Glycinamide, L-tyrosyl-D-alanyl-L-phenylalanyl-L-α-glutamyl-L-valyl-L-valyl-
| Title | Journal |
|---|---|
| Transport of the synthetic opioid peptide DADLE ([D-Ala2,D-Leu5]-enkephalin) in neuronal cells. | Journal of pharmaceutical sciences 20120101 |
| [Effect of opioid peptides on oxygen-dependent microbicidity of peripheral blood neutrophils]. | Fiziologiia cheloveka 20120101 |
| Activation of spinal mu- and delta-opioid receptors potently inhibits substance P release induced by peripheral noxious stimuli. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20110914 |
| Spinal activation of delta opioid receptors alleviates cancer-related bone pain. | Neuroscience 20110602 |
| Evidence for two different broad-specificity oligopeptide transporters in intestinal cell line Caco-2 and colonic cell line CCD841. | American journal of physiology. Cell physiology 20110601 |
| Transport of hepcidin, an iron-regulatory peptide hormone, into retinal pigment epithelial cells via oligopeptide transporters and its relevance to iron homeostasis. | Biochemical and biophysical research communications 20110211 |
| Opioid peptide deltorphin II simulates the cardioprotective effect of ischemic preconditioning: role of δ₂-opioid receptors, protein kinase C, and K(ATP) channels. | Bulletin of experimental biology and medicine 20101001 |
| Consequences of opioid receptor mutation on actions of univalent and bivalent kappa and delta ligands. | Psychopharmacology 20100601 |
| Protein kinase C mediates the synergistic interaction between agonists acting at alpha2-adrenergic and delta-opioid receptors in spinal cord. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20091021 |
| Regulation of interleukin-1beta and interleukin-8 production by agonists of mu and delta opiate receptors in vitro. | Neuroscience and behavioral physiology 20090701 |
| Differential noxious and motor tolerance of chronic delta opioid receptor agonists in rodents. | Neuroscience 20090630 |
| Activation of peripheral delta2 opioid receptors increases cardiac tolerance to ischemia/reperfusion injury Involvement of protein kinase C, NO-synthase, KATP channels and the autonomic nervous system. | Life sciences 20090508 |
| Functional identification of a novel transport system for endogenous and synthetic opioid peptides in the rabbit conjunctival epithelial cell line CJVE. | Pharmaceutical research 20090501 |
| Comparison with naloxone of two dynorphin A analogues with K- and delta-opioid antagonist activity. | Medicinal chemistry (Shariqah (United Arab Emirates)) 20090101 |
| Behavioral consequences of delta-opioid receptor activation in the periaqueductal gray of morphine tolerant rats. | Neural plasticity 20090101 |
| Design, data analysis, and simulation of in vitro drug transport kinetic experiments using a mechanistic in vitro model. | Drug metabolism and disposition: the biological fate of chemicals 20081201 |
| Removing TRPV1-expressing primary afferent neurons potentiates the spinal analgesic effect of delta-opioid agonists on mechano-nociception. | Neuropharmacology 20080801 |
| [Regulation of IL-1beta and IL-8 production by mu-, delta-opiate receptors agonists in vitro]. | Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova 20080701 |
| Distinct inhibition of voltage-activated Ca2+ channels by delta-opioid agonists in dorsal root ganglion neurons devoid of functional T-type Ca2+ currents. | Neuroscience 20080602 |
| Membrane partitioning of various delta-opioid receptor forms before and after agonist activations: the effect of cholesterol. | Biochimica et biophysica acta 20080601 |
| [Analysis of central mechanisms involved in gastric mucosal integrity]. | Neuropsychopharmacologia Hungarica : a Magyar Pszichofarmakologiai Egyesulet lapja = official journal of the Hungarian Association of Psychopharmacology 20080601 |
| Stimulation of Na+/Cl--coupled opioid peptide transport system in SK-N-SH cells by L-kyotorphin, an endogenous substrate for H+-coupled peptide transporter PEPT2. | Drug metabolism and pharmacokinetics 20080101 |
| Essential role of mu opioid receptor in the regulation of delta opioid receptor-mediated antihyperalgesia. | Neuroscience 20071219 |
| Trafficking of preassembled opioid mu-delta heterooligomer-Gz signaling complexes to the plasma membrane: coregulation by agonists. | Biochemistry 20071113 |
| Spinal administration of a delta opioid receptor agonist attenuates hyperalgesia and allodynia in a rat model of neuropathic pain. | European journal of pain (London, England) 20070801 |
| Mechanisms responsible for the enhanced antinociceptive effects of micro-opioid receptor agonists in the rostral ventromedial medulla of male rats with persistent inflammatory pain. | The Journal of pharmacology and experimental therapeutics 20070801 |
| Quantitative evaluation of human delta opioid receptor desensitization using the operational model of drug action. | Molecular pharmacology 20070501 |
| Differential modulation of sodium- and chloride-dependent opioid peptide transport system by small nonopioid peptides and free amino acids. | The Journal of pharmacology and experimental therapeutics 20070401 |
| Effects of opioid subtypes on detrusor overactivity in rats with cerebral infarction. | International journal of urology : official journal of the Japanese Urological Association 20070301 |
| Cholesterol reduction by methyl-beta-cyclodextrin attenuates the delta opioid receptor-mediated signaling in neuronal cells but enhances it in non-neuronal cells. | Biochemical pharmacology 20070215 |
| Morphine priming in rats with chronic inflammation reveals a dichotomy between antihyperalgesic and antinociceptive properties of deltorphin. | Neuroscience 20070105 |
| Behavioural and morphological evidence for the involvement of glial cell activation in delta opioid receptor function: implications for the development of opioid tolerance. | Molecular pain 20070101 |
| Peptide-labeled quantum dots for imaging GPCRs in whole cells and as single molecules. | Bioconjugate chemistry 20070101 |
| Repeated delta1-opioid receptor stimulation reduces delta2-opioid receptor responses in the SA node. | American journal of physiology. Heart and circulatory physiology 20061101 |
| Alkylation of opioid receptors by 5'-naltrindole-isothiocyanate injected into the nucleus accumbens of rats: receptor selectivity and anatomical diffusion. | Synapse (New York, N.Y.) 20061001 |
| Mu-delta opioid receptor functional interaction: Insight using receptor-G protein fusions. | The Journal of pharmacology and experimental therapeutics 20060801 |
| Reduction of lipopolysaccharide-induced interleukin-6 production by the kappa opioid U50,488 in a mouse monocyte-like cell line. | International immunopharmacology 20060601 |
| Effects of mu, kappa or delta opioids administered by pellet or pump on oral Salmonella infection and gastrointestinal transit. | European journal of pharmacology 20060318 |
| dextro- and levo-morphine attenuate opioid delta and kappa receptor agonist produced analgesia in mu-opioid receptor knockout mice. | European journal of pharmacology 20060215 |
| 24-hour pretreatment with delta opioid enhances survival from hemorrhagic shock. | Academic emergency medicine : official journal of the Society for Academic Emergency Medicine 20060201 |
| Peptidic delta opioid receptor agonists produce antidepressant-like effects in the forced swim test and regulate BDNF mRNA expression in rats. | Brain research 20060119 |
| A role for the distal carboxyl tails in generating the novel pharmacology and G protein activation profile of mu and delta opioid receptor hetero-oligomers. | The Journal of biological chemistry 20051118 |
| Morphine promotes phosphorylation of the human delta-opioid receptor at serine 363. | European journal of pharmacology 20050920 |
| Subpicomolar sensing of delta-opioid receptor ligands by molecular-imprinted polymers using plasmon-waveguide resonance spectroscopy. | Analytical chemistry 20050415 |
| Spinal G-protein-gated potassium channels contribute in a dose-dependent manner to the analgesic effect of mu- and delta- but not kappa-opioids. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20050406 |
| Polymorphisms in human organic anion-transporting polypeptide 1A2 (OATP1A2): implications for altered drug disposition and central nervous system drug entry. | The Journal of biological chemistry 20050311 |
| A Tyr-W-MIF-1 analog containing D-Pro2 acts as a selective mu2-opioid receptor antagonist in the mouse. | The Journal of pharmacology and experimental therapeutics 20050301 |
| Antinociception depends on the presence of G protein gamma2-subunits in brain. | European journal of pharmacology 20050131 |
| The non-peptidic delta opioid receptor agonist TAN-67 enhances dopamine efflux in the nucleus accumbens of freely moving rats via a mechanism that involves both glutamate and free radicals. | Neuroscience 20050101 |
| delta-opioid receptor-mediated actions on rostral ventromedial medulla neurons. | Neuroscience 20050101 |
| An efficient intrathecal delivery of small interfering RNA to the spinal cord and peripheral neurons. | Molecular pain 20050101 |
| Intrahypothalamic injection of deltorphin-II alters body temperature in rats. | Brain research 20040903 |
| Morphine-induced changes in delta opioid receptor trafficking are linked to somatosensory processing in the rat spinal cord. | The Journal of neuroscience : the official journal of the Society for Neuroscience 20040616 |
| Role of mu- and delta-opioid receptors in the nucleus accumbens in turning behaviour of rats. | Neuropharmacology 20040601 |
| Exploring deltorphin II binding to the third extracellular loop of the delta-opioid receptor. | The Journal of biological chemistry 20040514 |
| Deltorphin II enhances extracellular levels of dopamine in the nucleus accumbens via opioid receptor-independent mechanisms. | European journal of pharmacology 20040426 |
| The delta agonists DPDPE and deltorphin II recruit predominantly mu receptors to produce thermal analgesia: a parallel study of mu, delta and combinatorial opioid receptor knockout mice. | The European journal of neuroscience 20040401 |
| 2',6'-dimethylphenylalanine (Dmp) can mimic the N-terminal Tyr in opioid peptides. | Biological & pharmaceutical bulletin 20040201 |
| Identification of a novel Na+- and Cl--coupled transport system for endogenous opioid peptides in retinal pigment epithelium and induction of the transport system by HIV-1 Tat. | The Biochemical journal 20031001 |
| Pharmacological characterization of a 7-benzylidenenaltrexone-preferring opioid receptor in porcine ileal submucosa. | British journal of pharmacology 20031001 |
| Long-term effects on brain opioid and opioid receptor like-1 receptors after short periods of maternal separation in rats. | Neuroscience letters 20030724 |
| Buprenorphine blocks epsilon- and micro-opioid receptor-mediated antinociception in the mouse. | The Journal of pharmacology and experimental therapeutics 20030701 |
| Endomorphin-2, deltorphin II and their analogs suppress formalin-induced nociception and c-Fos expression in the rat spinal cord. | Life sciences 20030613 |
| Cardiac enkephalins interrupt vagal bradycardia via delta 2-opioid receptors in sinoatrial node. | American journal of physiology. Heart and circulatory physiology 20030501 |
| Identity of the putative delta1-opioid receptor as a delta-kappa heteromer in the mouse spinal cord. | European journal of pharmacology 20030425 |
| Design of novel chimeric melanotropin-deltorphin analogues. Discovery of the first potent human melanocortin 1 receptor antagonist. | Journal of medicinal chemistry 20030227 |
| Functional interactions between delta- and mu-opioid receptors in rat thermoregulation. | European journal of pharmacology 20030101 |
| Identification of a novel human organic anion transporting polypeptide as a high affinity thyroxine transporter. | Molecular endocrinology (Baltimore, Md.) 20021001 |
| The distribution of the anti-HIV drug, 2'3'-dideoxycytidine (ddC), across the blood-brain and blood-cerebrospinal fluid barriers and the influence of organic anion transport inhibitors. | Journal of neurochemistry 20020201 |
| alpha(2C)-Adrenergic receptors mediate spinal analgesia and adrenergic-opioid synergy. | The Journal of pharmacology and experimental therapeutics 20020101 |
| Localization of organic anion transporting polypeptide 4 (Oatp4) in rat liver and comparison of its substrate specificity with Oatp1, Oatp2 and Oatp3. | Pflugers Archiv : European journal of physiology 20011101 |
| Dexamethasone modulates hypotension induced by opioids in anaesthetised rats. | European journal of pharmacology 20011026 |
| The role of backbone conformation in deltorphin II binding: a QSAR study of new analogues modified in the 5-, 6-positions of the address domain. | Bioorganic & medicinal chemistry 20011001 |
| Administration of mu-, kappa- or delta2-receptor agonists via osmotic minipumps suppresses murine splenic antibody responses. | International immunopharmacology 20011001 |
| Fetal alveolar epithelial cells contain [D-Ala(2)]-deltorphin I-like immunoreactivity: delta- and mu-opiate receptors mediate opposite effects in developing lung. | American journal of respiratory cell and molecular biology 20011001 |
| Morphine-induced in vivo release of spinal cholecystokinin is mediated by delta-opioid receptors--effect of peripheral axotomy. | Journal of neurochemistry 20010701 |
| Supraspinal delta- and mu-opioid receptors mediate gastric mucosal protection in the rat. | The Journal of pharmacology and experimental therapeutics 20010601 |
| In vivo pharmacological characterization of SoRI 9409, a nonpeptidic opioid mu-agonist/delta-antagonist that produces limited antinociceptive tolerance and attenuates morphine physical dependence. | The Journal of pharmacology and experimental therapeutics 20010501 |
| Respiratory function in adult mice lacking the mu-opioid receptor: role of delta-receptors. | The European journal of neuroscience 20010501 |
| Activity of mu- and delta-opioid agonists in vas deferens from mice deficient in MOR gene. | British journal of pharmacology 20010401 |
| The role of delta-opioid receptor subtypes in neuropathic pain. | European journal of pharmacology 20010309 |
| Organic anion-transporting polypeptide B (OATP-B) and its functional comparison with three other OATPs of human liver. | Gastroenterology 20010201 |
| Dexamethasone blocking effects on mu- and delta-opioid-induced seizures involves kappa-opioid activity in the rabbit. | Neuropsychobiology 20010101 |
| Effect of opioids on oral Salmonella infection and immune function. | Advances in experimental medicine and biology 20010101 |
| Deltorphin II analogues with 6-hydroxy-2-aminotetralin-2-carboxylic acid in position 1. | Journal of medicinal chemistry 20000406 |
| A new opioid peptide predicted from cloned cDNAs from skin of Pachymedusa dacnicolor and Agalychnis annae. | FEBS letters 19980605 |
| Competitive and non-competitive NMDA antagonists block the development of antinociceptive tolerance to morphine, but not to selective mu or delta opioid agonists in mice. | Pain 19961201 |
| Nitric oxide modulates neuropeptide Y regulation of ion transport in mouse ileum. | The Journal of pharmacology and experimental therapeutics 19960701 |
| Inhibition of adenylyl cyclase activity by the cholecystokinin analog SNF 9007 in neuroblastoma x glioma NG108-15 hybrid cells. | Regulatory peptides 19960116 |
| Differential desensitization of mu- and delta- opioid receptors in selected neural pathways following chronic morphine treatment. | British journal of pharmacology 19960101 |
| Comparative conformational analyses of mu-selective dermorphin and delta-selective deltorphin-II in aqueous solution by 1H-NMR spectroscopy. | International journal of peptide and protein research 19940901 |
| Differential regulation of adenylyl cyclase activity by mu and delta opioids in rat caudate putamen and nucleus accumbens. | The Journal of pharmacology and experimental therapeutics 19931001 |
| In vitro potency, affinity and agonist efficacy of highly selective delta opioid receptor ligands. | The Journal of pharmacology and experimental therapeutics 19930801 |
| Agonist and antagonist profiles of [D-Ala2,Glu4]deltorphin and its [Cys4]- and [Ser4]-substituted derivatives: further evidence of opioid delta receptor multiplicity. | The Journal of pharmacology and experimental therapeutics 19930501 |
| Antidiarrheal and colonic antipropulsive effects of spinal and supraspinal administration of the natural delta opioid receptor agonist, [D-Ala2]deltorphin II, in the rat. | European journal of pharmacology 19920721 |
| Long-term sensitization to the activation of cerebral delta-opioid receptors by the deltorphin Tyr-D-Ala-Phe-Glu-Val-Val-Gly-NH2 in rats exposed to morphine. | Proceedings of the National Academy of Sciences of the United States of America 19920501 |
| Influence of peptidase inhibitors on the apparent agonist potency of delta selective opioid peptides in vitro. | Life sciences 19910101 |