substrate promiscuity.

Journal of molecular biology 20120907

Time-dependent density functional theory (TDDFT) modelling of Pechmann dyes: from accurate absorption maximum prediction to virtual dye screening.

Organic & biomolecular chemistry 20120907

π-Extended thiadiazoles fused with thienopyrrole or indole moieties: synthesis, structures, and properties.

The Journal of organic chemistry 20120907

Fluorinated alcohols as promoters for the metal-free direct substitution reaction of allylic alcohols with nitrogenated, silylated, and carbon nucleophiles.

The Journal of organic chemistry 20120907

Silver acetate catalyzed hydroamination of 1-(2-(sulfonylamino)phenyl)prop-2-yn-1-ols to (Z)-2-methylene-1-sulfonylindolin-3-ols.

The Journal of organic chemistry 20120907

Total synthesis of (±)-hirsutine: application of phosphine-catalyzed imine-allene [4 + 2] annulation.

Organic letters 20120907

A synthetic method for palladium-catalyzed stannylation at the 5- and 6-benzo positions of indoles.

Organic letters 20120907

Effect of acceptor heteroatoms on π-hydrogen bonding interactions: a study of indole···thiophene heterodimer in a supersonic jet.

The Journal of chemical physics 20120907

The role of site-specific hydrogen bonding interactions in the solvation dynamics of N-acetyltryptophanamide.

The journal of physical chemistry. B 20120906

Pd(II)-catalyzed regioselective 2-alkylation of indoles via a norbornene-mediated C-H activation: mechanism and applications.

Journal of the American Chemical Society 20120905

Strictosidinic acid, isolated from Psychotria myriantha Mull. Arg. (Rubiaceae), decreases serotonin levels in rat hippocampus.

Fitoterapia 20120901

Bioactivity guided isolation of antipsychotic constituents from the leaves of Rauwolfia tetraphylla L.

Fitoterapia 20120901

The molecular details of WPD-loop movement differ in the protein-tyrosine phosphatases YopH and PTP1B.

Archives of biochemistry and biophysics 20120901

An attenuated mutant of avian pathogenic Escherichia coli serovar O78: a possible live vaccine strain for prevention of avian colibacillosis.

Microbiology and immunology 20120901

Structural insights into cholinesterases inhibition by harmane β-carbolinium derivatives: a kinetics-molecular modeling approach.

Phytochemistry 20120901

The bacterial signalling molecule indole attenuates the virulence of the fungal pathogen Candida albicans.

Journal of applied microbiology 20120901

Characterization of three propane-inducible oxygenases in Mycobacterium sp. strain ENV421.

Letters in applied microbiology 20120901

Synthesis and biological evaluation of novel C-indolylxylosides as sodium-dependent glucose co-transporter 2 inhibitors.

European journal of medicinal chemistry 20120901

Indole-3-acetaldoxime-derived compounds restrict root colonization in the beneficial interaction between Arabidopsis roots and the endophyte Piriformospora indica.

Molecular plant-microbe interactions : MPMI 20120901

Indole alkaloids from two cultured cyanobacteria, Westiellopsis sp. and Fischerella muscicola.

Bioorganic & medicinal chemistry 20120901

Phenotypic and molecular characterization of a novel strongly hemolytic Brachyspira species, provisionally designated 'Brachyspira hampsonii'.

Journal of veterinary diagnostic investigation : official publication of the American Association of Veterinary Laboratory Diagnosticians, Inc 20120901

Diethyl 3,3'-(phenyl-methyl-ene)bis-(1H-indole-2-carboxyl-ate).

Acta crystallographica. Section E, Structure reports online 20120901

Simultaneous determination of alkaloids and flavonoids from aerial parts of Passiflora species and dietary supplements using UPLC-UV-MS and HPTLC.

Natural product communications 20120901

Hexafluoroisopropanol: a powerful solvent for the hydrogenation of indole derivatives. Selective access to tetrahydroindoles or cis-fused octahydroindoles.

Organic & biomolecular chemistry 20120828

Binding motifs of silver in prion octarepeat model peptides: a joint ion mobility, IR and UV spectroscopies, and theoretical approach.

Physical chemistry chemical physics : PCCP 20120828

Indole peroxygenase activity of indoleamine 2,3-dioxygenase.

Proceedings of the National Academy of Sciences of the United States of America 20120828

Evidence of preorganization in quinonoid intermediate formation from L-Trp in H463F mutant Escherichia coli tryptophan indole-lyase from effects of pressure and pH.

Biochemistry 20120821

A general method for palladium-catalyzed direct carbonylation of indole with alcohol and phenol.

Organic letters 20120817

Palladium-catalyzed cascade process consisting of isocyanide insertion and benzylic C(sp3)-H activation: concise synthesis of indole derivatives.

Organic letters 20120817

Goniomedines A and B: unprecedented bisindole alkaloids formed through fusion of two indole moieties via a dihydropyran unit.

Organic letters 20120817

DFT and surface-enhanced Raman scattering study of tryptophan-silver complex.

Journal of colloid and interface science 20120815

C3-heteroaroyl cannabinoids as photolabeling ligands for the CB2 cannabinoid receptor.

Bioorganic & medicinal chemistry letters 20120815

Metabolism and metabolites of dithiocarbamates in the plant pathogenic fungus Leptosphaeria maculans.

Journal of agricultural and food chemistry 20120815

The structure of 5-cyanoindole in the ground and the lowest electronically excited singlet states, deduced from rotationally resolved electronic spectroscopy and ab initio theory.

Physical chemistry chemical physics : PCCP 20120807

Using solid-state NMR to monitor the molecular consequences of Cryptococcus neoformans melanization with different catecholamine precursors.

Biochemistry 20120807

Al-catalyzed facile construction of quaternary C-C bonds by the allylic substitution of tertiary alcohols: a concise and formal synthesis of (±)-mersicarpine.

Chemistry (Weinheim an der Bergstrasse, Germany) 20120806

Nucleophilic addition of Grignard reagents to 3-acylindoles: stereoselective synthesis of highly substituted indoline scaffolds.

Organic letters 20120803

The novel indole compound SK228 induces apoptosis and FAK/Paxillin disruption in tumor cell lines and inhibits growth of tumor graft in the nude mouse.

International journal of cancer 20120801

Effects of feeding polydextrose on faecal characteristics, microbiota and fermentative end products in healthy adult dogs.

The British journal of nutrition 20120801

Detection of bioactive exometabolites produced by the filamentous marine cyanobacterium Geitlerinema sp.

Marine biotechnology (New York, N.Y.) 20120801

Influence of dietary protein content and source on colonic fermentative activity in dogs differing in body size and digestive tolerance.

Journal of animal science 20120801

Different scalding techniques do not affect boar taint.

Meat science 20120801

On the generation and quenching of reactive-oxygen-species by aqueous vitamin B2 and serotonin under visible-light irradiation.

Journal of photochemistry and photobiology. B, Biology 20120801

Neurotrophic actions initiated by proNGF in adult sensory neurons may require peri-somatic glia to drive local cleavage to NGF.

Journal of neurochemistry 20120801

Secondary metabolites from a marine-derived fungus Aspergillus carneus Blochwitz.

Phytochemistry 20120801

A three-step culture system to increase the xanthone production and antifungal activity of Hypericum perforatum subsp. angustifolium in vitro roots.

Plant physiology and biochemistry : PPB 20120801

Suppression of hydatidiform molar growth by inhibiting endogenous brain-derived neurotrophic factor/tyrosine kinase B signaling.

Endocrinology 20120801

Microbial transformation of azaarenes and potential uses in pharmaceutical synthesis.

Applied microbiology and biotechnology 20120801

Indole based cyclooxygenase inhibitors: synthesis, biological evaluation, docking and NMR screening.

European journal of medicinal chemistry 20120801

A labeled substrate approach to discovery of biocatalytic reactions: a proof of concept transformation with N-methylindole.

Journal of the American Chemical Society 20120801

Discovery of a novel azaindole class of antibacterial agents targeting the ATPase domains of DNA gyrase and Topoisomerase IV.

Bioorganic & medicinal chemistry letters 20120801

Structure of human Rack1 protein at a resolution of 2.45 Å.

Acta crystallographica. Section F, Structural biology and crystallization communications 20120801

Methyl 4-benz-yloxy-7-meth-oxy-1-methyl-1H-indole-2-carboxyl-ate.

Acta crystallographica. Section E, Structure reports online 20120801

Natural products from Antarctic colonial ascidians of the genera Aplidium and Synoicum: variability and defensive role.

Marine drugs 20120801

Straightforward acid-catalyzed synthesis of pyrrolyldipyrromethenes.

Angewandte Chemie (International ed. in English) 20120727

InCl3-mediated addition of indole to isatogens: an expeditious synthesis of 13-deoxy-isatisine A.

Chemistry (Weinheim an der Bergstrasse, Germany) 20120727

Mechanism inspired development of rationally designed dihydrofolate reductase inhibitors as anticancer agents.

Journal of medicinal chemistry 20120726

Are the wild and laboratory insect populations different in semiochemical emission? The case of the medfly sex pheromone.

Journal of agricultural and food chemistry 20120725

Access to electron-rich arene-fused hexahydroquinolizinones through a gold-catalysis-initiated cascade process.

Angewandte Chemie (International ed. in English) 20120716

Hyrtioreticulins A-E, indole alkaloids inhibiting the ubiquitin-activating enzyme, from the marine sponge Hyrtios reticulatus.

Bioorganic & medicinal chemistry 20120715

Cristatumins A-D, new indole alkaloids from the marine-derived endophytic fungus Eurotium cristatum EN-220.

Bioorganic & medicinal chemistry letters 20120715

A multicomponent synthetic strategy for two-carbon-tethered 1,3-oxathiole-indole pairs.

Organic & biomolecular chemistry 20120714

Human immunodeficiency virus type 1 alters brain-derived neurotrophic factor processing in neurons.

The Journal of neuroscience : the official journal of the Society for Neuroscience 20120711

Experimentally measured permanent dipoles induced by hydrogen bonding. The Stark spectrum of indole-NH3.

Physical chemistry chemical physics : PCCP 20120707

Study of N1-alkylation of indoles from the reaction of 2(or 3)-aminoindole-3-(or 2)carbonitriles with DMF-dialkylacetals.

Organic & biomolecular chemistry 20120707

Base-mediated selective synthesis of diversely substituted N-heterocyclic enamines and enaminones by the hydroamination of alkynes.

The Journal of organic chemistry 20120706

Lanthanide amido complexes incorporating amino-coordinate-lithium bridged bis(indolyl) ligands: synthesis, characterization, and catalysis for hydrophosphonylation of aldehydes and aldimines.

Inorganic chemistry 20120702

Caenispirillum salinarum sp. nov., a member of the family Rhodospirillaceae isolated from a solar saltern.

International journal of systematic and evolutionary microbiology 20120701

Role of conserved active site tryptophan-101 in functional activity and stability of phosphoserine aminotransferase from an enteric human parasite.

Amino acids 20120701

Altered expression level of Escherichia coli proteins in response to treatment with the antifouling agent zosteric acid sodium salt.

Environmental microbiology 20120701

Genetic parameters for androstenone, skatole, indole, and human nose scores as measures of boar taint and their relationship with finishing traits.

Journal of animal science 20120701

Tryptophan decarboxylase plays an important role in ajmalicine biosynthesis in Rauvolfia verticillata.

Planta 20120701

HPTLC method for the simultaneous determination of four indole alkaloids in Rauwolfia tetraphylla: a study of organic/green solvent and continuous/pulse sonication.

Journal of pharmaceutical and biomedical analysis 20120701

Finger-loop inhibitors of the HCV NS5b polymerase. Part 1: Discovery and optimization of novel 1,6- and 2,6-macrocyclic indole series.

Bioorganic & medicinal chemistry letters 20120701

UVA-induced oxidative degradation of melanins: fission of indole moiety in eumelanin and conversion to benzothiazole moiety in pheomelanin.

Pigment cell & melanoma research 20120701

Crystal structure of the lectin of Camptosema pedicellatum: implications of a conservative substitution at the hydrophobic subsite.

Journal of biochemistry 20120701

Synthesis and fungicidal activity of novel pimprinine analogues.

European journal of medicinal chemistry 20120701

Transdermal behaviors comparisons among Evodia rutaecarpa extracts with different purity of evodiamine and rutaecarpine and the effect of topical formulation in vivo.

Fitoterapia 20120701

Pharmacokinetics, pharmacodynamics and metabolism of a novel anticancer agent for prostate cancer.

International journal of oncology 20120701

Attenuation of the jasmonate burst, plant defensive traits, and resistance to specialist monarch caterpillars on shaded common milkweed (Asclepias syriaca).

Journal of chemical ecology 20120701

N'-[(E)-4-(Dimethyl-amino)-benz-ylidene]-2-(5-meth-oxy-2-methyl-1H-indol-3-yl)acetohydrazide.

Acta crystallographica. Section E, Structure reports online 20120701

(S)-(-)-2-(1H-Indol-3-yl)-N-(1-phenyl-eth-yl)acetamide.

Acta crystallographica. Section E, Structure reports online 20120701

3-(1H-Indol-3-yl)-2-(2-nitro-benzene-sulfonamido)-propanoic acid including an unknown solvate.

Acta crystallographica. Section E, Structure reports online 20120701

In-silico investigation of antitrypanosomal phytochemicals from Nigerian medicinal plants.

PLoS neglected tropical diseases 20120701

Determination of dimethyltryptamine and β-carbolines (ayahuasca alkaloids) in plasma samples by LC-MS/MS.

Bioanalysis 20120701

Alkaloids produced by endophytic fungi: a review.

Natural product communications 20120701

Enantioselective Friedel-Crafts alkylation of indoles with 2-enoylpyridine-N-oxides catalyzed by glucoBOX-Cu(II) complex.

Organic & biomolecular chemistry 20120628

The chemoselective reactions of tyrosine-containing G-protein-coupled receptor peptides with [Cp*Rh(H2O)3](OTf)2, including 2D NMR structures and the biological consequences.

Journal of the American Chemical Society 20120627

New quinoxaline derivatives as potential MT₁ and MT₂ receptor ligands.

Molecules (Basel, Switzerland) 20120625

Conformational, steric and electronic effects on the site- and chemoselectivity of the metal-catalyzed reaction of N-bis(trimethylsilyl)methyl, N-(2-indolyl)methyl α-diazoamides.

Organic & biomolecular chemistry 20120621

Designing allosteric control into enzymes by chemical rescue of structure.

Journal of the American Chemical Society 20120620

Sulfonyl-morpholino-pyrimidines: SAR and development of a novel class of selective mTOR kinase inhibitor.

Bioorganic & medicinal chemistry letters 20120615

Synthesis and evaluation of N(1)-alkylindole-3-ylalkylammonium compounds as nicotinic acetylcholine receptor ligands.

Bioorganic & medicinal chemistry 20120615

Prenylation at the indole ring leads to a significant increase of cytotoxicity of tryptophan-containing cyclic dipeptides.

Bioorganic & medicinal chemistry letters 20120615

Prenylation of a nonaromatic carbon of indolylbutenone by a fungal indole prenyltransferase.

Organic letters 20120615

Mechanism of the N-protecting group dependent annulations of 3-aryloxy alkynyl indoles under gold catalysis: a computational study.

Organic & biomolecular chemistry 20120614

Accurate prediction of cation-π interaction energy using substituent effects.

The journal of physical chemistry. A 20120614

Diazine indole acetic acids as potent, selective, and orally bioavailable antagonists of chemoattractant receptor homologous molecule expressed on Th2 cells (CRTH2) for the treatment of allergic inflammatory diseases.

Journal of medicinal chemistry 20120614

Palladium-catalyzed aerobic oxidative cyclization of N-aryl imines: indole synthesis from anilines and ketones.

Journal of the American Chemical Society 20120606

Total synthesis of Akuammiline alkaloid (-)-vincorine via intramolecular oxidative coupling.

Journal of the American Chemical Society 20120606

An acid-promoted novel skeletal rearrangement initiated by intramolecular ipso-Friedel-Crafts-type addition to 3-alkylidene indolenium cations.

Chemical communications (Cambridge, England) 20120604

Synthesis, characterization and biocidal activity of some transition metal(II) complexes with isatin salicylaldehyde acyldihydrazones.

Journal of enzyme inhibition and medicinal chemistry 20120601

Conformational and stereoelectronic investigation of tryptamine. An AIM/NBO study.

Journal of molecular modeling 20120601

Bufothionine, a possible effective component in cinobufocini injection for hepatocellular carcinoma.

Journal of ethnopharmacology 20120601

π-Cation interactions as the origin of the weak absorption at 532 nm observed in tryptophan-containing polypeptides.

Photochemical & photobiological sciences : Official journal of the European Photochemistry Association and the European Society for Photobiology 20120601

An exon-specific U1 small nuclear RNA (snRNA) strategy to correct splicing defects.

Human molecular genetics 20120601

Isorhynchophylline: A plant alkaloid with therapeutic potential for cardiovascular and central nervous system diseases.

Fitoterapia 20120601

Released products of pathogenic bacteria stimulate biofilm formation by Escherichia coli K-12 strains.

Antonie van Leeuwenhoek 20120601

Thermal disaggregation of type B yeast hexokinase by indole derivatives: a mechanistic study.

International journal of biological macromolecules 20120601

Cytotoxic dimeric indole alkaloids from Catharanthus roseus.

Fitoterapia 20120601

Multipotent MAO and cholinesterase inhibitors for the treatment of Alzheimer's disease: synthesis, pharmacological analysis and molecular modeling of heterocyclic substituted alkyl and cycloalkyl propargyl amine.

European journal of medicinal chemistry 20120601

Chemistry and biology of fascaplysin, a potent marine-derived CDK-4 inhibitor.

Mini reviews in medicinal chemistry 20120601

Meridianins: marine-derived potent kinase inhibitors.

Mini reviews in medicinal chemistry 20120601

Full evaporation dynamic headspace and gas chromatography-mass spectrometry for uniform enrichment of odor compounds in aqueous samples.

Journal of chromatography. A 20120601

Responses of Arabidopsis thaliana plant lines differing in hydroxylation of aliphatic glucosinolate side chains to feeding of a generalist and specialist caterpillar.

Plant physiology and biochemistry : PPB 20120601

Tryptophan oxygenation: mechanistic considerations.

Biochemical Society transactions 20120601

Modulation of imprinting efficiency in nanogels with catalytic activity in the Kemp elimination.

Journal of molecular recognition : JMR 20120601

3-(2-Methyl-2-nitro-prop-yl)-1H-indole.

Acta crystallographica. Section E, Structure reports online 20120601

5-Meth-oxy-2-[(5-meth-oxy-1H-indol-1-yl)carbon-yl]-1H-indole.

Acta crystallographica. Section E, Structure reports online 20120601

3-(1,2-Di-p-tolyl-vin-yl)-2-methyl-1H-indole.

Acta crystallographica. Section E, Structure reports online 20120601

Linear and non-linear quantitative structure-activity relationship models on indole substitution patterns as inhibitors of HIV-1 attachment.

Indian journal of biochemistry & biophysics 20120601

New indole alkaloid from Peschiera affinis (Apocynaceae).

Natural product communications 20120601

Indole alkaloids from Vinca major and V. minor growing in Turkey.

Natural product communications 20120601

Determination of the absolute configuration of 19-OH-(-)-eburnamonine using a combination of residual dipolar couplings, DFT chemical shift predictions, and chiroptics.

Natural product communications 20120601

Photoactivated [3+2] addition of 6,7-seco-angustilobine B to fullerene [C60].

Natural product communications 20120601

Secondary metabolite production by the basidiomycete, Lentinus strigellus, under different culture conditions.

Natural product communications 20120601

Synthesis and anticancer activity of novel 5-(indole-2-yl)-3-substituted 1,2,4-oxadiazoles.

Drug discoveries & therapeutics 20120601

[Chemical constituents of Rauvolfia verticillata].

Yao xue xue bao = Acta pharmaceutica Sinica 20120601

[The subcellular organelles of peroxisome, realization of biologic functions of trophology, homeostasis, endoecology and functional bond with mitochondrion: the lecture].

Klinicheskaia laboratornaia diagnostika 20120601

Identification of novel liver X receptor activators by structure-based modeling.

Journal of chemical information and modeling 20120525

A validated ultra-high performance liquid chromatography coupled to high resolution mass spectrometry analysis for the simultaneous quantification of the three known boar taint compounds.

Journal of chromatography. A 20120525

Indole alkaloids from Geissospermum reticulatum.

Journal of natural products 20120525

Perhentidines A-C: macroline-macroline bisindoles from Alstonia and the absolute configuration of perhentinine and macralstonine.

Journal of natural products 20120525

α-Glucosidase inhibitory constituents from Acanthopanax senticosus harm leaves.

Molecules (Basel, Switzerland) 20120525

Progress in palladium-based catalytic systems for the sustainable synthesis of annulated heterocycles: a focus on indole backbones.

Chemical Society reviews 20120521

Gold(I)-catalyzed rearrangement of 3-silyloxy-1,5-enynes: an efficient synthesis of benzo[b]thiophenes, dibenzothiophenes, dibenzofurans, and indole derivatives.

Chemistry (Weinheim an der Bergstrasse, Germany) 20120521

Synthesis of phidianidines A and B.

The Journal of organic chemistry 20120518

Total syntheses of anominine and tubingensin A.

Journal of the American Chemical Society 20120516

Structure-dependent activation of NR4A2 (Nurr1) by 1,1-bis(3'-indolyl)-1-(aromatic)methane analogs in pancreatic cancer cells.

Biochemical pharmacology 20120515

Silver triflate catalyzed tandem heterocyclization/alkynylation of 1-((2-tosylamino)aryl)but-2-yne-1,4-diols to 2-alkynyl indoles.

Chemistry (Weinheim an der Bergstrasse, Germany) 20120514

Pharmacokinetic evaluation and in vitro-in vivo correlation (IVIVC) of novel methylene-substituted 3,3' diindolylmethane (DIM).

European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20120512

A concise and versatile double-cyclization strategy for the highly stereoselective synthesis and arylative dimerization of Aspidosperma alkaloids.

Angewandte Chemie (International ed. in English) 20120507

Ketosulfonyl indoles in the regiodefined synthesis of tryptophols and related indole derivatives.

Organic & biomolecular chemistry 20120507

Total synthesis and absolute configuration of nocardioazine B.

Chemical communications (Cambridge, England) 20120507

Structure-based macrocyclization yields hepatitis C virus NS5B inhibitors with improved binding affinities and pharmacokinetic properties.

Angewandte Chemie (International ed. in English) 20120507

Concise total synthesis of (-)-mersicarpine.

Organic letters 20120504

Molecular dynamics simulations on the aggregation behavior of indole type organic dye molecules in dye-sensitized solar cells.

Journal of molecular modeling 20120501

Melatonin increases dendritogenesis in the hilus of hippocampal organotypic cultures.

Journal of pineal research 20120501

Effects of glucosinolates on a generalist and specialist leaf-chewing herbivore and an associated parasitoid.

Phytochemistry 20120501

Identification and characterization of an indigo-producing oxygenase involved in indole 3-acetic acid utilization by Acinetobacter baumannii.

Antonie van Leeuwenhoek 20120501

Inhibition of histone H3K9 methyltransferases by gliotoxin and related epipolythiodioxopiperazines.

The Journal of antibiotics 20120501

Deletion of penicillin-binding protein 1b impairs biofilm formation and motility in Escherichia coli.

Research in microbiology 20120501

Feeding dried chicory root to pigs decrease androstenone accumulation in fat by increasing hepatic 3β hydroxysteroid dehydrogenase expression.

The Journal of steroid biochemistry and molecular biology 20120501

Effects of koumine, an alkaloid of Gelsemium elegans Benth., on inflammatory and neuropathic pain models and possible mechanism with allopregnanolone.

Pharmacology, biochemistry, and behavior 20120501

Signaling-mediated bacterial persister formation.

Nature chemical biology 20120501

Overcoming fluconazole resistance in Candida albicans clinical isolates with tetracyclic indoles.

Bioorganic & medicinal chemistry letters 20120501

Manzamines: a potential for novel cures.

Cell cycle (Georgetown, Tex.) 20120501

Feeding Jerusalem artichoke reduced skatole level and changed intestinal microbiota in the gut of entire male pigs.

Animal : an international journal of animal bioscience 20120501

Potassium [1-(tert-but-oxy-carbon-yl)-1H-indol-3-yl]trifluoro-borate hemihydrate.

Acta crystallographica. Section E, Structure reports online 20120501

4-(4-Chloro-phen-yl)-2,6-bis-(1H-indol-3-yl)-1,4-dihydro-pyridine-3,5-dicarbo-nitrile ethanol monosolvate.

Acta crystallographica. Section E, Structure reports online 20120501

2,3,6,7-Tetra-bromo-9-butyl-9H-carbazole.

Acta crystallographica. Section E, Structure reports online 20120501

Ethyl 2-benzoyl-6-methyl-indolizine-7-carboxyl-ate.

Acta crystallographica. Section E, Structure reports online 20120501

6-Meth-oxy-1-(4-meth-oxy-phen-yl)-1,2,3,4-tetra-hydro-9H-β-carbolin-2-ium acetate.

Acta crystallographica. Section E, Structure reports online 20120501

[2-(1H-Indol-4-yl)eth-yl]dipropyl-amine.

Acta crystallographica. Section E, Structure reports online 20120501

(±)-trans-5-Benzoyl-2-(1H-indol-3-yl)-4-phenyl-4,5-dihydro-furan-3-carbonitrile.

Acta crystallographica. Section E, Structure reports online 20120501

6-Fluoro-1H-indole-3-carb-oxy-lic acid.

Acta crystallographica. Section E, Structure reports online 20120501

Volatiles from Michelia champaca flower: comparative analysis by simultaneous distillation-extraction and solid phase microextraction.

Natural product communications 20120501

Waikialoid A suppresses hyphal morphogenesis and inhibits biofilm development in pathogenic Candida albicans.

Journal of natural products 20120427

Is there no end to the total syntheses of strychnine? Lessons learned in strategy and tactics in total synthesis.

Angewandte Chemie (International ed. in English) 20120427

Fungal origins of the bicyclo[2.2.2]diazaoctane ring system of prenylated indole alkaloids.

Journal of natural products 20120427

Synthesis of new indole derivatives structurally related to donepezil and their biological evaluation as acetylcholinesterase inhibitors.

Molecules (Basel, Switzerland) 20120425

Site-specific synapsin I phosphorylation participates in the expression of post-tetanic potentiation and its enhancement by BDNF.

The Journal of neuroscience : the official journal of the Society for Neuroscience 20120425

Double C-H functionalization in sequential order: direct synthesis of polycyclic compounds by a palladium-catalyzed C-H alkenylation-arylation cascade.

Chemistry (Weinheim an der Bergstrasse, Germany) 20120423

Divergent total syntheses of (-)-aspidospermine and (+)-spegazzinine.

Organic letters 20120420

Insights into quinaldic acid moiety formation in thiostrepton biosynthesis facilitating fluorinated thiopeptide generation.

Chemistry & biology 20120420

Radical-mediated enzymatic methylation: a tale of two SAMS.

Accounts of chemical research 20120417

Total synthesis of exiguamines A and B inspired by catecholamine chemistry.

Chemistry (Weinheim an der Bergstrasse, Germany) 20120416

Total syntheses of the elusive welwitindolinones with bicyclo[4.3.1] cores.

Angewandte Chemie (International ed. in English) 20120416

Infrared multiple-photon dissociation spectroscopy of tripositive ions: lanthanum-tryptophan complexes.

Inorganic chemistry 20120416

Calcium/calmodulin inhibition of the Arabidopsis BRASSINOSTEROID-INSENSITIVE 1 receptor kinase provides a possible link between calcium and brassinosteroid signalling.

The Biochemical journal 20120415

Prospective acetylcholinesterase inhibitory activity of indole and its analogs.

Bioorganic & medicinal chemistry letters 20120415

Silver-promoted Friedel-Crafts reaction: concise total synthesis of (-)-ardeemin, (-)-acetylardeemin and (-)-formylardeemin.

Organic & biomolecular chemistry 20120414

Novel inhibitors of neurotropic alphavirus replication that improve host survival in a mouse model of acute viral encephalitis.

Journal of medicinal chemistry 20120412

Venting-while-heating microwave-assisted synthesis of 3-arylthioindoles.

ACS combinatorial science 20120409

Highly selective organic fluorescent probe for azide ion: formation of a 'molecular ring'.

The Analyst 20120407

Synthesis of dopamine and serotonin derivatives for immobilization on a solid support.

The Journal of organic chemistry 20120406

Total synthesis of (-)-herbindoles A, B, and C via transition-metal-catalyzed intramolecular [2 + 2 + 2] cyclization between ynamide and diynes.

Organic letters 20120406

Synthesis of tetrahydro-β-carbolines via isomerization of N-allyltryptamines: a metal-catalyzed variation on the Pictet-Spengler theme.

Chemical communications (Cambridge, England) 20120404

Palladium-catalyzed dehydrogenative β'-functionalization of β-keto esters with indoles at room temperature.

Journal of the American Chemical Society 20120404

Naucline, a new indole alkaloid from the bark of Nauclea officinalis.

Molecules (Basel, Switzerland) 20120402

9-hydroxycanthin-6-one induces penile erection and delays ejaculation.

The journal of sexual medicine 20120401

Emerging trends in research on spatial and temporal organization of terpenoid indole alkaloid pathway in Catharanthus roseus: a literature update.

Protoplasma 20120401

Antiplasmodial indole alkaloids from Leuconotis griffithii.

Journal of natural medicines 20120401

Weakly hydrated surfaces and the binding interactions of small biological solutes.

European biophysics journal : EBJ 20120401

A proximal pair of positive charges provides the dominant ligand-binding contribution to complement-like domains from the LRP (low-density lipoprotein receptor-related protein).

The Biochemical journal 20120401

Blocking epidermal growth factor receptor activation by 3,3'-diindolylmethane suppresses ovarian tumor growth in vitro and in vivo.

The Journal of pharmacology and experimental therapeutics 20120401

Serotypes, virulence genes, and intimin types of shiga toxin-producing Escherichia coli and enteropathogenic Escherichia coli isolated from mastitic milk relevant to human health in Egypt.

Vector borne and zoonotic diseases (Larchmont, N.Y.) 20120401

7-fluoroindole as an antivirulence compound against Pseudomonas aeruginosa.

FEMS microbiology letters 20120401

Novel and viable acetylcholinesterase target site for developing effective and environmentally safe insecticides.

Current drug targets 20120401

Non-systemic drugs: a critical review.

Current pharmaceutical design 20120401

GC-MS metabolomic differentiation of selected citrus varieties with different sensitivity to citrus huanglongbing.

Plant physiology and biochemistry : PPB 20120401

Effect of water coordination on competition between π and non-π cation binding sites in aromatic amino acids: L-phenylalanine, L-tyrosine, and L-tryptophan Li+, Na +, and K+ complexes.

Journal of biological inorganic chemistry : JBIC : a publication of the Society of Biological Inorganic Chemistry 20120401

An protocol for genetic transformation of Catharanthus roseus by Agrobacterium rhizogenes A4.

Applied biochemistry and biotechnology 20120401

Lathyrus cicera copper amine oxidase reactions with tryptamine.

Journal of inorganic biochemistry 20120401

Indeno[1,2-b]indole derivatives as a novel class of potent human protein kinase CK2 inhibitors.

Bioorganic & medicinal chemistry 20120401

Iodine-catalyzed condensation of isatin with indoles: a facile synthesis of di(indolyl)indolin-2-ones and evaluation of their cytotoxicity.

Bioorganic & medicinal chemistry letters 20120401

Nerve growth factor-mediated neuronal plasticity in spinal cord contributes to neonatal maternal separation-induced visceral hypersensitivity in rats.

European journal of pain (London, England) 20120401

Less is more: treatment with BTH and laminarin reduces herbivore-induced volatile emissions in maize but increases parasitoid attraction.

Journal of chemical ecology 20120401

Ligand-dependent conformations and dynamics of the serotonin 5-HT(2A) receptor determine its activation and membrane-driven oligomerization properties.

PLoS computational biology 20120401

Bis(6-meth-oxy-1-methyl-2,3,4,9-tetra-hydro-1H-β-carbolin-2-ium) tetra-chloridozincate(II) dihydrate.

Acta crystallographica. Section E, Structure reports online 20120401

4a-Methyl-2,3,4,4a-tetra-hydro-1H-carbazole-6-sulfonamide.

Acta crystallographica. Section E, Structure reports online 20120401

2-[(1H-Imidazol-1-yl)meth-yl]-1-[4-(trifluoro-meth-yl)phen-yl]-1H-indole.

Acta crystallographica. Section E, Structure reports online 20120401

5-Benzoyl-2-(1H-indol-3-yl)-4-(4-methyl-phen-yl)-4,5-dihydro-furan-3-carbonitrile.

Acta crystallographica. Section E, Structure reports online 20120401

5-Meth-oxy-1-[(5-meth-oxy-1H-indol-2-yl)meth-yl]-1H-indole.

Acta crystallographica. Section E, Structure reports online 20120401

Bacteriophages with the ability to degrade uropathogenic Escherichia coli biofilms.

Viruses 20120401

1-(2-Methyl-benz-yl)-1H-indole-3-carbaldehyde.

Acta crystallographica. Section E, Structure reports online 20120401

Plant insecticidal toxins in ecological networks.

Toxins 20120401

Identification of isomeric 5-hydroxytryptophan- and oxindolylalanine-containing peptides by mass spectrometry.

Journal of mass spectrometry : JMS 20120401

Structural insight into the unique substrate binding mechanism and flavin redox state of UDP-galactopyranose mutase from Aspergillus fumigatus.

The Journal of biological chemistry 20120330

Crystal structure of perakine reductase, founding member of a novel aldo-keto reductase (AKR) subfamily that undergoes unique conformational changes during NADPH binding.

The Journal of biological chemistry 20120330

pH-dependent complexation of histamine H1 receptor antagonists and human serum albumin studied by UV resonance Raman spectroscopy.

The journal of physical chemistry. B 20120329

Asymmetric hydrovinylation of vinylindoles. A facile route to cyclopenta[g]indole natural products (+)-cis-trikentrin A and (+)-cis-trikentrin B.

Journal of the American Chemical Society 20120328

Effect of an alkaloidal fraction of Tabernaemontana elegans (Stapf.) on selected micro-organisms.

Journal of ethnopharmacology 20120327

Alternative reaction pathways in domino reactions of hydrazinediidozirconium complexes with alkynes.

Chemistry (Weinheim an der Bergstrasse, Germany) 20120326

Analysis of organic volatile flavor compounds in fermented stinky tofu using SPME with different fiber coatings.

Molecules (Basel, Switzerland) 20120326

Rh-catalyzed intramolecular sp2 C-H bond difluoromethylenation.

Chemical communications (Cambridge, England) 20120325

Ultrafast photophysics of the isolated indole molecule.

The journal of physical chemistry. A 20120322

Structure-guided evolution of cyan fluorescent proteins towards a quantum yield of 93%.

Nature communications 20120320

Non-contiguous finished genome sequence and description of Anaerococcus senegalensis sp. nov.

Standards in genomic sciences 20120319

Rational design of an auxin antagonist of the SCF(TIR1) auxin receptor complex.

ACS chemical biology 20120316

Brønsted acid catalyzed enantioselective α-amidoalkylation in the synthesis of isoindoloisoquinolines.

The Journal of organic chemistry 20120316

Synthesis of the core of actinophyllic acid using a transannular acyl radical cyclization.

Organic letters 20120316

Biomimetic total synthesis of (-)-isatisine A.

Organic letters 20120316

High-pressure accelerated asymmetric organocatalytic Friedel-Crafts alkylation of indoles with enones: application to quaternary stereogenic centers construction.

Organic letters 20120316

Allosteric regulation of substrate channeling and catalysis in the tryptophan synthase bienzyme complex.

Archives of biochemistry and biophysics 20120315

β-Carboline alkaloids from the leaves of Trigonostemon lii Y.T. Chang.

Bioorganic & medicinal chemistry letters 20120315

N-1 and C-3 substituted indole Schiff bases as selective COX-2 inhibitors: synthesis and biological evaluation.

Bioorganic & medicinal chemistry letters 20120315

Indolyl and dihydroindolyl N-glycinamides as potent and in vivo active NPY5 antagonists.

Bioorganic & medicinal chemistry letters 20120315

Efficient synthesis of carbazoles via PtCl2-catalyzed RT cyclization of 1-(indol-2-yl)-2,3-allenols: scope and mechanism.

Organic & biomolecular chemistry 20120314

A novel class of highly potent irreversible hepatitis C virus NS5B polymerase inhibitors.

Journal of medicinal chemistry 20120308

Cyclooxygenase-1-selective inhibitors based on the (E)-2'-des-methyl-sulindac sulfide scaffold.

Journal of medicinal chemistry 20120308

Gold-containing indoles as anticancer agents that potentiate the cytotoxic effects of ionizing radiation.

Journal of medicinal chemistry 20120308

Total synthesis of (+)-scholarisine A.

Journal of the American Chemical Society 20120307

Theoretical study of photo-physical properties of indolylmaleimide derivatives.

Physical chemistry chemical physics : PCCP 20120307

Bioactivity-based liquid chromatography-coupled electrospray ionization tandem ion trap/time of flight mass spectrometry for β₂AR agonist identification in alkaloidal extract of Alstonia scholaris.

Journal of chromatography. A 20120302

Synthesis of reported and revised structures of amathamide D and synthesis of convolutamine F, H and lutamide A, C.

The Journal of organic chemistry 20120302

Oxidative 1,2- and 1,3-alkyl shift processes: developments and applications in synthesis.

The Journal of organic chemistry 20120302

A concise total synthesis of (±)-trigonoliimine B.

Organic letters 20120302

Substrate binding and translocation of the serotonin transporter studied by docking and molecular dynamics simulations.

Journal of molecular modeling 20120301

Indole inhibition of ColE1 replication contributes to stable plasmid maintenance.

Plasmid 20120301

Back to the future: lessons learned in modern target-based and whole-cell lead optimization of antimalarials.

Current topics in medicinal chemistry 20120301

Structure-activity relationships for the interaction of 5,10-dihydroindeno[1,2-b]indole derivatives with human and bovine carbonic anhydrase isoforms I, II, III, IV and VI.

European journal of medicinal chemistry 20120301

A water-soluble calix[4]resorcinarene with L-pipecolinic acid groups as a chiral NMR solvating agent.

Chirality 20120301

Binding of an indole alkaloid, vinblastine to double stranded DNA: a spectroscopic insight in to nature and strength of interaction.

Journal of photochemistry and photobiology. B, Biology 20120301

Brassinin induces G1 phase arrest through increase of p21 and p27 by inhibition of the phosphatidylinositol 3-kinase signaling pathway in human colon cancer cells.

International journal of oncology 20120301

3,5-Disubstituted indole derivatives as selective human neuronal nitric oxide synthase (nNOS) inhibitors.

Bioorganic & medicinal chemistry letters 20120301

1H NMR spectroscopic identification of protonable sites in cryptolepines with C-11 substituents containing two amino functionalities.

Magnetic resonance in chemistry : MRC 20120301

Histamine H4 receptor ligands and their potential therapeutic applications: an update.

Expert opinion on therapeutic patents 20120301

Tris(tetra-butyl-ammonium) hexa-kis-(tert-butane-thiol-ato-κS)hepta-μ(3)-chlorido-μ(3)-sulfido-hexa-molybdate dihydrate.

Acta crystallographica. Section E, Structure reports online 20120301

(E)-3-Phenyl-2-(1-tosyl-1H-indol-3-ylcarbon-yl)acrylonitrile.

Acta crystallographica. Section E, Structure reports online 20120301

(Z)-3-(1H-Indol-3-yl)-2-(3,4,5-tri-methoxy-phen-yl)acrylonitrile.

Acta crystallographica. Section E, Structure reports online 20120301

1'-Methyl-4'-phenyl-dispiro-[chromane-3,3'-pyrrolidine-2',3''-indoline]-2,2''-dione.

Acta crystallographica. Section E, Structure reports online 20120301

l-Tryptophan 4-nitro-phenol tris-olvate.

Acta crystallographica. Section E, Structure reports online 20120301

In vitro antiproliferative effects of the indole alkaloid vallesiachotamine on human melanoma cells.

Archives of pharmacal research 20120301

DNA binding studies of Vinca alkaloids: experimental and computational evidence.

Natural product communications 20120301

Isolation, identification & characterization of Proteus penneri--a missed rare pathogen.

The Indian journal of medical research 20120301

[New-type electrodeless excilamp for advanced treatment on nitrogen-heterocyclic compounds (NHCs) in aqueous solution].

Huan jing ke xue= Huanjing kexue 20120301

Geographical variation in antibiotic-resistant Escherichia coli isolates from stool, cow-dung and drinking water.

International journal of environmental research and public health 20120301

Mild synthetic approach to novel indole-1-carbinols and preliminary evaluation of their cytotoxicity in hepatocarcinoma cells.

Archiv der Pharmazie 20120301

Copper-catalyzed domino intramolecular cyclization: a facile and efficient approach to polycyclic indole derivatives.

Organic & biomolecular chemistry 20120227

Brønsted acid mediated cyclization of enaminones. Rapid and efficient access to the tetracyclic framework of the Strychnos alkaloids.

Journal of natural products 20120224

Melodinines M-U, cytotoxic alkaloids from Melodinus suaveolens.

Journal of natural products 20120224

Synthesis and evaluation of the cytotoxicities of tetraindoles: observation that the 5-hydroxy tetraindole (SK228) induces G₂ arrest and apoptosis in human breast cancer cells.

Journal of medicinal chemistry 20120223

Adsorption and properties of aromatic amino acids on single-walled carbon nanotubes.

Nanoscale 20120221

Asymmetric substitutions of O-Boc-protected Morita-Baylis-Hillman adducts with pyrrole and indole derivatives.

Organic & biomolecular chemistry 20120221

Regioselective preferential nucleophilic addition of N-heterocycles onto haloarylalkynes over N-arylation of aryl halides.

Organic letters 20120217

ZraP is a periplasmic molecular chaperone and a repressor of the zinc-responsive two-component regulator ZraSR.

The Biochemical journal 20120215

Bioactive metabolites from Chaetomium globosum L18, an endophytic fungus in the medicinal plant Curcuma wenyujin.

Phytomedicine : international journal of phytotherapy and phytopharmacology 20120215

Isolation and structural elucidation of indole alkaloids from Geissospermum vellosii by mass spectrometry.

Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20120215

Molecular dynamics simulations of the interaction of glucose with imidazole in aqueous solution.

Carbohydrate research 20120215

Quinol derivatives as potential trypanocidal agents.

Bioorganic & medicinal chemistry 20120215

Rapid access to polycyclic indolines related to the stephacidin alkaloids using a radical cascade.

Chemical communications (Cambridge, England) 20120214

DNA duplexes and triplex-forming oligodeoxynucleotides incorporating modified nucleosides forming stable and selective triplexes.

Organic & biomolecular chemistry 20120207

Femto to millisecond observations of indole-based squaraine molecules photodynamics in solution.

Physical chemistry chemical physics : PCCP 20120207

Synthesis of 6-substituted 2-pyrrolyl and indolyl benzoxazoles by intramolecular O-arylation in photostimulated reactions.

The Journal of organic chemistry 20120203

Complete reaction mechanism of indoleamine 2,3-dioxygenase as revealed by QM/MM simulations.

The journal of physical chemistry. B 20120202

K252a induces anoikis-sensitization with suppression of cellular migration in Epstein-Barr virus (EBV)--associated nasopharyngeal carcinoma cells.

Investigational new drugs 20120201

Analysis of heterologous taxadiene production in K- and B-derived Escherichia coli.

Applied microbiology and biotechnology 20120201

Rasamsonia, a new genus comprising thermotolerant and thermophilic Talaromyces and Geosmithia species.

Antonie van Leeuwenhoek 20120201

Indigo biosynthesis by Comamonas sp. MQ.

Biotechnology letters 20120201

The synthesis and spectral properties of a stimuli-responsive D-π-A charge transfer dye based on indole donor and dicyanomethylene acceptor moiety.

Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20120201

In vitro permeation of mesembrine alkaloids from Sceletium tortuosum across porcine buccal, sublingual, and intestinal mucosa.

Planta medica 20120201

Indole alkaloids from Ervatamia chinensis.

Phytochemistry 20120201

Synthesis of 3,5-diaryl substituted indole derivatives and its selective iodide ion chemosensing.

Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20120201

Novel Cβ-Cγ bond cleavages of tryptophan-containing peptide radical cations.

Journal of the American Society for Mass Spectrometry 20120201

Indole alkaloids from marine-derived fungus Aspergillus sydowii SCSIO 00305.

The Journal of antibiotics 20120201

Pyrrole alkanoic acid derivatives as nuisance inhibitors of microsomal prostaglandin E2 synthase-1.

European journal of medicinal chemistry 20120201

Metabolism of cryptolepine and 2-fluorocryptolepine by aldehyde oxidase.

The Journal of pharmacy and pharmacology 20120201

2'-Hy-droxy-methyl-1'-(4-methyl-phen-yl)-2'-nitro-1',2',5',6',7',7a'-hexa-hydro-spiro-[indoline-3,3'-pyrrolizin]-2-one.

Acta crystallographica. Section E, Structure reports online 20120201

Evodiamide.

Acta crystallographica. Section E, Structure reports online 20120201

3,3-Dimethyl-1,2,3,4-tetra-hydro-cyclo-penta-[b]indole-1,2-dione (bruceolline E).

Acta crystallographica. Section E, Structure reports online 20120201

2-(4-Bromo-1H-indol-3-yl)acetonitrile.

Acta crystallographica. Section E, Structure reports online 20120201

DOGS: reaction-driven de novo design of bioactive compounds.

PLoS computational biology 20120201

Growth promotion of Xanthium italicum by application of rhizobacterial isolates of Bacillus aryabhattai in microcosm soil.

Journal of microbiology (Seoul, Korea) 20120201

Indolinones as promising scaffold as kinase inhibitors: a review.

Mini reviews in medicinal chemistry 20120201

Two new tryptamine derivatives, leptoclinidamide and (-)-leptoclinidamine B, from an Indonesian ascidian Leptoclinides dubius.

Marine drugs 20120201

[Melatonin agonist: a possible disease-modifying agent for Alzheimer's disease].

Nihon rinsho. Japanese journal of clinical medicine 20120201

Implementation of a design of experiments to study the influence of the background electrolyte on separation and detection in non-aqueous capillary electrophoresis-mass spectrometry.

Electrophoresis 20120201

Physical properties and molecular conformations of indole alkaloids and model protein interactions--theoretical vs. experimental study.

Natural product communications 20120201

Chemical and bioactivity evaluation of the bark of Neonauclea purpurea.

Natural product communications 20120201

Pharmacokinetic comparisons of rutaecarpine and evodiamine after oral administration of Wu-Chu-Yu extracts with different purities to rats.

Journal of ethnopharmacology 20120131

In vitro antiplasmodial activity of indole alkaloids from the stem bark of Geissospermum vellosii.

Journal of ethnopharmacology 20120131

Structure-activity relationship (SAR) development and discovery of potent indole-based inhibitors of the hepatitis C virus (HCV) NS5B polymerase.

Journal of medicinal chemistry 20120126

Surprising repair activities of nonpolar analogs of 8-oxoG expose features of recognition and catalysis by base excision repair glycosylases.

Journal of the American Chemical Society 20120125

Scaffold tailoring by a newly detected Pictet-Spenglerase activity of strictosidine synthase: from the common tryptoline skeleton to the rare piperazino-indole framework.

Journal of the American Chemical Society 20120125

A unified route to the welwitindolinone alkaloids: total syntheses of (-)-N-methylwelwitindolinone C isothiocyanate, (-)-N-methylwelwitindolinone C isonitrile, and (-)-3-hydroxy-N-methylwelwitindolinone C isothiocyanate.

Journal of the American Chemical Society 20120125

A detailed study of the intramolecular hydroamination of N-(ortho-alkynyl)aryl-N'-substituted trifluoroacetamidines and bromodifluoroacetamidines.

Organic & biomolecular chemistry 20120121

Differential patterns of dehydroabietic acid biotransformation by Nicotiana tabacum and Catharanthus roseus cells.

Journal of biotechnology 20120120

Synthetic studies toward lapidilectine-type Kopsia alkaloids.

Organic letters 20120120

Synthesis of new 4,5-dihydrofuranoindoles and their evaluation as HCV NS5B polymerase inhibitors.

Organic letters 20120120

Biochemical characterization of NotB as an FAD-dependent oxidase in the biosynthesis of notoamide indole alkaloids.

Journal of the American Chemical Society 20120118

Evaluation of donor and steric properties of anionic ligands on high valent transition metals.

Inorganic chemistry 20120116

Bis-cyclometalated iridium(III) complexes bearing ancillary guanidinate ligands. Synthesis, structure, and highly efficient electroluminescence.

Inorganic chemistry 20120116

Induction of glandular stomach cancers in Helicobacter pylori-infected Mongolian gerbils by 1-nitrosoindole-3-acetonitrile.

International journal of cancer 20120115

Pro-nerve growth factor induces autocrine stimulation of breast cancer cell invasion through tropomyosin-related kinase A (TrkA) and sortilin protein.

The Journal of biological chemistry 20120113

Contribution of dynamic and static quenchers for the study of protein conformation in ionic liquids by steady-state fluorescence spectroscopy.

The journal of physical chemistry. B 20120112

Peculiarity of methoxy group-substituted phenylhydrazones in Fischer indole synthesis.

Proceedings of the Japan Academy. Series B, Physical and biological sciences 20120111

5-HT2A/C receptors mediate the antipsychotic-like effects of alstonine.

Progress in neuro-psychopharmacology & biological psychiatry 20120110

Biochemical characterization of indole prenyltransferases: filling the last gap of prenylation positions by a 5-dimethylallyltryptophan synthase from Aspergillus clavatus.

The Journal of biological chemistry 20120106

Total synthesis of hapalindoles J and U.

The Journal of organic chemistry 20120106

Stereoselective synthesis of brevianamide E.

Organic letters 20120106

Stereocontrolled synthesis of an indole moiety of sespendole and stereochemical assignment of the side chain.

Organic letters 20120106

Synthesis of highly functionalized chiral 3,3'-disubstituted oxindoles via an organocatalytic enantioselective Michael addition of nitroalkanes to indolylidenecyanoacetates.

Organic letters 20120106

A ridge walk between reaction modes: an unprecedented Pd-catalyzed domino sequence of diynyl-substituted bromoarenes.

Organic letters 20120106

Syntheses of strychnine, norfluorocurarine, dehydrodesacetylretuline, and valparicine enabled by intramolecular cycloadditions of Zincke aldehydes.

The Journal of organic chemistry 20120106

Green chemistry: solvent- and metal-free Prins cyclization. Application to sequential reactions.

Chemical communications (Cambridge, England) 20120104

Synthetic quorum-sensing circuit to control consortial biofilm formation and dispersal in a microfluidic device.

Nature communications 20120103

Exploiting the electrophilic properties of indole intermediates: new options in designing asymmetric reactions.

Angewandte Chemie (International ed. in English) 20120102

In vivo BDNF modulation of hippocampal mossy fiber plasticity induced by high frequency stimulation.

Hippocampus 20120101

Description of Christensenella minuta gen. nov., sp. nov., isolated from human faeces, which forms a distinct branch in the order Clostridiales, and proposal of Christensenellaceae fam. nov.

International journal of systematic and evolutionary microbiology 20120101

Two new indole alkaloids, 2-(3,3-dimethylprop-1-ene)-costaclavine and 2-(3,3-dimethylprop-1-ene)-epicostaclavine, from the marine-derived fungus Aspergillus fumigatus.

Journal of natural medicines 20120101

HPLC analysis of oxindole alkaloids in Uncaria tomentosa: sample preparation and analysis optimisation by factorial design.

Phytochemical analysis : PCA 20120101

Exercise and melatonin in humans: reciprocal benefits.

Journal of pineal research 20120101

Synthesis and comparison of antioxidant properties of indole-based melatonin analogue indole amino Acid derivatives.

Chemical biology & drug design 20120101

GABA(A) receptor blockade enhances memory consolidation by increasing hippocampal BDNF levels.

Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20120101

Alstonia scholaris R. Br. Significantly Inhibits Retinoid-Induced Skin Irritation In Vitro and In Vivo.

Evidence-based complementary and alternative medicine : eCAM 20120101

Indole prenylation in alkaloid synthesis.

Topics in current chemistry 20120101

Synthetic studies on amaryllidaceae and other terrestrially derived alkaloids.

Topics in current chemistry 20120101

Tumor angiogenesis as a target for dietary cancer prevention.

Journal of oncology 20120101

Natural products from ethnodirected studies: revisiting the ethnobiology of the zombie poison.

Evidence-based complementary and alternative medicine : eCAM 20120101

Biosynthesis and emission of insect herbivory-induced volatile indole in rice.

Phytochemistry 20120101

Early postnatal exposure of mice to side-steam tobacco smoke increases neuropeptide Y in lung.

American journal of physiology. Lung cellular and molecular physiology 20120101

Alternative splicing in oncogenic kinases: from physiological functions to cancer.

Journal of nucleic acids 20120101

Atrial natriuretic peptide enhances microvascular albumin permeability by the caveolae-mediated transcellular pathway.

Cardiovascular research 20120101

Indole alkaloids from Muntafara sessilifolia with antiplasmodial and cytotoxic activities.

Phytochemistry 20120101

Identification of a novel resistance mutation for benzimidazole inhibitors of the HCV RNA-dependent RNA polymerase.

Antiviral research 20120101

Indole RSK inhibitors. Part 2: optimization of cell potency and kinase selectivity.

Bioorganic & medicinal chemistry letters 20120101

Aminobenzoates as building blocks for natural product assembly lines.

Natural product reports 20120101

Electrochemical oxidation of nitrogen-heterocyclic compounds at boron-doped diamond electrode.

Chemosphere 20120101

Tryptophan side chain conformers monitored by NMR and time-resolved fluorescence spectroscopies.

Proteins 20120101

Indole RSK inhibitors. Part 1: discovery and initial SAR.

Bioorganic & medicinal chemistry letters 20120101

II. Novel HCV NS5B polymerase inhibitors: discovery of indole C2 acyl sulfonamides.

Bioorganic & medicinal chemistry letters 20120101

Isorhynchophylline, a natural alkaloid, promotes the degradation of alpha-synuclein in neuronal cells via inducing autophagy.

Autophagy 20120101

A novel, simple, and sensitive colorimetric method to determine aromatic amino acid aminotransferase activity using the Salkowski reagent.

Folia microbiologica 20120101

Splicing programs and cancer.

Journal of nucleic acids 20120101

Discovery of inhibitors and substrates of brassinin hydrolase: Probing selectivity with dithiocarbamate bioisosteres.

Bioorganic & medicinal chemistry 20120101

A photophysical study of the α-carboline (1-azacarbazole) aggregation process.

Photochemistry and photobiology 20120101

Principles of psychoneuroendocrinoimmunotherapy of cancer.

Immunotherapy 20120101

Conjugation of a 3-(1H-phenanthro[9,10-d]imidazol-2-yl)-1H-indole intercalator to a triplex oligonucleotide and to a three-way junction.

Bioorganic & medicinal chemistry 20120101

The indolic diet-derivative, 3,3'-diindolylmethane, induced apoptosis in human colon cancer cells through upregulation of NDRG1.

Journal of biomedicine & biotechnology 20120101

Indoxyl sulfate induces nephrovascular senescence.

Journal of renal nutrition : the official journal of the Council on Renal Nutrition of the National Kidney Foundation 20120101

A nexus of progression of chronic kidney disease: tryptophan, profibrotic cytokines, and charcoal.

Journal of renal nutrition : the official journal of the Council on Renal Nutrition of the National Kidney Foundation 20120101

Alternative Splicing of Fibroblast Growth Factor Receptor IgIII Loops in Cancer.

Journal of nucleic acids 20120101

New acetylcholinesterase inhibitors for Alzheimer's disease.

International journal of Alzheimer's disease 20120101

Development of new methods in organic synthesis and their applications to the synthesis of biologically interesting natural products.

Chemical & pharmaceutical bulletin 20120101

The role of indoleamine 2, 3 dioxygenase in regulating host immunity to leishmania infection.

Journal of biomedical science 20120101

The 5 alpha-reductase isozyme family: a review of basic biology and their role in human diseases.

Advances in urology 20120101

Using hydrophilic ionic liquid, [bmim]BF4-ethylene glycol system as a novel media for the rapid synthesis of copper nanoparticles.

PloS one 20120101

Functional evolution of duplicated odorant-binding protein genes, Obp57d and Obp57e, in Drosophila.

PloS one 20120101

Genome-wide association scan and phased haplotype construction for quantitative trait loci affecting boar taint in three pig breeds.

BMC genomics 20120101

A modular library of small molecule signals regulates social behaviors in Caenorhabditis elegans.

PLoS biology 20120101

New signaling chemicals spur worms to seek company.

PLoS biology 20120101

Global analysis of small molecule binding to related protein targets.

PLoS computational biology 20120101

Induction of VMAT-1 and TPH-1 expression induces vesicular accumulation of serotonin and protects cells and tissue from cooling/rewarming injury.

PloS one 20120101

Herbivore-mediated effects of glucosinolates on different natural enemies of a specialist aphid.

Journal of chemical ecology 20120101

5',11'-Dihydro-dispiro-[cyclo-hexane-1,6'-indolo[3,2-b]carbazole-12',1''-cyclo-hexa-ne].